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Otros inhibidores

Otros inhibidores

Esta categoría abarca una amplia variedad de inhibidores que no encajan en las clasificaciones estándar, pero que son fundamentales para diversas investigaciones bioquímicas y farmacológicas. Estos inhibidores pueden dirigirse a vías, enzimas e interacciones moleculares únicas o menos estudiadas, proporcionando herramientas valiosas para áreas de investigación especializadas. En CymitQuimica, ofrecemos una selección diversa de inhibidores de alta calidad que abarcan múltiples objetivos biológicos y disciplinas de investigación, lo que le permite explorar nuevas vías terapéuticas y profundizar su comprensión de los procesos biológicos complejos.

Se han encontrado 37902 productos de "Otros inhibidores"

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  • 18:0-LPS

    CAS:
    <p>18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.</p>
    Fórmula:C24H48NO9P
    Forma y color:Solid
    Peso molecular:525.613
  • O-Desmethyl Midostaurin

    CAS:
    O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.
    Fórmula:C34H28N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:556.61
  • Namitecan

    CAS:
    <p>Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.</p>
    Fórmula:C23H22N4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:434.44
  • Antibiotic LL Z1640-2

    CAS:
    <p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>
    Fórmula:C19H22O7
    Forma y color:Solid
    Peso molecular:362.38
  • Dexnebivolol

    CAS:
    <p>Dexnebivolol (R67138), a ß-adrenergic antagonist, is Nebivolol's enantiomer with β1 blocking and vasodilation properties.</p>
    Fórmula:C22H25F2NO4
    Forma y color:Solid
    Peso molecular:405.43
  • Oncopterin

    CAS:
    <p>Oncopterin is found in urine from patients with solid and blood cancers.</p>
    Fórmula:C12H18N6O3
    Forma y color:Solid
    Peso molecular:294.31
  • (±)-HIP-B

    CAS:
    <p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>
    Fórmula:C6H8N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:172.14
  • 9-Hydroxyoudemansin A

    CAS:
    <p>9-Hydroxyoudemansin A exhibits antifungal activity with a minimum inhibitory concentration (MIC) of 12.5 μg/mL against Saccharomyces cerevisiae. It shows resistance to fungi such as Candida albicans, Rhodotorula, Penicillium, and Streptomyces, with MIC values all exceeding 50 μg/mL. It does not possess antibacterial properties.</p>
    Fórmula:C16H20O4
    Forma y color:Solid
    Peso molecular:276.328
  • Granaticin B

    CAS:
    <p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>
    Fórmula:C28H30O12
    Forma y color:Solid
    Peso molecular:558.531
  • Chlorflavonin

    CAS:
    <p>Chlorflavonin exhibits antifungal activity against several fungi, including Aspergillus, yeast, and Botrytis cinerea, with exceptionally strong activity against Aspergillus nidulans, where the minimum inhibitory concentration is as low as 0.08 μg/mL.</p>
    Fórmula:C18H15ClO7
    Forma y color:Solid
    Peso molecular:378.761
  • FTI-2628

    CAS:
    <p>FTI-2628 is a novel inhibitor of protein farnesyltransferase (FT), inhibiting the growth of P. falciparum in red blood cells and suppressing parasitemia.</p>
    Fórmula:C31H34N4O3S
    Forma y color:Solid
    Peso molecular:542.69
  • Unoprostone isopropyl

    CAS:
    <p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>
    Fórmula:C25H44O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:424.61
  • Hetrombopag olamine

    CAS:
    <p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>
    Fórmula:C29H36N6O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:580.63
  • Ep vinyl quinidine

    CAS:
    <p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>
    Fórmula:C20H24N2O2
    Forma y color:Solid
    Peso molecular:324.42
  • GW311616

    CAS:
    <p>GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>
    Fórmula:C19H31N3O4S
    Forma y color:Solid
    Peso molecular:397.53
  • 12(S)-HEPE

    CAS:
    <p>12(S)-HEPE, made from EPA by 12-LO, is an anti-inflammatory ω-3 derivative affecting leukotriene formation.</p>
    Fórmula:C20H30O3
    Forma y color:Solid
    Peso molecular:318.45
  • HbF inducer-1


    <p>HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.</p>
    Fórmula:C18H19N3O3
    Forma y color:Solid
    Peso molecular:325.36
  • Leucomycin A7

    CAS:
    <p>Leucomycin A7 is a component of the leucomycin complex, isolated from *Streptomyces kitasatoensis*. It possesses antibacterial activity, effectively inhibiting the growth of gram-positive bacteria, while its inhibitory effect on gram-negative bacteria is comparatively weaker.</p>
    Fórmula:C38H63NO14
    Forma y color:Solid
    Peso molecular:757.905
  • Pyrrolomycin A

    CAS:
    <p>Pyrrolomycin A is a pyrrole antibiotic that exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>
    Fórmula:C4H2Cl2N2O2
    Forma y color:Solid
    Peso molecular:180.977
  • Pterulinic acid

    CAS:
    <p>Pterulinic acid is an inhibitor of coenzyme I:coenzyme Q oxidoreductase. It demonstrates IC50 values (μg/mL) of 50 for the mammalian cell line L1210, 20 for HL60, 25 for HeLaS3, and 100 for BHK.</p>
    Fórmula:C15H11ClO4
    Forma y color:Solid
    Peso molecular:290.70
  • Memnobotrin A

    CAS:
    <p>Memnobotrin A is an antibiotic with inhibitory effects on the NCI-460, MCF7, and SF-268 cell lines.</p>
    Fórmula:C25H33NO5
    Forma y color:Solid
    Peso molecular:427.53
  • DDCPPB-Glu

    CAS:
    <p>DDCPPB-Glu is a 6-5 fused ring heterocycle antifolate that shows antitumor activity.</p>
    Fórmula:C22H27N5O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:441.48
  • Ceclazepide

    CAS:
    <p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>
    Fórmula:C30H32N6O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:556.61
  • DMP 728

    CAS:
    <p>DMP 728 is an antagonist of Glycoprotein IIb-IIIa.</p>
    Fórmula:C26H40N8O10S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:656.71
  • NSC 357754

    CAS:
    <p>NSC 357754 is an inhibitor of Claudin. It can enhance transepithelial electrical resistance and reduce specific cation permeability. NSC 357754 is useful for research involving Claudin-2 and/or Claudin-15 mediated intestinal disorders.</p>
    Fórmula:C26H20N4O2
    Forma y color:Solid
    Peso molecular:420.463
  • (rel)-Myrislignan

    CAS:
    <p>(rel)-Myrislignan, a lignan compound with a relative configuration, has been isolated from Myristica fragrans Houtt.</p>
    Fórmula:C21H26O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:374.43
  • (R)-FL118

    CAS:
    <p>FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.</p>
    Fórmula:C21H16N2O6
    Forma y color:Solid
    Peso molecular:392.36
  • Orvepitant

    CAS:
    <p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>
    Fórmula:C31H35F7N4O2
    Forma y color:Solid
    Peso molecular:628.62
  • Feudomycin B

    CAS:
    <p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>
    Fórmula:C28H31NO10
    Forma y color:Solid
    Peso molecular:541.546
  • SORT1-IN-1

    CAS:
    <p>SORT1-IN-1 (compound 2) is a SORT1 inhibitor.</p>
    Fórmula:C17H13F3N2O4
    Forma y color:Solid
    Peso molecular:366.29
  • PD 113271

    CAS:
    <p>PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.</p>
    Fórmula:C19H27O10P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:446.39
  • Adecypenol

    CAS:
    <p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>
    Fórmula:C12H16N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:280.28
  • hCA IX-IN-1


    <p>hCA IX-IN-1 inhibits human carbonic anhydrases I, II, IX, and XII with Ki values of 331.4, 28.4, 9.4, 17.8 nM and exhibits anticancer properties.</p>
    Fórmula:C19H18N2O3S
    Forma y color:Solid
    Peso molecular:354.42
  • MDK-3298

    CAS:
    <p>MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).</p>
    Fórmula:C35H32BN3O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:617.46
  • S-1033

    CAS:
    <p>S-1033 is an FP receptor agonist.</p>
    Fórmula:C20H33NaO4
    Forma y color:Solid
    Peso molecular:360.4698
  • Leucomycin U

    CAS:
    <p>Leucomycin U is a macrolide antibiotic. It demonstrates significant activity against Gram-positive bacteria and also exhibits effects on spirochetes, rickettsiae, and chlamydiae.</p>
    Fórmula:C37H61NO14
    Forma y color:Solid
    Peso molecular:743.878
  • SLN124


    <p>SLN124, a GalNAc-siRNA targeting TMPRSS6, may normalize iron balance by restoring ferroregulation.</p>
    Forma y color:Solid
  • Mesulergine

    CAS:
    <p>Mesulergine is metabolized into dopaminergic agonists.</p>
    Fórmula:C18H26N4O2S
    Forma y color:Solid
    Peso molecular:362.49
  • Asperenone

    CAS:
    <p>Asperenone is a 15-lipoxygenase (15-LOX) inhibitor with an IC50 of 0.3 mM. Additionally, it acts as a platelet aggregation inhibitor with an IC50 of 0.23 mM. Asperenone also exhibits antifungal properties, inhibiting the growth of pathogenic fungi Ophiostoma crassivaginatum and O. piliferum, and may be utilized in research related to cardiovascular diseases and anti-infective treatments.</p>
    Fórmula:C20H22O
    Forma y color:Solid
    Peso molecular:278.388
  • C.I. Pigment Red 60

    CAS:
    <p>C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.</p>
    Fórmula:C17H9N2Na3O9S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:518.35
  • Gepotidacin hydrochloride

    CAS:
    <p>Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.</p>
    Fórmula:C24H29ClN6O3
    Forma y color:Solid
    Peso molecular:484.98
  • YKL-04-085

    CAS:
    <p>YKL-04-085 inhibits viral translation effectively, with strong antiviral action at much lower doses than those affecting host-cell growth.</p>
    Fórmula:C30H29N5O2
    Forma y color:Solid
    Peso molecular:491.6
  • Lycopodine

    CAS:
    <p>Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of</p>
    Fórmula:C16H25NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:247.38
  • KF-19418

    CAS:
    <p>KF-19418 is a follicle stimulant that directly activates follicles in vitro and promotes hair growth in vivo.</p>
    Fórmula:C21H14N4O
    Forma y color:Solid
    Peso molecular:338.36
  • Anti-Trypanosoma cruzi agent-1


    <p>Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.</p>
    Fórmula:C23H29N3O5
    Forma y color:Solid
    Peso molecular:427.49
  • Taprostene

    CAS:
    <p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>
    Fórmula:C24H30O5
    Forma y color:Solid
    Peso molecular:398.49
  • 8,9-Epoxyeicosatrienoic acid

    CAS:
    <p>8,9-Epoxyeicosatrienoic acid offers unique protective effects on the glomerulus. It inhibits the increase in glomerular albumin permeability caused by circulating permeability factors (FSPF). Additionally, 8,9-Epoxyeicosatrienoic acid is used in research related to glomerular dysfunction.</p>
    Fórmula:C20H32O3
    Forma y color:Solid
    Peso molecular:320.47
  • Ciprokiren

    CAS:
    <p>Ciprokiren, a renin inhibitor by Roche, halts human renin; IC50: 0.07/0.65 nmol/L. Lowers blood pressure in animals. Preclinical development ceased.</p>
    Fórmula:C37H55N5O8S
    Forma y color:Solid
    Peso molecular:729.93
  • Ornoprostil

    CAS:
    <p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>
    Fórmula:C23H38O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.54
  • (-)-15-Deoxyspergualin

    CAS:
    <p>(-)-15-Deoxyspergualin is a potent antitumor agent that demonstrates significant inhibition against mouse leukemia L-1210.</p>
    Fórmula:C17H37N7O3
    Forma y color:Solid
    Peso molecular:387.52
  • Butaprost

    CAS:
    <p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>
    Fórmula:C24H40O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:408.57
  • BE-10988

    CAS:
    <p>BE-10988 is a DNA topoisomerase (DNAtopoisomerase) inhibitor. It suppresses the growth of P388 murine leukemia cell lines that are resistant to Doxorubicin and Vinblastine by promoting the formation of DNA topoisomerase complexes.</p>
    Fórmula:C13H10N4O3S
    Forma y color:Solid
    Peso molecular:302.31
  • AMD-7049

    CAS:
    <p>AMD-7049 is a biochemical.</p>
    Fórmula:C25H39N5
    Forma y color:Solid
    Peso molecular:409.61
  • (S)-5-hydroxy-6-methoxy Duloxetine maleate


    <p>(S)-5-hydroxy-6-methoxy Duloxetine, an active metabolite of the (S)-duloxetine, functions as a serotonin (5-HT) and norepinephrine reuptake inhibitor.</p>
    Fórmula:C19H21NO3S·C4H4O4
    Forma y color:Solid
    Peso molecular:459.51
  • RS 2135

    CAS:
    <p>RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.</p>
    Fórmula:C18H21ClN2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:332.83
  • Erizepine

    CAS:
    <p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>
    Fórmula:C20H22N2
    Forma y color:Solid
    Peso molecular:290.4
  • OM-153

    CAS:
    <p>OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.</p>
    Fórmula:C28H24FN7O2
    Forma y color:Solid
    Peso molecular:509.53
  • SARS-CoV-2-IN-6


    <p>SARS-CoV-2-IN-6 is an inhibitor of SARS-CoV-2 3CLpro with the IC 50 value of 73 nM.</p>
    Fórmula:C17H13ClN2O2
    Forma y color:Solid
    Peso molecular:312.75
  • Detajmium

    CAS:
    <p>Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.</p>
    Fórmula:C27H42N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:456.64
  • LK-732

    CAS:
    <p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>
    Fórmula:C25H29N5O3S
    Forma y color:Solid
    Peso molecular:479.59
  • THR-β agonist 4

    CAS:
    <p>THR-β agonist 4 is a potent agonist of THR-β.</p>
    Fórmula:C16H11Cl2F2N5O6S
    Forma y color:Solid
    Peso molecular:510.26
  • Cedarmycin B

    CAS:
    <p>Cedarmycin B exhibits activity against Candida, Cryptococcus neoformans, and Aspergillus fumigatus, with a minimum inhibitory concentration (MIC) ranging from 12.5 to 50 μg/mL.</p>
    Fórmula:C12H18O4
    Forma y color:Solid
    Peso molecular:226.269
  • (25S)-δ7-Dafachronic acid

    CAS:
    <p>(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.</p>
    Fórmula:C27H42O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:414.62
  • nNOS-IN-25

    CAS:
    <p>nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.</p>
    Fórmula:C21H22N4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:330.43
  • (6S)-CP-470711

    CAS:
    <p>(6S)-CP-470711 (Compound 8) acts as an inhibitor of sorbitol dehydrogenase (SDH) in both humans and rats, exhibiting inhibitory concentrations (IC50) of 19 nM and 27 nM, respectively. Additionally, (6S)-CP-470711 has been shown to ameliorate diabetes in rats induced by Streptozotocin.</p>
    Fórmula:C18H26N6O2
    Forma y color:Solid
    Peso molecular:358.44
  • AT-IAP

    CAS:
    AT-IAP is an effective dual antagonist of XIAP and cIAP1.
    Fórmula:C29H40FN5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:509.66
  • Ici D1542

    CAS:
    <p>Ici D1542: potent TXS inhibitor &amp; TXA2 receptor antagonist, effective thromboxane blocker in vitro.</p>
    Fórmula:C25H30N2O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:470.51
  • SSTR5 antagonist 2 TFA

    CAS:
    <p>Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.</p>
    Fórmula:C34H36F4N2O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:660.65
  • L 671776

    CAS:
    <p>L 671776 is an inositol monophosphatase inhibitor.</p>
    Fórmula:C23H32O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:388.5
  • SARS-CoV-2 nsp3-IN-1


    <p>Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.</p>
    Fórmula:C17H15N5O2
    Forma y color:Solid
    Peso molecular:321.33
  • Rafutrombopag

    CAS:
    <p>Rafutrombopag is a thrombopoietin (TPO) agonist.</p>
    Fórmula:C25H22N4O5
    Forma y color:Solid
    Peso molecular:458.47
  • SB 204070 hydrochloride

    CAS:
    <p>SB 204070 hydrochloride is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.</p>
    Fórmula:C19H27ClN2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:382.88
  • ONO-DI-004

    CAS:
    <p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>
    Fórmula:C24H38O6
    Forma y color:Solid
    Peso molecular:422.55
  • Ro-51

    CAS:
    <p>dual P2X3 and P2X2/3 antagonist</p>
    Fórmula:C17H23IN4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:474.29
  • Chloroquinocin

    CAS:
    <p>Chloroquinocin exhibits moderate activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA).</p>
    Fórmula:C17H15ClO5
    Forma y color:Solid
    Peso molecular:334.751
  • AM-3189

    CAS:
    <p>AM-3189: potent, selective GPR40 agonist with low CNS penetration, good pharmacokinetics, and efficacy mirroring AMG 837.</p>
    Fórmula:C27H25ClN2O3
    Forma y color:Solid
    Peso molecular:460.95
  • AGN-795

    CAS:
    <p>AGN-795 is a biochemical.</p>
    Fórmula:C14H20N2
    Forma y color:Solid
    Peso molecular:216.328
  • SARS-CoV-2 nsp14-IN-2


    <p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>
    Fórmula:C21H21N5O5S
    Forma y color:Solid
    Peso molecular:455.49
  • Cofpropamine

    CAS:
    <p>Cofpropamine, a caffeine derivative that inhibits polyadenylation, enhances the suppressive effects of Cyclophosphamide in animal models of rat adjuvant arthritis and mouse collagen-induced arthritis.</p>
    Fórmula:C13H21N5O3
    Forma y color:Solid
    Peso molecular:295.34
  • FW 34569

    CAS:
    <p>FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.</p>
    Fórmula:C30H43N5O7S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:617.76
  • 16(S)-Iloprost

    CAS:
    <p>Iloprost, a potent prostacyclin analog, binds to human IP &amp; EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>
    Fórmula:C22H32O4
    Forma y color:Solid
    Peso molecular:360.49
  • Aspochalasin M

    CAS:
    <p>Aspochalasin M shows moderate activity on HL-60 cells (IC50=20.0 μ M). Aspochalasin M has research potential in leukemia diseases.</p>
    Fórmula:C24H35NO4
    Forma y color:Solid
    Peso molecular:401.54
  • RORγt Inverse agonist 2

    CAS:
    <p>RORγt Inverse agonist 2 is a selective, orally active inverse agonist of RORγt(EC50 of 119 nM).</p>
    Fórmula:C27H25F8NO5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:627.54
  • IMR687

    CAS:
    <p>IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.</p>
    Fórmula:C21H26N6O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:394.47
  • IMP-321

    CAS:
    IMP-321 is a soluble dimeric recombinant form of LAG-3 and first-in-class antigen presenting cell activator.
    Fórmula:C56H78N18O14S
    Forma y color:Solid
    Peso molecular:1259.4
  • DGY-08-097

    CAS:
    <p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>
    Fórmula:C60H76N10O14
    Forma y color:Solid
    Peso molecular:1161.3
  • BILA 1906 BS

    CAS:
    BILA 1906 BS is an inhibitor of substrate analog protease.
    Fórmula:C41H52N6O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:724.95
  • NUCC-555

    CAS:
    <p>NUCC-555 is a first-in-class antagonist of activin. It opens a completely new approach to inhibiting the activity of TGF-beta receptor superfamily members.</p>
    Fórmula:C25H25N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:443.5
  • BSc5367

    CAS:
    <p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>
    Fórmula:C20H15N3O2
    Forma y color:Soild
    Peso molecular:329.35
  • Fonsartan free acid

    CAS:
    <p>Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.</p>
    Fórmula:C26H32N4O5S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:544.69
  • SARS-CoV-2-IN-22

    CAS:
    <p>SARS-CoV-2-IN-22 is a SARS-CoV-2 pseudovirus inhibitor (IC50: 16.96 μM).</p>
    Fórmula:C27H24N2O3S
    Forma y color:Solid
    Peso molecular:456.56
  • T-3861174

    CAS:
    <p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>
    Fórmula:C26H25FN6O2
    Forma y color:Solid
    Peso molecular:472.51
  • CEP-2563

    CAS:
    <p>CEP-2563 is a prodrug of CEP-751. It also used as an antitumor agent, inhibiting protein kinases.</p>
    Fórmula:C36H41ClN6O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:689.20
  • ZL-Pin13

    CAS:
    <p>ZL-Pin13: potent Pin1 inhibitor (IC50: 67 nM), halts MDA-MB-231 cell growth, reduces Pin1 substrates.</p>
    Fórmula:C24H23ClN2O3S
    Forma y color:Soild
    Peso molecular:454.97
  • TLR7/8 antagonist 2


    <p>TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.</p>
    Fórmula:C22H26FN5
    Forma y color:Solid
    Peso molecular:379.47
  • PZ-3022

    CAS:
    <p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>
    Fórmula:C20H21N5O
    Forma y color:Solid
    Peso molecular:347.41
  • Cbl-b-IN-1

    CAS:
    <p>Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 &lt;100 nM) with potential anticancer activity for the study of intestinal inflammation.</p>
    Fórmula:C29H34N6O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:498.631
  • L-739750

    CAS:
    <p>L-739,750 is an inhibitor (FTI) of peptidomimetic farnesyltransferase.</p>
    Fórmula:C23H39N3O6S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:517.7
  • Antitumor agent-47


    <p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>
    Fórmula:C30H27NO11
    Forma y color:Solid
    Peso molecular:577.54
  • MSK-195

    CAS:
    <p>MSK-195 is an effective TRPV1 agonist.</p>
    Fórmula:C28H40N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:484.63
  • Chitinase-IN-4


    <p>Chitinase-IN-4 (compound 8f) is a potent and selective inhibitor of OfChi-h with an IC50 value of 0.1 μM and good insecticidal activity.</p>
    Fórmula:C21H24ClN7
    Forma y color:Solid
    Peso molecular:409.92
  • L-Tyrosyl-L-glutamic acid

    CAS:
    <p>L-Tyrosyl-L-glutamic acid acts as an inhibitor of the amino acid permease GAP1.</p>
    Fórmula:C14H18N2O6
    Forma y color:Solid
    Peso molecular:310.3
  • Kaitocephalin

    CAS:
    <p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>
    Fórmula:C18H21Cl2N3O9
    Forma y color:Solid
    Peso molecular:494.28
  • 4-Chloropyridine

    CAS:
    <p>4-Chloropyridine acts as an inhibitor of Nicotinamide N-methyltransferase (NNMT). Serving as a substrate for NNMT, this compound enhances the electrophilicity at the C4 position through methylation of the pyridine nitrogen. This modification facilitates an aromatic nucleophilic substitution reaction with the non-catalytic cysteine (C159) in NNMT, ultimately leading to suicidal activity inhibition of the enzyme. 4-Chloropyridine is a promising candidate for the development of activity-based probes targeting NNMT functions.</p>
    Fórmula:C5H4ClN
    Forma y color:Solid
    Peso molecular:113.55
  • Pim-1 kinase inhibitor 3

    CAS:
    <p>Pim-1 kinase inhibitor 3 (Compound H5) is a potent inhibitor of Pim-1 kinase, demonstrating an inhibitory concentration (IC50) of 35.13 nM [1].</p>
    Fórmula:C20H25N3O2
    Forma y color:Solid
    Peso molecular:339.43
  • ASB14780


    <p>ASB14780 is a 4-phenoxy derivative and an inhibitor of cytoplasmic phospholipase cPLA2α (IC50: 20 nM).</p>
    Forma y color:Solid
  • Pyrisulfoxin B

    CAS:
    <p>Pyrisulfoxin B is an antibiotic produced by the bacterium Streptomyces (BS-75).</p>
    Fórmula:C13H11N3O2S
    Forma y color:Solid
    Peso molecular:273.31
  • BRD-9526

    CAS:
    <p>BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).</p>
    Fórmula:C26H31Cl2N3O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:584.51
  • L 767679

    CAS:
    <p>L 767679 is an antagonist of the fibrinogen receptors.</p>
    Fórmula:C20H24N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:384.43
  • Pateamine A

    CAS:
    <p>Pateamine A: marine-sourced macrolide from Mycale hentscheli; anticancer, antiviral, and translation inhibitor.</p>
    Fórmula:C31H45N3O4S
    Forma y color:Solid
    Peso molecular:555.77
  • SSR-182289A (Free)

    CAS:
    <p>SSR-182289A (Free) is a thrombin inhibitor.</p>
    Fórmula:C30H33F2N5O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:597.68
  • Dinordrin

    CAS:
    <p>Dinordrin is an implantation inhibitor and hormone.</p>
    Fórmula:C27H36O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:424.57
  • U 75875

    CAS:
    <p>U 75875 is a protease inhibitor.</p>
    Fórmula:C45H61N7O7
    Forma y color:Solid
    Peso molecular:812.01
  • L 365209

    CAS:
    <p>L 365209 is an oxytocin antagonist.</p>
    Fórmula:C40H50N8O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:738.88
  • MEIS-IN-1

    CAS:
    <p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>
    Fórmula:C24H21F3N2O4
    Forma y color:Solid
    Peso molecular:458.43
  • SX 3202

    CAS:
    <p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>
    Fórmula:C17H11BrFN3O4
    Forma y color:Solid
    Peso molecular:420.19
  • 14,15-dehydro Leukotriene B4

    CAS:
    <p>LTB4 is a leukocyte-activating fatty acid via 5-lipoxygenase. Two receptors, BLT1 and BLT2, bind it. 14,15-dehydro LTB4 is a stronger BLT1 antagonist.</p>
    Fórmula:C20H30O4
    Forma y color:Solid
    Peso molecular:334.45
  • Rpi 856 C

    CAS:
    <p>Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.</p>
    Fórmula:C39H56N6O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:768.90
  • Anticancer agent 79


    <p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>
    Fórmula:C20H12F3NO5
    Forma y color:Solid
    Peso molecular:403.31
  • Gypsetin

    CAS:
    <p>Gypsetin inhibits the activity of acyl-CoA:cholesterol acyltransferase (ACAT), showing inhibitory effects on rat liver microsomal ACAT with an IC50 of 18 μM, and competes with oleoyl-CoA substrate, possessing a Ki value of 5.5 μM. Additionally, Gypsetin prevents the formation of cholesterol esters from oleic acid with an IC50 of 0.65 μM.</p>
    Fórmula:C32H36N4O4
    Forma y color:Solid
    Peso molecular:540.653
  • AVE 0991

    CAS:
    <p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>
    Fórmula:C29H32N4O5S2
    Pureza:98.69%
    Forma y color:Solid
    Peso molecular:580.72
  • Leucomycin V

    CAS:
    <p>Leucomycin V is a macrolide antibiotic. Leucomycin A9 exhibits strong activity against Gram-positive bacteria and also affects spirochetes, rickettsiae, and chlamydiae.</p>
    Fórmula:C35H59NO13
    Forma y color:Solid
    Peso molecular:701.842
  • MDL-28050

    CAS:
    <p>MDL-28050 is a synthetic analog of hirudin 55-65 C-terminal fragment and a peptide inhibitor.</p>
    Fórmula:C61H88N10O23
    Forma y color:Solid
    Peso molecular:1329.4
  • SORT1-IN-3

    CAS:
    <p>SORT1-IN-3 (compound 5) is a SORT1 inhibitor characterized by its ability to permeate the blood-brain barrier.</p>
    Fórmula:C16H26ClNO3
    Forma y color:Solid
    Peso molecular:315.84
  • Dinalbuphine sebacate

    CAS:
    <p>Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.</p>
    Fórmula:C52H68N2O10
    Forma y color:Solid
    Peso molecular:881.1
  • Flusoxolol

    CAS:
    <p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>
    Fórmula:C22H30FNO4
    Forma y color:Solid
    Peso molecular:391.48
  • Iroxanadine hydrobromide

    CAS:
    <p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>
    Fórmula:C14H21BrN4O
    Forma y color:Solid
    Peso molecular:341.25
  • CE-2072

    CAS:
    <p>CE-2072 is a synthetic host serine proteases inhibitor.</p>
    Fórmula:C33H41N5O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:603.71
  • NRX-2663

    CAS:
    <p>NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).</p>
    Fórmula:C20H13F3N2O5
    Forma y color:Solid
    Peso molecular:418.32
  • DS69910557


    <p>DS69910557: potent hPTHR1 antagonist, IC50 0.08 μM, oral, for hyperparathyroidism &amp; osteoporosis research.</p>
    Fórmula:C32H33Cl2FN4O3
    Forma y color:Solid
    Peso molecular:611.53
  • P7170

    CAS:
    <p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>
    Fórmula:C21H16F3N9
    Forma y color:Solid
    Peso molecular:451.42
  • LPA5 antagonist 1


    <p>LPA5 antagonist 1: selective, potent (IC50=32 nM), high brain permeability, studies inflammatory/neuropathic pain.</p>
    Fórmula:C28H26N2O4S
    Forma y color:Solid
    Peso molecular:486.58
  • GSK340


    <p>GSK340 is a BET inhibitor.</p>
    Fórmula:C26H31N3O2
    Forma y color:Solid
    Peso molecular:417.55
  • KCa2 channel modulator 2


    Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.
    Fórmula:C16H15ClFN5
    Forma y color:Solid
    Peso molecular:331.78
  • PCSK9-IN-17

    CAS:
    <p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>
    Fórmula:C16H19N5OS
    Forma y color:Solid
    Peso molecular:329.42
  • Ro 31-8472

    CAS:
    <p>Ro 31-8472 is an angiotensin-converting enzyme (ACE) inhibitor and an analog of cilazaprilat.</p>
    Fórmula:C20H27N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:405.44
  • BMS-748730

    CAS:
    <p>BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.</p>
    Fórmula:C22H26ClN7O3S
    Forma y color:Solid
    Peso molecular:504.01
  • ChemR23-IN-3


    <p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>
    Fórmula:C31H33N5O5S2
    Forma y color:Solid
    Peso molecular:619.75
  • METTL3-IN-3

    CAS:
    METTL3-IN-3 is a polyheterocyclic compound, acts as METTL3 inhibitor .
    Fórmula:C26H28BrFN6O2
    Forma y color:Solid
    Peso molecular:555.44
  • A 70450

    CAS:
    <p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>
    Fórmula:C42H71ClN6O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:775.50
  • Alkannin

    CAS:
    <p>Alkannin: potent, tumor-specific PKM2 inhibitor; non-inhibitory to PKM1/PKL; potential anticancer agent.</p>
    Fórmula:C16H16O5
    Forma y color:Solid
    Peso molecular:288.3
  • Agosterol A

    CAS:
    <p>Agosterol A is isolated from marine sponge Spongia.</p>
    Fórmula:C33H52O8
    Forma y color:Solid
    Peso molecular:576.76
  • mPGES-1-IN-1


    <p>MPGES-1, potential anti-inflammatory drug target, has IC50 of 0.03 μM with mPGES-1-IN-1.</p>
    Fórmula:C21H14N4O2S
    Forma y color:Solid
    Peso molecular:386.43
  • Pulvomycin

    CAS:
    <p>Pulvomycin is a protein biosynthesis inhibitor preventing ternary complex formation between elongation factor Tu, GTP, and aminoacyl-tRNA.</p>
    Fórmula:C47H66O13
    Pureza:98%
    Forma y color:Solid
    Peso molecular:839.032
  • Mimocine

    CAS:
    <p>Mimosine, a plant amino acid, is known to act as a normoxic inducer of hypoxia-inducible factor (HIF).</p>
    Fórmula:C15H14N2O5
    Forma y color:Solid
    Peso molecular:302.28
  • LA-810

    CAS:
    <p>LA-810 is a nitrous oxide donor.</p>
    Fórmula:C15H25N5O7S
    Forma y color:Solid
    Peso molecular:419.45
  • MSX-3 free acid

    CAS:
    <p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>
    Fórmula:C21H23N4O7P
    Forma y color:Solid
    Peso molecular:474.40
  • ZD6021

    CAS:
    <p>ZD6021 is an antagonist of neurokinin 1 receptor.</p>
    Fórmula:C35H35Cl2N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:632.64
  • Anticancer agent 80


    <p>Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).</p>
    Fórmula:C19H12BrNO5
    Forma y color:Solid
    Peso molecular:414.21
  • PAD2-IN-1 hydrochloride


    <p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>
    Fórmula:C25H30ClFN6O3
    Forma y color:Solid
    Peso molecular:517
  • NB-533

    CAS:
    <p>NB-533 is a macrocyclic peptidic BACE-1 inhibitor.</p>
    Fórmula:C33H55N3O4
    Forma y color:Solid
    Peso molecular:557.81
  • HOE-288

    CAS:
    <p>HOE-288 is a converting enzyme (CE) inhibitor.</p>
    Fórmula:C27H38N2O5
    Forma y color:Solid
    Peso molecular:470.60
  • Org-31710

    CAS:
    <p>Org-31710 is a progesterone receptor antagonist potentially for contraception.</p>
    Fórmula:C30H39NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:445.64
  • SSM3 TFA

    CAS:
    <p>SSM3 TFA is a potent furin inhibitor, blocking furin-dependent cell surface processing of anthrax protective antigen-83 in vitro..</p>
    Fórmula:C22H32N12O2
    Forma y color:Solid
    Peso molecular:496.57
  • EP-7041 HCl

    CAS:
    <p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>
    Fórmula:C19H27ClN4O4
    Forma y color:Solid
    Peso molecular:410.89
  • Cortistatin A

    CAS:
    <p>Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.</p>
    Fórmula:C30H36N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:472.62
  • GSK3527497

    CAS:
    <p>GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).</p>
    Fórmula:C17H16ClFN4O4S
    Forma y color:Solid
    Peso molecular:426.85
  • VU6028418


    <p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>
    Forma y color:Liquid
  • Olanzapine/Samidorphan

    CAS:
    <p>Olanzapine/Samidorphan, a tablet blending olanzapine and samidorphan, targets schizophrenia and bipolar I, curbing weight gain.</p>
    Fórmula:C38H46N6O4S
    Forma y color:Solid
    Peso molecular:682.88
  • Miyakamide A2

    CAS:
    <p>Miyakamide A2 is an antibiotic with insecticidal properties. It inhibits the growth of brine shrimp and exhibits weak activity against Xanthomonas species. The IC50 for inhibiting P388 cells is 12.2 μg/mL.</p>
    Fórmula:C31H32N4O3
    Forma y color:Solid
    Peso molecular:508.611
  • Carazostatin

    CAS:
    <p>Carazostatin is an antioxidant, free radical scavenger, and potent lipid peroxidation inhibitor.</p>
    Fórmula:C20H25NO
    Pureza:98%
    Forma y color:Pale Yellow Solid
    Peso molecular:295.42
  • Antiangiogenic agent 3


    <p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>
    Fórmula:C19H20O7
    Forma y color:Solid
    Peso molecular:360.36
  • Revamilast sodium

    CAS:
    <p>Revamilast sodium, also known as GRC4039 sodium, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritis</p>
    Fórmula:C18H8Cl2F2N3NaO4
    Forma y color:Solid
    Peso molecular:462.17
  • Freselestat

    CAS:
    <p>Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.</p>
    Fórmula:C23H28N6O4
    Forma y color:Solid
    Peso molecular:452.51
  • GDC-6036-NH

    CAS:
    <p>GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.</p>
    Fórmula:C26H30ClF4N7O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:568.01
  • U 80215

    CAS:
    <p>U 80215 is an enzyme-competitive inhibitor.</p>
    Fórmula:C42H60N8O6S
    Forma y color:Solid
    Peso molecular:805.04
  • PKG1α activator 3


    <p>PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).</p>
    Fórmula:C27H26Cl2N2O6
    Forma y color:Solid
    Peso molecular:545.41
  • GNE-203

    CAS:
    <p>GNE-203 is a Met inhibitor.</p>
    Fórmula:C30H29Cl2F3N8O3
    Forma y color:Solid
    Peso molecular:677.50
  • Fusarochromanone

    CAS:
    <p>Fusarochromanone (FC-101) is a mycotoxin produced by Fusarium oxysporum with potent antiangiogenic, anticancer and antimalarial activities.</p>
    Fórmula:C15H20N2O4
    Pureza:95.31% - 96%
    Forma y color:Solid
    Peso molecular:292.33
  • DSP-6952

    CAS:
    <p>DSP-6952 is a 5-HT4 receptor partial agonist, inhibiting visceral hypersensitivity and ameliorating gastrointestinal dysfunction.</p>
    Fórmula:C21H32BrClN4O5
    Forma y color:Solid
    Peso molecular:535.86
  • ONO-8809

    CAS:
    <p>ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.</p>
    Fórmula:C30H46BrNO4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:596.66
  • Antiallergic agent-1


    <p>Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.</p>
    Fórmula:C27H19F6N5O
    Forma y color:Solid
    Peso molecular:543.46
  • Methyl Streptonigrin

    CAS:
    <p>Methyl Streptonigrin is an ABCG2 transporter function inhibitor.</p>
    Fórmula:C26H24N4O8
    Pureza:98%
    Forma y color:Solid
    Peso molecular:520.49
  • GR-71251

    CAS:
    <p>GR-71251 is a Tachykinin receptor antagonist.</p>
    Fórmula:C74H105N19O13
    Forma y color:Solid
    Peso molecular:1468.74
  • MtDTBS-IN-1


    <p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>
    Fórmula:C16H16N4O5
    Forma y color:Solid
    Peso molecular:344.32
  • SphK2-IN-2


    <p>SphK2-IN-2 (21g) is a potent and selective inhibitor of SphK2 (IC50: 0.23 μM).</p>
    Fórmula:C21H25ClN10O
    Forma y color:Solid
    Peso molecular:468.94
  • PARP1-IN-5


    <p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>
    Fórmula:C25H24N2O5S
    Forma y color:Solid
    Peso molecular:464.53
  • Anti-TSWV agent 1


    <p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>
    Fórmula:C22H27ClN4OS3
    Forma y color:Solid
    Peso molecular:495.12
  • GSK579289A

    CAS:
    <p>GSK579289A is an inhibitor of benzimidazole thiophene.</p>
    Fórmula:C26H27ClN4O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:511.04
  • Ekatetrone

    CAS:
    <p>Ekatetrone displays activity against both Gram-positive and Gram-negative bacteria, with particularly strong inhibitory effects on Mycobacterium tuberculosis.</p>
    Fórmula:C19H13NO7
    Forma y color:Solid
    Peso molecular:367.309
  • Gilvusmycin

    CAS:
    <p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>
    Fórmula:C38H34N6O8
    Forma y color:Solid
    Peso molecular:702.712
  • Anti-inflammatory agent 16


    <p>Compound 14 is a peptidomimetic that significantly lowers TNFα, NO, CD40, and CD86, showcasing strong anti-inflammatory effects.</p>
    Fórmula:C21H23N5O3
    Forma y color:Solid
    Peso molecular:393.44
  • Retelliptine

    CAS:
    Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.
    Fórmula:C25H32N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:404.55
  • LASSBio-1632


    <p>LASSBio-1632: Novel anti-asthmatic, blocks PDE4A/D, reduces AHR &amp; lung TNF-α, crosses BBB.</p>
    Fórmula:C18H20N2O6S
    Forma y color:Solid
    Peso molecular:392.43
  • L 739749

    CAS:
    <p>L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.</p>
    Fórmula:C24H41N3O6S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:531.73
  • Naltalimide

    CAS:
    <p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>
    Fórmula:C28H28N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:472.53
  • Pamiparib maleate

    CAS:
    <p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>
    Fórmula:C44H42F2N8O14
    Pureza:98%
    Forma y color:Solid
    Peso molecular:944.859
  • Piperazinomycin

    CAS:
    <p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>
    Fórmula:C18H20N2O2
    Forma y color:Solid
    Peso molecular:296.36
  • Basroparib

    CAS:
    <p>Basroparib is an inhibitor of ribose polymerase (PARP) and has shown antitumour effects.</p>
    Fórmula:C18H21F2N7O3
    Forma y color:Solid
    Peso molecular:421.4
  • KF 20274

    CAS:
    <p>KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.</p>
    Fórmula:C21H29N5O
    Forma y color:Solid
    Peso molecular:367.49
  • PARP10/15-IN-1


    <p>PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].</p>
    Fórmula:C13H10N2O3S
    Forma y color:Solid
    Peso molecular:274.3
  • Ambelline

    CAS:
    <p>Ambelline has antitumor activity.</p>
    Fórmula:C18H21NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:331.36
  • PKCiota-IN-1

    CAS:
    <p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>
    Fórmula:C25H22FN5O
    Forma y color:Solid
    Peso molecular:427.47
  • CYP2C1/CYP2C19-IN-2


    <p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Fórmula:C27H28N2O6S
    Forma y color:Solid
    Peso molecular:508.59
  • GSK945237

    CAS:
    <p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>
    Fórmula:C24H26FN5O3
    Forma y color:Solid
    Peso molecular:451.49
  • Tuvatidine

    CAS:
    <p>Tuvatidine is a histamine 2 receptor antagonist.</p>
    Fórmula:C10H17N9O2S3
    Forma y color:Solid
    Peso molecular:391.5
  • Keap1-Nrf2-IN-1 TFA


    <p>Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.</p>
    Fórmula:C26H25F3N2O9S
    Forma y color:Solid
    Peso molecular:598.54
  • (±)-ANAP hydrochloride (1185251-08-4 free base)


    <p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>
    Fórmula:C15H17ClN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:308.76
  • 7-Hydroxyguanine

    CAS:
    <p>7-Hydroxyguanine is an antibiotic that inhibits the growth of L1210 leukemia cells.</p>
    Fórmula:C5H5N5O2
    Forma y color:Solid
    Peso molecular:167.126
  • Leustroducsin B

    CAS:
    <p>Leustroducsin B is a novel colony-stimulating factor (CSF) inducer extracted from Streptomyces platensis SANK 60191.</p>
    Fórmula:C34H56NO10P
    Forma y color:Solid
    Peso molecular:669.78