Receptor de adenosina
Los receptores de adenosina son una clase de GPCR que responden al nucleósido endógeno adenosina. Estos receptores están involucrados en la regulación de diversos procesos fisiológicos, incluidos la función cardiovascular, los ciclos sueño-vigilia y las respuestas inmunitarias. Los moduladores de los receptores de adenosina tienen un potencial terapéutico en el tratamiento de afecciones como las arritmias cardíacas, la inflamación y las enfermedades neurodegenerativas. En CymitQuimica, ofrecemos una selección de moduladores de receptores de adenosina de alta calidad para apoyar su investigación en biología cardiovascular, neurociencia e inmunología.
Se han encontrado 251 productos de "Receptor de adenosina"
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VUF 5574
CAS:VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.Fórmula:C21H17N5O2Pureza:99.53%Forma y color:SolidPeso molecular:371.39Neladenoson dalanate HCl
CAS:Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).Fórmula:C35H35Cl2N7O4S2Pureza:98%Forma y color:SolidPeso molecular:752.73Cirazoline hydrochloride
CAS:Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.Fórmula:C13H17ClN2OPureza:99.863%Forma y color:SolidPeso molecular:252.74Naxifylline
CAS:Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.Fórmula:C18H24N4O3Forma y color:SolidPeso molecular:344.41A3AR antagonist 1
CAS:A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.Fórmula:C32H24N4O4SForma y color:SolidPeso molecular:560.62A2AR-antagonist-1
CAS:Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Fórmula:C27H25N5O2Pureza:98%Forma y color:SolidPeso molecular:451.52WRC-0571
CAS:WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.Fórmula:C17H26N6OPureza:98%Forma y color:SolidPeso molecular:330.43Adenosine receptor antagonist 2
CAS:Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.Fórmula:C23H21FN8OForma y color:SolidPeso molecular:444.46Bamifylline Hydrochloride
CAS:Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.Fórmula:C20H28ClN5O3Forma y color:SolidPeso molecular:421.92VUF8504
CAS:VUF8504 is a novel ligand of adenosine A3 receptor.Fórmula:C22H17N3O2Forma y color:SolidPeso molecular:355.39MRS1067
CAS:MRS1067 is an antagonist of A3 adenosine receptor.Fórmula:C19H16Cl2O3Forma y color:SolidPeso molecular:363.23CAY10498
CAS:A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.Fórmula:C18H20N6Forma y color:SolidPeso molecular:320.39VUF8507
CAS:Vuf8507 is an allosteric regulator of adenosine receptor.Fórmula:C21H15N3OForma y color:SolidPeso molecular:325.36PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFórmula:C14H12F3NOSPureza:98%Forma y color:SolidPeso molecular:299.31Sipagladenant
CAS:Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.Fórmula:C20H19N3O4SForma y color:SolidPeso molecular:397.45SCH-202676 HBr
CAS:SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.Fórmula:C15H13N3SPureza:98%Forma y color:SolidPeso molecular:267.35A3AR antagonist 2
CAS:A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.Fórmula:C22H16N6O3Forma y color:SolidPeso molecular:412.4TH-162
CAS:TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.Fórmula:C19H23N5O4Forma y color:SolidPeso molecular:385.42PQ-69
CAS:PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.Fórmula:C20H19FN4OForma y color:SolidPeso molecular:350.39MRS 1523
CAS:MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.Fórmula:C23H29NO3SPureza:98%Forma y color:SolidPeso molecular:399.55Inupadenant
CAS:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].Fórmula:C25H26F2N8O4S2Forma y color:SolidPeso molecular:604.65CAY10680
CAS:CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.Fórmula:C18H16N2O2SForma y color:SolidPeso molecular:324.4FR-194921
CAS:FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.Fórmula:C23H23N5OForma y color:SolidPeso molecular:385.46CVT-2759
CAS:CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.Fórmula:C17H24N6O6Forma y color:SolidPeso molecular:408.41Adenosine receptor inhibitor 2
CAS:Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.Fórmula:C17H20BrN5O2Forma y color:SolidPeso molecular:406.28Acefylline piperazine
CAS:Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.Fórmula:C9H10N4O4·xC4H10N2Forma y color:SolidPeso molecular:562.54JNJ-40255293
CAS:JNJ-40255293 is an antagonist of adenosine A2A/A1.Fórmula:C23H22N4O3Pureza:98%Forma y color:SolidPeso molecular:402.45AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Fórmula:C22H21N3O4Forma y color:SolidPeso molecular:391.42ATL-801
CAS:ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.Fórmula:C24H25N7O3Forma y color:SolidPeso molecular:459.5N-[(4-Aminophenyl)methyl]adenosine
CAS:N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Fórmula:C17H20N6O4Pureza:98.75%Forma y color:SolidPeso molecular:372.38Ref: TM-T16166
1mg52,00€5mg111,00€1mL*10mM (DMSO)141,00€10mg166,00€25mg318,00€50mg504,00€100mg803,00€ISAM-140
CAS:ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.Fórmula:C19H19N3O3Pureza:99.51%Forma y color:SolidPeso molecular:337.37APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Fórmula:C18H22N6O4Pureza:99.88%Forma y color:SolidPeso molecular:386.41N6-Cyclopentyladenosine
CAS:N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFórmula:C15H21N5O4Pureza:99.95%Forma y color:SolidPeso molecular:335.36FK-453
CAS:FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Fórmula:C23H25N3O2Pureza:99.44%Forma y color:SolidPeso molecular:375.46Selodenoson
CAS:Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Fórmula:C17H24N6O4Pureza:99.39%Forma y color:SolidPeso molecular:376.41GS-9667
CAS:GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFórmula:C21H24FN5O4SPureza:99.77% - 99.96%Forma y color:SolidPeso molecular:461.51N 0861
CAS:N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Fórmula:C13H17N5Pureza:98.78%Forma y color:SolidPeso molecular:243.31Ref: TM-T70722
1mg164,00€2mg234,00€5mg389,00€10mg532,00€25mg820,00€50mg1.063,00€100mg1.423,00€200mg1.945,00€KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Fórmula:C23H18N2O2Pureza:98.33%Forma y color:SolidPeso molecular:354.4Ref: TM-T9238
2mg35,00€5mg55,00€1mL*10mM (DMSO)62,00€10mg95,00€25mg172,00€50mg264,00€100mg399,00€200mg560,00€BAY 60-6583
CAS:BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Fórmula:C19H17N5O2SPureza:98.46% - 99.8%Forma y color:SolidPeso molecular:379.44Ref: TM-T14506
1mg39,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)101,00€10mg116,00€25mg233,00€50mg376,00€100mg567,00€200mg797,00€LAS38096
CAS:LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Fórmula:C17H12N6OPureza:99.18% - 99.95%Forma y color:SolidPeso molecular:316.322'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Fórmula:C16H22ClN5O4Pureza:99.93%Forma y color:SolidPeso molecular:383.83Sonedenoson
CAS:Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.Fórmula:C18H20ClN5O5Pureza:99.79%Forma y color:SolidPeso molecular:421.84A2A receptor antagonist 1
CAS:A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Fórmula:C16H12FN5OPureza:99.52% - 99.93%Forma y color:SolidPeso molecular:309.3Ref: TM-T37792
2mgA consultar200mgA consultar1mL*10mM (DMSO)47,00€5mg62,00€10mg87,00€25mg183,00€50mg280,00€100mg416,00€GW-493838
CAS:GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgiaFórmula:C21H21ClFN7O4Pureza:99.11% - 99.58%Forma y color:SolidPeso molecular:489.89Ref: TM-T27509
1mg143,00€5mg346,00€1mL*10mM (DMSO)399,00€10mg492,00€25mg740,00€50mg999,00€100mg1.350,00€500mg2.647,00€MRS1220
CAS:MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFórmula:C21H14ClN5O2Pureza:98.43%Forma y color:SolidPeso molecular:403.82ANR 94
CAS:ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Fórmula:C9H13N5OPureza:98.9%Forma y color:SolidPeso molecular:207.23Ref: TM-T22031
5mg46,00€1mL*10mM (DMSO)46,00€10mg71,00€25mg130,00€50mg219,00€100mg309,00€200mg434,00€N6-(2-Phenylethyl)adenosine
CAS:N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFórmula:C18H21N5O4Pureza:99.83%Forma y color:SolidPeso molecular:371.39ST-1535
CAS:ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.Fórmula:C12H16N8Pureza:99.64% - 99.69%Forma y color:SolidPeso molecular:272.31Adenosine antagonist-1
CAS:Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
Fórmula:C18H13N7SPureza:99.28% - 99.95%Forma y color:SolidPeso molecular:359.41Evodenoson
CAS:Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Fórmula:C23H29N7O6Pureza:99.75% - 99.83%Forma y color:SolidPeso molecular:499.52
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