Receptor de bradicinina
Los receptores de bradicinina son GPCR que median los efectos de la bradicinina, un péptido involucrado en las respuestas inflamatorias, la sensación de dolor y la regulación de la presión arterial. Hay dos tipos principales de receptores de bradicinina, B1 y B2, cada uno con roles distintos en procesos fisiopatológicos. Los antagonistas de los receptores de bradicinina se utilizan en el tratamiento de afecciones como el angioedema hereditario, el dolor crónico y la hipertensión. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de bradicinina de alta calidad para apoyar su investigación en inflamación, manejo del dolor y biología cardiovascular.
Se han encontrado 59 productos de "Receptor de bradicinina"
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NPC 567
CAS:<p>NPC 567 is an antagonist of the bradykinin receptor.</p>Fórmula:C60H87N19O13Pureza:98%Forma y color:SolidPeso molecular:1282.48L 366811
CAS:<p>L 366811 is a potent oxytocin antagonist.</p>Fórmula:C43H56N8O6Forma y color:SolidPeso molecular:780.95FR167344 free base
CAS:<p>FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.</p>Fórmula:C30H28BrCl2N5O4Pureza:98%Forma y color:SolidPeso molecular:673.38Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Fórmula:C16H28N6O4Pureza:98%Forma y color:SolidPeso molecular:368.43JMV-1645
CAS:<p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>Fórmula:C49H69N13O12SPureza:98%Forma y color:SolidPeso molecular:1064.23Lys-[Des-Arg9]Bradykinin TFA
CAS:<p>Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.</p>Fórmula:C54H75F6N13O15Forma y color:SolidPeso molecular:1260.24MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Fórmula:C60H90N20O11SPureza:98%Forma y color:SolidPeso molecular:1299.56Methionyl-Lysyl-Bradykinin
CAS:<p>Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .</p>Fórmula:C61H94N18O13SForma y color:SolidPeso molecular:1319.58Bradykinin (1-7)
CAS:<p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>Fórmula:C35H52N10O9Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:756.85Bradykinin (1-6)
CAS:<p>Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.</p>Fórmula:C30H45N9O8Pureza:98%Forma y color:SolidPeso molecular:659.73Lys-[Des-Arg9]Bradykinin
CAS:<p>Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.</p>Fórmula:C50H73N13O11Pureza:98%Forma y color:SolidPeso molecular:1032.21Retrobradykinin
CAS:<p>Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.</p>Fórmula:C50H73N15O11Forma y color:SolidPeso molecular:1060.228Lys-[Hyp3]-Bradykinin
CAS:<p>Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.</p>Fórmula:C56H85N17O13Forma y color:SolidPeso molecular:1204.38Bradykinin (1-5)
CAS:<p>Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.</p>Fórmula:C27H40N8O6Forma y color:SolidPeso molecular:572.66Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
<p>Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to</p>Fórmula:C49H70N12O13Pureza:99.93%Forma y color:SolidPeso molecular:1035.15Icatibant Acetate
CAS:<p>Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.</p>Fórmula:C61H93N19O15SPureza:99.68%Forma y color:SolidPeso molecular:1364.575-Hydroxy-1-methylhydantoin
CAS:<p>5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.</p>Fórmula:C4H6N2O3Pureza:99.99%Forma y color:SolidPeso molecular:130.1Bradykinin
CAS:<p>Bradykinin is an inflammatory mediator.</p>Fórmula:C50H73N15O11Pureza:99.68%Forma y color:SolidPeso molecular:1060.21Emorfazone
CAS:<p>Emorfazone (PH011085) has an anti-nociceptive effect.</p>Fórmula:C11H17N3O3Pureza:99.89%Forma y color:SolidPeso molecular:239.27ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Fórmula:C29H29ClN4O2Pureza:99.88%Forma y color:SolidPeso molecular:501.02
![Lys-[Des-Arg9]Bradykinin TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT73646.webp&w=3840&q=75)
![Lys-[Des-Arg9]Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1918.webp&w=3840&q=75)
![Lys-[Hyp3]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76293.webp&w=3840&q=75)
![Sar-[D-Phe8]-des-Arg9-Bradykinin acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1917L1.webp&w=3840&q=75)
