Otros inhibidores
Esta categoría abarca una amplia variedad de inhibidores que no encajan en las clasificaciones estándar, pero que son fundamentales para diversas investigaciones bioquímicas y farmacológicas. Estos inhibidores pueden dirigirse a vías, enzimas e interacciones moleculares únicas o menos estudiadas, proporcionando herramientas valiosas para áreas de investigación especializadas. En CymitQuimica, ofrecemos una selección diversa de inhibidores de alta calidad que abarcan múltiples objetivos biológicos y disciplinas de investigación, lo que le permite explorar nuevas vías terapéuticas y profundizar su comprensión de los procesos biológicos complejos.
Se han encontrado 36533 productos de "Otros inhibidores"
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9-cis-13,14-Dihydroretinoic acid
CAS:<p>9-cis-13,14-Dihydroretinoic acid (9CDHRA) is a selective retinoid X receptor (RXR) agonist with a Kd of 90 nM. It can ameliorate memory deficits caused by impaired RXR signaling in vivo. This compound shows potential for research in the fields of neuroscience and metabolic diseases.</p>Fórmula:C20H30O2Forma y color:SolidPeso molecular:302.451Glidobactin G
CAS:<p>Glidobactin G is an antitumor antibiotic with activity against pathogenic fungi and yeasts. Additionally, Glidobactin G prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Fórmula:C27H44N4O7Forma y color:SolidPeso molecular:536.6612-Hydroxygentamicin B
CAS:<p>2-Hydroxygentamicin B is an aminoglycoside antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C19H38N4O11Forma y color:SolidPeso molecular:498.52511-Deacetoxywortmannin
CAS:11-Deacetoxywortmannin is an antibiotic with potent antibacterial and anti-inflammatory properties, and it also exhibits anti-edema effects.Fórmula:C21H22O6Forma y color:SolidPeso molecular:370.3963-O-Demethylmonensin A
CAS:3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).Fórmula:C35H60O11Forma y color:SolidPeso molecular:656.84GSK-1264
CAS:<p>GSK-1264: allosteric HIV integrase inhibitor, halts viral replication & abnormal protein multimerization.</p>Fórmula:C26H28FNO5Forma y color:SolidPeso molecular:453.5Dykellic acid
CAS:<p>Dykellic acid is a RhoA inhibitor. It can suppress the migration and motility of B16 cells and inhibit the tubular formation of HUVECs. Dykellic acid shows potential for use in cancer research.</p>Fórmula:C14H16O4Forma y color:SolidPeso molecular:248.274Exophilin A
CAS:<p>Exophilin A is an antibiotic that exhibits activity against Gram-positive bacteria.</p>Fórmula:C30H56O10Forma y color:SolidPeso molecular:576.76Herbimycin B
CAS:Herbimycin B, an ansamycin antibiotic, functions as an inhibitor of Src family kinases. It exhibits herbicidal effects on most monocotyledonous and dicotyledonous plants and can inhibit the activity of tobacco mosaic virus (TMV), HeLa cells, and Ehrlich cells.Fórmula:C29H40N2O7Forma y color:SolidPeso molecular:528.637Eulicin
CAS:<p>Eulicin is an antifungal agent that inhibits human immunodeficiency virus (HIV) infection and replication. It demonstrates broad-spectrum activity against both Gram-positive and Gram-negative bacteria and can be found in Streptomyces.</p>Fórmula:C24H52N8O2Forma y color:SolidPeso molecular:484.722Fluvirucin A1
CAS:<p>Fluvirucin A1 is a novel antibiotic effective against the Influenza A virus.</p>Fórmula:C23H44N2O5Forma y color:SolidPeso molecular:428.61Anti-ToCV agent 1
Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.Fórmula:C22H19FN2O5SForma y color:SolidPeso molecular:442.46Cytochalasin M
CAS:Cytochalasin M exhibits various biological activities, including reversible inhibition of cytoplasmic division and the suppression of both endocytosis and exocytosis in macrophages.Fórmula:C30H37NO6Forma y color:SolidPeso molecular:507.618Micacocidin B
CAS:<p>Micacocidin B is an antibiotic that exhibits exceptional activity against Mycoplasma species.</p>Fórmula:C27H37CuN3O4S3Forma y color:SolidPeso molecular:627.34Calphostin B
CAS:Calphostins, PKC inhibitors from Cladosporium fungus, include A, B, C, D, I; C is most potent.Fórmula:C37H34O11Forma y color:SolidPeso molecular:654.66GR-112000
CAS:GR-112000 is a peptide-based tachykinin NK2 receptor antagonist.Fórmula:C30H36N6O3Forma y color:SolidPeso molecular:528.65Juglomycin A
CAS:<p>Juglomycin A exhibits broad-spectrum antibacterial and anti-mycobacterial activity and can inhibit Ehrlich ascites carcinoma in mice.</p>Fórmula:C14H10O6Forma y color:SolidPeso molecular:274.2263-Methoxy-2,5-toluquinone
CAS:<p>3-Methoxy-2,5-toluquinone is an antimicrobial agent that exhibits moderate antibacterial and antifungal properties.</p>Fórmula:C8H8O3Forma y color:SolidPeso molecular:152.147Resorthiomycin
CAS:<p>Resorthiomycin is an antitumor antibiotic that can inhibit L5178Y leukemia cells in vitro.</p>Fórmula:C14H20O4SForma y color:SolidPeso molecular:284.371Lp-PLA2-IN-5
CAS:<p>Lp-PLA2-IN-5 inhibits Lp-PLA2 and PAF-AH, potentially useful in Alzheimer's and atherosclerosis studies.</p>Fórmula:C23H18F5N3O4Forma y color:SolidPeso molecular:495.4Carpetimycin A
CAS:<p>Carpetimycin A exhibits potent activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. It also acts as a strong inhibitor of β-lactamase.</p>Fórmula:C14H18N2O6SForma y color:SolidPeso molecular:342.368MRS2279 diammonium
CAS:<p>MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.</p>Fórmula:C13H24ClN7O8P2Forma y color:SolidPeso molecular:503.77Elacestrant S enantiomer
<p>Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.</p>Fórmula:C30H38N2O2Pureza:98%Forma y color:SolidPeso molecular:458.63Trichodermin
CAS:<p>Trichodermin is a naturally occurring sesquiterpene antibiotic (antibiotic) and a powerful inhibitor of protein synthesis (protein synthesis). It binds to eukaryotic ribosomes, inhibiting protein translation by interacting with peptidyl transferase. Trichodermin suppresses oral cancer growth by inducing apoptosis (apoptosis)-related mitochondrial dysfunction and HDAC-2-mediated signaling. It exhibits potent antimicrobial activity against filamentous fungi, yeasts, and bacteria.</p>Fórmula:C17H24O4Forma y color:SolidPeso molecular:292.37Fluoropolyoxin M
CAS:Fluoropolyoxin M exhibits inhibitory activity against Escherichia coli and Enterococcus faecium.Fórmula:C16H22FN5O11Forma y color:SolidPeso molecular:479.371Cryptosporiopsin
CAS:<p>Cryptosporiopsin can be isolated from strains of Cryptosporiopsis sp. and Sporormia affinis. It exhibits antimicrobial activity against various basidiomycetes, alga fungi, ascomycetes, and glaucomycetes responsible for wood decay. Additionally, it inhibits the germination of Phytophthora potatoes spores. Cryptosporiopsin also shows some activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C10H10Cl2O4Forma y color:SolidPeso molecular:265.09NSC 357754
CAS:NSC 357754 is an inhibitor of Claudin. It can enhance transepithelial electrical resistance and reduce specific cation permeability. NSC 357754 is useful for research involving Claudin-2 and/or Claudin-15 mediated intestinal disorders.Fórmula:C26H20N4O2Forma y color:SolidPeso molecular:420.463Polyoxin A
CAS:<p>Polyoxin A is a nucleoside-based antifungal antibiotic.</p>Fórmula:C23H32N6O14Forma y color:SolidPeso molecular:616.532Chrymutasin A
CAS:<p>Chrymutasin A is a glycoside antitumor antibiotic, known for its cytotoxic properties.</p>Fórmula:C33H33NO13Forma y color:SolidPeso molecular:651.614Sannamycin F
CAS:Sannamycin F is an aminoglycoside antibiotic that exhibits mild antibacterial activity against both Gram-positive and Gram-negative bacteria.Fórmula:C18H35N5O6Forma y color:SolidPeso molecular:417.5Quadrilineatin
CAS:<p>Quadrilineatin exhibits antifungal and antibacterial properties.</p>Fórmula:C10H10O4Forma y color:SolidPeso molecular:194.184Seldomycin factor 3
CAS:<p>Seldomycin factor 3 (XK 88-3) is an aminoglycoside antibiotic with broad-spectrum antibacterial activity.</p>Fórmula:C17H35N5O9Forma y color:SolidPeso molecular:453.488Emimycin
CAS:<p>Emimycin exhibits activity against Gram-positive and Gram-negative bacteria, as well as fungi like Saccharomyces cerevisiae (brewer's yeast).</p>Fórmula:C4H4N2O2Forma y color:SolidPeso molecular:112.087Vps34-IN-3
Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .Fórmula:C14H20N4O2Forma y color:SolidPeso molecular:276.33Melithiazole C
CAS:<p>Melithiazol C is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA) with antifungal properties.</p>Fórmula:C16H21NO5SForma y color:SolidPeso molecular:339.407Methyl 5-thia-6,8,11,14-eicosatetraenoate
CAS:Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.Fórmula:C20H32O2SForma y color:SolidPeso molecular:336.53Hydroxymycotrienin A
CAS:Hydroxymycotrienin A is an ansamycin antibiotic with the ability to inhibit human neck tumor cell lines. Its inhibitory effect is more pronounced on HPV-positive neck tumor cells (such as HeLa, CaSKi, and SiHa) compared to HPV-negative cells.Fórmula:C36H48N2O9Forma y color:SolidPeso molecular:652.774Phyllosinol
CAS:Phyllosinol is an antifungal antibiotic.Fórmula:C7H8O4Forma y color:SolidPeso molecular:156.13610-Decarbomethoxyaclacinomycin A
CAS:<p>10-Decarbomethoxyaclacinomycin A is an anthracycline antibiotic produced by the mutant strain Streptomyces galilaeus MA144-Mlt KE303. This compound exhibits antibacterial activity.</p>Fórmula:C40H51NO13Forma y color:SolidPeso molecular:753.832PLAP-IN-1
CAS:<p>PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.</p>Fórmula:C25H21Cl2N3O5Forma y color:SoildPeso molecular:514.36Gentamicin A
CAS:<p>Gentamicin A is an antibiotic exhibiting effective antibacterial activity against both Gram-positive and Gram-negative bacteria, and it also demonstrates activity against most methicillin-sensitive staphylococci.</p>Fórmula:C18H36N4O10Forma y color:SolidPeso molecular:468.499Cytochalasin L
CAS:<p>Cytochalasin L possesses reversible biological activities, including the inhibition of cytoplasmic division, as well as the suppression of both endocytosis and exocytosis in phagocytic macrophages.</p>Fórmula:C32H37NO7Forma y color:SolidPeso molecular:547.6396"'-Deamino-6"'-hydroxyneomycin B
CAS:6"'-Deamino-6"'-hydroxyneomycin B is an aminoglycoside antibiotic produced by [Streptomyces fradiaeUC 75]. It is effective against both Gram-positive and Gram-negative bacteria and serves as an intermediate in the biosynthesis of neomycin.Fórmula:C23H45N5O14Forma y color:SolidPeso molecular:615.628Epoxyquinomicin C
CAS:<p>Epoxyquinomicin C is an antibiotic that can be isolated from Amycolatopsis sp. It exhibits anti-inflammatory properties against collagen-induced arthritis and is also utilized in the synthesis of the NF-κB inhibitor DHMEQ.</p>Fórmula:C14H13NO6Forma y color:SolidPeso molecular:291.256Diaporthin
CAS:<p>Diaporthin is a phytotoxin that can be isolated from Cryphonectria parasitica. It exhibits antibacterial activity.</p>Fórmula:C13H14O5Forma y color:SolidPeso molecular:250.247Diphenicillin
CAS:<p>Diphenicillin (Ancillin (free acid); 2-Biphenylyl penicillin (free acid); SKF-12141 (free acid)) is a penicillin that resists Penicillinase and exhibits antibacterial activity. It shows effective activity against Gram-positive cocci. Diphenicillin is promising for research on infectious diseases caused by Gram-positive bacteria such as staphylococci, pneumococci, and group A streptococci.</p>Fórmula:C21H20N2O4SForma y color:SolidPeso molecular:396.459Pluracidomycin B
CAS:<p>Pluracidomycin B, a carbapenem antibiotic, exhibits activity against both Gram-positive and Gram-negative bacteria and also functions as an inhibitor of β-lactamase enzymes.</p>Fórmula:C11H13NO10S2Forma y color:SolidPeso molecular:383.352Epoxyquinomicin D
CAS:<p>Epoxyquinomicin D is an antibiotic that can be isolated from Amycolatopsis sp. It exhibits anti-inflammatory properties against collagen-induced arthritis.</p>Fórmula:C14H12ClNO6Forma y color:SolidPeso molecular:325.701Deacetylravidomycin N-oxide
CAS:<p>Deacetylravidomycin N-oxide is an antibiotic produced by [Streptomyces ravidus S50905] that exhibits activity against Gram-positive bacteria but is inactive against Gram-negative bacteria. Additionally, Deacetylravidomycin N-oxide demonstrates antitumor properties against P388 leukemia and methylcholanthrene A fibrosarcoma.</p>Fórmula:C31H33NO10Forma y color:SolidPeso molecular:579.594Kigamicin B
CAS:<p>Kigamicin B exhibits activity against gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>Fórmula:C40H45NO15Forma y color:SolidPeso molecular:779.78Nemotinic acid
CAS:<p>Nemotinic acid exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while also displaying weaker activity against Gram-negative bacteria.</p>Fórmula:C11H10O3Forma y color:SolidPeso molecular:190.195Cycloleucomelone
CAS:<p>Cycloleucomelone is a secondary metabolite and a fungal pigment.</p>Fórmula:C18H10O7Forma y color:SolidPeso molecular:338.268Inactone
CAS:<p>Inactone is a biologically active molecule with a 3-pentanoylimino group that inhibits the large ribosomal subunit.</p>Fórmula:C15H21NO4Forma y color:SolidPeso molecular:279.332Antidepressant agent 2
<p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>Fórmula:C21H22ClFN2O3SForma y color:SolidPeso molecular:436.935-cis Carbaprostacyclin
CAS:5-cis Carbaprostacyclin: a PGI2 stable analog; poor human platelet aggregation inhibitor (IC50: 2.8 μM); weakens rabbit artery relaxation (EC50: 104 μM).Fórmula:C21H34O4Forma y color:SolidPeso molecular:350.49Epicorazine B
CAS:<p>Epicorazine B exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, with an MIC of 25 μg/mL.</p>Fórmula:C18H16N2O6S2Forma y color:SolidPeso molecular:420.459Pyralomicin 2c
CAS:<p>Pyralomicin 2c is an antibiotic with antibacterial properties.</p>Fórmula:C19H19Cl2NO8Forma y color:SolidPeso molecular:460.262Glidobactin F
CAS:<p>Glidobactin F is an antitumor antibiotic effective against pathogenic fungi and yeasts. It has been shown to increase the survival time of mice inoculated with leukemia P388 cells.</p>Fórmula:C25H40N4O6Forma y color:SolidPeso molecular:492.608CY208-243 Mandelate
CAS:CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.Fórmula:C27H26N2O3Forma y color:SolidPeso molecular:426.52Nnc 09-0026
CAS:Nnc 09-0026 is a neuronal calcium channel blockerFórmula:C25H35Cl2F3N2OForma y color:SolidPeso molecular:507.46Cirramycin B1
CAS:Cirramycin B1 exhibits activity against both Gram-positive bacteria, Gram-negative bacteria, and mycoplasmas.Fórmula:C37H59NO12Forma y color:SolidPeso molecular:709.864Collinone
CAS:Collinone is a recombinant polyketide antibiotic with antimicrobial activity against Gram-positive bacteria and exhibits cytotoxicity.Fórmula:C27H18O12Forma y color:SolidPeso molecular:534.425Glucosylquestiomycin
CAS:<p>Glucosylquestiomycin exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and yeast.</p>Fórmula:C18H18N2O7Forma y color:SolidPeso molecular:374.345Korormicin
CAS:<p>Korormicin is effective against marine Gram-negative bacteria but does not work against marine Gram-positive bacteria or common bacteria.</p>Fórmula:C25H39NO5Forma y color:SolidPeso molecular:433.581Porothramycin A
CAS:<p>Porothramycin A is an antibiotic effective against Gram-positive bacteria and anaerobic bacteria.</p>Fórmula:C18H21N3O4Forma y color:SolidPeso molecular:343.377Menoxymycin B
CAS:Menoxymycin B is an antibiotic with cytotoxic properties, inhibiting KB and N18-RE-105 cells with IC50 values of 0.22 μM and 0.023 μM, respectively.Fórmula:C25H31NO9Forma y color:SolidPeso molecular:489.515CL656
CAS:<p>CL656 is a stimulator of interferon genes (STING) activator.</p>Fórmula:C20H21F2N9O9P2S2Pureza:98%Forma y color:SolidPeso molecular:695.51Cilengitide hydrochloride
CAS:Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Fórmula:C27H41ClN8O7Forma y color:SolidPeso molecular:625.12Methylenomycin B
CAS:<p>Methylenomycin B is a cyclopentanone-derived antibiotic effective against both Gram-negative and Gram-positive bacteria.</p>Fórmula:C8H10OForma y color:SolidPeso molecular:122.164GSK2945 hydrochloride
<p>GSK2945 HCl is a specific Rev-erbα antagonist, EC50: 21.5 μM (mouse), 20.8 μM (human), increases cholesterol 7α-hydroxylase.</p>Fórmula:C20H19Cl3N2O2SForma y color:SolidPeso molecular:457.8Steroid sulfatase-IN-4
Steroid sulfatase-IN-4 irreversibly inhibits human STS with a 25 nM IC50, useful for endometriosis research.Fórmula:C19H17ClN2O5SForma y color:SolidPeso molecular:420.87Fredericamycin A
CAS:<p>Fredericamycin A exhibits activity against gram-positive bacteria and fungi, demonstrating potent antitumor effects both in vivo and in vitro.</p>Fórmula:C30H21NO9Forma y color:SolidPeso molecular:539.489Jietacin A
CAS:<p>Jietacin A exhibits nematocidal activity, capable of killing Burs helenchus Lignicolus at a concentration of 0.25 μg/mL.</p>Fórmula:C18H34N2O2Forma y color:SolidPeso molecular:310.475Dehydroindapamide
CAS:Dehydroindapamide, an indole form of Indapamide, is utilized to quantify the turnover rate of Indapamide in CYP3A4, which is approximately 10 times higher than that of Indoline, with slightly enhanced affinity for CYP3A4.Fórmula:C16H14ClN3O3SForma y color:SolidPeso molecular:363.82Fosfocytocin
CAS:<p>Fosfocytocin can be found in the Pseudomonas fluorescens strain PK-52 and exhibits very weak antibacterial activity.</p>Fórmula:C12H20N4O13P2Forma y color:SolidPeso molecular:490.254SLC7A11-IN-2
CAS:SLC7A11-IN-2 (Compound 1) is an inhibitor of SLC7A11/xCT. It disrupts the oxidative balance in HeLa cells by decreasing intracellular glutathione levels and increasing oxidative stress, thereby inducing cell death with an IC50 of 10.23 μM. Molecular dynamics simulations have demonstrated that SLC7A11-IN-2 exhibits a stronger binding affinity to SLC7A11 compared to Erastin. This compound is useful for research in the field of cervical cancer.Fórmula:C19H24N4O3Forma y color:SolidPeso molecular:356.42Cyclophellitol
CAS:<p>Cyclophellitol is an inhibitor of β-glycosidase, with an IC50 of 0.8 μg/mL.</p>Fórmula:C7H12O5Forma y color:SolidPeso molecular:176.1676"'-Deamino-6"'-hydroxyparomomycin I
CAS:<p>6"'-Deamino-6"'-hydroxyparomomycin I is an aminoglycoside antibiotic produced by Streptomyces rimosus forma paromomycinus A67 15, exhibiting activity against both Gram-positive and Gram-negative bacteria. It serves as an intermediate in the biosynthesis of paromomycin.</p>Fórmula:C23H44N4O15Forma y color:SolidPeso molecular:616.613PARP1-IN-5
<p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>Fórmula:C25H24N2O5SForma y color:SolidPeso molecular:464.53Chrymutasin B
CAS:<p>Chrymutasin B is a glycoside antitumor antibiotic known for its cytotoxic properties.</p>Fórmula:C32H31NO13Forma y color:SolidPeso molecular:637.587Anti-inflammatory agent 12
<p>Pentacyclic triterpene, anti-inflammatory agent 12, inhibits LPS inflammation (IC50: 2.22 μM). May benefit inflammatory disease studies.</p>Fórmula:C30H50O4Forma y color:SolidPeso molecular:474.72Sannamycin G
CAS:<p>Sannamycin G (Istamycin X0) is an aminoglycoside antibiotic that exhibits only weak antibacterial activity against a limited range of bacteria.</p>Fórmula:C14H30N4O4Forma y color:SolidPeso molecular:318.412NB-216
CAS:NB-216 is a macrocyclic peptidic BACE-1 inhibitor.Fórmula:C35H45N3O4Forma y color:SolidPeso molecular:571.75PX-316
CAS:PX-316: AKT inhibitor, reduces Akt activity by 78% in HT-29 xenografts, effective against MCF-7 and HT-29 cancers, well-tolerated intravenously.Fórmula:C28H57O10PForma y color:SolidPeso molecular:584.72Topoisomerase II inhibitor 5
Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.Fórmula:C26H27N5O4Forma y color:SolidPeso molecular:473.52Neoenactin A
CAS:Neoenactin A exhibits potent activity against yeasts and filamentous fungi.Fórmula:C19H36N2O5Forma y color:SolidPeso molecular:372.5Ezomycin A2
CAS:Ezomycin A2 is an antifungal antibiotic. It is primarily effective against plant pathogens such as Sclerotinia and Botrytis, showing efficacy in controlling crop diseases like sclerotinia rot, botrytis blight, and candidiasis.Fórmula:C19H26N6O12Forma y color:SolidPeso molecular:530.443DS88790512
CAS:DS88790512, IC50 at 11 nM, is an effective, selective, oral bioeffective TRPC6 inhibitor.Fórmula:C22H29N3O2Pureza:98%Forma y color:SolidPeso molecular:367.48AFM-30a hydrochloride
AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.Fórmula:C24H28ClFN6O3Forma y color:SolidPeso molecular:502.97ASP-8731
CAS:ASP8731 is a selective inhibitor of BACH1 that prevents inflammation and vascular occlusion, and induces fetal hemoglobin in sickle cell disease.Fórmula:C20H21N5O4Forma y color:SolidPeso molecular:395.41AX15910
AX15910 is a potent inhibitor of BRD4 and ERK5.Fórmula:C32H38N6O3Forma y color:SolidPeso molecular:554.7STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Fórmula:C17H12N4O4Forma y color:SolidPeso molecular:336.3TY 11223
CAS:TY 11223: stable homoisocarbacyclin analog, potently inhibits platelet aggregation with lasting effect and selective activity.Fórmula:C24H34O5Forma y color:SolidPeso molecular:402.52MRS2179 tetrasodium hydrate
MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.Fórmula:C11H15N5Na4O10P2Forma y color:SolidPeso molecular:576.21BMS-554417
CAS:BMS-554417 inhibits IGF-IR/insulin receptors, curbing cell proliferation and tumor growth, with IC50 values of 120 nm–>8.5 μmol/L.Fórmula:C28H30ClN7O2Forma y color:SolidPeso molecular:532.04LLS30
CAS:<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Fórmula:C34H33Cl4N5O3Forma y color:SolidPeso molecular:701.47PF-06305591 dihydrate
PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADMEFórmula:C15H26N4O3Forma y color:SolidPeso molecular:310.39Epoxyquinomicin B
CAS:Epoxyquinomicin B is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus, with a minimum inhibitory concentration (MIC) of 6.25-12.5 µg/mL. It also shows cytotoxicity in cancer cells L1210, with an IC50 of 16.3 µg/mL. Additionally, Epoxyquinomicin B demonstrates anti-inflammatory effects on collagen-induced arthritis.Fórmula:C14H11NO6Forma y color:SolidPeso molecular:289.24BGC-638
CAS:BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.Fórmula:C32H33N5O9Forma y color:SolidPeso molecular:631.63Balanol
CAS:Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.Fórmula:C28H26N2O10Forma y color:SolidPeso molecular:550.51CI 922
CAS:<p>CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.</p>Fórmula:C26H30N10O6Forma y color:SolidPeso molecular:578.58Carbacyclin
CAS:Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.Fórmula:C21H34O4Pureza:98%Forma y color:SolidPeso molecular:350.49LIT-001 free base
CAS:LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.Fórmula:C28H33N7O2SPureza:98%Forma y color:SolidPeso molecular:531.67Antitrypanosomal agent 6
<p>Compound 18a: potent vs. T. brucei (IC50: 0.47 μM), >2x efficacy compared to Nifurtimox, good ADME, binds AT-rich DNA.</p>Fórmula:C22H29Cl2N5OForma y color:SolidPeso molecular:450.4CHNQD-01255
CAS:<p>CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).</p>Fórmula:C23H29NO6Forma y color:SolidPeso molecular:415.48Sekdel sequence
CAS:Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.Fórmula:C29H49N7O14Forma y color:SolidPeso molecular:719.74Thalicarpine
CAS:<p>Thalicarpine, a natural anticancer alkaloid, inhibits p-glycoprotein and induces DNA damage, arresting cell cycle.</p>Fórmula:C41H48N2O8Forma y color:SolidPeso molecular:696.83OM-153
CAS:OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.Fórmula:C28H24FN7O2Forma y color:SolidPeso molecular:509.53Oudemansin A
CAS:<p>Oudemansin A is an antibiotic that targets fungi, inhibiting the synthesis of proteins, RNA, and DNA.</p>Fórmula:C17H22O4Forma y color:SolidPeso molecular:290.35Npc 12626
CAS:Npc 12626 is a N-methyl-D-aspartate receptor antagonist; NPC 17742, the (2R,4R,5S)-isomer, is the most potent isomer in the mixture NPC 12626.Fórmula:C11H22NO5PForma y color:SolidPeso molecular:279.27Methylenomycin A
CAS:<p>Methylenomycin A is a cyclopentanone-derived antibiotic effective against both Gram-negative and Gram-positive bacteria.</p>Fórmula:C9H10O4Forma y color:SolidPeso molecular:182.173AZD-3199 dihydrobromide
CAS:<p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>Fórmula:C32H44Br2N4O4SForma y color:SolidPeso molecular:740.59Epicorazine A
CAS:<p>Epicorazine A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, showing an MIC of 25 μg/mL.</p>Fórmula:C18H16N2O6S2Forma y color:SolidPeso molecular:420.459NCATS-SM4487
CAS:NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).Fórmula:C25H24ClFN8O2Forma y color:SolidPeso molecular:522.963'-GMP
CAS:<p>3'-GMP is a nucleotide that can be isolated from the tubers of Helianthus tuberosus L. (Jerusalem artichoke).</p>Fórmula:C10H14N5O8PForma y color:SolidPeso molecular:363.221Fistupyrone
CAS:<p>Fistupyrone, an antibiotic, is a microbial metabolite found in Streptomyces (TP-A0569). It has the ability to inhibit infections caused by Alternaria brassicicola in Chinese cabbage.</p>Fórmula:C10H14O3Forma y color:SolidPeso molecular:182.216Calphostin A
CAS:Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.Fórmula:C44H38O12Forma y color:SolidPeso molecular:758.77Miyakamide B2
CAS:Miyakamide B2 is an antibiotic with insecticidal properties. It suppresses the growth of brine shrimp and shows weak activity against Xanthomonas species. The IC50 for inhibition of P388 cells by Miyakamide B2 is 7.6 μg/mL.Fórmula:C31H32N4O4Forma y color:SolidPeso molecular:524.61Sapintoxin D
CAS:Sapintoxin D is a fluorescent phorbol ester and selective activator of protein kinase C.Fórmula:C30H37NO8Forma y color:SolidPeso molecular:539.62Deoxyfuconojirimycin hydrochloride
CAS:Deoxyfuconojirimycin hydrochloride acts as a specific competitive inhibitor targeting human liver α-L-fucosidase.Fórmula:C6H14ClNO3Forma y color:SolidPeso molecular:183.63LPM4870108
<p>LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.</p>Fórmula:C20H19FN6O3Forma y color:SolidPeso molecular:410.4Oberadilol
CAS:Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory actionFórmula:C25H30ClN5O3Forma y color:SolidPeso molecular:483.99Eilatine
CAS:Eilatine is a novel marine alkaloid inhibits in vitro proliferation of progenitor cells in chronic myeloid leukemia patients.Fórmula:C24H12N4Forma y color:SolidPeso molecular:356.38Cinatrin C1
CAS:Cinatrin C1 is a phospholipase A2 (PLA2) inhibitor that can be extracted from the Circinotrichum falcatisporum strain RF-641.Fórmula:C18H30O8Forma y color:SolidPeso molecular:374.426MPro N3
CAS:Mpro inhibitor blocks MHV-A29, HCoV-229E, FOPV (IC50: 2.7–8.8 μM), and SARS-CoV-2 (IC50: 16.8 μM) in plaque assays.Fórmula:C35H48N6O8Forma y color:SolidPeso molecular:680.79Longicoricin
CAS:<p>Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.</p>Fórmula:C37H68O6Forma y color:SolidPeso molecular:608.93KT2-962
CAS:<p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>Fórmula:C23H27ClNNaO5S2Forma y color:SolidPeso molecular:520.04Paulomycin A2
CAS:Paulomycin A2 exhibits antibacterial activity against Gram-positive bacteria and specifically inhibits Staphylococcus aureus that is resistant to penicillin, streptomycin, neomycin, and macrolide antibiotics.Fórmula:C34H46N2O17SForma y color:SolidPeso molecular:786.797Pegcantratinib
CAS:Pegcantratinib is a tropomyosin receptor kinase inhibitor for treatment for inherited CYLD defective skin tumours.Fórmula:C32H28N4O7Forma y color:SolidPeso molecular:580.59C20 Sphingomyelin (d18:1/20:1)
CAS:C20 Sphingomyelin (d18:1/20:1) (Compound SM:20:1) is a type of sphingolipid. This compound shows potential for research related to motor neuron diseases, such as amyotrophic lateral sclerosis (ALS) and primary lateral sclerosis (PLS).Fórmula:C43H85N2O6PForma y color:SolidPeso molecular:757.119Hydroxynybomycin
CAS:Hydroxynybomycin is an antibiotic with activity against Gram-negative bacteria.Fórmula:C16H14N2O5Forma y color:SolidPeso molecular:314.293Lactaroviolin
CAS:Lactaroviolin is an aromatic derivative antibiotic that can inhibit the growth of Mycobacterium tuberculosis.Fórmula:C15H14OForma y color:SolidPeso molecular:210.271Chloronectrin
CAS:<p>Chloronectrin exhibits activity against Gram-positive bacteria.</p>Fórmula:C25H33ClO6Forma y color:SolidPeso molecular:464.979Milbemycin α11
CAS:<p>Milbemycin α11 (Meilingmycin A) is an antibiotic known for its ability to eliminate nematodes and mites.</p>Fórmula:C36H50O9Forma y color:SolidPeso molecular:626.78Griseochelin
CAS:<p>Griseochelin exhibits activity against Gram-negative bacteria and inhibits Coccidioides.</p>Fórmula:C33H60O7Forma y color:SolidPeso molecular:568.825Halomicin B
CAS:<p>Halomicin B is an ansamycin-type antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C43H58N2O12Forma y color:SolidPeso molecular:794.927Macquarimicin C
CAS:Macquarimicin C is an antibiotic.Fórmula:C22H26O5Forma y color:SolidPeso molecular:370.439Fluvirucin B2
CAS:<p>Fluvirucin B2 is a novel antibiotic effective against the influenza A virus.</p>Fórmula:C25H48N2O5Forma y color:SolidPeso molecular:456.66LGB-321 HCl
CAS:LGB-321: potent, selective PIM kinase inhibitor, active against PIM2, halts diverse blood cancers' growth, orally effective in mice.Fórmula:C23H23ClF3N5O2Forma y color:SolidPeso molecular:493.919-O-Demethyltrigonostemone
CAS:<p>9-O-Demethyltrigonostemone is a natural IDO1 inhibitor, cytotoxic and antiplasmodial agent from the Roots of Strophioblachia fimbricalyx.</p>Fórmula:C19H20O4Forma y color:SolidPeso molecular:312.36Chelocardin
CAS:Chelocardin exhibits activity against Gram-positive and Gram-negative bacteria.Fórmula:C22H21NO7Forma y color:SolidPeso molecular:411.405Polyoxin E
CAS:<p>Polyoxin E is a nucleoside antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight.</p>Fórmula:C17H23N5O13Forma y color:SolidPeso molecular:505.39Medermycin
CAS:<p>Lactoquinomycin A is a quinone antibiotic displaying activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy is weaker against the latter and it is ineffective against fungi. It inhibits various cell lines, including lymphoma L5178Y progenitor cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, murine leukemia L-1210 cells, and murine leukemia P388 cells, with ID50 values (μg/mL) of 0.02, 0.006, 0.008, 0.033, 0.013, and 0.03, respectively.</p>Fórmula:C24H27NO8Forma y color:SolidPeso molecular:457.473HR-546
CAS:HR-546 is a prostaglandin E2 and prostaglandin F2alpha antagonist.Fórmula:C26H44O6Forma y color:SolidPeso molecular:452.62Mutalomycin
CAS:Mutalomycin is a polyether antibiotic with activity against Gram-positive bacteria, mycoplasma, and coccidia.Fórmula:C41H70O12Forma y color:SolidPeso molecular:754.987Pacidamycin D
CAS:<p>Pacidamycin D is an antibiotic of the Pacidamycin class, demonstrating activity against Pseudomonas aeruginosa with a minimum inhibitory concentration (MIC) of 4-16 μg/mL. It shows no efficacy against other Gram-negative or Gram-positive bacteria, nor does it affect drug-resistant strains of Pseudomonas aeruginosa.</p>Fórmula:C32H41N9O10Forma y color:SolidPeso molecular:711.722Phellinsin
CAS:<p>Phellinsin selectively inhibits the activity of chitin synthase I and II, with IC50 values of 76 and 28 μg/mL, respectively. It also exhibits antimicrobial effects against pathogens such as anthracnose, rice blast fungus, Aspergillus fumigatus, and Trichophyton mentagrophytes, with a MIC ranging from 12.5 to 50 μg/mL.</p>Fórmula:C18H14O8Forma y color:SolidPeso molecular:358.302-Hydroxygentamicin A3
CAS:<p>2-Hydroxygentamicin A3 is an aminoglycoside antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C18H36N4O11Forma y color:SolidPeso molecular:484.499Antitumor agent-50
Antitumor agent-50 (compound 1a) is a thiazolidinone.Fórmula:C17H14FNO3SForma y color:SolidPeso molecular:331.36Fosfazinomycin B
CAS:<p>Fosfazinomycin B exhibits activity against plant pathogenic fungi such as the rice blast pathogen (Xanthomonas oryzae).</p>Fórmula:C10H23N6O6PForma y color:SolidPeso molecular:354.3Nanaomycin E
CAS:<p>Nanaomycin E is an antibiotic with activity against Gram-positive bacteria and fungi.</p>Fórmula:C16H14O7Forma y color:SolidPeso molecular:318.278Kigamicin A
CAS:<p>Kigamicin A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>Fórmula:C34H35NO13Forma y color:SolidPeso molecular:665.64Seldomycin factor 1
CAS:Seldomycin factor 1 (XK 88-1) is an aminoglycoside antibiotic known for its broad-spectrum antibacterial activity.Fórmula:C17H34N4O10Forma y color:SolidPeso molecular:454.473Pyrisulfoxin A
CAS:<p>Pyrisulfoxin A is an antibiotic that can be found in Streptomyces callfornicus [BS-75].</p>Fórmula:C13H13N3O3SForma y color:SolidPeso molecular:291.326SBI-581
SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.Fórmula:C24H21N3O2Forma y color:SolidPeso molecular:383.44Monensin C
CAS:Monensin C is an oxygenated heterocyclic polyether antibiotic. It exhibits activity against bacteria, mycobacteria, fungi, and protozoa, though it is less effective against Gram-negative bacteria. Additionally, it shows inhibitory effects on HeLa cells.Fórmula:C37H64O11Forma y color:SolidPeso molecular:684.898Ophiobolin D
CAS:Ophiobolin D is a terpene antibiotic with mild inhibitory effects on Staphylococcus aureus.Fórmula:C25H36O4Forma y color:SolidPeso molecular:400.55AVE-1330A free acid
CAS:AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.Fórmula:C7H11N3O6SForma y color:SolidPeso molecular:265.24Napyradiomycin C2
CAS:<p>Napyradiomycin C2 is an antibiotic with activity against Gram-positive bacteria and mycobacteria.</p>Fórmula:C25H27Cl3O5Forma y color:SolidPeso molecular:513.8384"-Demethylgentamicin C1
CAS:<p>4"-Demethylgentamicin C1 exhibits antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H41N5O7Forma y color:SolidPeso molecular:463.57Fudecalone
CAS:<p>Fudecalone is produced by the Penicillium strain FO-2030. It completely inhibits the coccidian parasite Eimeria Tenella that is resistant to Monensin.</p>Fórmula:C15H22O3Forma y color:SolidPeso molecular:250.33TrxR-IN-2
TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.Fórmula:C22H22N4O4Forma y color:SolidPeso molecular:406.43Carnostatine
<p>Carnostatine (SAN9812), a potent CN1 inhibitor with 11 nM K i, may boost renal carnosine to treat DN.</p>Fórmula:C10H16N4O4Pureza:98%Forma y color:SolidPeso molecular:256.26Chitinase-IN-4
Chitinase-IN-4 (compound 8f) is a potent and selective inhibitor of OfChi-h with an IC50 value of 0.1 μM and good insecticidal activity.Fórmula:C21H24ClN7Forma y color:SolidPeso molecular:409.92Gilvocarcin E
CAS:<p>Gilvocarcin E exhibits activity against Gram-positive bacteria and is capable of inhibiting Sarcoma 180 and P388 leukemia cells.</p>Fórmula:C27H28O9Forma y color:SolidPeso molecular:496.506Memnobotrin B
CAS:Memnobotrin B is an antibiotic that exhibits inhibitory effects on the NCI-460, MCF7, and SF-268 cell lines.Fórmula:C27H37NO6Forma y color:SolidPeso molecular:471.59Pyrrolomycin E
CAS:<p>Pyrrolomycin E is a pyrrole-based antibiotic with activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>Fórmula:C10H5Cl3N2O3Forma y color:SolidPeso molecular:307.5174-Nitrochalcone
CAS:<p>4-Nitrochalcone (2-(4-Nitrobenzylidene)acetophenone) inhibits proteasomes and suppresses TNFα-induced NF-κB activity.</p>Fórmula:C15H11NO3Forma y color:SolidPeso molecular:253.25Flavipucine
CAS:<p>Flavipucine (Flavipucin) is a glutarimide antibiotic found in the Aspergillus flavipes F-2090/7 strain. It exhibits antibacterial activity against Bacillus subtilis, possesses antiprotozoal properties, and demonstrates cytotoxic effects on various cancer cells.</p>Fórmula:C12H15NO4Forma y color:SolidPeso molecular:237.252ER272
CAS:<p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>Fórmula:C24H34O6Forma y color:SolidPeso molecular:418.52O-Demethylpaulomycin A
CAS:<p>O-Demethylpaulomycin A is an antibiotic known for its antibacterial properties. It is particularly effective against Gram-positive bacteria, including Staphylococcus aureus.</p>Fórmula:C33H44N2O17SForma y color:SolidPeso molecular:772.771Chitinovorin C
CAS:Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.Fórmula:C15H20N4O8SForma y color:SolidPeso molecular:416.406STAT3-IN-7
CAS:STAT3-IN-7, an orally active aryl sulfonamido azetidine compound, serves as a STAT3 inhibitor with anticancer activities.Fórmula:C30H26F5N5O4SForma y color:SolidPeso molecular:647.62Deoxyfrenolicin
CAS:<p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>Fórmula:C18H18O6Forma y color:SolidPeso molecular:330.332RSK4-IN-1
CAS:RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.Fórmula:C19H20F2N4O3Forma y color:SolidPeso molecular:390.38Ayapin
CAS:<p>Ayapin, found in sunflowers, is a primary plant phytoalexin. It inhibits the growth of S. scerorotiorum, with an IC50 of 0.16 mM indicating 50% inhibition. Ayapin is utilized in studies on controlling sclerotinia stem rot.</p>Fórmula:C10H6O4Forma y color:SolidPeso molecular:190.15Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Fórmula:C21H36O7Forma y color:SolidPeso molecular:400.506ACT-281959
CAS:<p>ACT-281959, a prodrug of ACT-246475, is a potent P2Y12 antagonist, better than Clopidogrel, effective orally, and in human trials.</p>Fórmula:C38H55N6O14PForma y color:SolidPeso molecular:850.85Lactoquinomycin B
CAS:<p>Lactoquinomycin B is a quinone antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy against Gram-negative species is weaker and it does not affect fungi. It inhibits various cell lines, including lymphoma L5178Y parental cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, and murine leukemia L-1210 and P388 cells, with ID50 (μg/mL) values of 0.43, 0.21, 0.19, 0.16, 0.2, and 0.12, respectively.</p>Fórmula:C24H27NO9Forma y color:SolidPeso molecular:473.473Halomicin D
CAS:Halomicin D is an ansamycin-class antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.Fórmula:C43H56N2O12Forma y color:SolidPeso molecular:792.91111-Demethyltomaymycin
CAS:<p>11-Demethyltomaymycin is an antibiotic that exhibits antiviral activity against Escherichia coli T1 and T3 bacteriophages, along with antibacterial properties against Gram-positive bacteria. Furthermore, it shows cytotoxic effects on leukemia L1210 cells.</p>Fórmula:C15H18N2O4Forma y color:SolidPeso molecular:290.314Narbomycin
CAS:<p>Narbomycin exhibits activity against Gram-positive bacteria.</p>Fórmula:C28H47NO7Forma y color:SolidPeso molecular:509.675TTK inhibitor 3
CAS:TTK inhibitor 3 is a potent and selective TTK (an essential spindle assembly checkpoint enzyme) inhibitor with an IC 50 value of 3.0 nM.Fórmula:C42H49N9O3Forma y color:SolidPeso molecular:727.9MraY-IN-1
MraY-IN-1 inhibits MraY (IC50: 140μM), fights E. coli K12, B. subtilis W23, P. fluorescens (MIC50: 7-46μg/ml), for antimicrobial research.Fórmula:C35H46N3O5Forma y color:SolidPeso molecular:588.76AZ0108
CAS:<p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>Fórmula:C24H20F4N6O2Forma y color:SolidPeso molecular:500.4518:0-LPS
CAS:18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.Fórmula:C24H48NO9PForma y color:SolidPeso molecular:525.613Feudomycin B
CAS:Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.Fórmula:C28H31NO10Forma y color:SolidPeso molecular:541.546Rimegepant sulfate hydrate
CAS:<p>Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.</p>Fórmula:C56H64F4N12O13SForma y color:SolidPeso molecular:1221.2526Fumaryl-DL-alanine
CAS:Fumaryl-DL-alanine exhibits activity against Gram-positive bacteria.Fórmula:C7H9NO5Forma y color:SolidPeso molecular:187.15AGN-795
CAS:<p>AGN-795 is a biochemical.</p>Fórmula:C14H20N2Forma y color:SolidPeso molecular:216.328Nanaomycin B
CAS:<p>Nanaomycin B is an antibiotic with activity against Gram-positive bacteria, mycobacteria, mycoplasma, and fungi.</p>Fórmula:C16H16O7Forma y color:SolidPeso molecular:320.294Endophenazine A
CAS:<p>Endophenazine A exhibits activity against Gram-positive bacteria and filamentous fungi such as Mucor and Penicillium, but demonstrates limited herbicidal effect on Lemna.</p>Fórmula:C18H16N2O2Forma y color:SolidPeso molecular:292.332Pterulinic acid
CAS:<p>Pterulinic acid is an inhibitor of coenzyme I:coenzyme Q oxidoreductase. It demonstrates IC50 values (μg/mL) of 50 for the mammalian cell line L1210, 20 for HL60, 25 for HeLaS3, and 100 for BHK.</p>Fórmula:C15H11ClO4Forma y color:SolidPeso molecular:290.70Cystothiazole A
CAS:<p>Cystothiazole A exhibits antifungal properties, effectively inhibiting Candida albicans, Saccharomyces cerevisiae, and Aspergillus fumigatus with minimum inhibitory concentrations (MIC) of 0.4 μg/mL, 0.1 μg/mL, and 1.6 μg/mL, respectively. It also demonstrates inhibitory activity against human tumor cells such as HPT-116 and K562, with MIC values of 130 ng/mL and 110 ng/mL. However, it shows no antibacterial activity.</p>Fórmula:C20H26N2O4S2Forma y color:SolidPeso molecular:422.561SphK2-IN-1
CAS:<p>SphK2-IN-1 is an SphK2 inhibitor with an IC50 value of 0.359 μM. SphK2-IN-1 can be used to study cancer, inflammation, neurological and cardiovascular diseases.</p>Fórmula:C23H22ClF3N8OForma y color:SolidPeso molecular:518.92OUN58101
CAS:<p>OUN58101, also MDK-8101/BI-D, is an RSV L-protein inhibitor with no formal name, first reported in patent WO 2005042530.</p>Fórmula:C32H36N6O6Forma y color:SolidPeso molecular:600.662-Hydroxygentamicin C2
CAS:2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.Fórmula:C20H41N5O8Forma y color:SolidPeso molecular:479.568Formadicin B
CAS:<p>Formadicin B exhibits significant activity against various species of Pseudomonas, Proteus, and Alcaligenes.</p>Fórmula:C30H34N4O15Forma y color:SolidPeso molecular:690.61Menoxymycin A
CAS:<p>Menoxymycin A is an antibiotic with cytotoxic properties. It inhibits the growth of KB and N18-RE-105 cells, with IC50 values of 0.86 μM and 0.14 μM, respectively.</p>Fórmula:C24H27NO9Forma y color:SolidPeso molecular:473.473
