Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Se han encontrado 447 productos de "Proteasa del VIH"
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Probenecid
CAS:<p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>Fórmula:C13H19NO4SPureza:98.95% - 99.84%Forma y color:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Peso molecular:285.36(S)-(+)-N-3-Benzylnirvanol
CAS:<p>(S)-(+)-N-3-Benzylnirvanol is a cytochrome P450 CYP2C19 inhibitor with a ki value of 82.5μM for CYP2C9 and 0.25μM for CYP2C19.Cost-effective and quality-assured.</p>Fórmula:C18H18N2O2Pureza:98.90%Forma y color:SoildPeso molecular:294.35(Rac)-Telinavir
CAS:<p>N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.</p>Fórmula:C33H44N6O5Pureza:99.30%Forma y color:SolidPeso molecular:604.74Islatravir
CAS:<p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>Fórmula:C12H12FN5O3Pureza:98.77%Forma y color:SolidPeso molecular:293.25Salicylanilide
CAS:<p>Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.</p>Fórmula:C13H11NO2Pureza:99.55%Forma y color:White To Off-White Crystalline PowderPeso molecular:213.23Dolutegravir intermediate-1
CAS:<p>Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.</p>Fórmula:C13H17NO8Pureza:99.52%Forma y color:SolidPeso molecular:315.28Ibalizumab
CAS:<p>Ibalizumab(TMB-355) is a humanized IgG4 monoclonal antibody that acts as a CD4 receptor inhibitor, blocking the entry of HIV-1 into cells by binding to the CD4</p>Pureza:SDS-PAGE:96.4%;SEC-HPLC:97.7%Forma y color:LiquidPeso molecular:147.3 kDaGSK2838232
CAS:<p>GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.</p>Fórmula:C48H73ClN2O6Pureza:97.97%Forma y color:SolidPeso molecular:809.56Elsulfavirine
CAS:<p>Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.</p>Fórmula:C24H17BrCl2FN3O5SPureza:99.66%Forma y color:SolidPeso molecular:629.28Zalcitabine
CAS:<p>Zalcitabine (ddC) is a nucleoside analog inhibiting HIV by blocking reverse transcriptase and halting viral DNA synthesis.</p>Fórmula:C9H13N3O3Pureza:99.08% - ≥95%Forma y color:White To Off-White Crystalline PowderPeso molecular:211.223-Deazaadenosine hydrochloride
CAS:<p>3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.</p>Fórmula:C11H15ClN4O4Pureza:98.48%Forma y color:SolidPeso molecular:302.71Nevirapine
CAS:<p>Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor.</p>Fórmula:C15H14N4OPureza:99.58% - 99.59%Forma y color:White Or Off-White Crystalline PowderPeso molecular:266.3Fostemsavir Tris
CAS:<p>Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.</p>Fórmula:C29H37N8O11PPureza:99.45%Forma y color:SolidPeso molecular:704.62BRD-6929
CAS:<p>BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.</p>Fórmula:C19H17N3O2SPureza:98.01% - 99.05%Forma y color:SolidPeso molecular:351.42Pepstatin
CAS:<p>Pepstatin (Pepsin Inhibitor S 735A) is a specific and orally aspartate protease inhibitor that also inhibits HIV protease activity. Cost effective and quality assured.</p>Fórmula:C34H63N5O9Pureza:96.74% - 99.94%Forma y color:SolidPeso molecular:685.89Benfotiamine
CAS:<p>Benfotiamine (S-Benzoylthiamine O-monophosphate) is a synthetic S-acyl derivative of thiamine (vitamin B1), used as an antioxidant dietary supplement.</p>Fórmula:C19H23N4O6PSPureza:99.2% - 99.91%Forma y color:Shinning Black PowderPeso molecular:466.45Atazanavir
CAS:<p>Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.</p>Fórmula:C38H52N6O7Pureza:98% - 99.95%Forma y color:Crystalline SolidPeso molecular:704.86Ritonavir
CAS:<p>Ritonavir (ABT 538) inhibits HIV-1/2 proteases; serum proteins limit it but it enhances other HIV drugs by hindering P450 degradation.</p>Fórmula:C37H48N6O5S2Pureza:99.38% - 99.96%Forma y color:White PowderPeso molecular:720.94Tenofovir diphosphate TEA
CAS:<p>Tenofovir diphosphate TEA (TFV-DP TEA) is an ATP-competitive DNA polymerase inhibitor that inhibits HIV-1 reverse transcriptase that\has anti-HIV/HBV potential.</p>Fórmula:C9H16N5O10P3·C6H15NPureza:93.45% - 98.51%Forma y color:SolidPeso molecular:548.36Hck-IN-1
CAS:<p>Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; >20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.</p>Fórmula:C16H11ClN6O3SPureza:99.07%Forma y color:SolidPeso molecular:402.81Atazanavir sulfate
CAS:<p>Atazanavir sulfate, an azapeptide HIV-protease inhibitor, treats HIV/AIDS alongside other anti-HIV drugs.</p>Fórmula:C38H52N6O7·H2SO4Pureza:99.31% - 99.40%Forma y color:SolidPeso molecular:802.93TERT-IN-1
CAS:<p>TERT-IN-1 has anti-HIV activity and can be used to study HIV infection.</p>Fórmula:C16H20ClN3SPureza:99.31%Forma y color:SoildPeso molecular:321.87NBD-556
CAS:<p>NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.</p>Fórmula:C17H24ClN3O2Pureza:99.79%Forma y color:SolidPeso molecular:337.84PF-3450074
CAS:<p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>Fórmula:C27H27N3O2Pureza:99.92%Forma y color:SolidPeso molecular:425.52L 754394
CAS:<p>L 754394 is an effective and specific inhibitor of the HIV-1 protease.</p>Fórmula:C38H47N5O5Forma y color:SolidPeso molecular:653.81HIV p17 Gag (77-85)
CAS:<p>Targeting HIV Gag p17 (77-85) with intracellular Ab cDNA disrupts viral replication pre/post-integration.</p>Fórmula:C44H72N10O15Pureza:98%Forma y color:SolidPeso molecular:981.1Bictegravir Sodium
CAS:<p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>Fórmula:C21H17F3N3NaO5Pureza:99.97%Forma y color:SolidPeso molecular:471.36Globotriaosylceramides (porcine)
CAS:<p>Globotriaosylceramides, cell membrane glycosphingolipids, act as Shiga toxin receptors and accumulate in Fabry disease, resisting HIV by blocking gp120.</p>Fórmula:C60H113NO18Forma y color:SolidPeso molecular:1136.553HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Forma y color:Odour SolidHIV-1 inhibitor-81
<p>HIV-1inhibitor-81 (Compound 14g) is an HIV-1 protease inhibitor with a Ki of 1.6 nM. This compound exhibits antiviral activity against HIV-1, with an EC50 value of 250 nM.</p>Fórmula:C32H44N2O8SForma y color:SolidPeso molecular:616.77HIV-1 protease-IN-10
<p>HIV-1 protease-IN-10 (Compound 2), exhibiting HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to the PKCδ C1b domain (IC50: 0.69 μM) and</p>Fórmula:C23H40O5Pureza:98%Forma y color:SolidPeso molecular:396.56Protease Inhibitor Library
<p>A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening;</p>Forma y color:Odour SolidScirpusin A
CAS:<p>Scirpusin A is a hydroxystilbene dimer from the rhizome of Scirpus fluviatilis and Xinjiang wine grape.</p>Fórmula:C28H22O7Forma y color:SolidPeso molecular:470.47HIV gag peptide (197-205)
CAS:<p>HIV gag peptide (197-205) is a H-2Kd-restricted epitope derived from the p24 portion of the HIV-1 gag protein and composed of the amino acid 197-205 (AMQMLKETI</p>Fórmula:C45H81N11O14S2Pureza:98%Forma y color:SolidPeso molecular:1064.32Peptide T TFA
CAS:<p>Peptide T (TFA), an octapeptide from HIV-1 gp120, inhibits HIV binding to CD4.</p>Fórmula:C37H56F3N9O18Pureza:98%Forma y color:SolidPeso molecular:971.89HIV-1 inhibitor-11
<p>HIV-1 inhibitor-11, a fused pyridine ring derivative, is a HIV-1 inhibitor.</p>Fórmula:C42H36ClF10N7O5S2Forma y color:SolidPeso molecular:1008.35Kuguacin N
<p>Kuguacin N is a useful organic compound for research related to life sciences and the catalog number is T126345.</p>Fórmula:C30H46O4Forma y color:SolidPeso molecular:470.694MPG, HIV related
CAS:<p>MPG: 27-amino acid peptide from HIV-1 gp41 & SV40 T antigen, delivers nucleic acids into cells efficiently.</p>Fórmula:C126H201N35O33SPureza:98%Forma y color:SolidPeso molecular:2766.22NF279
CAS:<p>P2X1 antagonist</p>Fórmula:C49H36N6Na6O23S6Pureza:98%Forma y color:SolidPeso molecular:1407.17VIR-165
<p>VIR-165, a derivative of VIRIP (353-372 of alpha1-antitrypsin), blocks several HIV-1 strains.</p>Fórmula:C109H158N22O25S2Pureza:98%Forma y color:SolidPeso molecular:2240.7Delavirdine
CAS:<p>Delavirdine, an NNRTI for HIV-1, is used in HAART.</p>Fórmula:C22H28N6O3SForma y color:SolidPeso molecular:456.56NNRT-IN-6
<p>NNRT-IN-6 (Compound 13a) is a non-nucleoside reverse transcriptase inhibitor (NNRT) used to inhibit HIV-1 reverse transcriptase (HIV-1RT), with an IC50 of 0.41 μM. It effectively suppresses both wild-type HIV-1 and mutants L100I, K103N, Y181C, Y188L, E138K, F227L/V106A, and RES056, with an EC50 range of 6.2-250 nM.</p>Fórmula:C32H31N9O3SForma y color:SolidPeso molecular:621.71Peptide T
CAS:<p>Peptide T, an HIV-1 derived octapeptide, may inhibit gp120 binding to CD4 and cytokines, and affect VIP receptors.</p>Fórmula:C35H55N9O16Pureza:98%Forma y color:SolidPeso molecular:857.86Cys-TAT(47-57)
CAS:<p>Cys-TAT(47-57): arginine-rich peptide from HIV-1 TAT protein's transduction domain.</p>Fórmula:C67H124N34O14SPureza:98%Forma y color:SolidPeso molecular:1661.99MB-66
<p>MB-66 (MAPP-66) is a fully human IgG1 antibody targeting HSV and HIV. It is a monoclonal antibody membrane intended for vaginal application. The isotype control for MB-66 can be referred to as HumanIgG1kappa, Isotype Control.</p>Forma y color:Odour LiquidSPD-756
CAS:<p>SPD-756, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Fórmula:C12H16N6O3Pureza:98%Forma y color:SolidPeso molecular:292.29HIV-1 inhibitor-59
<p>HIV-1 Inhibitor-59 (Compound I-5b) effectively inhibits both wild-type and mutant strains of HIV-1, with EC50 values ranging from 5.62 to 171 nM.</p>Fórmula:C28H28FN5O3SForma y color:SolidPeso molecular:533.62Clavirolide L
<p>Clavirolide L (Compound 3), a dolabellane-type diterpenoid isolated from Clavularia viridis, demonstrates significant inhibition against HIV-1 without</p>Fórmula:C20H28O3Forma y color:SolidPeso molecular:316.43HIV-1 inhibitor-6
CAS:<p>HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing</p>Fórmula:C14H10N4O4SPureza:99.33%Forma y color:SolidPeso molecular:330.32Hinnuliquinone
CAS:Hinnuliquinone is an anti-HIV agent.Fórmula:C32H30N2O4Pureza:98%Forma y color:SolidPeso molecular:506.59
