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Receptor GNRH

Receptor GNRH

Los receptores de la hormona liberadora de gonadotropinas (GnRH) son GPCR que se unen a la GnRH, una hormona responsable de regular la liberación de la hormona luteinizante (LH) y la hormona foliculoestimulante (FSH) de la glándula pituitaria. Estos receptores son cruciales para la función reproductiva y son el objetivo de terapias para condiciones como el cáncer de próstata, la endometriosis y la infertilidad. Los agonistas y antagonistas de los receptores de GnRH también se utilizan en tecnologías de reproducción asistida. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de GnRH de alta calidad para apoyar su investigación en salud reproductiva, endocrinología y terapia hormonal.

Se han encontrado 91 productos para "Receptor GNRH".

productos por página.
  • Fertirelin

    CAS:
    Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).
    Fórmula:C55H76N16O12
    Pureza:>99.99%
    Forma y color:White Solid
    Peso molecular:1153.2919
  • Elagolix sodium

    CAS:
    Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
    Fórmula:C32H29F5N3NaO5
    Pureza:99.71%
    Forma y color:White Solid
    Peso molecular:653.5715
  • Linzagolix

    CAS:
    Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei
    Fórmula:C22H15F3N2O7S
    Pureza:99.33% - 99.95%
    Forma y color:White Solid
    Peso molecular:508.424
  • Goserelin acetate

    CAS:
    Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
    Fórmula:C61H88N18O16
    Pureza:99.77% - >99.99%
    Forma y color:Solid
    Peso molecular:1329.46
  • Cetrorelix diacetate

    CAS:
    Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.
    Fórmula:C74H100ClN17O18
    Pureza:98.38%
    Forma y color:White Solid
    Peso molecular:1551.142
  • Relugolix

    CAS:
    Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with
    Fórmula:C29H27F2N7O5S
    Pureza:98.64% - 99.97%
    Forma y color:White Solid
    Peso molecular:623.63
  • Ganirelix Acetate

    CAS:
    Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
    Fórmula:C82H117ClN18O15
    Pureza:96.05%
    Forma y color:Solid
    Peso molecular:1630.4
  • LGnRH-III, lamprey acetate


    LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion
    Fórmula:C61H78N18O16
    Pureza:96.65%
    Forma y color:Solid
    Peso molecular:1319.38
  • Fertirelin acetate

    CAS:
    Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.
    Fórmula:C55H74N16O13
    Forma y color:Solid
    Peso molecular:1167.29
  • Argtide

    CAS:
    Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.
    Fórmula:C80H104ClN21O14
    Forma y color:Solid
    Peso molecular:1619.27
  • NBI-42902

    CAS:
    NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.
    Fórmula:C27H24F3N3O3
    Forma y color:Solid
    Peso molecular:495.49
  • Cetrorelix Acetate

    CAS:
    Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
    Fórmula:C72H96ClN17O16
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:1491.09
  • BAY 1214784

    CAS:
    BAY 1214784 is a selective and orally active human GnRH-R antagonist, which can effectively reduce plasma luteinizing hormone levels by up to 49%.
    Fórmula:C29H26ClF4N3O5S2
    Pureza:100% - 99.77%
    Forma y color:White Solid
    Peso molecular:672.11
  • EA-230

    CAS:
    Ea-230 is an immunomodulator that may be used in the treatment of renal failure.
    Fórmula:C15H27N5O6
    Forma y color:Solid
    Peso molecular:373.4
  • Opigolix

    CAS:
    Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
    Fórmula:C25H19F3N4O5S
    Pureza:98.60% - 99.77%
    Forma y color:Solid
    Peso molecular:544.5
  • BAY-298

    CAS:
    BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.
    Fórmula:C27H21ClFN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.926
  • 5α-Pregnane-3α,20α-diol

    CAS:
    5α-Pregnane-3α,20α-diol is a progesterone metabolite that modulates LH and FSH release under specific endocrine conditions in animal studies.
    Fórmula:C21H36O2
    Forma y color:Solid
    Peso molecular:320.51
  • BAY-784

    CAS:
    BAY-784 is a potent GnRH receptor antagonist with nanomolar activity in human and rat receptors, widely used in endocrine and reproductive research.
    Fórmula:C29H26ClF4N3O5S2
    Pureza:99.22% - 99.75%
    Forma y color:White Solid
    Peso molecular:672.11
  • [D-Ala6]-LH-RH

    CAS:
    [D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].
    Fórmula:C56H77N17O13
    Forma y color:Solid
    Peso molecular:1196.32
  • T 98475

    CAS:
    gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active
    Fórmula:C37H37F2N3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:657.77