
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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Lenperone HCl
CAS:<p>Lenperone HCl is a dopamine antagonist and an antipsychotic agent.</p>Fórmula:C22H24ClF2NO2Pureza:98%Forma y color:SolidPeso molecular:407.88(-)-GSK598809
CAS:<p>(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.</p>Fórmula:C22H23F4N5OSPureza:98%Forma y color:SolidPeso molecular:481.51Tesofensine
CAS:<p>Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.</p>Fórmula:C17H23Cl2NOPureza:98%Forma y color:SolidPeso molecular:328.28Acetophenazine
CAS:<p>Acetophenazine is an anxiolytic compound that is used in the study of depression.</p>Fórmula:C23H29N3O2SPureza:99.30%Forma y color:SoildPeso molecular:411.56GBR 12783
CAS:<p>GBR 12783 enhances memory, boosts rat hippocampal acetylcholine, and is a potent dopamine uptake inhibitor with IC50s of 1.8/1.2 nM in rats/mice.</p>Fórmula:C28H32N2OPureza:98%Forma y color:SolidPeso molecular:412.57ST-836
CAS:<p>ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .</p>Fórmula:C23H34N4OSPureza:98%Forma y color:SolidPeso molecular:414.61Org-10490
CAS:<p>Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.</p>Fórmula:C17H19NOPureza:98%Forma y color:SolidPeso molecular:253.34L 741742 hydrochloride
CAS:<p>L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.</p>Fórmula:C23H26Cl2N2OPureza:99.9%Forma y color:SolidPeso molecular:417.37A68930
CAS:<p>A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.</p>Fórmula:C16H17NO3Forma y color:SolidPeso molecular:271.31Remoxipride
CAS:<p>Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.</p>Fórmula:C16H23BrN2O3Pureza:98%Forma y color:SolidPeso molecular:371.27PF-06256142
CAS:<p>PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).</p>Fórmula:C21H16N4O2Pureza:98%Forma y color:SolidPeso molecular:356.38YQA14
CAS:<p>YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.</p>Fórmula:C23H27ClN4O3Pureza:99.52%Forma y color:SolidPeso molecular:442.94PF-592379
CAS:<p>PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).</p>Fórmula:C13H21N3OPureza:98%Forma y color:SolidPeso molecular:235.33PD 119819
CAS:<p>PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.</p>Fórmula:C21H25Cl2N3O3Pureza:98%Forma y color:SolidPeso molecular:438.35ADR-851 HCl
CAS:<p>ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.</p>Fórmula:C14H19Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:332.23CAD031
CAS:<p>CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.</p>Fórmula:C18H14F6N2O2Forma y color:SolidPeso molecular:404.31R-SKF-38393A HCl
CAS:<p>R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.</p>Fórmula:C16H18ClNO2Pureza:98%Forma y color:SolidPeso molecular:291.77Mosapramine
CAS:<p>Mosapramine is a dopamine D2-receptor antagonist.</p>Fórmula:C28H35ClN4OPureza:98%Forma y color:SolidPeso molecular:479.06Sultopride
CAS:<p>Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.</p>Fórmula:C17H26N2O4SForma y color:SolidPeso molecular:354.46U-101958 Maleate
CAS:<p>U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.</p>Fórmula:C25H33N3O5Pureza:98%Forma y color:SolidPeso molecular:455.55NGB 2904 hydrochloride
CAS:<p>dopamine D3 receptor antagonist</p>Fórmula:C28H30Cl3N3OPureza:98%Forma y color:SolidPeso molecular:530.92Oxiperomide
CAS:<p>Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.</p>Fórmula:C20H23N3O2Pureza:98%Forma y color:SolidPeso molecular:337.42PD-89211
CAS:<p>PD 89211 selectively blocks dopamine D4.2 receptor >800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).</p>Fórmula:C19H21ClN4OPureza:98%Forma y color:SolidPeso molecular:356.85R(+)-6-Bromo-APB HBr
CAS:<p>R(+)-6-Bromo-APB HBr is used as a D1 Dopamine receptor agonist.</p>Fórmula:C19H21Br2NO2Pureza:98%Forma y color:SolidPeso molecular:455.18SKF 83959 hydrobromide
CAS:<p>SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.</p>Fórmula:C18H21BrClNO2Pureza:98%Forma y color:SolidPeso molecular:398.72CGP 25454A
CAS:<p>CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.</p>Fórmula:C15H21Cl2N3O2Forma y color:SolidPeso molecular:346.25ST-198
CAS:<p>ST-198 is a dopamine D3 receptor antagonist.</p>Fórmula:C22H26N2OPureza:98%Forma y color:SolidPeso molecular:334.45Piperidine-MO-1
CAS:<p>Piperidine-MO-1 is a dopamine receptor modulator, with an ED50 of 68 μmol/kg on increase of DOPAC in the rat striatum.</p>Fórmula:C14H21ClFNO2SPureza:99.88%Forma y color:SolidPeso molecular:321.84SKF83822 hydrobromide
CAS:<p>SKF83822 hydrobromide is a dopamine D1-like receptor agonist.</p>Fórmula:C20H23BrClNO2Pureza:98%Forma y color:SolidPeso molecular:424.76CL-216303 HCl
CAS:<p>CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.</p>Fórmula:C11H12Cl3NPureza:98%Forma y color:SolidPeso molecular:264.58SKF-82958
CAS:<p>SKF 82958 is a D1/D5 receptor full agonist.</p>Fórmula:C19H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:329.82Dopamine D2 receptor antagonist-1
CAS:<p>Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.</p>Fórmula:C14H17N3SPureza:99.86%Forma y color:SolidPeso molecular:259.37(+)-UH 232 maleate
CAS:<p>D2 antagonist</p>Fórmula:C18H29NOPureza:98%Forma y color:SolidPeso molecular:275.43A412997
CAS:<p>A412997 is a selective agonist of dopamine D4 receptor.</p>Fórmula:C19H23N3OPureza:98%Forma y color:SolidPeso molecular:309.41S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Fórmula:C16H20ClN3OSForma y color:SolidPeso molecular:337.87FR 64822
CAS:<p>FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.</p>Fórmula:C11H14N4OForma y color:SolidPeso molecular:218.26SV-156
CAS:<p>SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).</p>Fórmula:C21H23BrN2O2Forma y color:SolidPeso molecular:415.32Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Fórmula:C22H26ClNPureza:98%Forma y color:SolidPeso molecular:339.9Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Fórmula:C20H25BrN4OForma y color:SolidPeso molecular:417.34SKF-104557
CAS:<p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>Fórmula:C13H18N2OForma y color:SolidPeso molecular:218.29A 68930 hydrochloride
CAS:<p>A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].</p>Fórmula:C16H18ClNO3Forma y color:Off-White SolidPeso molecular:307.77SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Forma y color:SolidPeso molecular:376.29Tau-aggregation-IN-1
CAS:<p>Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).</p>Fórmula:C28H37N5O2SForma y color:SolidPeso molecular:507.69DOV-216,303 Free Base
CAS:<p>DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.</p>Fórmula:C11H11Cl2NPureza:96.7%Forma y color:SolidPeso molecular:228.12Octoclothepin maleate salt
CAS:<p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>Fórmula:C23H25ClN2O4SForma y color:SolidPeso molecular:460.97RTI 336
CAS:<p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>Fórmula:C24H26Cl2N2OPureza:98%Forma y color:SolidPeso molecular:429.38SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Fórmula:C17H20BrNO2Forma y color:SolidPeso molecular:350.25UNC9995
CAS:<p>UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).</p>Fórmula:C20H21Cl2N3OSPureza:98%Forma y color:SolidPeso molecular:422.37NPEC-caged-dopamine
CAS:<p>Dopamine receptor agonist</p>Fórmula:C17H18N2O6Pureza:98%Forma y color:SolidPeso molecular:346.33RBI-257 Maleate
CAS:<p>RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.</p>Fórmula:C25H32IN3O5Forma y color:SolidPeso molecular:581.44
