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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • Sumanirole maleate

    CAS:
    <p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>
    Fórmula:C15H17N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:319.31
  • UCSF924

    CAS:
    <p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>
    Fórmula:C20H22N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:322.4
  • Pramipexole dihydrochloride

    CAS:
    <p>Pramipexole dihydrochloride could be used to treat Parkinson disease.</p>
    Fórmula:C10H18ClN3S
    Pureza:98%
    Forma y color:White Crystalline Powder
    Peso molecular:247.79
  • cis-(Z)-Flupentixol dihydrochloride

    CAS:
    <p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.07%
    Forma y color:Solid
    Peso molecular:507.44
  • PD128907 HCl

    CAS:
    <p>PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.</p>
    Fórmula:C14H20ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:285.77
  • Aramisulpride

    CAS:
    <p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>
    Fórmula:C17H27N3O4S
    Forma y color:Solid
    Peso molecular:369.48
  • Eticlopride hydrochloride

    CAS:
    <p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>
    Fórmula:C17H25ClN2O3·HCl
    Pureza:98%
    Forma y color:Solid
    Peso molecular:377.31
  • SKF-82958 hydrobromide

    CAS:
    <p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>
    Fórmula:C19H21BrClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.73
  • (-)-Apomorphine hydrochloride hydrate

    CAS:
    <p>(-)-Apomorphine hydrochloride hydrate is a broad-spectrum dopamine agonist and ferroptosis inhibitor.</p>
    Fórmula:C17H17NO2HClXH2O
    Forma y color:Solid
    Peso molecular:303.8
  • Tiapride-d3


    <p>Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.</p>
    Fórmula:C15H21D3N2O4S
    Forma y color:Solid
    Peso molecular:331.45
  • Clomipramine D3 hydrochloride

    CAS:
    <p>Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).</p>
    Fórmula:C19H24Cl2N2
    Forma y color:Solid
    Peso molecular:354.33
  • ABT-724

    CAS:
    <p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>
    Fórmula:C17H19N5
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:293.37
  • Nomifensine maleate

    CAS:
    <p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>
    Fórmula:C20H22N2O4
    Pureza:98.46%
    Forma y color:Solid
    Peso molecular:354.4
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Forma y color:Solid
    Peso molecular:433.57
  • Alizapride hydrochloride

    CAS:
    <p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>
    Fórmula:C16H21N5O2·HCl
    Pureza:99.35% - 99.48%
    Forma y color:Coa
    Peso molecular:351.83
  • GBR 12935

    CAS:
    <p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>
    Fórmula:C28H34N2O
    Forma y color:Solid
    Peso molecular:414.58
  • Azaperone

    CAS:
    <p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>
    Fórmula:C19H22FN3O
    Pureza:98.73%
    Forma y color:White Or Off-White Crystalline
    Peso molecular:327.4
  • Raclopride tartrate

    CAS:
    <p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>
    Fórmula:C19H26Cl2N2O9
    Forma y color:Solid
    Peso molecular:497.32
  • Bisacodyl

    CAS:
    <p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>
    Fórmula:C22H19NO4
    Pureza:99.45% - 99.78%
    Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline Powder
    Peso molecular:361.39
  • BisfluoroModafinil

    CAS:
    <p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>
    Fórmula:C15H13F2NO2S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:309.33