Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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BMS-986121
CAS:<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Fórmula:C15H9Cl2N3O2SPureza:99.67%Forma y color:SolidPeso molecular:366.22Asimadoline
CAS:<p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54LY2940094 tartrate
CAS:<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Fórmula:C26H29ClF2N4O8SForma y color:SolidPeso molecular:631.04Naloxegol (NKTR-118)
CAS:<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Fórmula:C34H53NO11Forma y color:SolidPeso molecular:651.78b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Fórmula:C25H31N3O7Pureza:98.99%Forma y color:SolidPeso molecular:485.53BMS986187
CAS:<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Fórmula:C31H34O4Pureza:99.09%Forma y color:SolidPeso molecular:470.6N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Fórmula:C30H39N5O8Pureza:>99.99%Forma y color:SolidPeso molecular:597.66Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Fórmula:C51H73N15O11Pureza:98.59%Forma y color:SolidPeso molecular:1072.22Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Fórmula:C21H26ClNO3Pureza:98% - 99.85%Forma y color:SolidPeso molecular:375.89Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Fórmula:C19H23NO4Pureza:99.02% - 99.73%Forma y color:White PowderPeso molecular:329.39Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Fórmula:C51H68N12O13Pureza:99.66%Forma y color:SolidPeso molecular:1057.16Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Fórmula:C31H40F3N5O9Pureza:98.79%Forma y color:SolidPeso molecular:683.67EST73502 hydrochloride
CAS:<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Fórmula:C19H27ClF2N2O2Forma y color:SolidPeso molecular:388.88Naloxegol oxalate
CAS:<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Fórmula:C36H55NO15Pureza:99.67% - >99.99%Forma y color:SolidPeso molecular:741.83Corydaline
CAS:<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Fórmula:C22H27NO4Pureza:98.97% - 99.86%Forma y color:SolidPeso molecular:369.45GR 89696 free base
CAS:<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Fórmula:C19H25Cl2N3O3Forma y color:SolidPeso molecular:414.33Sec-O-Glucosylhamaudol
CAS:<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Fórmula:C21H26O10Pureza:99.79%Forma y color:SolidPeso molecular:438.43Nociceptin
CAS:<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Fórmula:C79H129N27O22Pureza:99.35%Forma y color:SolidPeso molecular:1809.04Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Fórmula:C63H101F3N22O17Pureza:97.64%Forma y color:SolidPeso molecular:1495.61MCOPPB
CAS:<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Fórmula:C26H40N4Forma y color:SolidPeso molecular:408.62
