Receptor GNRH
Los receptores de la hormona liberadora de gonadotropinas (GnRH) son GPCR que se unen a la GnRH, una hormona responsable de regular la liberación de la hormona luteinizante (LH) y la hormona foliculoestimulante (FSH) de la glándula pituitaria. Estos receptores son cruciales para la función reproductiva y son el objetivo de terapias para condiciones como el cáncer de próstata, la endometriosis y la infertilidad. Los agonistas y antagonistas de los receptores de GnRH también se utilizan en tecnologías de reproducción asistida. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de GnRH de alta calidad para apoyar su investigación en salud reproductiva, endocrinología y terapia hormonal.
Se han encontrado 85 productos para "Receptor GNRH".
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Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Fórmula:C66H86N18O15Pureza:99.59% - 99.90%Forma y color:White SolidPeso molecular:1371.53Ref: TM-T21410
5mg52,00€10mg78,00€1mL*10mM (DMSO)116,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Fórmula:C32H29F5N3NaO5Pureza:99.71%Forma y color:White SolidPeso molecular:653.57Ref: TM-T5031
2mg34,00€5mg50,00€1mL*10mM (DMSO)71,00€10mg75,00€25mg137,00€50mg215,00€100mg340,00€200mg504,00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Fórmula:C68H87N17O15Pureza:99.98%Forma y color:SolidPeso molecular:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFórmula:C22H15F3N2O7SPureza:99.33% - 99.95%Forma y color:White SolidPeso molecular:508.42Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.Fórmula:C61H88N18O16Pureza:99.77% - >99.99%Forma y color:SolidPeso molecular:1329.46EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Fórmula:C15H27N5O6Forma y color:SolidPeso molecular:373.4Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Fórmula:C55H74N16O13Forma y color:SolidPeso molecular:1167.29Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Fórmula:C70H92ClN17O14·xC2H4O2Pureza:99.97%Forma y color:SolidPeso molecular:1491.11Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Fórmula:C80H104ClN21O14Forma y color:SolidPeso molecular:1619.27BAY 1214784
CAS:BAY 1214784 is a selective and orally active human GnRH-R antagonist, which can effectively reduce plasma luteinizing hormone levels by up to 49%.Fórmula:C29H26ClF4N3O5S2Pureza:100% - 99.77%Forma y color:White SolidPeso molecular:672.11NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Fórmula:C27H24F3N3O3Forma y color:SolidPeso molecular:495.49Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Fórmula:C25H19F3N4O5SPureza:98.60% - 98.97%Forma y color:SolidPeso molecular:544.55α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFórmula:C21H36O2Forma y color:SolidPeso molecular:320.51DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Fórmula:C11H17Cl2NOSForma y color:SolidPeso molecular:282.22BAY-784
CAS:BAY-784 is a potent GnRH receptor antagonist with nanomolar activity in human and rat receptors, widely used in endocrine and reproductive research.Fórmula:C29H26ClF4N3O5S2Pureza:99.22% - 99.75%Forma y color:White SolidPeso molecular:672.11BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Fórmula:C27H21ClFN3O2Pureza:98%Forma y color:SolidPeso molecular:473.93T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFórmula:C37H37F2N3O4SPureza:98%Forma y color:SolidPeso molecular:657.77[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Fórmula:C56H77N17O13Forma y color:SolidPeso molecular:1196.32Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Fórmula:C80H102ClN15O14Forma y color:SolidPeso molecular:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Fórmula:C36H35F7N4O6Forma y color:SolidPeso molecular:752.68
