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<p>8-Benzyloxy-5-((R)-2-bromo-1-hydroxyethyl)-1H-quinolinone is a potassium channel blocker. It binds to the central cavity of the channel pore and blocks potassium ion flux, inhibiting the function of potassium channels. 8-Benzyloxy-5-(2-(R)-bromo-1,3-dihydroxypropyl)quinolinone has been shown to inhibit voltage gated channels in a number of different tissues, including cardiomyocytes from rat hearts.</p>

<p>6-Bromo-pyrazolo[1,5-a]pyrimidine is a bone morphogenetic protein (BMP) inhibitor. It has been shown to be a potent inhibitor of the tyrosine kinase activity of BMP receptors and may be useful for the development of new strategies for the treatment of osteoporosis. 6-Bromo-pyrazolo[1,5-a]pyrimidine is also an effective inhibitor of the proliferation and survival of cancer cells. It inhibits cell growth by interfering with cellular signaling pathways that regulate these processes. 6-Bromo-pyrazolo[1,5-a]pyrimidine was also found to inhibit the production of bone morphogenetic protein 2 (BMP2) in mouse calvaria cells without affecting other bone metabolism markers such as alkaline phosphatase or osteocalcin.</p>

<p>1H-Indazole-5-boronic acid is a potent compound that belongs to the class of indazole compounds. It has been shown to inhibit protein phosphorylation and induce morphological changes in cells. This compound also inhibits the activity of a number of different cellular enzymes, including protein phosphatases, protein kinases, and protein tyrosine phosphatases. 1H-Indazole-5-boronic acid has been shown to be a promising lead compound for the discovery of novel inhibitors of these enzymes.</p>

<p>4,4'-Dimethyl-2,2'-bipyridine is a molecule that belongs to the group of p2 metal complexes. It has been shown to have synergistic effects with ruthenium complexes in analytical chemistry and electrochemical studies. Theoretical calculations have been performed for 4,4'-dimethyl-2,2'-bipyridine and its derivatives. These calculations show that the molecule is planar and that it can be considered as a diazonium salt. The photochemical properties of 4,4'-dimethyl-2,2'-bipyridine have also been studied in detail. This substance emits light when excited by ultraviolet light or visible light, which makes it an excellent candidate for use as a luminescent material in optical displays.</p>

<p>Please enquire for more information about 1-Boc-5-Cyano-3-hydroxymethylindole including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>4-Chloro-6,7-dimethoxyquinoline (4C6DMQ) is a potent inhibitor of the growth of prostate cancer cells. 4C6DMQ is an analog of chloropropyl chloride, which inhibits the growth of epidermal growth factor receptor (EGFR). The binding site for 4C6DMQ on EGFR is the same as that for chloropropyl chloride. 4C6DMQ inhibits EGFR by preventing the activation of downstream signaling cascades, leading to a decrease in cell proliferation and tumor size. The IC50 values for 4C6DMQ are approximately 10 times higher than those for chloropropyl chloride. This drug has been shown to be more potent than other inhibitors of EGFR such as erlotinib and gefitinib.</p>

<p>Benzo[a]phenanthrene is a polycyclic aromatic hydrocarbon that is found in petroleum and coal tar. It has been shown to be a potent inducer of enzymes involved in the detoxification of xenobiotics, such as chrysene-inducible cytochrome P450 1A1 (CYP1A1), s-phenylmercapturic acid-inducible cytochrome P450 2E1 (CYP2E1), and benzo[a]pyrene-inducible glutathione S-transferase (GST). The optimum concentration for benzo[a]phenanthrene is determined by measuring the amount of enzyme activity in rat liver microsomes following the addition of benzo[a]phenanthrene. A fluorescence detector can be used to measure the fluorescence emission from benzo[a]phenanthrene at an excitation wavelength of 300 nm and an emission wavelength of 400 nm.</p>

<p>Please enquire for more information about 1-Boc-4-aminoindole including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>6-Chloroindole-3-carboxaldehyde is a natural compound with the molecular formula C8H6ClNO2. It has been shown to have anticancer activity against lung cancer cells and has been found to inhibit the growth of metastatic lung cancer cells in mice. 6-Chloroindole-3-carboxaldehyde inhibits the proliferation of human lung cancer cells by arresting cells in the G1 phase of the cell cycle, which may be due to its ability to bind to deoxyhexose and form a complex. This compound also has antimicrobial activity against bacterial strains such as Streptococcus pneumoniae and Mycoplasma pneumoniae.</p>

<p>Please enquire for more information about (1S,4S)-2-Oxa-5-azabicyclo[2.2.1]heptane hydrochloride including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>8-Quinolinesulfonyl chloride (8QSC) is a quinoline derivative that has been shown to have anticancer activity. 8QSC binds to the receptor site of cells and inhibits the production of amines, which are important for cell growth and proliferation. It also binds to hydrogen bonds, which may be involved in the cytotoxicity observed in pancreatic cancer cells. 8QSC shows significant cytotoxicity against Panc-1 cells, but not against NIH 3T3 cells. This may be due to its ability to form supramolecular aggregates with copper ions and quinoline derivatives.</p>

<p>Please enquire for more information about Oxindole-4-boronic acid, pinacol ester including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>7-Bromo-1H-indazole is a brominated indazole with an unusual amino acid sequence. It can be used as a building block for the synthesis of new compounds that have potential as medicines. 7-Bromo-1H-indazole has been investigated in cancer cell lines, and it has been shown to inhibit the growth of these cells by inhibiting the production of chloride ions. The molecular modeling of this compound has also shown that it may bind to the chloride channel on cancer cells, preventing chloride ions from entering or leaving the cell. The X-ray crystal structures show that 7-bromoindazole binds with hydrogen bonds to azobisisobutyronitrile (AIBN) and ruthenium complex, which are both potential anticancer drugs.</p>

<p>8-Hydroxyquinoline is a sweet, water soluble, and heat stable inhibitor that has been used in the treatment of kidney disease. 8-Hydoxyquinoline has been shown to inhibit the growth of the rootstock Asiaticus by interfering with cell metabolism. It is also an insecticide that kills insects by causing damage to their cells. 8-Hydoxyquinoline inhibits polymerase chain reaction (PCR) by binding to DNA polymerase, blocking its activity and reducing its ability to synthesize DNA. This drug is also a potent blocker of angiotensinogen synthesis, which leads to reduced blood pressure levels.</p>

<p>2,9-Bis(2-phenylethyl)anthraquinone (BPAQ) is a synthetic compound that is used as an fluorescent probe to study biological processes. BPAQ binds to peptides and inhibits their binding to the surface of cells. This property has been used in diagnostic tests for stenosis, infantum, and other conditions. BPAQ has also been shown to inhibit HIV-1 replication in human cells by binding to the HIV-1 envelope protein gp120 and blocking its interaction with CD4 receptors on host cells. The discovery of the antiviral activity of BPAQ was based on its ability to inhibit leishmania growth in animals.</p>

<p>Please enquire for more information about 5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)indoline including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>Marmesinin is a furanocoumarin compound, which is a type of phytochemical derived from certain plant species. It is specifically obtained from the plant Aegle marmelos, commonly known as the bael tree. Marmesinin acts primarily through mechanisms that are characteristic of coumarins, such as influencing biochemical pathways involved in cellular growth and immune response modulation.</p>

<p>(+)-Peucedanol is a sesquiterpene compound, which is a type of natural organic compound composed of three isoprene units resulting in a 15-carbon backbone. It is derived from various species within the plant genus Peucedanum, known for their rich content of bioactive compounds. The stereoisomerism indicated by the "(+)" suggests a specific three-dimensional configuration that may influence its biological activity.</p>

<p>Please enquire for more information about [4,4'-Di-t-butyl-2,2'-bipyridine][bis[5-(t-butyl)-2-[4-(t-butyl)-2-pyridinyl-kN]phenyl-kC]iridium(III) hexafluorophosphate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>H-Tyr-L-1,2,3,4-tetrahydroisoquinoline-3-carboxamide·HCl is a monoclinic crystalline compound. It has a molecular weight of 607.14 and contains the dipeptide Tyr-Lys in its structure. H-Tyr-L-1,2,3,4-tetrahydroisoquinoline-3-carboxamide·HCl crystallizes in the P21/c space group and has an asymmetric unit cell with dimensions a=8.851 Å, b=7.965 Å and c=5.98 Å. This compound has been shown to have antibacterial properties against methicillin resistant Staphylococcus aureus (MRSA) isolates and Clostridium perfringens strains by inhibiting bacterial protein synthesis through inhibition of peptidyl transferase activity.</p>