
Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Se han encontrado 449 productos de "Proteasa del VIH"
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HIV-1 inhibitor-31
CAS:<p>HIV-1 inhibitor-31 (compound 4) is a potent inhibitor of HIV-1. HIV-1 inhibitor-31 can be used in the study of AIDS.</p>Fórmula:C21H13Cl2N3O2Forma y color:SolidPeso molecular:410.25Deaminase inhibitor-1
CAS:<p>Deaminase inhibitor-1 is an APOBEC3G DNA Deaminase inhibitor with an IC 50 value of 18.9 μM [1].</p>Fórmula:C11H12BrN3OSForma y color:SolidPeso molecular:314.2HIV-1 inhibitor-50
CAS:<p>HIV-1 inhibitor-50 is a non-nucleoside reverse transcriptase inhibitor (NNRTI) that targets HIV-1 reverse transcriptase (IC50 = 50 nM).</p>Fórmula:C24H18FN5O2Forma y color:SolidPeso molecular:427.43S-1360
CAS:<p>S-1360 is an inhibitor of HIV-1 integrase.</p>Fórmula:C16H12FN3O3Pureza:98%Forma y color:SolidPeso molecular:313.28PF-46396
CAS:<p>PF-46396 is a HIV maturation inhibitor and can be used against HIV-1 clade B and C.</p>Fórmula:C27H29F3N2OForma y color:SolidPeso molecular:454.53HIV-1 inhibitor-39
CAS:<p>HIV-1 inhibitor-39: blocks HIV-1, anti-RT (IC50=15.75 μM), toxic to MT-4 cells (CC50=112.9 μM).</p>Fórmula:C20H17ClN4O4S4Forma y color:SolidPeso molecular:541.09Antiviral agent 9
<p>Antiviral agent 9: EC50 0.006 nM vs HIV-1, 300x more selective than TAF.</p>Fórmula:C38H50N7O8PForma y color:SolidPeso molecular:763.82HIV-1 inhibitor-48
CAS:<p>HIV-1 inhibitor-48 is a novel non-nucleoside reverse transcriptase inhibitor (NNRTI) and exhibits anti-HIV-1 activity .</p>Fórmula:C19H16BrN5Forma y color:SolidPeso molecular:394.27HIV-1 inhibitor-35
CAS:<p>HIV-1 inhibitor-35, potent against HIV (EC50: 80 nM LTR, 70 nM CMV), also suppresses HepG2 cells (CC50: 40 nM), may reverse HIV-1 latency.</p>Fórmula:C13H12Cl3N5OSForma y color:SolidPeso molecular:392.69HIV-1 inhibitor-9
CAS:<p>HIV-1 inhibitor-9 potently blocks WT and NNRTI-resistant HIV strains at low nanomolar levels.</p>Fórmula:C24H21N5OForma y color:SolidPeso molecular:395.46HIV-1 inhibitor-56
CAS:<p>HIV-1 inhibitor-56 (compound 12126065) is a potent non-nucleoside reverse transcriptase inhibitor with significant antiviral activity against wild-type HIV-1,</p>Fórmula:C22H14ClN7O2SForma y color:SolidPeso molecular:475.91Cgp 53820
CAS:<p>CGP 53820 is a pseudosymmetric inhibitor of HIV-1 Protease.</p>Fórmula:C31H51N5O5Forma y color:SolidPeso molecular:573.77HIV-1 inhibitor-33
CAS:<p>HIV-1 inhibitor-33, potent against HIV-1 (EC50: 8.6 nM), low toxicity to MT-4 cells (CC50: 18 μM), useful for AIDS research.</p>Fórmula:C25H28N6OForma y color:SolidPeso molecular:428.53ML67-33
CAS:<p>ML67-33 selectively activates K2P channels; EC50: 36.3 μM (cell-free), 9.7 μM (HEK293). Reversible TREK-1 modulation.</p>Fórmula:C18H17Cl2N5Pureza:98%Forma y color:SolidPeso molecular:374.27HEPT
CAS:<p>HEPT is a non-nucleoside inhibitor of HIV-1 reverse transcription.</p>Fórmula:C14H16N2O4SPureza:98%Forma y color:SolidPeso molecular:308.35L-Ristosamine nucleoside
CAS:<p>L-Ristosamine nucleoside shows antiviral activity.</p>Fórmula:C21H21N3O7Forma y color:SolidPeso molecular:427.41Suberosol
CAS:<p>Suberosol possesses anti-HIV replication activity.</p>Fórmula:C31H50O2Pureza:98%Forma y color:SolidPeso molecular:454.73ZP7
CAS:<p>ZP7 is a HIV-1 replication inhibitor.</p>Fórmula:C15H9Br2ClN4OS2Pureza:98%Forma y color:SolidPeso molecular:520.65APA-APA-MPO
CAS:<p>APA-APA-MPO is a PCAF bromodomain/Tat-AcK50 association inhibitor.</p>Fórmula:C12H25Cl2N5OPureza:98%Forma y color:SolidPeso molecular:326.27Ingenol 3-Hexanoate
CAS:<p>Ingenol 3-Hexanoate is a novel potent reactivator of latent HIV-1.</p>Fórmula:C26H38O6Pureza:98%Forma y color:SolidPeso molecular:446.58
