
Receptor de glucagón
Los receptores de glucagón son GPCR que median los efectos del glucagón, una hormona involucrada en la regulación de la homeostasis de la glucosa al promover la descomposición del glucógeno y la liberación de glucosa desde el hígado. Estos receptores son cruciales en la gestión de los niveles de azúcar en sangre y son de particular interés en el estudio de la diabetes y los trastornos metabólicos. Los antagonistas de los receptores de glucagón se están explorando como posibles tratamientos para la hiperglucemia en la diabetes tipo 2. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de glucagón de alta calidad para apoyar su investigación en endocrinología, diabetes y regulación metabólica.
Se han encontrado 164 productos de "Receptor de glucagón"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Albiglutide TFA (782500-75-8 free base)
<p>Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).</p>Fórmula:C150H225F3N40O47Pureza:>99.99%Forma y color:SolidPeso molecular:3397.63Teduglutide acetate
<p>Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy.</p>Fórmula:C166H256N44O56SPureza:97.39%Forma y color:SoildPeso molecular:3812.13ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Fórmula:C23H31N3O3SPureza:99.75%Forma y color:SolidPeso molecular:429.58Exenatide
CAS:<p>Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.</p>Fórmula:C186H286N50O62SPureza:99.42%Forma y color:SolidPeso molecular:4247Glucagon-like peptide 1 (1-37), human acetate
<p>Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.</p>Pureza:98%Forma y color:LiquidPeso molecular:N/ACotadutide acetate
<p>Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.</p>Fórmula:C169H256N42O57Pureza:98.28%Forma y color:SolidPeso molecular:3788.14GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Fórmula:C151H228N40O47Pureza:98.89%Forma y color:SolidPeso molecular:3355.67Avexitide
CAS:<p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>Fórmula:C149H234N40O47SPureza:98% - 99.65%Forma y color:SolidPeso molecular:3369.76GLP-1 receptor agonist 9
CAS:<p>1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.</p>Fórmula:C32H31ClFN3O5Pureza:98%Forma y color:SolidPeso molecular:592.06PF-06291874
CAS:<p>PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.</p>Fórmula:C26H28F3N3O4Pureza:99.12% - 99.27%Forma y color:SolidPeso molecular:503.51NNC-0640
CAS:<p>NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.</p>Fórmula:C29H31N7O4SPureza:97.04%Forma y color:SolidPeso molecular:573.67Glucagon receptor antagonists-5
CAS:<p>Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.</p>Fórmula:C30H29ClF3N3O3Pureza:98%Forma y color:SolidPeso molecular:572.02BAY-27-9955
CAS:<p>BAY-27-9955 is a glucagon receptor antagonist.</p>Fórmula:C23H31FOForma y color:SolidPeso molecular:342.49(R)-V-0219
<p>(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.</p>Fórmula:C20H25F3N4O2Forma y color:SolidPeso molecular:410.43GLP-1R agonist 1
CAS:<p>GLP-1R agonist 1, an imidazole derivative and potent GLP-1R activator, may aid diabetes research.</p>Fórmula:C32H29ClFN3O5Forma y color:SolidPeso molecular:590.04Glucagon receptor antagonists-2
CAS:<p>Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.</p>Fórmula:C22H30FNO2Pureza:98%Forma y color:SolidPeso molecular:359.48MS012
CAS:<p>MS012 is a Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase (Kd = 46 ± 15 nM).</p>Fórmula:C22H35N5O2Forma y color:SolidPeso molecular:401.55(S)-V-0219
<p>(S)-V-0219: oral, GLP-1R PAM, boosts calcium in hGLP-1R HEK cells, lowers glucose, curbs hunger in mice.</p>Fórmula:C20H25F3N4O2Forma y color:SolidPeso molecular:410.43GCGR antagonist 2
CAS:<p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>Fórmula:C28H26N4O2Forma y color:SolidPeso molecular:450.53NNC 92-1687
CAS:<p>NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.</p>Fórmula:C15H12N2O3SPureza:98.70% - 99.70%Forma y color:SolidPeso molecular:300.33

