Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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Cariprazine hydrochloride
CAS:<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Forma y color:SolidPeso molecular:463.87Domperidone monomaleate
CAS:<p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>Fórmula:C26H28ClN5O6Forma y color:SolidPeso molecular:541.98Mesdopetam
CAS:<p>Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.</p>Fórmula:C12H18FNO3SForma y color:SolidPeso molecular:275.34Dimethocaine
CAS:<p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>Fórmula:C16H26N2O2Pureza:99.52%Forma y color:SolidPeso molecular:278.39Rotundine
CAS:<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Fórmula:C21H25NO4Pureza:99.8% - 99.91%Forma y color:Off-White SolidPeso molecular:355.43Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Forma y color:Off-White To Pale Yellow SolidPeso molecular:440.94Thozalinone
CAS:<p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>Fórmula:C11H12N2O2Pureza:99.68%Forma y color:SolidPeso molecular:204.23Clebopride malate
CAS:<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Fórmula:C24H30ClN3O7Pureza:99.52%Forma y color:SolidPeso molecular:507.96Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Fórmula:C21H24Cl2FNO2Forma y color:SolidPeso molecular:412.33Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Forma y color:SolidPeso molecular:417.97JNJ-37822681
CAS:<p>JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.</p>Fórmula:C17H17F5N4Pureza:99.84%Forma y color:SolidPeso molecular:372.34Zuclopenthixol
CAS:<p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>Fórmula:C22H25ClN2OSPureza:98.9% - 99.82%Forma y color:SolidPeso molecular:400.96Clozapine N-Oxide
CAS:<p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>Fórmula:C18H19ClN4OPureza:98.43% - 99.94%Forma y color:SolidPeso molecular:342.82Fenoldopam mesylate
CAS:<p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>Fórmula:C16H16ClNO3·CH4O3SPureza:99.19%Forma y color:SolidPeso molecular:401.86Lurasidone hydrochloride
CAS:<p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.</p>Fórmula:C28H36N4O2S·HClPureza:99.51%Forma y color:SolidPeso molecular:529.14GBR 12935 dihydrochloride
CAS:<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Fórmula:C28H36Cl2N2OPureza:99.09% - ≥95%Forma y color:SolidPeso molecular:487.5Loxapine
CAS:<p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>Fórmula:C18H18ClN3OPureza:99.88%Forma y color:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.81Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Forma y color:White SolidPeso molecular:463Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Forma y color:White Or Off-White CrystallinePeso molecular:327.4Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Forma y color:SolidPeso molecular:433.57Alizapride
CAS:<p>Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].</p>Fórmula:C16H21N5O2Forma y color:SolidPeso molecular:315.37A-381393
CAS:<p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>Fórmula:C20H24N4Pureza:99.00%Forma y color:SolidPeso molecular:320.43Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Fórmula:C19H21NO2Pureza:98.76% - 99.79%Forma y color:SolidPeso molecular:295.38Zuclopenthixol dihydrochloride
CAS:<p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>Fórmula:C22H27Cl3N2OSPureza:98%Forma y color:SolidPeso molecular:473.89Protein deglycase DJ-1 against-1
CAS:<p>Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.</p>Fórmula:C24H23N3O4Pureza:97.23%Forma y color:SolidPeso molecular:417.46Dexpramipexole
CAS:<p>Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.</p>Fórmula:C10H17N3SPureza:99.78%Forma y color:SolidPeso molecular:211.33Trazpiroben
CAS:<p>Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.</p>Fórmula:C31H39N3O4Pureza:99.41% - >99.99%Forma y color:SolidPeso molecular:517.66Ropinirole
CAS:<p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>Fórmula:C16H24N2OPureza:99.68%Forma y color:SolidPeso molecular:260.38L-745870
CAS:<p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>Fórmula:C18H19ClN4Pureza:98%Forma y color:SolidPeso molecular:326.82Vanoxerine
CAS:<p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>Fórmula:C28H32F2N2OPureza:98%Forma y color:SolidPeso molecular:450.56Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Fórmula:C12H15N3O2Pureza:98%Forma y color:SolidPeso molecular:233.27A23887
CAS:<p>A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.</p>Fórmula:C22H24ClNPureza:98%Forma y color:SolidPeso molecular:337.89SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Fórmula:C21H22ClNO5Pureza:98%Forma y color:SolidPeso molecular:403.86Quinpirole Hydrochloride
CAS:<p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>Fórmula:C13H22ClN3Pureza:98%Forma y color:SolidPeso molecular:255.79Fallypride
CAS:<p>Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.</p>Fórmula:C20H29FN2O3Pureza:98.97% - >99.99%Forma y color:SolidPeso molecular:364.45CP-226269
CAS:<p>CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.</p>Fórmula:C18H19FN4Pureza:99.08%Forma y color:SolidPeso molecular:310.37PD 120697
CAS:<p>PD 120697 is a dopamine antagonist with central dopamine agonist properties.</p>Fórmula:C11H15N3SPureza:98%Forma y color:SolidPeso molecular:221.32Talipexole
CAS:<p>Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.</p>Fórmula:C10H15N3SPureza:98%Forma y color:SolidPeso molecular:209.31Foscarbidopa
CAS:<p>Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.</p>Fórmula:C10H15N2O7PPureza:96.17% - 97.27%Forma y color:SolidPeso molecular:306.21Nafadotride
CAS:<p>Nafadotride is a dopamine D3 receptor antagonist.</p>Fórmula:C22H27N3O2Forma y color:SolidPeso molecular:365.47PD168,077
CAS:<p>PD168,077 is an agonist of dopamine D4 receptor. It has a facilitatory effect on memory consolidation.</p>Fórmula:C20H22N4OPureza:98%Forma y color:SolidPeso molecular:334.41Fluphenazine Decanoate Dihydrochloride
CAS:<p>Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.</p>Fórmula:C32H46Cl2F3N3O2SPureza:98%Forma y color:SolidPeso molecular:664.69Roxindole hydrochloride
CAS:<p>Dopamine D2 autoreceptor agonist</p>Fórmula:C23H27ClN2OPureza:98%Forma y color:SolidPeso molecular:382.93Dopamine D4 receptor antagonist-1
CAS:<p>Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.</p>Fórmula:C18H19ClN4Forma y color:SolidPeso molecular:326.82JHW 007 hydrochloride
CAS:<p>JHW 007 hydrochloride is a Dopamine uptake inhibitor.</p>Fórmula:C24H30ClF2NOPureza:98%Forma y color:SolidPeso molecular:421.95Indatraline hydrochloride
CAS:<p>Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)</p>Fórmula:C16H16Cl3NPureza:98%Forma y color:SolidPeso molecular:328.662-CMDO
CAS:<p>2-CMDO is a Dopamine D2-like receptor antagonist.</p>Fórmula:C23H23ClN2O5Pureza:98%Forma y color:SolidPeso molecular:442.89JPC-211
CAS:<p>JPC-211 is an agonist of dopamine-receptor.</p>Fórmula:C17H27NO2Pureza:98%Forma y color:SolidPeso molecular:277.4GBR 13069 dihydrochloride
CAS:<p>GBR 13069 dihydrochloride is a dopamine uptake inhibitor.</p>Fórmula:C28H32Cl2F2N2OPureza:98%Forma y color:SolidPeso molecular:521.47SB269652
CAS:<p>SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.</p>Fórmula:C27H30N4OPureza:98%Forma y color:SolidPeso molecular:426.55Lenperone HCl
CAS:<p>Lenperone HCl is a dopamine antagonist and an antipsychotic agent.</p>Fórmula:C22H24ClF2NO2Pureza:98%Forma y color:SolidPeso molecular:407.88(-)-GSK598809
CAS:<p>(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.</p>Fórmula:C22H23F4N5OSPureza:98%Forma y color:SolidPeso molecular:481.51Tesofensine
CAS:<p>Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.</p>Fórmula:C17H23Cl2NOPureza:98%Forma y color:SolidPeso molecular:328.28Acetophenazine
CAS:<p>Acetophenazine is an anxiolytic compound that is used in the study of depression.</p>Fórmula:C23H29N3O2SPureza:99.30%Forma y color:SoildPeso molecular:411.56GBR 12783
CAS:<p>GBR 12783 enhances memory, boosts rat hippocampal acetylcholine, and is a potent dopamine uptake inhibitor with IC50s of 1.8/1.2 nM in rats/mice.</p>Fórmula:C28H32N2OPureza:98%Forma y color:SolidPeso molecular:412.57ST-836
CAS:<p>ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .</p>Fórmula:C23H34N4OSPureza:98%Forma y color:SolidPeso molecular:414.61Org-10490
CAS:<p>Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.</p>Fórmula:C17H19NOPureza:98%Forma y color:SolidPeso molecular:253.34L 741742 hydrochloride
CAS:<p>L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.</p>Fórmula:C23H26Cl2N2OPureza:99.9%Forma y color:SolidPeso molecular:417.37A68930
CAS:<p>A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.</p>Fórmula:C16H17NO3Forma y color:SolidPeso molecular:271.31Remoxipride
CAS:<p>Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.</p>Fórmula:C16H23BrN2O3Pureza:98%Forma y color:SolidPeso molecular:371.27PF-06256142
CAS:<p>PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).</p>Fórmula:C21H16N4O2Pureza:98%Forma y color:SolidPeso molecular:356.38YQA14
CAS:<p>YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.</p>Fórmula:C23H27ClN4O3Pureza:99.52%Forma y color:SolidPeso molecular:442.94PF-592379
CAS:<p>PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).</p>Fórmula:C13H21N3OPureza:98%Forma y color:SolidPeso molecular:235.33PD 119819
CAS:<p>PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.</p>Fórmula:C21H25Cl2N3O3Pureza:98%Forma y color:SolidPeso molecular:438.35ADR-851 HCl
CAS:<p>ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.</p>Fórmula:C14H19Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:332.23CAD031
CAS:<p>CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.</p>Fórmula:C18H14F6N2O2Forma y color:SolidPeso molecular:404.31R-SKF-38393A HCl
CAS:<p>R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.</p>Fórmula:C16H18ClNO2Pureza:98%Forma y color:SolidPeso molecular:291.77Mosapramine
CAS:<p>Mosapramine is a dopamine D2-receptor antagonist.</p>Fórmula:C28H35ClN4OPureza:98%Forma y color:SolidPeso molecular:479.06Sultopride
CAS:<p>Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.</p>Fórmula:C17H26N2O4SForma y color:SolidPeso molecular:354.46U-101958 Maleate
CAS:<p>U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.</p>Fórmula:C25H33N3O5Pureza:98%Forma y color:SolidPeso molecular:455.55NGB 2904 hydrochloride
CAS:<p>dopamine D3 receptor antagonist</p>Fórmula:C28H30Cl3N3OPureza:98%Forma y color:SolidPeso molecular:530.92Oxiperomide
CAS:<p>Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.</p>Fórmula:C20H23N3O2Pureza:98%Forma y color:SolidPeso molecular:337.42PD-89211
CAS:<p>PD 89211 selectively blocks dopamine D4.2 receptor >800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).</p>Fórmula:C19H21ClN4OPureza:98%Forma y color:SolidPeso molecular:356.85R(+)-6-Bromo-APB HBr
CAS:<p>R(+)-6-Bromo-APB HBr is used as a D1 Dopamine receptor agonist.</p>Fórmula:C19H21Br2NO2Pureza:98%Forma y color:SolidPeso molecular:455.18SKF 83959 hydrobromide
CAS:<p>SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.</p>Fórmula:C18H21BrClNO2Pureza:98%Forma y color:SolidPeso molecular:398.72CGP 25454A
CAS:<p>CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.</p>Fórmula:C15H21Cl2N3O2Forma y color:SolidPeso molecular:346.25ST-198
CAS:<p>ST-198 is a dopamine D3 receptor antagonist.</p>Fórmula:C22H26N2OPureza:98%Forma y color:SolidPeso molecular:334.45Piperidine-MO-1
CAS:<p>Piperidine-MO-1 is a dopamine receptor modulator, with an ED50 of 68 μmol/kg on increase of DOPAC in the rat striatum.</p>Fórmula:C14H21ClFNO2SPureza:99.88%Forma y color:SolidPeso molecular:321.84SKF83822 hydrobromide
CAS:<p>SKF83822 hydrobromide is a dopamine D1-like receptor agonist.</p>Fórmula:C20H23BrClNO2Pureza:98%Forma y color:SolidPeso molecular:424.76CL-216303 HCl
CAS:<p>CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.</p>Fórmula:C11H12Cl3NPureza:98%Forma y color:SolidPeso molecular:264.58SKF-82958
CAS:<p>SKF 82958 is a D1/D5 receptor full agonist.</p>Fórmula:C19H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:329.82Dopamine D2 receptor antagonist-1
CAS:<p>Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.</p>Fórmula:C14H17N3SPureza:99.86%Forma y color:SolidPeso molecular:259.37(+)-UH 232 maleate
CAS:<p>D2 antagonist</p>Fórmula:C18H29NOPureza:98%Forma y color:SolidPeso molecular:275.43A412997
CAS:<p>A412997 is a selective agonist of dopamine D4 receptor.</p>Fórmula:C19H23N3OPureza:98%Forma y color:SolidPeso molecular:309.41S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Fórmula:C16H20ClN3OSForma y color:SolidPeso molecular:337.87FR 64822
CAS:<p>FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.</p>Fórmula:C11H14N4OForma y color:SolidPeso molecular:218.26SV-156
CAS:<p>SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).</p>Fórmula:C21H23BrN2O2Forma y color:SolidPeso molecular:415.32Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Fórmula:C22H26ClNPureza:98%Forma y color:SolidPeso molecular:339.9Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Fórmula:C20H25BrN4OForma y color:SolidPeso molecular:417.34SKF-104557
CAS:<p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>Fórmula:C13H18N2OForma y color:SolidPeso molecular:218.29A 68930 hydrochloride
CAS:<p>A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].</p>Fórmula:C16H18ClNO3Forma y color:Off-White SolidPeso molecular:307.77SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Forma y color:SolidPeso molecular:376.29Tau-aggregation-IN-1
CAS:<p>Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).</p>Fórmula:C28H37N5O2SForma y color:SolidPeso molecular:507.69DOV-216,303 Free Base
CAS:<p>DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.</p>Fórmula:C11H11Cl2NPureza:96.7%Forma y color:SolidPeso molecular:228.12Octoclothepin maleate salt
CAS:<p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>Fórmula:C23H25ClN2O4SForma y color:SolidPeso molecular:460.97RTI 336
CAS:<p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>Fórmula:C24H26Cl2N2OPureza:98%Forma y color:SolidPeso molecular:429.38SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Fórmula:C17H20BrNO2Forma y color:SolidPeso molecular:350.25UNC9995
CAS:<p>UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).</p>Fórmula:C20H21Cl2N3OSPureza:98%Forma y color:SolidPeso molecular:422.37NPEC-caged-dopamine
CAS:<p>Dopamine receptor agonist</p>Fórmula:C17H18N2O6Pureza:98%Forma y color:SolidPeso molecular:346.33RBI-257 Maleate
CAS:<p>RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.</p>Fórmula:C25H32IN3O5Forma y color:SolidPeso molecular:581.44Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Forma y color:SolidPeso molecular:282.81SKF-83822
CAS:<p>SKF-83822 is an agonist of dopamine D1-like receptor.</p>Fórmula:C20H22ClNO2Pureza:98%Forma y color:SolidPeso molecular:343.85BRD5814
CAS:<p>BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.</p>Fórmula:C21H23ClF3NO2Forma y color:SolidPeso molecular:413.86SB-277011 dihydrochloride
CAS:<p>SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.</p>Fórmula:C28H32Cl2N4OPureza:98%Forma y color:SolidPeso molecular:511.49PF2562
CAS:<p>PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).</p>Fórmula:C19H17N5OPureza:98%Forma y color:SolidPeso molecular:331.37Odapipam
CAS:<p>Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).</p>Fórmula:C19H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:329.82Lenperone
CAS:<p>Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic.</p>Fórmula:C22H23F2NO2Forma y color:SolidPeso molecular:371.42BAK2-66
CAS:<p>BAK2-66 is a selective antagonist of the dopamine D3 receptor.</p>Fórmula:C23H24Cl2FN3O2Pureza:98%Forma y color:SolidPeso molecular:464.36Brl 20596
CAS:<p>Brl 20596 is a central dopamine antagonist in the class of anilide.</p>Fórmula:C20H24ClN3O2Pureza:98%Forma y color:SolidPeso molecular:373.88FAUC-3019
CAS:<p>FAUC-3019 is a partial agonist of the dopamine D(4) receptor.</p>Fórmula:C22H24N2OForma y color:SolidPeso molecular:332.44Lergotrile
CAS:<p>Lergotrile is used as an enzyme Inhibitor (Prolactin).</p>Fórmula:C17H18ClN3Pureza:98%Forma y color:SolidPeso molecular:299.8CJB-090 2HCl
CAS:<p>CJB-090 2HCl is a partial agonist of the dopamine D3 receptor.</p>Fórmula:C26H30Cl4N4OForma y color:SolidPeso molecular:556.35Gyki 32887
CAS:<p>Gyki 32887 is a dopamine agonist.</p>Fórmula:C23H28N6O6SPureza:98%Forma y color:SolidPeso molecular:516.57Amitifadine free base
CAS:<p>Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.</p>Fórmula:C11H11Cl2NForma y color:SolidPeso molecular:228.12A 69024
CAS:<p>A 69024 is a highly selective antagonist of dopamine D-1 receptor.</p>Fórmula:C20H24BrNO4Pureza:98%Forma y color:SolidPeso molecular:422.31Seproxetine HCl
CAS:<p>Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.</p>Fórmula:C16H17ClF3NOPureza:98%Forma y color:SolidPeso molecular:331.76Lergotrile mesylate
CAS:<p>Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.</p>Fórmula:C18H22ClN3O3SForma y color:SolidPeso molecular:395.9Bromperidol decanoate
CAS:<p>Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.</p>Fórmula:C31H41BrFNO3Forma y color:SolidPeso molecular:574.56LY 171859
CAS:<p>LY 171859 is an agonist of D2-receptor.</p>Fórmula:C17H14O5Pureza:98%Forma y color:SolidPeso molecular:298.29Nor-SCH-12679 Maleate
CAS:<p>Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.</p>Fórmula:C22H25NO6Pureza:98%Forma y color:SolidPeso molecular:399.44Clothixamide
CAS:<p>Clothixamide（Clotixamide） is a thioxanthene derivative with antipsychotic activity.</p>Fórmula:C24H28ClN3OSPureza:95.51%Forma y color:SolidPeso molecular:442.02CI-943
CAS:<p>CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.</p>Fórmula:C12H17N5Pureza:98%Forma y color:SolidPeso molecular:231.33'-Fluorobenzylspiperone maleate
CAS:<p>ligand for the D2 receptor</p>Fórmula:C34H35F2N3O6Pureza:98%Forma y color:SolidPeso molecular:619.66Butaclamol free base
CAS:<p>Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.</p>Fórmula:C25H31NOPureza:98%Forma y color:SolidPeso molecular:361.52PD 118440
CAS:<p>PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.</p>Fórmula:C11H17N3SPureza:98%Forma y color:SolidPeso molecular:223.34Sch 24518
CAS:<p>Sc h24518 is an antagonist of D1 receptor.</p>Fórmula:C16H17BrClNOPureza:98%Forma y color:SolidPeso molecular:354.67Dicarbine
CAS:<p>Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.</p>Fórmula:C13H18N2Pureza:98%Forma y color:SolidPeso molecular:202.3L-750,667 Trihydrochloride
CAS:<p>L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.</p>Fórmula:C18H22Cl3IN4Pureza:99.63%Forma y color:SolidPeso molecular:527.666-Chloromelatonin
CAS:<p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>Fórmula:C13H15ClN2O2Pureza:98.01% - 99.25%Forma y color:SolidPeso molecular:266.72A-77636
CAS:<p>A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50</p>Fórmula:C20H27NO3Pureza:98%Forma y color:SolidPeso molecular:329.43D4R agonist-1
CAS:<p>D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.</p>Fórmula:C19H22N4SPureza:98.44%Forma y color:SolidPeso molecular:338.47PG 01037 dihydrochloride
CAS:<p>PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.</p>Fórmula:C26H28Cl4N4OPureza:99.89%Forma y color:SolidPeso molecular:554.34SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Fórmula:C18H20ClNO2Pureza:98.68%Forma y color:SolidPeso molecular:317.81WAY-260022
CAS:<p>WAY-260022 is the norepinephrine transporter inhibitor.</p>Fórmula:C21H31F3N2O2Pureza:97.61% - 99.41%Forma y color:SolidPeso molecular:400.48UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Fórmula:C23H28Cl2N4O2Pureza:98.78% - 98.78%Forma y color:SolidPeso molecular:463.4Medifoxamine
CAS:<p>Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine</p>Fórmula:C16H19NO2Pureza:97.14%Forma y color:SolidPeso molecular:257.33Halopemide
CAS:<p>Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).</p>Fórmula:C21H22ClFN4O2Pureza:96.57%Forma y color:SolidPeso molecular:416.88Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Forma y color:SolidPeso molecular:381.44SB-277011
CAS:<p>SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).</p>Fórmula:C28H30N4OPureza:99.39%Forma y color:SolidPeso molecular:438.56Milenperone
CAS:<p>Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.</p>Fórmula:C22H23ClFN3O2Pureza:98.09% - 99.84%Forma y color:SolidPeso molecular:415.89PF-00217830
CAS:<p>PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.</p>Fórmula:C26H30N4O2Pureza:98.72%Forma y color:SolidPeso molecular:430.54U 99194 maleate
CAS:<p>U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.</p>Fórmula:C21H31NO6Pureza:99.45%Forma y color:SolidPeso molecular:393.47PD 168568 dihydrochloride
CAS:<p>PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).</p>Fórmula:C22H29Cl2N3OPureza:99.71%Forma y color:SolidPeso molecular:422.39NGD 94-1
CAS:<p>NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.</p>Fórmula:C18H20N6Pureza:99.61%Forma y color:SolidPeso molecular:320.39MLS1547
CAS:<p>MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).</p>Fórmula:C19H19ClN4OPureza:99.64%Forma y color:SolidPeso molecular:354.837-Hydroxy-DPAT hydrobromide
CAS:<p>7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.</p>Fórmula:C16H26BrNOPureza:99.73%Forma y color:SolidPeso molecular:328.29GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Fórmula:C28H34Cl2N2OPureza:98.08%Forma y color:SolidPeso molecular:485.49Seridopidine
CAS:<p>Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.</p>Fórmula:C14H20FNO2SPureza:99.65%Forma y color:SolidPeso molecular:285.38Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Fórmula:C14H20FNO2SPureza:99.39%Forma y color:SolidPeso molecular:285.38Molindone
CAS:<p>Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.</p>Fórmula:C16H24N2O2Pureza:99.37% - 99.46%Forma y color:Off-White SolidPeso molecular:276.37A-437203
CAS:<p>A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.</p>Fórmula:C20H27F3N6OSPureza:98.80%Forma y color:SolidPeso molecular:456.53BP14979
CAS:<p>BP14979 is D3R-selective partial agonist.</p>Fórmula:C23H34N4O2Pureza:98.29% - 99.73%Forma y color:SolidPeso molecular:398.54SK609 HCl
CAS:<p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>Fórmula:C10H15Cl2NPureza:99.02%Forma y color:SolidPeso molecular:220.14Remoxipride hydrochloride
CAS:<p>Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-</p>Fórmula:C16H24BrClN2O3Pureza:99.88%Forma y color:SolidPeso molecular:407.73CyPPA
CAS:<p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>Fórmula:C16H23N5Pureza:99.88%Forma y color:SolidPeso molecular:285.39Fananserin
CAS:<p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>Fórmula:C23H24FN3O2SPureza:99.88%Forma y color:SolidPeso molecular:425.52CCG 203769
CAS:<p>CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.</p>Fórmula:C8H14N2O2SPureza:99.88%Forma y color:SolidPeso molecular:202.27Sonepiprazole
CAS:<p>Sonepiprazole (PNU-101387G) is a chemical compound known for its selective antagonistic properties toward D4 dopamine receptors, exhibiting dissociation</p>Fórmula:C21H27N3O3SPureza:99.81%Forma y color:SolidPeso molecular:401.52CY 208-243
CAS:<p>CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.</p>Fórmula:C19H18N2Pureza:98%Forma y color:SolidPeso molecular:274.36Timiperone
CAS:<p>Timiperone exhibits a high affinity for cerebral dopamine D2 receptors, demonstrating antipsychotic activity as it mitigates stereotyped behavior.</p>Fórmula:C22H24FN3OSPureza:98%Forma y color:SolidPeso molecular:397.51ABT-670
CAS:<p>ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.</p>Fórmula:C19H23N3O2Pureza:98%Forma y color:SolidPeso molecular:325.4SKF 81297
CAS:<p>SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].</p>Fórmula:C16H16ClNO2Pureza:98%Forma y color:SolidPeso molecular:289.76FAUC-312
CAS:<p>FAUC-312 is a potent and selective agonist of the dopamine D4 receptor.</p>Fórmula:C21H26N4Pureza:98%Forma y color:SolidPeso molecular:334.46LY3154885
CAS:<p>LY3154885 is an orally active dopamine D1 receptor orthosteric modulator (PAM) that reduces the risk of drug-drug interactions (DDI).</p>Fórmula:C23H23Cl2N3O2Forma y color:SolidPeso molecular:444.35Quinpirole dihydrochloride
CAS:<p>Quinpirole dihydrochloride is an agonist of the D2-like dopamine receptor.</p>Fórmula:C13H23Cl2N3Pureza:98%Forma y color:SolidPeso molecular:292.25Pentiapine
CAS:<p>Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.</p>Fórmula:C15H17N5SPureza:99.35%Forma y color:SolidPeso molecular:299.39AJ-76 hydrochloride
CAS:<p>AJ-76 hydrochloride ((+)-AJ 76 hydrochloride) serves as a dopamine autoreceptor antagonist, exhibiting pK i values of 6.95 for hD3, 6.67 for hD4, 6.37 for hD2S, 6.21 for hD2L, and 6.07 for rD2 receptors, indicating its binding affinity strength across these receptor types.</p>Fórmula:C15H24ClNOForma y color:SolidPeso molecular:269.81Carbidine dihydrochloride
CAS:<p>Carbidine, a gamma-carboline derivative, is an atypical antipsychotic that modulates dopamine release and tyrosine hydroxylase activity.</p>Fórmula:C13H20Cl2N2Pureza:98.59%Forma y color:SolidPeso molecular:275.217UWA-101 hydrochloride
CAS:<p>UWA-101 hydrochloride is a selective, non-cytotoxic inhibitor of DAT/SERT, demonstrating EC50 values of 3.6 µM for DAT and 2.3 µM for SERT inhibition. It mitigates motor disorders and other side effects associated with dopaminergic agent use (e.g., L-DOPA) without exhibiting psychotropic effects. This compound is utilized in research focused on neurodegenerative conditions like Parkinson's disease [1] [2].</p>Fórmula:C13H18ClNO2Forma y color:SolidPeso molecular:255.74SB-414796
CAS:<p>SB-414796 is a selective antagonist of the dopamine D3 receptor.</p>Fórmula:C29H36N4O4SPureza:98%Forma y color:SolidPeso molecular:536.69Naxagolide free base
CAS:<p>Naxagolide is a sustained release formulation. It is a dopamine agonist.</p>Fórmula:C15H21NO2Pureza:98%Forma y color:SolidPeso molecular:247.33Dihydrexidine
CAS:<p>Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.</p>Fórmula:C17H17NO2Pureza:98%Forma y color:SolidPeso molecular:267.32Z1078601926
CAS:<p>Z1078601926 is an allosteric inhibitor of the human dopamine transporter (hDAT) and exhibits a synergistic effect when combined with Nomifensine [1].</p>Fórmula:C14H19FN2OForma y color:SolidPeso molecular:250.31Carmoxirole hydrochloride
CAS:<p>Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity in vivo.</p>Fórmula:C24H27ClN2O2Pureza:99.37% - 99.62%Forma y color:SolidPeso molecular:410.94PW0464
CAS:<p>PW0464 ((Rac)-Razpipadon) is a non-catechol D1R agonist and potent omplete G protein biased ligand with an EC50 (Gs-cAMP)=5.8 nM for neurological disorders.</p>Fórmula:C19H17F2N3O4Pureza:98.78%Forma y color:SolidPeso molecular:389.35LBT 999
CAS:<p>LBT 999 is used as a dopamine reuptake inhibitor.</p>Fórmula:C20H26FNO2Forma y color:SolidPeso molecular:331.42JNJ-37822681 dihydrochloride
CAS:<p>JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的，可快速解离的多巴胺 D2受体拮抗剂，与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。</p>Fórmula:C17H19Cl2F5N4Pureza:99.78%Forma y color:SolidPeso molecular:445.26(+)-Dihydrexidine hydrochloride
CAS:<p>(+)-Dihydrexidine hydrochloride is an agonist of dopamine D1 receptor(EC50 of 72± 21 nM).</p>Fórmula:C17H18ClNO2Pureza:98%Forma y color:SolidPeso molecular:303.78Brilaroxazine
CAS:<p>Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.</p>Fórmula:C22H25Cl2N3O3Pureza:99.36%Forma y color:SolidPeso molecular:450.36LY-368975
CAS:<p>LY-368975 is a potent and selective inhibitor of the norepinephrine (NE) reuptake site. LY-368975 reduces food consumption in rodents.</p>Fórmula:C17H21NOSForma y color:SolidPeso molecular:287.42SKF 81297 hydrobromide
CAS:<p>SKF 81297 hydrobromide, a selective agonist of the dopamine D1-like receptor，exhibits central activity and is widely used to study the neuromodulatory effects.</p>Fórmula:C16H17BrClNO2Pureza:99.52%Forma y color:SolidPeso molecular:370.67CP-293019
CAS:<p>CP-293019 is a potent, selective antagonist of dopamine D4 receptor.</p>Fórmula:C19H22F2N4OPureza:98%Forma y color:SolidPeso molecular:360.44-Amino-PPHT Hydrobromide
CAS:<p>4-Amino-PPHT Hydrobromide is a precursor for fluorescent labeled Dopamine D2 receptors agonist.</p>Fórmula:C21H28N2OPureza:98%Forma y color:SolidPeso molecular:324.46PAOPA
CAS:<p>dopamine D2 receptor modulator</p>Fórmula:C11H18N4O3Pureza:>99.99%Forma y color:SolidPeso molecular:254.29NMI 8739
CAS:<p>NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.</p>Fórmula:C30H41NO3Pureza:98.51%Forma y color:SolidPeso molecular:463.65Lumateperone
CAS:<p>Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).</p>Fórmula:C24H28FN3OPureza:99.68% - 99.91%Forma y color:SolidPeso molecular:393.5Dopamine D3 receptor antagonist-1
<p>Dopamine D3 receptor antagonist-1 is a dopamine D3 receptor selective or multi-targeting ligand with a Ki value of 1.58 nM that has demonstrated therapeutic</p>Fórmula:C31H35Cl2N3O3Forma y color:SolidPeso molecular:568.53D4R antagonist-1
<p>Potent, selective D4R antagonist; IC50 = 6.87 µM; potential in Parkinson’s disease research.</p>Fórmula:C21H25F2NO2Forma y color:SolidPeso molecular:361.43CM699
CAS:<p>CM699 is an effective dual inhibitor of the dopamine transporter (DAT) and Sigma receptor (σR), with IC50 values of 311 nM and 14.1 nM, respectively.</p>Fórmula:C24H29N3O2Forma y color:SolidPeso molecular:391.51Dopamine D3 receptor ligand-1
<p>Dopamine D 3 receptor ligand is a potent, selective, high-affinity dopamine D3 receptor ligand that is 89 times more selective for D3 (Ki: 8 nM) than D2 (Ki:</p>Fórmula:C27H29N5OForma y color:SolidPeso molecular:439.55D1R antagonist 1
CAS:<p>Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].</p>Fórmula:C22H26BrNO4Pureza:98%Forma y color:SolidPeso molecular:448.35Dopamine D3 receptor antagonist-2
<p>Dopamine D3 receptor antagonist-2 is a dopamine D3 receptor selective (Ki=2.16 nM) or multi-targeting dual ligand that shows potential effects in CNS disorders.</p>Fórmula:C23H27Cl2N3O3Forma y color:SolidPeso molecular:464.38UNC10099984A
CAS:<p>UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, exhibiting a Ki value of 4.6 nM and an EC50 of 6.2 nM for β-arrestin. This compound is useful for research into central nervous system diseases related to the D2 receptor.</p>Fórmula:C24H29Cl2N3O2Forma y color:SolidPeso molecular:462.41Neflumozide
CAS:<p>Neflumozide (HRP 913) is an orally effective derivative of benzisoxazole, characterized by its potent dopamine antagonist properties and antipsychotic activity. It is utilized in research related to psychiatric disorders.</p>Fórmula:C22H23FN4O2Forma y color:SolidPeso molecular:394.44NMDAR antagonist 5
CAS:<p>NMDAR antagonist 5 (Compound A17) is a multi-target antagonist that acts on NMDAR and monoamine transporters (SERT, DAT, and NET). It demonstrates strong NMDAR antagonistic efficacy (IC50= 0.3 μM) and effective activity on monoamine transporters (SERT IC50= 1.1 μM, DAT IC50= 0.7 μM, NET IC50= 2.7 μM). NMDAR antagonist 5 exhibits high safety with low toxicity (hepatic and renal toxicity IC50> 100 μM; cardiac toxicity IC50= 24.5 μM). It has antidepressant properties and is useful for depression research.</p>Fórmula:C17H21N3Forma y color:SolidPeso molecular:267.369D4R antagonis-2
<p>Potent D4R antagonist-2: selective, IC50=6.52 μM, good in vitro PK and brain penetration, potential for Parkinson's research.</p>Fórmula:C21H23ClF2N2O2Forma y color:SolidPeso molecular:408.87Lisuride
CAS:<p>Lisuride: an oral D2 dopamine agonist, ergot derivative, used in Parkinson's, migraine, and high prolactin research.</p>Fórmula:C20H26N4OForma y color:SolidPeso molecular:338.45Cendifensine
CAS:<p>Cendifensine functions as a monoamine reuptake inhibitor, targeting the serotonin transporter (SERT), norepinephrine transporter (NET), and dopamine transporter (DAT).</p>Fórmula:C14H17Cl2NOForma y color:SolidPeso molecular:286.197Disulergine
CAS:<p>Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.</p>Fórmula:C17H24N4O2SPureza:98%Forma y color:SolidPeso molecular:348.46Dinoxyline
CAS:<p>Dinoxyline is a potent dopamine receptor agonist, with dissociation constants (Ki values) for D1, D2, D3, and D4 receptors being 7 nM, 6 nM, 5 nM, and 43 nM, respectively. It is utilized in neuroscience research.</p>Fórmula:C15H13NO3Forma y color:SolidPeso molecular:255.27
