Receptor GNRH
Los receptores de la hormona liberadora de gonadotropinas (GnRH) son GPCR que se unen a la GnRH, una hormona responsable de regular la liberación de la hormona luteinizante (LH) y la hormona foliculoestimulante (FSH) de la glándula pituitaria. Estos receptores son cruciales para la función reproductiva y son el objetivo de terapias para condiciones como el cáncer de próstata, la endometriosis y la infertilidad. Los agonistas y antagonistas de los receptores de GnRH también se utilizan en tecnologías de reproducción asistida. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de GnRH de alta calidad para apoyar su investigación en salud reproductiva, endocrinología y terapia hormonal.
Se han encontrado 69 productos de "Receptor GNRH"
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LGnRH-III, lamprey acetate(147859-97-0 free base)
<p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>Fórmula:C61H78N18O16Pureza:99.66%Forma y color:SolidPeso molecular:1319.38Cetrorelix Acetate
CAS:<p>Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.</p>Fórmula:C70H92ClN17O14·xC2H4O2Pureza:97.96%Forma y color:SolidPeso molecular:1491.11NBI-42902
CAS:<p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>Fórmula:C27H24F3N3O3Forma y color:SolidPeso molecular:495.49BAY 1214784
CAS:<p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>Fórmula:C29H26ClF4N3O5S2Forma y color:SolidPeso molecular:672.11Argtide
CAS:<p>Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.</p>Fórmula:C80H104ClN21O14Forma y color:SolidPeso molecular:1619.27Opigolix
CAS:<p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>Fórmula:C25H19F3N4O5SPureza:98.60% - 98.97%Forma y color:SolidPeso molecular:544.5BAY-298
CAS:<p>BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.</p>Fórmula:C27H21ClFN3O2Pureza:98%Forma y color:SolidPeso molecular:473.93[D-Ala6]-LH-RH
CAS:<p>[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].</p>Fórmula:C56H77N17O13Forma y color:SolidPeso molecular:1196.32T 98475
CAS:<p>gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active</p>Fórmula:C37H37F2N3O4SPureza:98%Forma y color:SolidPeso molecular:657.77BAY-784
CAS:<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Fórmula:C29H26ClF4N3O5S2Pureza:98%Forma y color:SolidPeso molecular:672.11DCOIT
CAS:<p>DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].</p>Fórmula:C11H17Cl2NOSForma y color:SolidPeso molecular:282.22Abarelix acetate
CAS:<p>Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.</p>Fórmula:C72H95ClN14O14·xC2H4O2Forma y color:SolidPeso molecular:1476.14BAY-899
CAS:<p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>Fórmula:C25H19F2N5O2Pureza:98%Forma y color:SolidPeso molecular:459.45Acyline
CAS:<p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>Fórmula:C80H102ClN15O14Forma y color:SolidPeso molecular:1533.21Merigolix
CAS:<p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>Fórmula:C36H35F7N4O6Forma y color:SolidPeso molecular:752.68GnRH-R antagonist 1
CAS:<p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>Fórmula:C31H28F5N7O6SPureza:98%Forma y color:SolidPeso molecular:721.65GnRH antagonist 2
CAS:<p>GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.</p>Fórmula:C28H27F2N9O5Pureza:98.08%Forma y color:SolidPeso molecular:607.57(R)-BAY-899
<p>(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.</p>Fórmula:C25H19F2N5O2Forma y color:SolidPeso molecular:459.45Dimethandrolone Undecanoate
CAS:<p>Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.</p>Fórmula:C31H50O3Pureza:99.65% - >99.99%Forma y color:SolidPeso molecular:470.73Ref: TM-T27176
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