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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Forma y color:Solid
    Peso molecular:463.87
  • Domperidone monomaleate

    CAS:
    <p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>
    Fórmula:C26H28ClN5O6
    Forma y color:Solid
    Peso molecular:541.98
  • Mesdopetam

    CAS:
    <p>Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.</p>
    Fórmula:C12H18FNO3S
    Forma y color:Solid
    Peso molecular:275.34
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:417.89
  • Veralipride

    CAS:
    <p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>
    Fórmula:C17H25N3O5S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:383.46
  • Dimethocaine

    CAS:
    <p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>
    Fórmula:C16H26N2O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:278.39
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Fórmula:C21H25NO4
    Pureza:99.8% - 99.91%
    Forma y color:Off-White Solid
    Peso molecular:355.43
  • Clebopride malate

    CAS:
    <p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>
    Fórmula:C24H30ClN3O7
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:507.96
  • Haloperidol hydrochloride

    CAS:
    <p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>
    Fórmula:C21H24Cl2FNO2
    Forma y color:Solid
    Peso molecular:412.33
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Forma y color:Solid
    Peso molecular:417.97
  • JNJ-37822681

    CAS:
    <p>JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.</p>
    Fórmula:C17H17F5N4
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:372.34
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Forma y color:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • Thozalinone

    CAS:
    <p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>
    Fórmula:C11H12N2O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:204.23
  • Fenoldopam mesylate

    CAS:
    <p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>
    Fórmula:C16H16ClNO3·CH4O3S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:401.86
  • Lurasidone hydrochloride

    CAS:
    <p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia &amp; bipolar, affects dopamine, serotonin &amp; adrenergic receptors.</p>
    Fórmula:C28H36N4O2S·HCl
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:529.14
  • GBR 12935 dihydrochloride

    CAS:
    <p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>
    Fórmula:C28H36Cl2N2O
    Pureza:99.09% - ≥95%
    Forma y color:Solid
    Peso molecular:487.5
  • Loxapine

    CAS:
    <p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>
    Fórmula:C18H18ClN3O
    Pureza:99.88%
    Forma y color:Pale Yellowish Crystals From Petroleum Ether Solid
    Peso molecular:327.81
  • Zuclopenthixol

    CAS:
    <p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>
    Fórmula:C22H25ClN2OS
    Pureza:98.9% - 99.82%
    Forma y color:Solid
    Peso molecular:400.96
  • Azaperone

    CAS:
    <p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>
    Fórmula:C19H22FN3O
    Pureza:98.73%
    Forma y color:White Or Off-White Crystalline
    Peso molecular:327.4
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Forma y color:Solid
    Peso molecular:433.57