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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Fórmula:C21H25NO4
    Pureza:99.8% - 99.91%
    Forma y color:Off-White Solid
    Peso molecular:355.43
  • Lurasidone

    CAS:
    <p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>
    Fórmula:C28H36N4O2S
    Pureza:99.78% - 99.91%
    Forma y color:Solid
    Peso molecular:492.68
  • L-DOPA methyl ester (hydrochloride)

    CAS:
    <p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>
    Fórmula:C10H14ClNO4
    Pureza:98.69% - 99.81%
    Forma y color:White Solid
    Peso molecular:247.675
  • Zuclopenthixol dihydrochloride

    CAS:
    <p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>
    Fórmula:C22H27Cl3N2OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.89
  • AHN 1-055 hydrochloride

    CAS:
    <p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>
    Fórmula:C21H24ClF2NO
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:379.87
  • L-745870 hydrochloride

    CAS:
    <p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>
    Fórmula:C18H20Cl2N4
    Pureza:97.36%
    Forma y color:Solid
    Peso molecular:363.28
  • FAUC-365

    CAS:
    <p>FAUC-365 is a D3 dopamine receptor agonist.</p>
    Fórmula:C23H25Cl2N3OS
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:462.44
  • Tetrahydropalmatine hydrochloride

    CAS:
    <p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>
    Fórmula:C21H26ClNO4
    Pureza:98% - 99.59%
    Forma y color:Solid
    Peso molecular:391.888
  • Mesdopetam hemitartrate

    CAS:
    <p>Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.</p>
    Fórmula:C28H42F2N2O12S2
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:700.77
  • (+)-PD 128907 hydrochloride

    CAS:
    <p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>
    Fórmula:C14H20ClNO3
    Pureza:97.76%
    Forma y color:Solid
    Peso molecular:285.77
  • Metergoline

    CAS:
    <p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Forma y color:Solid
    Peso molecular:403.52
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Forma y color:Solid
    Peso molecular:538.64
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Forma y color:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • Fenoldopam mesylate

    CAS:
    <p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>
    Fórmula:C16H16ClNO3·CH4O3S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:401.86
  • Clebopride malate

    CAS:
    <p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>
    Fórmula:C24H30ClN3O7
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:507.96
  • Flupentixol dihydrochloride

    CAS:
    <p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.76% - >99.99%
    Forma y color:White Or Off-White Solid
    Peso molecular:507.43
  • Decynium 22

    CAS:
    <p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>
    Fórmula:C23H23IN2
    Pureza:99.92%
    Forma y color:Dark Red Crystals
    Peso molecular:454.35
  • Domperidone monomaleate

    CAS:
    <p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>
    Fórmula:C26H28ClN5O6
    Forma y color:Solid
    Peso molecular:541.98
  • GBR 12935 dihydrochloride

    CAS:
    <p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>
    Fórmula:C28H36Cl2N2O
    Pureza:99.09% - ≥95%
    Forma y color:Solid
    Peso molecular:487.5
  • Thozalinone

    CAS:
    <p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>
    Fórmula:C11H12N2O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:204.23