
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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PF-06256142
CAS:<p>PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).</p>Fórmula:C21H16N4O2Pureza:98%Forma y color:SolidPeso molecular:356.38YQA14
CAS:<p>YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.</p>Fórmula:C23H27ClN4O3Pureza:99.52%Forma y color:SolidPeso molecular:442.94PF-592379
CAS:<p>PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).</p>Fórmula:C13H21N3OPureza:98%Forma y color:SolidPeso molecular:235.33PD 119819
CAS:<p>PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.</p>Fórmula:C21H25Cl2N3O3Pureza:98%Forma y color:SolidPeso molecular:438.35ADR-851 HCl
CAS:<p>ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.</p>Fórmula:C14H19Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:332.23CAD031
CAS:<p>CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.</p>Fórmula:C18H14F6N2O2Forma y color:SolidPeso molecular:404.31R-SKF-38393A HCl
CAS:<p>R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.</p>Fórmula:C16H18ClNO2Pureza:98%Forma y color:SolidPeso molecular:291.77Mosapramine
CAS:<p>Mosapramine is a dopamine D2-receptor antagonist.</p>Fórmula:C28H35ClN4OPureza:98%Forma y color:SolidPeso molecular:479.06Sultopride
CAS:<p>Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.</p>Fórmula:C17H26N2O4SForma y color:SolidPeso molecular:354.46U-101958 Maleate
CAS:<p>U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.</p>Fórmula:C25H33N3O5Pureza:98%Forma y color:SolidPeso molecular:455.55NGB 2904 hydrochloride
CAS:<p>dopamine D3 receptor antagonist</p>Fórmula:C28H30Cl3N3OPureza:98%Forma y color:SolidPeso molecular:530.92Oxiperomide
CAS:<p>Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.</p>Fórmula:C20H23N3O2Pureza:98%Forma y color:SolidPeso molecular:337.42PD-89211
CAS:<p>PD 89211 selectively blocks dopamine D4.2 receptor >800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).</p>Fórmula:C19H21ClN4OPureza:98%Forma y color:SolidPeso molecular:356.85R(+)-6-Bromo-APB HBr
CAS:<p>R(+)-6-Bromo-APB HBr is used as a D1 Dopamine receptor agonist.</p>Fórmula:C19H21Br2NO2Pureza:98%Forma y color:SolidPeso molecular:455.18SKF 83959 hydrobromide
CAS:<p>SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.</p>Fórmula:C18H21BrClNO2Pureza:98%Forma y color:SolidPeso molecular:398.72CGP 25454A
CAS:<p>CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.</p>Fórmula:C15H21Cl2N3O2Forma y color:SolidPeso molecular:346.25ST-198
CAS:<p>ST-198 is a dopamine D3 receptor antagonist.</p>Fórmula:C22H26N2OPureza:98%Forma y color:SolidPeso molecular:334.45Piperidine-MO-1
CAS:<p>Piperidine-MO-1 is a dopamine receptor modulator, with an ED50 of 68 μmol/kg on increase of DOPAC in the rat striatum.</p>Fórmula:C14H21ClFNO2SPureza:99.88%Forma y color:SolidPeso molecular:321.84SKF83822 hydrobromide
CAS:<p>SKF83822 hydrobromide is a dopamine D1-like receptor agonist.</p>Fórmula:C20H23BrClNO2Pureza:98%Forma y color:SolidPeso molecular:424.76CL-216303 HCl
CAS:<p>CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.</p>Fórmula:C11H12Cl3NPureza:98%Forma y color:SolidPeso molecular:264.58
