
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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Sumanirole maleate
CAS:<p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>Fórmula:C15H17N3O5Pureza:98%Forma y color:SolidPeso molecular:319.31UCSF924
CAS:<p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>Fórmula:C20H22N2O2Pureza:98%Forma y color:SolidPeso molecular:322.4Pramipexole dihydrochloride
CAS:<p>Pramipexole dihydrochloride could be used to treat Parkinson disease.</p>Fórmula:C10H18ClN3SPureza:98%Forma y color:White Crystalline PowderPeso molecular:247.79cis-(Z)-Flupentixol dihydrochloride
CAS:<p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>Fórmula:C23H27Cl2F3N2OSPureza:98.07%Forma y color:SolidPeso molecular:507.44PD128907 HCl
CAS:<p>PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.</p>Fórmula:C14H20ClNO3Pureza:98%Forma y color:SolidPeso molecular:285.77Aramisulpride
CAS:<p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>Fórmula:C17H27N3O4SForma y color:SolidPeso molecular:369.48Eticlopride hydrochloride
CAS:<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Fórmula:C17H25ClN2O3·HClPureza:98%Forma y color:SolidPeso molecular:377.31SKF-82958 hydrobromide
CAS:<p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>Fórmula:C19H21BrClNO2Pureza:98%Forma y color:SolidPeso molecular:410.73(-)-Apomorphine hydrochloride hydrate
CAS:<p>(-)-Apomorphine hydrochloride hydrate is a broad-spectrum dopamine agonist and ferroptosis inhibitor.</p>Fórmula:C17H17NO2HClXH2OForma y color:SolidPeso molecular:303.8Tiapride-d3
<p>Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.</p>Fórmula:C15H21D3N2O4SForma y color:SolidPeso molecular:331.45Clomipramine D3 hydrochloride
CAS:<p>Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).</p>Fórmula:C19H24Cl2N2Forma y color:SolidPeso molecular:354.33ABT-724
CAS:<p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>Fórmula:C17H19N5Pureza:99.73%Forma y color:SolidPeso molecular:293.37Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Fórmula:C20H22N2O4Pureza:98.46%Forma y color:SolidPeso molecular:354.4Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Forma y color:SolidPeso molecular:433.57Alizapride hydrochloride
CAS:<p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>Fórmula:C16H21N5O2·HClPureza:99.35% - 99.48%Forma y color:CoaPeso molecular:351.83GBR 12935
CAS:<p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>Fórmula:C28H34N2OForma y color:SolidPeso molecular:414.58Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Forma y color:White Or Off-White CrystallinePeso molecular:327.4Raclopride tartrate
CAS:<p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>Fórmula:C19H26Cl2N2O9Forma y color:SolidPeso molecular:497.32Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Fórmula:C22H19NO4Pureza:99.45% - 99.78%Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39BisfluoroModafinil
CAS:<p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>Fórmula:C15H13F2NO2SPureza:99.19%Forma y color:SolidPeso molecular:309.33
