Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Se han encontrado 450 productos de "Proteasa del VIH"
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Antiviral agent 55
CAS:Antiviralagent 55 (Compound 95) is an inhibitor of human immunodeficiency viruses 1 and 2 (HIV1 and HIV2), demonstrating antiviral activity.Fórmula:C21H20N2O4Forma y color:SolidPeso molecular:364.39Zinlirvimab
CAS:<p>Zinlirvimab is a humanized IgG1-λ2 monoclonal antibody that neutralizes HIV by targeting the HIV-1 gp120 envelope glycoprotein, specifically the IIIB gp120 V3</p>Forma y color:LiquidGCA-186
CAS:GCA-186 is an effective non-nucleoside HIV-1 reverse transcriptase inhibitor.Fórmula:C19H26N2O3Pureza:98%Forma y color:SolidPeso molecular:330.42APOBEC3G-IN-1
CAS:<p>APOBEC3G-IN-1 (MN136.0185) is a targeted APOBEC3G inhibitor with anti-HIV activity for the study of infectious diseases and cancer.</p>Fórmula:C15H11NO3Pureza:96.54%Forma y color:SolidPeso molecular:253.25HIV-IN-6
CAS:<p>HIV-IN-6, an anti-HIV agent, blocks replication by targeting SFKs like Hck involved with Nef protein.</p>Fórmula:C20H16N4O3SPureza:97.12%Forma y color:SolidPeso molecular:392.43HIV-1 inhibitor-49
<p>HIV-1 inhibitor-49, an oral HEPT analog, has strong pharmacokinetics, potent reverse transcriptase inhibition (IC50=30nM), and is safe in mice.</p>Fórmula:C21H18F2N2O3SForma y color:SolidPeso molecular:416.44MK-2048
CAS:<p>MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.</p>Fórmula:C21H21ClFN5O4Pureza:98%Forma y color:SolidPeso molecular:461.87HIV-1 inhibitor-22
CAS:<p>HIV-1 inhibitor-22 effectively blocks HIV-1 RT (IC50=3.63 μM) with low cytotoxicity (CC50 > 227 μM).</p>Fórmula:C30H26N6O3SForma y color:SolidPeso molecular:550.63HIV-1 integrase inhibitor 4
CAS:<p>HIV-1 integrase inhibitor 4 is an HIV-1 integrase strand transfer (INST) inhibitor (IC50: 3.7 nM).</p>Fórmula:C24H20F2N4O5SPureza:98%Forma y color:SolidPeso molecular:514.5HIV-1 inhibitor-29
CAS:<p>HIV-1 inhibitor-29: Blocks HIV-1 IIIB (EC50: 2.18μM), resists F227L/V106A (EC50: 0.974μM), low toxicity (CC50: 211μM), for AIDS research.</p>Fórmula:C30H36N6O5Forma y color:SolidPeso molecular:560.64D77
CAS:D77 is anti-HIV-1 inhibitor. D77 inhibits HIV-1(IIIB) replication by EC50 value of 23.8 μg/ml in MT-4 cell (5.03 μg/ml for C8166 cells).Fórmula:C28H22BrNO7SPureza:98%Forma y color:SolidPeso molecular:596.45HIV-1 inhibitor-34
CAS:<p>HIV-1 inhibitor-34 (5q): potent, selective; EC50: 6.4 nM; MT-4 CC50: 16 μM; useful in AIDS research.</p>Fórmula:C26H27N7OForma y color:SolidPeso molecular:453.54HIV-IN-4
CAS:<p>HIV-IN-4 (Compound 12) is a potent HIV inhibitor that exhibits promising anti-HIV activities [1].</p>Fórmula:C14H18N2O3Forma y color:SolidPeso molecular:262.3HIV-1 inhibitor-16
CAS:<p>HIV-1 inhibitor-16: potent with EC50 1.3 nM for wild-type; inhibits K103N, E138K, Y181C, L100I strains; good solubility; stable; low CYP impact; non-toxic.</p>Fórmula:C23H16F2N6Forma y color:SolidPeso molecular:414.41HIV-1 inhibitor-57
CAS:<p>HIV-1 Inhibitor-57 (Compound 12g) is an antiviral agent that potently inhibits both wild-type and five common NNRTI-resistant strains of HIV-1, exhibiting EC50</p>Fórmula:C25H24FN5O3SForma y color:SolidPeso molecular:493.55SARS-CoV-IN-3
CAS:SARS-CoV-IN-3 is an effective SARS-CoV replication inhibitor.Fórmula:C25H28ClFeN3OPureza:98%Forma y color:SolidPeso molecular:477.81Mesoxalic acid
CAS:<p>Mesoxalic acid is a dicarboxylic acid and a ketonic acid which blocks RT translocation.</p>Fórmula:C3H2O5Pureza:98%Forma y color:SolidPeso molecular:118.04SAMT-247
CAS:<p>SAMT-247 is an HIV inhibitor that acts by modifying the nucleocapsid NCp7 region of Gag in infected cells and blocking Gag processing and reducing infectivity.</p>Fórmula:C12H14N2O3SForma y color:SolidPeso molecular:266.32TMC310911
CAS:TMC310911 is an oral HIV-1 protease inhibitor with an EC50 of 2.2-14.2 nM, effective against various HIV-1 strains.Fórmula:C38H53N5O7S2Pureza:98%Forma y color:SolidPeso molecular:755.99Reverse transcriptase-IN-3
<p>Reverse transcriptase-IN-3, a pyrimidine carboxamide, inhibits HIV-1 including mutant strains.</p>Fórmula:C28H31N7O4SForma y color:SolidPeso molecular:561.66
