Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Se han encontrado 449 productos de "Proteasa del VIH"
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Aureothin
CAS:<p>Aureothin: a nitroaryl polyketide with antitumor, antifungal & insecticidal properties; inhibits NADH:oxidoreductase (IC50s: 0.07-22 nmol/mg).</p>Fórmula:C22H23NO6Forma y color:SolidPeso molecular:397.42Kadsuralignan A
CAS:<p>Kadsuralignan A (compound 1), a dibenzocyclooctadiene lignan extracted from the leaves and stems of Schisandra lancifolia, exhibits anti-HIV activity, with an</p>Fórmula:C22H26O7Forma y color:SolidPeso molecular:402.44HIV protease-IN-1
CAS:<p>HIV protease-IN-1 (compound 1·succinate), a potent non-peptidic inhibitor of HIV protease, is utilized for AIDS research [1].</p>Fórmula:C39H40ClF7N10O7Forma y color:SolidPeso molecular:929.24VIR-165
<p>VIR-165, a derivative of VIRIP (353-372 of alpha1-antitrypsin), blocks several HIV-1 strains.</p>Fórmula:C109H158N22O25S2Pureza:98%Forma y color:SolidPeso molecular:2240.7PROTAC Vif degrader-1
<p>PROTACVif degrader-1 (Compound L15) is a Vif-targeted PROTAC degrader exhibiting anti-HIV-1 virucidal activity, with an EC50 of 33.35 μM against HIV-1IIIB.</p>Forma y color:Odour SolidMPG, HIV related
CAS:<p>MPG: 27-amino acid peptide from HIV-1 gp41 & SV40 T antigen, delivers nucleic acids into cells efficiently.</p>Fórmula:C126H201N35O33SPureza:98%Forma y color:SolidPeso molecular:2766.22Pol (476-484), HIV-1 RT Epitope
CAS:<p>Pol (476-484), HIV-1 RT Epitope is a biologically active peptide and represents the dominant HLA A*0201-restricted epitope within HIV-1 reverse transcriptase (</p>Fórmula:C46H78N12O12Forma y color:SolidPeso molecular:991.18BNM-III-170
CAS:<p>BNM-III-170 is able to inhibit HIV-1 viral entry into target cells.</p>Fórmula:C25H26ClF7N6O6Forma y color:SolidPeso molecular:674.96Peptide T
CAS:<p>Peptide T, an HIV-1 derived octapeptide, may inhibit gp120 binding to CD4 and cytokines, and affect VIP receptors.</p>Fórmula:C35H55N9O16Pureza:98%Forma y color:SolidPeso molecular:857.86Interiorin
CAS:<p>Interiorin, extracted from Kadsura heteroclita, exhibits moderate anti-HIV activity, exhibiting an EC_50 of 1.6 μg/mL [1].</p>Fórmula:C27H30O8Forma y color:SolidPeso molecular:482.52Globotriaosylceramides (porcine)
CAS:<p>Globotriaosylceramides, cell membrane glycosphingolipids, act as Shiga toxin receptors and accumulate in Fabry disease, resisting HIV by blocking gp120.</p>Fórmula:C60H113NO18Forma y color:SolidPeso molecular:1136.553Enfuvirtide
CAS:<p>Enfuvirtide (INN) is an HIV fusion inhibitor, the first of a class of antiretroviral drugs used in combination therapy for the treatment of HIV-1 infection.</p>Fórmula:C204H301N51O64Pureza:98%Forma y color:White To Off-White Amorphous SolidPeso molecular:4491.945GP120, HIV-1 MN
GP120, HIV-1 MN, a peptide, is utilized in researching HIV infection [1] [2].Fórmula:C135H221N45O33Forma y color:SolidPeso molecular:3002.5Ac-Ser-Gln-Asn-Tyr-Pro-Val-Val-NH2
CAS:<p>Ac-Ser-Gln-Asn-Tyr-Pro-Val-Val-NH2, a peptide substrate for HIV-1 protease, is used in inhibition assays.</p>Fórmula:C38H58N10O12Forma y color:SolidPeso molecular:846.93HIV-1 inhibitor-75
<p>HIV-1inhibitor-75 is a human immunodeficiency virus 1 (HIV-1) inhibitor with an EC50 range of 0.0039-0.338 μM. Its target is the reverse transcriptase, exhibiting an IC50 value of 0.055 μM. Additionally, HIV-1inhibitor-75 demonstrates good metabolic stability in vitro, presenting moderate clearance rates and an extended half-life in human plasma and liver microsomes.</p>Fórmula:C25H20ClN3O3SForma y color:SolidPeso molecular:477.964-Acetylbutyric acid
CAS:<p>4-Acetylbutyric acid is a ketone acid widely used in biochemical experiments and drug synthesis research.</p>Fórmula:C6H10O3Pureza:99.88%Forma y color:SolidPeso molecular:130.14(±)-BI-D
CAS:<p>(±)-BI-D is an effective ALLINI(An allosteric IN inhibitor) that binds integrase at the LEDGF/p75 binding site (IC50: 2.4–2.9 μM).</p>Fórmula:C25H27NO4Forma y color:SolidPeso molecular:405.49gardiquimod TFA salt
CAS:<p>Gardiquimod diTFA is a TLR7/8 agonist that may block HIV-1 in macrophages and PBMCs, active under 10 μM.</p>Fórmula:C21H25F6N5O5Forma y color:SolidPeso molecular:541.44Dideoxyadenosine
CAS:<p>2',3'-Dideoxyadenosine is an inhibitor of HIV replication with antiretroviral activity and antiviral efficacy [1].</p>Fórmula:C10H13N5O2Pureza:99.28%Forma y color:Physical Description Off-White Powder (Ntp 1992)Peso molecular:235.242'-Deoxy-2'-fluoroarabinoadenosine
CAS:<p>2'-Deoxy-2'-fluoroarabinoadenosine is a nucleoside analogue with extensive anti-tumor activity and can be used for the study of tumor diseases.</p>Fórmula:C10H12FN5O3Pureza:99.95%Forma y color:SolidPeso molecular:269.23
