Receptor GNRH
Los receptores de la hormona liberadora de gonadotropinas (GnRH) son GPCR que se unen a la GnRH, una hormona responsable de regular la liberación de la hormona luteinizante (LH) y la hormona foliculoestimulante (FSH) de la glándula pituitaria. Estos receptores son cruciales para la función reproductiva y son el objetivo de terapias para condiciones como el cáncer de próstata, la endometriosis y la infertilidad. Los agonistas y antagonistas de los receptores de GnRH también se utilizan en tecnologías de reproducción asistida. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de GnRH de alta calidad para apoyar su investigación en salud reproductiva, endocrinología y terapia hormonal.
Se han encontrado 84 productos de "Receptor GNRH"
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Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Fórmula:C56H78N16O12Pureza:99.81% - >99.99%Forma y color:White PowderPeso molecular:1167.34Ref: TM-T1494
5mg58,00€10mg95,00€25mg115,00€50mg156,00€100mg180,00€500mg452,00€1mL*10mM (DMSO)120,00€Degarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Fórmula:C84H107ClN18O18Pureza:98.66%Forma y color:SolidPeso molecular:1692.34(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Fórmula:C32H30F5N3O5Pureza:99.08%Forma y color:SolidPeso molecular:631.59Ref: TM-T11174
5mg52,00€10mg80,00€25mg144,00€50mg205,00€100mg324,00€200mg477,00€1mL*10mM (DMSO)73,00€Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Fórmula:C72H95ClN14O14Pureza:>99.99%Forma y color:SolidPeso molecular:1416.06[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Fórmula:C58H82N16O12Peso molecular:1195.37Onvitrelin ucalontide
CAS:Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.Fórmula:C163H243N43O32Peso molecular:3316.94Kisspeptin-54(human)
CAS:Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.Fórmula:C258H401N79O78Pureza:98%Forma y color:SolidPeso molecular:5857.49AG 045572
CAS:AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 isFórmula:C30H37NO5Pureza:99.96%Forma y color:SolidPeso molecular:491.62LHRH
CAS:Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFórmula:C55H74N16O14Pureza:98%Forma y color:SolidPeso molecular:1183.27LGnRH-III, lamprey
CAS:GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Fórmula:C59H74N18O14Pureza:98%Forma y color:SolidPeso molecular:1259.33MI 1544
CAS:MI 1544 is a LHRH antagonist.Fórmula:C71H94ClN17O13Forma y color:SolidPeso molecular:1429.09Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS:LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.Fórmula:C60H73N15O13Pureza:98%Forma y color:SolidPeso molecular:1212.31Phoenixin-14
CAS:<p>Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/</p>Fórmula:C75H110N18O20Pureza:98%Forma y color:SolidPeso molecular:1583.78RS 18286
CAS:RS 18286 is a LHRH antagonist.Fórmula:C74H101Cl2N17O14Forma y color:SolidPeso molecular:1523.6LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Fórmula:C56H77N17O13Forma y color:SolidPeso molecular:1196.32Avorelin
CAS:Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.Fórmula:C65H85N17O12Pureza:98%Forma y color:SolidPeso molecular:1296.48(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Fórmula:C64H81N17O14Peso molecular:1312.43APTAA-LHRH
CAS:APTAA-LHRH is a gonadorelin antagonist.Fórmula:C69H91Cl2N17O14Pureza:98%Forma y color:SolidPeso molecular:1453.47Azaline
CAS:Azaline is a gonadorelin antagonist.Fórmula:C74H106ClN23O12Pureza:98%Forma y color:SolidPeso molecular:1545.26Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Fórmula:C27H28F3N3O8SPureza:99.64%Forma y color:SolidPeso molecular:611.59LH-RH (4-10)
CAS:LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Fórmula:C33H53N11O9Peso molecular:747.84Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Fórmula:C58H79N15O15Peso molecular:1226.34(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS:(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Fórmula:C53H62N12O11Peso molecular:1043.13Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Fórmula:C44H80N14O15Peso molecular:1044.59276Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Fórmula:C74H92ClN17O13Pureza:98%Forma y color:SolidPeso molecular:1463.08[D-Phe2,6, Pro3]-LH-RH
CAS:[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Fórmula:C59H80N14O13Peso molecular:1193.35Human follicular gonadotropin releasing peptide
CAS:Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)Fórmula:C68H94N22O27Peso molecular:1651.61Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Fórmula:C162H26N56O44SPeso molecular:3724.17Prolactin Releasing Peptide (1-31), human
CAS:Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).Fórmula:C160H252N56O42SPureza:98%Forma y color:SolidPeso molecular:3664.15Surfagon
CAS:Surfagon is an effective LHRH agonist.Fórmula:C56H78N16O12Pureza:98%Forma y color:SolidPeso molecular:1167.34[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.Fórmula:C67H84N16O13Forma y color:SolidPeso molecular:1321.48[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Fórmula:C54H71N15O14Pureza:98%Forma y color:SolidPeso molecular:1154.23Fsh receptor-binding inhibitor fragment(bi-10)
CAS:FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.Fórmula:C42H67N13O19Forma y color:SolidPeso molecular:1058.06Zebrafish Kisspeptin-1
CAS:Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.Fórmula:C58H84N16O15Forma y color:SolidPeso molecular:1245.39GnRH Associated Peptide (1-24), human
CAS:GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.Fórmula:C117H190N32O43Forma y color:SolidPeso molecular:2732.95LH-RH (7-10)
CAS:LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.Fórmula:C19H36N8O4Forma y color:SolidPeso molecular:440.54(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:<p>Analog of LHRH, stimulates LH and FSH release, controls reproduction.</p>Fórmula:C59H84N18O14Forma y color:SolidPeso molecular:1269.41Kisspeptin-54(human) TFA
Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.Fórmula:C258H401N79O78·C2HF3O2Forma y color:SolidPeso molecular:5971.45sGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Fórmula:C64H83N17O12Forma y color:SolidPeso molecular:1282.45Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Fórmula:C75H110N18O20·xC2HF3O2Pureza:99.11%Forma y color:SolidPeso molecular:1583.78 (free base)Kisspeptin 13
CAS:<p>Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.</p>Fórmula:C78H107N21O18Forma y color:SolidPeso molecular:1626.81Azaline B
CAS:Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.Fórmula:C80H102ClN23O12Forma y color:SolidPeso molecular:1613.27A 76154
CAS:A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Fórmula:C70H93FN12O12Forma y color:SolidPeso molecular:1313.584Wy 43657
CAS:Wy 43657 is a gonadorelin antagonist.Fórmula:C71H86N14O13Pureza:98%Forma y color:SolidPeso molecular:1343.554LUF5771
CAS:LUF5771: potent allosteric recLH & Org 43553 inhibitor, partial LH receptor activator with low efficacy.Fórmula:C24H23NO2Forma y color:SolidPeso molecular:357.44Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Fórmula:C59H84N16O12Forma y color:SolidPeso molecular:1209.4Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFórmula:C61H88N16O14Pureza:98.1%Forma y color:SolidPeso molecular:1269.45Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFórmula:C29H27F2N7O5SPureza:98.64% - 99.97%Forma y color:SolidPeso molecular:623.63Ref: TM-T3630
2mg42,00€5mg62,00€10mg87,00€25mg170,00€50mg264,00€100mg430,00€200mg618,00€1mL*10mM (DMSO)86,00€Sufugolix
CAS:Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.Fórmula:C36H31F2N5O4SPureza:97.78%Forma y color:SolidPeso molecular:667.72Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Fórmula:C23H31FO5Pureza:99.47%Forma y color:CoaPeso molecular:406.49Ref: TM-T21335
2mg47,00€5mg71,00€10mg101,00€25mg188,00€50mg276,00€100mg394,00€200mg520,00€1mL*10mM (DMSO)85,00€Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Fórmula:C55H76N16O12Pureza:>99.99%Forma y color:SolidPeso molecular:1153.29Ref: TM-TP1288
1mg47,00€2mg63,00€5mg96,00€10mg135,00€50mg177,00€100mg264,00€200mg393,00€1mL*10mM (DMSO)170,00€Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Fórmula:C74H100ClN17O18Pureza:98.38%Forma y color:SolidPeso molecular:1551.17Ref: TM-T5520L
1mg52,00€5mg90,00€10mg150,00€25mg291,00€50mg437,00€100mg642,00€500mg1.359,00€1mL*10mM (DMSO)251,00€Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFórmula:C82H117ClN18O15Pureza:96.05%Forma y color:SolidPeso molecular:1630.4LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFórmula:C61H78N18O16Pureza:99.66%Forma y color:SolidPeso molecular:1319.38Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Fórmula:C68H90N18O14Pureza:99.92%Forma y color:SolidPeso molecular:1383.55Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Fórmula:C66H87N17O14Pureza:99.84%Forma y color:SolidPeso molecular:1342.5Buserelin Acetate (57982-77-1 free base)
CAS:Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Fórmula:C62H90N16O15Pureza:99.31% - 99.78%Forma y color:SolidPeso molecular:1299.48Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Fórmula:C66H86N18O15Pureza:99.90%Forma y color:White PowderPeso molecular:1371.53Ref: TM-T21410
5mg55,00€10mg82,00€25mg126,00€50mg182,00€100mg273,00€200mg409,00€1mL*10mM (DMSO)123,00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Fórmula:C32H29F5N3NaO5Pureza:99.71%Forma y color:SolidPeso molecular:653.57Ref: TM-T5031
2mg35,00€5mg52,00€10mg80,00€25mg144,00€50mg227,00€100mg359,00€200mg532,00€1mL*10mM (DMSO)74,00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Fórmula:C68H87N17O15Pureza:99.98%Forma y color:SolidPeso molecular:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFórmula:C22H15F3N2O7SPureza:99.33%Forma y color:SolidPeso molecular:508.42Goserelin acetate
CAS:<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Fórmula:C61H88N18O16Pureza:99.77% - >99.99%Forma y color:White Crystalline PowderPeso molecular:1329.46Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Fórmula:C70H92ClN17O14·xC2H4O2Pureza:97.96%Forma y color:SolidPeso molecular:1491.11Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Fórmula:C55H74N16O13Forma y color:SolidPeso molecular:1167.29Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Fórmula:C80H104ClN21O14Forma y color:SolidPeso molecular:1619.27NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Fórmula:C27H24F3N3O3Forma y color:SolidPeso molecular:495.49EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Fórmula:C15H27N5O6Forma y color:SolidPeso molecular:373.4BAY 1214784
CAS:BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.Fórmula:C29H26ClF4N3O5S2Forma y color:SolidPeso molecular:672.11Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Fórmula:C25H19F3N4O5SPureza:98.60% - 98.97%Forma y color:SolidPeso molecular:544.5BAY-784
CAS:<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Fórmula:C29H26ClF4N3O5S2Pureza:98%Forma y color:SolidPeso molecular:672.115α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFórmula:C21H36O2Forma y color:SolidPeso molecular:320.51T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFórmula:C37H37F2N3O4SPureza:98%Forma y color:SolidPeso molecular:657.77BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Fórmula:C27H21ClFN3O2Pureza:98%Forma y color:SolidPeso molecular:473.93DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Fórmula:C11H17Cl2NOSForma y color:SolidPeso molecular:282.22[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Fórmula:C56H77N17O13Forma y color:SolidPeso molecular:1196.32Abarelix acetate
CAS:Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Fórmula:C72H95ClN14O14·xC2H4O2Forma y color:SolidPeso molecular:1476.14BAY-899
CAS:BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.Fórmula:C25H19F2N5O2Pureza:98%Forma y color:SolidPeso molecular:459.45(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Fórmula:C25H19F2N5O2Forma y color:SolidPeso molecular:459.45GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Fórmula:C31H28F5N7O6SPureza:98%Forma y color:SolidPeso molecular:721.65GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Fórmula:C28H27F2N9O5Pureza:98.08%Forma y color:SolidPeso molecular:607.57Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Fórmula:C80H102ClN15O14Forma y color:SolidPeso molecular:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Fórmula:C36H35F7N4O6Forma y color:SolidPeso molecular:752.68Goserelin acetate(65807-02-5 Free base)
<p>Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.</p>Pureza:99.77%Forma y color:Odour SolidDimethandrolone Undecanoate
CAS:Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Fórmula:C31H50O3Pureza:99.65% - >99.99%Forma y color:SolidPeso molecular:470.73Ref: TM-T27176
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