
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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SKF-82958
CAS:<p>SKF 82958 is a D1/D5 receptor full agonist.</p>Fórmula:C19H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:329.82Dopamine D2 receptor antagonist-1
CAS:<p>Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.</p>Fórmula:C14H17N3SPureza:99.86%Forma y color:SolidPeso molecular:259.37(+)-UH 232 maleate
CAS:<p>D2 antagonist</p>Fórmula:C18H29NOPureza:98%Forma y color:SolidPeso molecular:275.43A412997
CAS:<p>A412997 is a selective agonist of dopamine D4 receptor.</p>Fórmula:C19H23N3OPureza:98%Forma y color:SolidPeso molecular:309.41S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Fórmula:C16H20ClN3OSForma y color:SolidPeso molecular:337.87FR 64822
CAS:<p>FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.</p>Fórmula:C11H14N4OForma y color:SolidPeso molecular:218.26SV-156
CAS:<p>SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).</p>Fórmula:C21H23BrN2O2Forma y color:SolidPeso molecular:415.32Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Fórmula:C22H26ClNPureza:98%Forma y color:SolidPeso molecular:339.9Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Fórmula:C20H25BrN4OForma y color:SolidPeso molecular:417.34SKF-104557
CAS:<p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>Fórmula:C13H18N2OForma y color:SolidPeso molecular:218.29A 68930 hydrochloride
CAS:<p>A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].</p>Fórmula:C16H18ClNO3Forma y color:Off-White SolidPeso molecular:307.77SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Forma y color:SolidPeso molecular:376.29Tau-aggregation-IN-1
CAS:<p>Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).</p>Fórmula:C28H37N5O2SForma y color:SolidPeso molecular:507.69DOV-216,303 Free Base
CAS:<p>DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.</p>Fórmula:C11H11Cl2NPureza:96.7%Forma y color:SolidPeso molecular:228.12Octoclothepin maleate salt
CAS:<p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>Fórmula:C23H25ClN2O4SForma y color:SolidPeso molecular:460.97RTI 336
CAS:<p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>Fórmula:C24H26Cl2N2OPureza:98%Forma y color:SolidPeso molecular:429.38SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Fórmula:C17H20BrNO2Forma y color:SolidPeso molecular:350.25UNC9995
CAS:<p>UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).</p>Fórmula:C20H21Cl2N3OSPureza:98%Forma y color:SolidPeso molecular:422.37NPEC-caged-dopamine
CAS:<p>Dopamine receptor agonist</p>Fórmula:C17H18N2O6Pureza:98%Forma y color:SolidPeso molecular:346.33RBI-257 Maleate
CAS:<p>RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.</p>Fórmula:C25H32IN3O5Forma y color:SolidPeso molecular:581.44
