Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Se han encontrado 449 productos de "Proteasa del VIH"
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gardiquimod TFA salt
CAS:<p>Gardiquimod diTFA is a TLR7/8 agonist that may block HIV-1 in macrophages and PBMCs, active under 10 μM.</p>Fórmula:C21H25F6N5O5Forma y color:SolidPeso molecular:541.44Saquinavir mesylate
CAS:Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapyFórmula:C39H54N6O8SPureza:99.19%Forma y color:White Or Pale Yellow PowderPeso molecular:766.9Betulin diacetate
CAS:<p>Betulin diacetate is a bioactive chemical.</p>Fórmula:C34H54O4Forma y color:SolidPeso molecular:526.8Ditiocarb sodium
CAS:<p>Ditiocarb sodium (Sodium diethyldithiocarbamate) (sodium diethiocarbamate) is a copper reagent, which reacts with Cu2 + solution to form a complex and improves</p>Fórmula:C5H10NNaS2Pureza:98.04%Forma y color:White Solid CrystallinePeso molecular:171.26Amprenavir
CAS:<p>Amprenavir (KVX-478) is a synthetic derivative of hydroxyethylamine sulfonamide that selectively binds to and inhibits human immunodeficiency virus (HIV)</p>Fórmula:C25H35N3O6SPureza:99.60% - 99.87%Forma y color:Off-White To Pale YellowPeso molecular:505.63Delavirdine mesylate
CAS:<p>Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).</p>Fórmula:C23H32N6O6S2Pureza:99.99%Forma y color:Light Brown SolidPeso molecular:552.67Tenofovir alafenamide
CAS:<p>Tenofovir alafenamide (GS-7340) is a nucleotide reverse transcriptase inhibitor (NRTI) and a novel ester prodrug of the antiretroviral tenofovir.</p>Fórmula:C21H29N6O5PPureza:99.68% - 99.81%Forma y color:SolidPeso molecular:476.47Dolutegravir sodium
CAS:<p>Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature</p>Fórmula:C20H18F2N3NaO5Pureza:98% - 99.46%Forma y color:SolidPeso molecular:441.36Escin IA
CAS:<p>Escin IA (Escin IA;Aescin IA) is a triterpene saponin isolated from horse chestnut, which inhibits HIV-1 protease with IC50 values of 35 μM.</p>Fórmula:C55H86O24Pureza:98.97% - 99.81%Forma y color:SolidPeso molecular:1131.26Doravirine
CAS:<p>Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.</p>Fórmula:C17H11ClF3N5O3Pureza:99.65% - 99.79%Forma y color:SolidPeso molecular:425.75Cobicistat
CAS:<p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>Fórmula:C40H53N7O5S2Pureza:97.36% - 99.62%Forma y color:SolidPeso molecular:776.02Lopinavir
CAS:<p>Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation.</p>Fórmula:C37H48N4O5Pureza:98% - 99.62%Forma y color:White Crystalline SolidPeso molecular:628.8Raltegravir sodium
CAS:<p>Raltegravir (MK 0518) sodium is a potent, orally active HIV integrase (IN) inhibitor.</p>Fórmula:C20H20FN6NaO5Forma y color:SolidPeso molecular:466.405Amylmetacresol
CAS:<p>Amylmetacresol treats sore throat, pharyngitis, tonsillitis, laryngitis, influenza A, and SARS-CoV.</p>Fórmula:C12H18OPureza:99.66%Forma y color:SolidPeso molecular:178.27Dolutegravir
CAS:<p>Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.</p>Fórmula:C20H19F2N3O5Pureza:98.97% - 99.75%Forma y color:White To Pale Yellow SolidPeso molecular:419.38Didanosine
CAS:<p>Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).</p>Fórmula:C10H12N4O3Pureza:99.64%Forma y color:White Crystalline PowderPeso molecular:236.23Ganoderic acid B
CAS:<p>Ganoderic acid B: quality marker for G. lucidum products, inhibits telomerase & EBV activation, moderates HIV-1 protease.</p>Fórmula:C30H44O7Pureza:99.09% - 99.95%Forma y color:SolidPeso molecular:516.67Darunavir
CAS:<p>Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.</p>Fórmula:C27H37N3O7SPureza:99.67% - 99.76%Forma y color:White Amorphous SolidPeso molecular:547.66Temsavir
CAS:<p>Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.</p>Fórmula:C24H23N7O4Pureza:99.14%Forma y color:SolidPeso molecular:473.48BMS-707035
CAS:<p>BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.</p>Fórmula:C17H19FN4O5SPureza:99.78%Forma y color:SolidPeso molecular:410.42TAT
CAS:<p>TAT peptide (YGRKKRRQRRR), originating from the human immunodeficiency virus-1 (HIV-1) transactivator of transcription (TAT), enhances the solubility and</p>Fórmula:C64H118N32O14Pureza:>99.99%Forma y color:SolidPeso molecular:1559.83Raltegravir
CAS:<p>Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIV</p>Fórmula:C20H21FN6O5Pureza:99.86% - >99.99%Forma y color:SolidPeso molecular:444.42NBD-557
CAS:<p>NBD-557 is a potentially HIV-1 inhibitor.</p>Fórmula:C17H24BrN3O2Pureza:99.52%Forma y color:SolidPeso molecular:382.3I-XW-053 sodium
CAS:<p>I-XW-053 sodium inhibits the replication of a diverse panel of primary HIV-1 isolates in Peripheral blood mononuclear cell with no appreciable cytotoxicity.</p>Fórmula:C22H16N2NaO2Forma y color:SolidPeso molecular:363.372LDC4297 hydrochloride
CAS:<p>LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.</p>Fórmula:C23H29ClN8OForma y color:SolidPeso molecular:468.98Darunavir Ethanolate
CAS:<p>Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.</p>Fórmula:C29H43N3O8SPureza:99.84% - 99.86%Forma y color:SolidPeso molecular:593.742,4-Dihydroxypyridine
CAS:<p>2,4-Dihydroxypyridine: a pyridine derivative, chelates metals, assesses ion levels, measures enzymatic reactions, and quantifies biomolecules.</p>Fórmula:C5H5NO2Pureza:97.79%Forma y color:White To Yellow-Beige Crystals OrPeso molecular:111.1Rosamultin
CAS:<p>Rosamultin has antioxidant, antiinflammatory/antinociceptive properties,and has anti-human immunodeficiency virus (HIV) activity.</p>Fórmula:C36H58O10Pureza:98% - 99.83%Forma y color:SolidPeso molecular:650.84Thiamine disulfide
CAS:<p>Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.</p>Fórmula:C24H34N8O4S2Pureza:99.81%Forma y color:CoaPeso molecular:562.71Inosine pranobex
CAS:<p>Inosine pranobex (Delimmun) has a lot of immunomodulatory effects, including inducing T-lymphocyte differentiation, augmenting macrophage and NK cell functions.</p>Fórmula:C52H78N10O17Pureza:99.78% - 99.91%Forma y color:SolidPeso molecular:1115.23Raltegravir potassium
CAS:<p>Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.</p>Fórmula:C20H20FN6O5·KPureza:98% - 99.55%Forma y color:Off-White SolidPeso molecular:482.51Rolipram
CAS:<p>Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.</p>Fórmula:C16H21NO3Pureza:99.22% - >99.99%Forma y color:SolidPeso molecular:275.34IMB-301
CAS:<p>IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.</p>Fórmula:C19H17Cl2FN2OPureza:99.72%Forma y color:SolidPeso molecular:379.26PMEDAP
CAS:<p>PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiency</p>Fórmula:C8H13N6O4PPureza:99.77%Forma y color:SolidPeso molecular:288.2Dimercaprol
CAS:<p>Dimercaprol (Dicaptol) is an anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-</p>Fórmula:C3H8OS2Pureza:98.91% - 99.64%Forma y color:Viscous Oily LiquidPeso molecular:124.22PTACH
CAS:<p>PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).</p>Fórmula:C20H26N2O2S2Pureza:87.44% - 99.74%Forma y color:SolidPeso molecular:390.56Peldesine dihydrochloride
CAS:<p>Peldesine (BCX 34) dihydrochloride is an inhibitor of PNP in humans, rats, and mice, also hindering T-cell proliferation, used in lymphoma and HIV research.</p>Fórmula:C12H13Cl2N5OForma y color:SolidPeso molecular:314.17Fostemsavir
CAS:<p>Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.</p>Fórmula:C25H26N7O8PPureza:98.95%Forma y color:SolidPeso molecular:583.49Bictegravir
CAS:<p>Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).</p>Fórmula:C21H18F3N3O5Pureza:97.6% - 99.51%Forma y color:SolidPeso molecular:449.38HODHBt
CAS:<p>HODHBt is a STAT5-SUMO protein-protein interaction inhibitor.</p>Fórmula:C7H5N3O2Pureza:99.45% - 99.95%Forma y color:Off-White To Yellow SolidPeso molecular:163.13Rilpivirine
CAS:<p>Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatment</p>Fórmula:C22H18N6Pureza:97.22% - 98.83%Forma y color:SolidPeso molecular:366.42Tenofovir alafenamide hemifumarate
CAS:<p>Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.</p>Fórmula:C21H29N6O5PC4H4O4Pureza:99.33% - 99.96%Forma y color:SolidPeso molecular:534.51Des(benzylpyridyl) Atazanavi
CAS:<p>The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.</p>Fórmula:C26H43N5O7Pureza:98% - 99.75%Forma y color:SolidPeso molecular:537.65Saquinavir
CAS:<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Fórmula:C38H50N6O5Pureza:99.50% - >99.99%Forma y color:SolidPeso molecular:670.84Dexelvucitabine
CAS:<p>Dexelvucitabine (RVT), a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Fórmula:C9H10FN3O3Pureza:98.25%Forma y color:SolidPeso molecular:227.19HIV-1 Inhibitor 18A
CAS:<p>HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.</p>Fórmula:C14H11N5O2SPureza:99.79%Forma y color:SolidPeso molecular:313.33Etravirine
CAS:<p>Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.</p>Fórmula:C20H15BrN6OPureza:97.61% - 99.74%Forma y color:White To Off-White SolidPeso molecular:435.28HIV-1 Nef-IN-1
CAS:<p>HIV-1 Nef-IN-1 is an inhibitor of HIV-1 Nef protein. It efficiently competes for Nef-SH3Hck interactions(Kd : 6.7 μM).</p>Fórmula:C18H16O2Pureza:99.90%Forma y color:SolidPeso molecular:264.32Elvitegravir
CAS:<p>Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.</p>Fórmula:C23H23ClFNO5Pureza:98.43% - 99.57%Forma y color:SolidPeso molecular:447.88Obefazimod
CAS:<p>Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).</p>Fórmula:C16H10ClF3N2OPureza:99.86%Forma y color:SolidPeso molecular:338.71
