Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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Spiperone
CAS:<p>Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.</p>Fórmula:C23H26FN3O2Pureza:99.34% - 99.91%Forma y color:SolidPeso molecular:395.47Bromperidol
CAS:<p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>Fórmula:C21H23BrFNO2Pureza:99.89%Forma y color:Tan SolidPeso molecular:420.32Itopride hydrochloride
CAS:<p>Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.</p>Fórmula:C20H27ClN2O4Pureza:99.59%Forma y color:White Or Pale Brownish CrystalPeso molecular:394.9ONC206
CAS:<p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>Fórmula:C23H22F2N4OPureza:99.38% - 99.81%Forma y color:SolidPeso molecular:408.44Quetiapine hemifumarate
CAS:<p>Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.</p>Fórmula:C46H54N6O8S2Pureza:99.32% - >99.99%Forma y color:White Crystalline SolidPeso molecular:883.09Pipamperone
CAS:<p>Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.</p>Fórmula:C21H30FN3O2Pureza:99.85%Forma y color:White PowderPeso molecular:375.48Oxidopamine hydrobromide
CAS:<p>Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.</p>Fórmula:C8H12BrNO3Pureza:98.22% - 99.88%Forma y color:Beige To Brown Fine Crystalline PowderPeso molecular:250.09UCM-1306
CAS:<p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>Fórmula:C14H14FNO2SPureza:99.98%Forma y color:SoildPeso molecular:279.33Haloperidol
CAS:<p>Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.</p>Fórmula:C21H23ClFNO2Pureza:98.69% - 98.97%Forma y color:Crystals SolidPeso molecular:375.86Fluphenazine dihydrochloride
CAS:<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Fórmula:C22H28Cl2F3N3OSPureza:99.23%Forma y color:Off-White SolidPeso molecular:510.44D5R agonist 1
<p>D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.</p>Forma y color:Odour SolidDETQ
CAS:<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Fórmula:C22H25Cl2NO3Forma y color:SolidPeso molecular:422.34Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Fórmula:C27H22F4N4O3SPureza:98.83%Forma y color:SolidPeso molecular:558.55Vanicoside E
CAS:<p>Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .</p>Fórmula:C53H52O22Forma y color:SolidPeso molecular:1040.97Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Forma y color:Odour SolidFenoldopam
CAS:<p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>Fórmula:C16H16ClNO3Pureza:98%Forma y color:SolidPeso molecular:305.767-Hydroxy-PIPAT maleate
CAS:<p>7-Hydroxy-PIPAT maleate is a D3R agonist.</p>Fórmula:C16H22INOForma y color:SolidPeso molecular:371.262[18F]-Labeled L-dopa precursor
CAS:<p>[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].</p>Fórmula:C35H36N2O7Forma y color:SolidPeso molecular:596.67Neuromedin N
CAS:<p>Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.</p>Fórmula:C38H63N7O8Pureza:98%Forma y color:SolidPeso molecular:745.95ABT 724 trihydrochloride
CAS:<p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>Fórmula:C17H22Cl3N5Pureza:99.91%Forma y color:SolidPeso molecular:402.75Octodrine
CAS:<p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>Fórmula:C8H19NPureza:99.98%Forma y color:Clear Colorless To Light Yellow LiquidPeso molecular:129.24Clomipramine D3
CAS:<p>Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).</p>Fórmula:C19H23ClN2Pureza:98%Forma y color:SolidPeso molecular:317.87MLS1082
CAS:<p>MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.</p>Fórmula:C24H23N3O2Pureza:99.53%Forma y color:SolidPeso molecular:385.46D3R/MOR antagonist 1
<p>Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM</p>Fórmula:C22H27Cl2N3OPureza:98%Forma y color:SolidPeso molecular:420.38Dopamine D2 receptor agonist-2
CAS:<p>Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.</p>Fórmula:C25H31Cl2N5OSPureza:98.93%Forma y color:SoildPeso molecular:520.52ADTN hydrobromide
CAS:<p>ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).</p>Fórmula:C10H14BrNO2Forma y color:SolidPeso molecular:260.13Amisulpride hydrochloride
CAS:<p>Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.</p>Fórmula:C17H28ClN3O4SForma y color:SolidPeso molecular:405.94MOR agonist-2
<p>Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.</p>Fórmula:C37H47Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:680.71LE 300
CAS:<p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>Fórmula:C20H22N2Pureza:97.91% - 98.79%Forma y color:SolidPeso molecular:290.4Moperone
CAS:<p>Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.</p>Fórmula:C22H26FNO2Forma y color:SolidPeso molecular:355.45D3R ligand 1
<p>D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.</p>Fórmula:C27H37NO5Pureza:98%Forma y color:SolidPeso molecular:455.59ADTN
CAS:<p>ADTN is an agonist of the dopamine receptor.</p>Fórmula:C10H13NO2Pureza:98%Forma y color:SolidPeso molecular:179.22Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Fórmula:C26H37N5O2Pureza:97.69% - 99.86%Forma y color:White Crystalline SolidPeso molecular:451.6A 77636 hydrochloride
CAS:<p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>Fórmula:C20H28ClNO3Pureza:99.57%Forma y color:SolidPeso molecular:365.89O-2172
CAS:<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Fórmula:C14H16Cl2O2Forma y color:SolidPeso molecular:287.18(R)-Preclamol hydrochloride
CAS:<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Haloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Preclamol hydrochloride
CAS:<p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Secretoneurin, rat
CAS:<p>Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).</p>Fórmula:C159H252N40O58Pureza:98%Forma y color:SolidPeso molecular:3651.95Fluphenazine free base
CAS:<p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>Fórmula:C22H26F3N3OSForma y color:SolidPeso molecular:437.52Adrogolide HCl
CAS:<p>Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.</p>Fórmula:C22H26ClNO4SForma y color:SolidPeso molecular:435.96N-0500 HCl
CAS:<p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>Fórmula:C15H22ClNO2Pureza:98.85% - 99.54%Forma y color:SolidPeso molecular:283.79(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Fórmula:C22H24ClF4N5OSPureza:98.36%Forma y color:SoildPeso molecular:517.97Quinelorane
CAS:<p>Quinelorane is dextrorotary isomer.</p>Fórmula:C14H22N4Forma y color:SolidPeso molecular:246.35PF-4363467
CAS:<p>PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.</p>Fórmula:C22H30N2O3SForma y color:SolidPeso molecular:402.55D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Fórmula:C25H31ClN2OPureza:98%Forma y color:SolidPeso molecular:410.98ST-836 hydrochloride
CAS:<p>ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .</p>Fórmula:C23H35ClN4OSPureza:98%Forma y color:SolidPeso molecular:451.07cis-(Z)-Flupentixol dihydrochloride
CAS:<p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>Fórmula:C23H27Cl2F3N2OSPureza:98.07%Forma y color:SolidPeso molecular:507.44Haloperidol (D4')
CAS:<p>Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.</p>Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Eticlopride hydrochloride
CAS:<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Fórmula:C17H25ClN2O3·HClPureza:98%Forma y color:SolidPeso molecular:377.31
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