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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • PF-06256142

    CAS:
    <p>PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).</p>
    Fórmula:C21H16N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.38
  • YQA14

    CAS:
    <p>YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.</p>
    Fórmula:C23H27ClN4O3
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:442.94
  • PF-592379

    CAS:
    <p>PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).</p>
    Fórmula:C13H21N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:235.33
  • PD 119819

    CAS:
    <p>PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.</p>
    Fórmula:C21H25Cl2N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.35
  • ADR-851 HCl

    CAS:
    <p>ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.</p>
    Fórmula:C14H19Cl2N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:332.23
  • CAD031

    CAS:
    <p>CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.</p>
    Fórmula:C18H14F6N2O2
    Forma y color:Solid
    Peso molecular:404.31
  • R-SKF-38393A HCl

    CAS:
    <p>R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.</p>
    Fórmula:C16H18ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:291.77
  • Mosapramine

    CAS:
    <p>Mosapramine is a dopamine D2-receptor antagonist.</p>
    Fórmula:C28H35ClN4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:479.06
  • Sultopride

    CAS:
    <p>Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.</p>
    Fórmula:C17H26N2O4S
    Forma y color:Solid
    Peso molecular:354.46
  • U-101958 Maleate

    CAS:
    <p>U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.</p>
    Fórmula:C25H33N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:455.55
  • NGB 2904 hydrochloride

    CAS:
    <p>dopamine D3 receptor antagonist</p>
    Fórmula:C28H30Cl3N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:530.92
  • Oxiperomide

    CAS:
    <p>Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.</p>
    Fórmula:C20H23N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:337.42
  • PD-89211

    CAS:
    <p>PD 89211 selectively blocks dopamine D4.2 receptor &gt;800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).</p>
    Fórmula:C19H21ClN4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.85
  • R(+)-6-Bromo-APB HBr

    CAS:
    <p>R(+)-6-Bromo-APB HBr is used as a D1 Dopamine receptor agonist.</p>
    Fórmula:C19H21Br2NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:455.18
  • SKF 83959 hydrobromide

    CAS:
    <p>SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.</p>
    Fórmula:C18H21BrClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:398.72
  • CGP 25454A

    CAS:
    <p>CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.</p>
    Fórmula:C15H21Cl2N3O2
    Forma y color:Solid
    Peso molecular:346.25
  • ST-198

    CAS:
    <p>ST-198 is a dopamine D3 receptor antagonist.</p>
    Fórmula:C22H26N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:334.45
  • Piperidine-MO-1

    CAS:
    <p>Piperidine-MO-1 is a dopamine receptor modulator, with an ED50 of 68 μmol/kg on increase of DOPAC in the rat striatum.</p>
    Fórmula:C14H21ClFNO2S
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:321.84
  • SKF83822 hydrobromide

    CAS:
    <p>SKF83822 hydrobromide is a dopamine D1-like receptor agonist.</p>
    Fórmula:C20H23BrClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:424.76
  • CL-216303 HCl

    CAS:
    <p>CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.</p>
    Fórmula:C11H12Cl3N
    Pureza:98%
    Forma y color:Solid
    Peso molecular:264.58