
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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Rotundine
CAS:<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Fórmula:C21H25NO4Pureza:99.8% - 99.91%Forma y color:Off-White SolidPeso molecular:355.43Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Forma y color:SolidPeso molecular:492.68L-DOPA methyl ester (hydrochloride)
CAS:<p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>Fórmula:C10H14ClNO4Pureza:98.69% - 99.81%Forma y color:White SolidPeso molecular:247.675Zuclopenthixol dihydrochloride
CAS:<p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>Fórmula:C22H27Cl3N2OSPureza:98%Forma y color:SolidPeso molecular:473.89AHN 1-055 hydrochloride
CAS:<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Fórmula:C21H24ClF2NOPureza:99.89%Forma y color:SolidPeso molecular:379.87L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Fórmula:C18H20Cl2N4Pureza:97.36%Forma y color:SolidPeso molecular:363.28FAUC-365
CAS:<p>FAUC-365 is a D3 dopamine receptor agonist.</p>Fórmula:C23H25Cl2N3OSPureza:99.62%Forma y color:SolidPeso molecular:462.44Tetrahydropalmatine hydrochloride
CAS:<p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>Fórmula:C21H26ClNO4Pureza:98% - 99.59%Forma y color:SolidPeso molecular:391.888Mesdopetam hemitartrate
CAS:<p>Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.</p>Fórmula:C28H42F2N2O12S2Pureza:99.98%Forma y color:SolidPeso molecular:700.77(+)-PD 128907 hydrochloride
CAS:<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Fórmula:C14H20ClNO3Pureza:97.76%Forma y color:SolidPeso molecular:285.77Metergoline
CAS:<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Forma y color:SolidPeso molecular:403.52WAY-100635 Monomaleate
CAS:<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Forma y color:SolidPeso molecular:538.64Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Forma y color:Off-White To Pale Yellow SolidPeso molecular:440.94Fenoldopam mesylate
CAS:<p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>Fórmula:C16H16ClNO3·CH4O3SPureza:99.19%Forma y color:SolidPeso molecular:401.86Clebopride malate
CAS:<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Fórmula:C24H30ClN3O7Pureza:99.52%Forma y color:SolidPeso molecular:507.96Flupentixol dihydrochloride
CAS:<p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>Fórmula:C23H27Cl2F3N2OSPureza:98.76% - >99.99%Forma y color:White Or Off-White SolidPeso molecular:507.43Decynium 22
CAS:<p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>Fórmula:C23H23IN2Pureza:99.92%Forma y color:Dark Red CrystalsPeso molecular:454.35Domperidone monomaleate
CAS:<p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>Fórmula:C26H28ClN5O6Forma y color:SolidPeso molecular:541.98GBR 12935 dihydrochloride
CAS:<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Fórmula:C28H36Cl2N2OPureza:99.09% - ≥95%Forma y color:SolidPeso molecular:487.5Thozalinone
CAS:<p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>Fórmula:C11H12N2O2Pureza:99.68%Forma y color:SolidPeso molecular:204.23
