Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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DPI-3290
CAS:<p>DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent</p>Fórmula:C30H34FN3O2Pureza:98%Forma y color:SolidPeso molecular:487.61Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Fórmula:C34H48N6O10Pureza:98%Forma y color:SolidPeso molecular:700.78Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Fórmula:C30H34FN5O5Pureza:98%Forma y color:SolidPeso molecular:563.62Icalcaprant
CAS:<p>Icalcaprant is a kappa-opioid receptor antagonist [1].</p>Fórmula:C23H26N4O3Pureza:98%Forma y color:SolidPeso molecular:406.48μ opioid receptor agonist 1
CAS:<p>μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that can</p>Fórmula:C26H38N4OForma y color:SolidPeso molecular:422.61Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Fórmula:C38H43ClN4O6Pureza:98%Forma y color:SolidPeso molecular:687.22ICI 204448
CAS:<p>ICI 204448 is a potent and peripherally selective κ-opioid agonist.</p>Fórmula:C23H26Cl2N2O4Forma y color:SolidPeso molecular:465.37N-Benzylnaltrindole hydrochloride
CAS:<p>δ2 opioid receptor antagonist</p>Fórmula:C33H33ClN2O3Pureza:98%Forma y color:SolidPeso molecular:541.08Trap-101 hydrochloride
CAS:<p>nociceptin/orphanin FQ (NOP) receptor antagonist</p>Fórmula:C24H36ClN3O2Pureza:98%Forma y color:SolidPeso molecular:434.02ADL-08-0011
CAS:<p>ADL-08-0011 is an metabolite of alvimopan.</p>Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.49FK 33-824
CAS:<p>FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.</p>Fórmula:C29H41N5O7SPureza:98%Forma y color:SolidPeso molecular:603.73J-113397
CAS:<p>J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).</p>Fórmula:C24H37N3O2Pureza:98%Forma y color:SolidPeso molecular:399.57BNTX
CAS:<p>BNTX (7-Benzylidenenaltrexone) is a selective δ1-opioid receptor antagonist. It competitively counteracts the antisecretory effects of DPDPE, Deltorphin 2, and DAMGO. BNTX is applicable in research focused on antinociceptive effects.</p>Fórmula:C27H27NO4Forma y color:SolidPeso molecular:429.508Mu opioid receptor antagonist 4
<p>Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki & EC50: 0.38 nM; useful for OUD research.</p>Fórmula:C25H28N2O4SForma y color:SolidPeso molecular:452.57SB-612111 hydrochloride
<p>SB-612111 is a potent ORL-1 antagonist, with high affinity (Ki: 0.33 nM) and µ-receptor activity (Ki: 57.6 nM), blocking Nociceptin-induced pain.</p>Fórmula:C24H30Cl3NOForma y color:SolidPeso molecular:454.86RX 809055AX
CAS:<p>RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.</p>Fórmula:C29H29ClN2O4Forma y color:SolidPeso molecular:505SC13
CAS:<p>SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.</p>Fórmula:C26H30N2O5Forma y color:SolidPeso molecular:450.53BU09059
CAS:<p>BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).</p>Fórmula:C28H37N3O5Pureza:98%Forma y color:SolidPeso molecular:495.61Mu opioid receptor antagonist 3
<p>Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.</p>Fórmula:C25H28N2O4SForma y color:SolidPeso molecular:452.57Allyphenyline oxalate
CAS:<p>The pKi values of Allyphenyline oxalate (compound 9) for the α2-adrenergic receptor subtypes α2A, α2B, and α2C are 7.24, 6.47, and 7.07, respectively.</p>Fórmula:C16H20N2O5Forma y color:SolidPeso molecular:320.34
