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Receptor de glucagón

Receptor de glucagón

Los receptores de glucagón son GPCR que median los efectos del glucagón, una hormona involucrada en la regulación de la homeostasis de la glucosa al promover la descomposición del glucógeno y la liberación de glucosa desde el hígado. Estos receptores son cruciales en la gestión de los niveles de azúcar en sangre y son de particular interés en el estudio de la diabetes y los trastornos metabólicos. Los antagonistas de los receptores de glucagón se están explorando como posibles tratamientos para la hiperglucemia en la diabetes tipo 2. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de glucagón de alta calidad para apoyar su investigación en endocrinología, diabetes y regulación metabólica.

Se han encontrado 164 productos de "Receptor de glucagón"

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  • Anti-GCGR Antibody (7J909)


    <p>Anti-GCGR Antibody (7J909) is an antibody targeting GCGR. Anti-GCGR Antibody (7J909) can be used in ELISA.</p>
    Forma y color:Odour Liquid
  • SCO-267

    CAS:
    <p>SCO-267 is a full agonist of GPR40/FFAR1, stimulating insulin secretion and GLP-1 release in diabetic rats, improving glucose tolerance,type 2 diabetes.</p>
    Fórmula:C36H46N4O5
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:614.77
  • GLP-1R modulator C5

    CAS:
    <p>GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.</p>
    Fórmula:C24H21NO3
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:371.43
  • Liraglutide

    CAS:
    <p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>
    Fórmula:C172H265N43O51
    Pureza:97.65% - 99.04%
    Forma y color:Solid
    Peso molecular:3751.25
  • PF-06882961 Tris

    CAS:
    <p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>
    Fórmula:C35H41FN6O7
    Pureza:98.74% - 99.79%
    Forma y color:Solid
    Peso molecular:676.7
  • GRA Ex-25

    CAS:
    <p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>
    Fórmula:C29H36F3N3O5
    Pureza:98.2% - 98.88%
    Forma y color:Solid
    Peso molecular:563.61
  • Shanzhiside methyl ester

    CAS:
    <p>Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.</p>
    Fórmula:C17H26O11
    Pureza:98.998% - 99.32%
    Forma y color:Solid
    Peso molecular:406.38
  • Lixisenatide acetate (320367-13-3 free base)

    CAS:
    <p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>
    Fórmula:C215H347N61O65S·6C2H4O2
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:5218.88
  • BETP

    CAS:
    <p>BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).</p>
    Fórmula:C20H17F3N2O2S
    Pureza:98.51%
    Forma y color:Solid
    Peso molecular:406.42
  • HAEGTFTSDVSSYLE


    <p>HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.</p>
    Fórmula:C71H103N17O28
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1642.71
  • GLP-1(7-36), amide

    CAS:
    <p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>
    Fórmula:C149H226N40O45
    Pureza:99.85%
    Forma y color:White Powder
    Peso molecular:3297.63
  • Exendin-4

    CAS:
    <p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>
    Fórmula:C184H282N50O60S
    Pureza:97.71% - 99.78%
    Forma y color:Solid
    Peso molecular:4186.57
  • Semaglutide

    CAS:
    <p>Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).</p>
    Fórmula:C187H291N45O59
    Pureza:96.92% - 99.78%
    Forma y color:Solid
    Peso molecular:4114
  • Exendin-4 acetate

    CAS:
    <p>Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).</p>
    Fórmula:C186H286N50O62S
    Pureza:98.48% - 99.78%
    Forma y color:Solid
    Peso molecular:4247
  • Oxyntomodulin acetate


    <p>Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].</p>
    Pureza:99.24%
    Forma y color:Liquid
    Peso molecular:N/A
  • Bay 55-9837 acetate


    <p>Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.</p>
    Pureza:98.27%
    Forma y color:Liquid
    Peso molecular:N/A
  • Secretin (33-59), rat

    CAS:
    <p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>
    Fórmula:C129H216N42O42
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:3027.35
  • Glucagon (19-29), human acetate


    <p>Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.</p>
    Fórmula:C63H93N15O20S
    Pureza:98.11%
    Forma y color:Solid
    Peso molecular:1412.57
  • HAEGTFT acetate(926018-95-3 free base)


    <p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>
    Fórmula:C35H51N9O14
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:821.84
  • Tirzepatide Acetate(2023788-19-2 free base)


    Tirzepatide (LY3298176) Acetate (2023788-19-2 free base) is a new molecule that can control blood glucose levels.Cost-effective and quality-assured.
    Fórmula:C227H352N48O70
    Pureza:97.3% - 98.05%
    Forma y color:Solid
    Peso molecular:4873.5