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Receptor de glucagón

Receptor de glucagón

Los receptores de glucagón son GPCR que median los efectos del glucagón, una hormona involucrada en la regulación de la homeostasis de la glucosa al promover la descomposición del glucógeno y la liberación de glucosa desde el hígado. Estos receptores son cruciales en la gestión de los niveles de azúcar en sangre y son de particular interés en el estudio de la diabetes y los trastornos metabólicos. Los antagonistas de los receptores de glucagón se están explorando como posibles tratamientos para la hiperglucemia en la diabetes tipo 2. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de glucagón de alta calidad para apoyar su investigación en endocrinología, diabetes y regulación metabólica.

Se han encontrado 164 productos de "Receptor de glucagón"

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  • HAEGTFTSDVS

    CAS:
    <p>HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.</p>
    Fórmula:C48H71N13O20
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1150.18
  • Pal-Glu(OSu)-OH

    CAS:
    <p>Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.</p>
    Fórmula:C25H42N2O7
    Forma y color:Solid
    Peso molecular:482.618
  • TT-OAD2

    CAS:
    <p>TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.</p>
    Fórmula:C50H49Cl4N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:929.75
  • GLP-2(1-33)(human)

    CAS:
    <p>GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.</p>
    Fórmula:C165H254N44O55S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3766.19
  • HAEGTFT

    CAS:
    <p>HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.</p>
    Fórmula:C33H47N9O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:761.78
  • GLP-1R agonist 29


    <p>GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.</p>
    Forma y color:Odour Solid
  • GLP-1 moiety from Dulaglutide


    <p>GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist.</p>
    Fórmula:C149H221N37O49
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3314.62
  • Apraglutide

    CAS:
    <p>Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.</p>
    Fórmula:C172H263N43O52
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3765.25
  • Dulaglutide

    CAS:
    <p>Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).</p>
    Forma y color:Solid
  • Taspoglutide

    CAS:
    <p>Taspoglutide is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist(EC50 value of 0.06 nM),and for treatment of type 2 diabetes</p>
    Fórmula:C152H232N40O45
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3339.763
  • LSN3160440

    CAS:
    <p>LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.</p>
    Fórmula:C27H27Cl2N3O
    Forma y color:Solid
    Peso molecular:480.43
  • GLP-1 receptor agonist 13


    <p>Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].</p>
    Fórmula:C25H23ClF2N6O
    Forma y color:Solid
    Peso molecular:496.94
  • Secretin, porcine

    CAS:
    <p>Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.</p>
    Fórmula:C130H220N44O41·xC2H4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:N/A
  • TT-OAD2 free base

    CAS:
    <p>TT-OAD2 free base, a non-peptide GLP-1 receptor agonist, can treat diabetes; has an EC50 of 5 nM.</p>
    Fórmula:C50H47Cl2N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:856.83
  • Tirzepatide

    CAS:
    <p>Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.</p>
    Fórmula:C225H348N48O68
    Pureza:99.52% - 99.99%
    Forma y color:Solid
    Peso molecular:4813.45
  • {Val1}-Exendin-3/4


    <p>{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.</p>
    Fórmula:NA
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3241.7
  • GLP-1R agonist 14

    CAS:
    <p>GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].</p>
    Fórmula:C45H42F2N10O5
    Forma y color:Solid
    Peso molecular:840.88
  • GIP/GLP-1 dual receptor agonist-1

    CAS:
    <p>Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.</p>
    Forma y color:Solid
  • VU0453379

    CAS:
    <p>VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).</p>
    Fórmula:C26H34N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:434.57
  • Glucagon receptor antagonists-1

    CAS:
    <p>Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.</p>
    Fórmula:C29H34FNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:447.58