Otros inhibidores
Esta categoría abarca una amplia variedad de inhibidores que no encajan en las clasificaciones estándar, pero que son fundamentales para diversas investigaciones bioquímicas y farmacológicas. Estos inhibidores pueden dirigirse a vías, enzimas e interacciones moleculares únicas o menos estudiadas, proporcionando herramientas valiosas para áreas de investigación especializadas. En CymitQuimica, ofrecemos una selección diversa de inhibidores de alta calidad que abarcan múltiples objetivos biológicos y disciplinas de investigación, lo que le permite explorar nuevas vías terapéuticas y profundizar su comprensión de los procesos biológicos complejos.
Se han encontrado 37926 productos de "Otros inhibidores"
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eIF4A3-IN-4
<p>eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).</p>Fórmula:C24H20N2O5Forma y color:SolidPeso molecular:416.43Citrinin hydrate
CAS:<p>Citrinin hydrate is an inhibitor of human rhinovirus (HRV) 3C protease, with an IC50 of 1.0 mM.</p>Fórmula:C13H16O6Forma y color:SolidPeso molecular:268.263Pluracidomycin C1
CAS:<p>Pluracidomycin C1 is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria and also possesses β-lactamase inhibitory properties.</p>Fórmula:C10H13NO10S2Forma y color:SolidPeso molecular:371.341Epithienamycin F
CAS:<p>Epithienamycin F is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C13H18N2O8S2Forma y color:SolidPeso molecular:394.421Melanocin A
CAS:<p>Melanocin A is an inhibitor of melanin biosynthesis. It suppresses the synthesis of melanin and tyrosinase with an IC50 of 9.0 nM and MIC of 0.9 μM. Additionally, Melanocin A exhibits antioxidant properties.</p>Fórmula:C18H14N2O5Forma y color:SolidPeso molecular:338.31Melithiazole B
CAS:<p>Melithiazol B is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA), with both antifungal and cytotoxic properties.</p>Fórmula:C20H24N2O4S2Forma y color:SolidPeso molecular:420.546C20 Sphingomyelin (d18:1/20:1)
CAS:<p>C20 Sphingomyelin (d18:1/20:1) (Compound SM:20:1) is a type of sphingolipid. This compound shows potential for research related to motor neuron diseases, such as amyotrophic lateral sclerosis (ALS) and primary lateral sclerosis (PLS).</p>Fórmula:C43H85N2O6PForma y color:SolidPeso molecular:757.119Nanaomycin D
CAS:<p>Nanaomycin D is an antibiotic with antibacterial properties.</p>Fórmula:C16H12O6Forma y color:SolidPeso molecular:300.263FW 34569
CAS:<p>FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.</p>Fórmula:C30H43N5O7SPureza:98%Forma y color:SolidPeso molecular:617.76ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Fórmula:C23H26Cl2N2O3Forma y color:SolidPeso molecular:449.37Hydroxynybomycin
CAS:<p>Hydroxynybomycin is an antibiotic with activity against Gram-negative bacteria.</p>Fórmula:C16H14N2O5Forma y color:SolidPeso molecular:314.293Lactaroviolin
CAS:<p>Lactaroviolin is an aromatic derivative antibiotic that can inhibit the growth of Mycobacterium tuberculosis.</p>Fórmula:C15H14OForma y color:SolidPeso molecular:210.271Exatecan-amide-cyclopropanol
CAS:<p>Exatecan-amide-cyclopropanol potently inhibits SK-BR-3 and U87 cancer cells (IC50 0.12 and 0.23 nM)</p>Fórmula:C28H26FN3O6Pureza:98.308%Forma y color:SolidPeso molecular:519.52U 75875
CAS:<p>U 75875 is a protease inhibitor.</p>Fórmula:C45H61N7O7Forma y color:SolidPeso molecular:812.01Sdz 210-096
CAS:<p>Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.</p>Fórmula:C27H31NO2Forma y color:SolidPeso molecular:401.54Fujianmycin A
CAS:<p>Fujianmycin A exhibits activity against Bacillus subtilis (hay bacillus).</p>Fórmula:C19H14O5Forma y color:SolidPeso molecular:322.311Diospyrin
CAS:<p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>Fórmula:C22H14O6Forma y color:SolidPeso molecular:374.34Thiomuscimol hydrobromide
CAS:<p>Thiomuscimol hydrobromide is an agonist of GABAA receptor.</p>Fórmula:C4H6N2OSPureza:98%Forma y color:SolidPeso molecular:130.17Diazaquinomycin A
CAS:<p>Diazaquinomycin A (DAQA) is a diazaquinomycin antibiotic that acts as an inhibitor of thymidylate synthase. DAQA induces DNA damage, cell cycle arrest, and apoptosis through cleavage of PARP.</p>Fórmula:C20H22N2O4Forma y color:SolidPeso molecular:354.4Butaprost
CAS:<p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>Fórmula:C24H40O5Pureza:98%Forma y color:SolidPeso molecular:408.57NA 382
CAS:<p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>Fórmula:C31H28N4O6Forma y color:SolidPeso molecular:552.58(R)-FL118
CAS:<p>FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.</p>Fórmula:C21H16N2O6Forma y color:SolidPeso molecular:392.36TLN-232
CAS:<p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>Fórmula:C36H49N9O7S2Forma y color:SolidPeso molecular:783.96Halomicin B
CAS:<p>Halomicin B is an ansamycin-type antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C43H58N2O12Forma y color:SolidPeso molecular:794.927Polyoxin E
CAS:<p>Polyoxin E is a nucleoside antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight.</p>Fórmula:C17H23N5O13Forma y color:SolidPeso molecular:505.39L2H2-6OTD
CAS:<p>L2H2-6OTD is a telomerase inhibitor with G-quadruplex loops; IC50: 15 nM.</p>Fórmula:C30H30N10O8Forma y color:SolidPeso molecular:658.62MCTR2
CAS:<p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>Fórmula:C27H40N2O6SForma y color:SolidPeso molecular:520.68Epoxyquinomicin A
CAS:<p>Epoxyquinomicin A is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus with MIC values of 3-12.5 µg/mL. Additionally, it shows cytotoxicity in cancer cells L1210, B16, and S180, with an IC50 of 2-8 µg/mL. Furthermore, Epoxyquinomicin A demonstrates anti-inflammatory effects in collagen-induced arthritis.</p>Fórmula:C14H10ClNO6Forma y color:SolidPeso molecular:323.685Mutalomycin
CAS:<p>Mutalomycin is a polyether antibiotic with activity against Gram-positive bacteria, mycoplasma, and coccidia.</p>Fórmula:C41H70O12Forma y color:SolidPeso molecular:754.987Kigamicin A
CAS:<p>Kigamicin A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>Fórmula:C34H35NO13Forma y color:SolidPeso molecular:665.64Nebramycin Ⅳ
CAS:<p>Nebramycin IV is an aminoglycoside antibiotic with a broad antimicrobial spectrum, demonstrating significant efficacy against Gram-positive bacteria, Gram-negative bacteria, and mycobacteria.</p>Fórmula:C19H38N6O11Forma y color:SolidPeso molecular:526.539SCP1-IN-1
CAS:<p>SCP1-IN-1 (SH T-62) is a potent inhibitor of SCP1, promoting REST degradation and potentially aiding glioblastoma research.</p>Fórmula:C20H19F3N2O7S2Pureza:99.53%Forma y color:SoildPeso molecular:520.5CEP-7055
CAS:<p>CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.</p>Fórmula:C32H35N3O4Forma y color:SolidPeso molecular:525.64RSV-IN-5
CAS:<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Fórmula:C28H37N7O2Forma y color:SolidPeso molecular:503.64ErSO-DFP
<p>ErSO-DFP activates a-UPR, targets ERα+ cancer cells with high selectivity, and effectively reduces MCF-7 tumours.</p>Fórmula:C20H17F5N2O2Forma y color:SolidPeso molecular:412.35PTP1B-IN-16
<p>PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.</p>Fórmula:C26H18ClN3O4SForma y color:SolidPeso molecular:503.96Glucosylquestiomycin
CAS:<p>Glucosylquestiomycin exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and yeast.</p>Fórmula:C18H18N2O7Forma y color:SolidPeso molecular:374.345DC41SMe
CAS:<p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>Fórmula:C38H36ClN5O4S2Pureza:98%Forma y color:SolidPeso molecular:726.31Pradimicin T2
CAS:<p>Pradimicin T2 is an antibiotic with activity against filamentous fungi and yeast-like fungi.</p>Fórmula:C37H37NO19Forma y color:SolidPeso molecular:799.6852-Hydroxygentamicin B1
CAS:<p>2-Hydroxygentamicin B1 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H40N4O11Forma y color:SolidPeso molecular:512.552BXL0124
CAS:<p>BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.</p>Fórmula:C32H44F6O4Forma y color:SolidPeso molecular:606.68Ophiobolin D
CAS:<p>Ophiobolin D is a terpene antibiotic with mild inhibitory effects on Staphylococcus aureus.</p>Fórmula:C25H36O4Forma y color:SolidPeso molecular:400.55Sinulatumolin E
CAS:<p>Sinulatumolin E, a terpenoid, inhibits TNF-α (IC 50: 3.6 μM); has anti-inflammatory properties.</p>Fórmula:C15H22O2Forma y color:SolidPeso molecular:234.33Antitumor agent-51
<p>Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.</p>Fórmula:C23H25N5O2SForma y color:SolidPeso molecular:435.54Napyradiomycin C2
CAS:<p>Napyradiomycin C2 is an antibiotic with activity against Gram-positive bacteria and mycobacteria.</p>Fórmula:C25H27Cl3O5Forma y color:SolidPeso molecular:513.838Tandutinib (MLN518) HCl
<p>Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.</p>Fórmula:C31H43ClN6O4Pureza:98%Forma y color:SolidPeso molecular:599.16Fudecalone
CAS:<p>Fudecalone is produced by the Penicillium strain FO-2030. It completely inhibits the coccidian parasite Eimeria Tenella that is resistant to Monensin.</p>Fórmula:C15H22O3Forma y color:SolidPeso molecular:250.33Octahydrocyclopenta[c]pyrrole
CAS:<p>Octahydrocyclopenta[c]pyrrole has demonstrated promising applications in the fields of anti-inflammatory, anti-tumor, and neuroprotection. The unique structure-activity relationship of Octahydrocyclopenta[c]pyrrole offers fresh insights for the design of new drugs.</p>Fórmula:C7H13NForma y color:SolidPeso molecular:111.18Pim-1 kinase inhibitor 3
CAS:<p>Pim-1 kinase inhibitor 3 (Compound H5) is a potent inhibitor of Pim-1 kinase, demonstrating an inhibitory concentration (IC50) of 35.13 nM [1].</p>Fórmula:C20H25N3O2Forma y color:SolidPeso molecular:339.433'-O-Decarbamoylirumamycin
CAS:<p>3'-O-Decarbamoylirumamycin is a 20-membered macrolide antibiotic produced by Streptomyces subflavus subsp. irumaensis. It exhibits inhibitory effects against plant pathogenic fungi, such as Pyricularia oryzae and Sclerotinia.</p>Fórmula:C40H64O11Forma y color:SolidPeso molecular:720.93Ezomycin B2
CAS:<p>Ezomycin B2 is an antibiotic with antifungal activity.</p>Fórmula:C19H25N5O13Forma y color:SolidPeso molecular:531.4271,6-Dihydroxy-2-chlorophenazine
CAS:<p>1,6-Dihydroxy-2-chlorophenazine exhibits weak antifungal and anti-yeast activity.</p>Fórmula:C12H7ClN2O2Forma y color:SolidPeso molecular:246.65Scytalol A
CAS:<p>Scytalol A selectively inhibits the biosynthesis of dihydroxynaphthalene melanin in Lachnellula sp. A32-89, while not affecting the growth of the strain.</p>Fórmula:C15H18O6Forma y color:SolidPeso molecular:294.35(S),6(S)-DiHETE
CAS:<p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>Fórmula:C20H32O4Forma y color:SolidPeso molecular:336.47AY-22,252
CAS:<p>AY-22,252 is an inhibitor of beef heart & rat brain nucleoside-3',5'- monophosphate phosphodiesterase.</p>Fórmula:C27H37NaO7Forma y color:SolidPeso molecular:496.574-Nitrochalcone
CAS:<p>4-Nitrochalcone (2-(4-Nitrobenzylidene)acetophenone) inhibits proteasomes and suppresses TNFα-induced NF-κB activity.</p>Fórmula:C15H11NO3Forma y color:SolidPeso molecular:253.25Dermostatin B
CAS:<p>Dermostatin B is a polyene antibiotic with antifungal properties, suitable for research on fungal infections.</p>Fórmula:C41H66O11Forma y color:SolidPeso molecular:734.956Evategrel
CAS:<p>Evategrel is an inhibitor of platelet aggregation.</p>Fórmula:C21H26ClNO7SForma y color:SolidPeso molecular:471.95Deoxyfrenolicin
CAS:<p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>Fórmula:C18H18O6Forma y color:SolidPeso molecular:330.332Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Fórmula:C21H36O7Forma y color:SolidPeso molecular:400.506Isobetanin
CAS:<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Fórmula:C24H26N2O13Forma y color:SolidPeso molecular:550.47Lactoquinomycin B
CAS:<p>Lactoquinomycin B is a quinone antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy against Gram-negative species is weaker and it does not affect fungi. It inhibits various cell lines, including lymphoma L5178Y parental cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, and murine leukemia L-1210 and P388 cells, with ID50 (μg/mL) values of 0.43, 0.21, 0.19, 0.16, 0.2, and 0.12, respectively.</p>Fórmula:C24H27NO9Forma y color:SolidPeso molecular:473.473Ornoprostil
CAS:<p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>Fórmula:C23H38O6Pureza:98%Forma y color:SolidPeso molecular:410.54Halomicin D
CAS:<p>Halomicin D is an ansamycin-class antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C43H56N2O12Forma y color:SolidPeso molecular:792.911Detoxin D1
CAS:<p>Detoxin D1 is a selective blasticidin S antagonist.</p>Fórmula:C28H41N3O8Pureza:98%Forma y color:SolidPeso molecular:547.64Formadicin A
CAS:<p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>Fórmula:C30H34N4O16Forma y color:SolidPeso molecular:706.608rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Fórmula:C25H24Cl2FN3O3Forma y color:SolidPeso molecular:504.38Narbomycin
CAS:<p>Narbomycin exhibits activity against Gram-positive bacteria.</p>Fórmula:C28H47NO7Forma y color:SolidPeso molecular:509.675DG013A
CAS:<p>DG013A inhibits ERAP1 & ERAP2 (IC50: 33 nM & 11 nM) to research autoimmune diseases & cancer.</p>Fórmula:C27H37N4O4PForma y color:SolidPeso molecular:512.58Porothramycin A
CAS:<p>Porothramycin A is an antibiotic effective against Gram-positive bacteria and anaerobic bacteria.</p>Fórmula:C18H21N3O4Forma y color:SolidPeso molecular:343.377Haliangicin B
CAS:<p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>Fórmula:C22H32O5Forma y color:SolidPeso molecular:376.49DLCI-1
CAS:<p>DLCI-1 is a potent and selective oral inhibitor of cytochrome P450 2A6 (CYP2A6), significantly reducing self-administered nicotine doses in both male and female mice.</p>Fórmula:C12H14N2SForma y color:SolidPeso molecular:218.32Cervicarcin
CAS:<p>Cervicarcin is an antitumor antibiotic (antibiotic) exhibiting strong inhibitory effects on sarcoma 180 and sarcoma NF, while showing weaker activity against sarcoma 37, Ehrlich ascites carcinoma, and Freund leukemia.</p>Fórmula:C19H20O9Forma y color:SolidPeso molecular:392.35718:0-LPS
CAS:<p>18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.</p>Fórmula:C24H48NO9PForma y color:SolidPeso molecular:525.613Feudomycin B
CAS:<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Fórmula:C28H31NO10Forma y color:SolidPeso molecular:541.546Bacithrocin D
CAS:<p>Bacithrocin D (Thiolstatin D) inhibits various proteases and has the capability to prolong clotting time. It exhibits IC50 values of 124, 9, 0.85, and 0.01 μM against thrombin, factor Xa, trypsin, and papain, respectively.</p>Fórmula:C17H25N5O3Forma y color:SolidPeso molecular:347.4127(Z),11(Z)-Nonacosadiene
CAS:<p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>Fórmula:C29H56Forma y color:SolidPeso molecular:404.75Cetoniacytone B
CAS:<p>Cetoniacytone B inhibits the growth of HEPG2 and MCF7 human tumor cell lines, with a GI50 of 4.4 μM.</p>Fórmula:C7H9NO4Forma y color:SolidPeso molecular:171.151Furaprevir
CAS:<p>Furaprevir is an HCV NS3/4A Inhibitor</p>Fórmula:C47H56N6O10SForma y color:SolidPeso molecular:897.05CGC 11144
CAS:<p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>Fórmula:C40H100Cl10N10Forma y color:SolidPeso molecular:1075.82Lasonolide A
CAS:<p>Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.</p>Fórmula:C41H60O9Forma y color:SolidPeso molecular:696.91IACS-8779 disodium
CAS:<p>IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.</p>Fórmula:C21H23N9Na2O10P2S2Forma y color:SolidPeso molecular:733.52P-gp inhibitor 2
CAS:<p>Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.</p>Fórmula:C29H26N2O6Forma y color:SolidPeso molecular:498.53Vindeburnol
CAS:<p>Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.</p>Fórmula:C17H20N2OForma y color:SolidPeso molecular:268.35Tetrahydrouridine dihydrate
<p>THU dihydrate, a potent CDA inhibitor, outperforms cytidine by blocking the enzyme's active site.</p>Fórmula:C9H20N2O8Forma y color:SolidPeso molecular:284.26Metocurine chloride
CAS:<p>Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.</p>Fórmula:C40H48Cl2N2O6Forma y color:SolidPeso molecular:723.72Dienomycin B
CAS:<p>Dienomycin B exhibits mild antibacterial activity.</p>Fórmula:C18H23NO2Forma y color:SolidPeso molecular:285.38Fusarin C
CAS:<p>Fusarin C is a mutagenic compound found in strains of the Fusarium genus.</p>Fórmula:C23H29NO7Forma y color:SolidPeso molecular:431.479Exfoliamycin
CAS:<p>Exfoliamycin is a naphthoquinone antibiotic found in the Streptomyces strain Exfoliamycin Tu 1424, and it exhibits activity against Gram-positive bacteria.</p>Fórmula:C22H26O9Forma y color:SolidPeso molecular:434.436Oximidine Ⅲ
CAS:<p>Oximidine III is an antitumor antibiotic that selectively inhibits the growth of rat fibroblast 3Y1 cells and induces mutations in various tumor genes. The inhibitory effects of Oximidine III on vH-ras-3Y1, v-src-3Y1 cells, and normal 3Y1 cells have IC50 values of 14 nM, 4.5 nM, and 140 nM, respectively. Additionally, Oximidine III arrests cells with RAS or SRC mutations in the G1 phase of the cell cycle and increases the expression of p21WAF1.</p>Fórmula:C23H24N2O6Forma y color:SolidPeso molecular:424.459-cis-13,14-Dihydroretinoic acid
CAS:<p>9-cis-13,14-Dihydroretinoic acid (9CDHRA) is a selective retinoid X receptor (RXR) agonist with a Kd of 90 nM. It can ameliorate memory deficits caused by impaired RXR signaling in vivo. This compound shows potential for research in the fields of neuroscience and metabolic diseases.</p>Fórmula:C20H30O2Forma y color:SolidPeso molecular:302.451Glidobactin G
CAS:<p>Glidobactin G is an antitumor antibiotic with activity against pathogenic fungi and yeasts. Additionally, Glidobactin G prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Fórmula:C27H44N4O7Forma y color:SolidPeso molecular:536.6613-O-Demethylmonensin A
CAS:<p>3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).</p>Fórmula:C35H60O11Forma y color:SolidPeso molecular:656.84Eulicin
CAS:<p>Eulicin is an antifungal agent that inhibits human immunodeficiency virus (HIV) infection and replication. It demonstrates broad-spectrum activity against both Gram-positive and Gram-negative bacteria and can be found in Streptomyces.</p>Fórmula:C24H52N8O2Forma y color:SolidPeso molecular:484.722Curromycin A
CAS:<p>Curromycin A exhibits antibacterial activity against Gram-positive bacteria such as Bacillus subtilis. Additionally, it can inhibit the replication of the human immunodeficiency virus (HIV) and suppresses the growth of mouse melanoma B16 and leukemia P388 cells.</p>Fórmula:C38H55N3O10Forma y color:SolidPeso molecular:713.857Fluvirucin A1
CAS:<p>Fluvirucin A1 is a novel antibiotic effective against the Influenza A virus.</p>Fórmula:C23H44N2O5Forma y color:SolidPeso molecular:428.61Cytochalasin M
CAS:<p>Cytochalasin M exhibits various biological activities, including reversible inhibition of cytoplasmic division and the suppression of both endocytosis and exocytosis in macrophages.</p>Fórmula:C30H37NO6Forma y color:SolidPeso molecular:507.618Micacocidin B
CAS:<p>Micacocidin B is an antibiotic that exhibits exceptional activity against Mycoplasma species.</p>Fórmula:C27H37CuN3O4S3Forma y color:SolidPeso molecular:627.343-O-Demethylmonensin B
CAS:<p>3-O-Demethylmonensin B is a polyether antibiotic produced by the bacterium *Streptomyces cinnamoneus* LO-63.</p>Fórmula:C34H58O11Forma y color:SolidPeso molecular:642.82Kinamycin A
CAS:<p>Kinamycin A possesses antibacterial and antimycobacterial properties, yet it exhibits reduced efficacy against Gram-negative bacteria.</p>Fórmula:C24H20N2O10Forma y color:SolidPeso molecular:496.423Clavamycin C
CAS:<p>Clavamycin C exhibits significant antifungal activity against Candida species, which can be antagonized by dipeptides or tripeptides, though not by amino acids. It lacks antibacterial properties and does not inhibit β-lactamase activity.</p>Fórmula:C13H22N4O8Forma y color:SolidPeso molecular:362.336Polyoxin F
CAS:<p>Polyoxin F is a nucleoside-type antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight disease.</p>Fórmula:C23H30N6O15Forma y color:SolidPeso molecular:630.52Human carbonic anhydrase II-IN-1
<p>Compound S-13: Potent hCA II inhibitor, Kis 4.4, 9.2, 480.2, 14.7 nM for hCA II, I, IV, IX. Used in glaucoma research.</p>Fórmula:C20H25N3O4SForma y color:SolidPeso molecular:403.5Rhodomycin B
CAS:<p>Rhodomycin B exhibits activity against Gram-positive bacteria, while its effects on Gram-negative bacteria and fungi are relatively weak.</p>Fórmula:C28H33NO10Forma y color:SolidPeso molecular:543.562Phoslactomycin A
CAS:<p>Phoslactomycin A exhibits weaker activity against Gram-positive bacteria, yet it shows stronger efficacy against fungi.</p>Fórmula:C29H46NO10PForma y color:SolidPeso molecular:599.65Endophenazine C
CAS:<p>Endophenazine C is a type of phenazine antibiotic.</p>Fórmula:C19H20N2O2Forma y color:SolidPeso molecular:308.37Baumycin C1
CAS:<p>Baumycin C1 is an antitumor antibiotic (antibiotic).</p>Fórmula:C28H29NO11Forma y color:SolidPeso molecular:555.53Nocardicin B
CAS:<p>Nocardicin B was originally isolated from Nocardia uniformis subsp. tsugamanensis [ATCC 21806], showing weak antibacterial activity against Proteus and Corynebacterium species.</p>Fórmula:C23H24N4O9Forma y color:SolidPeso molecular:500.46Emimycin
CAS:<p>Emimycin exhibits activity against Gram-positive and Gram-negative bacteria, as well as fungi like Saccharomyces cerevisiae (brewer's yeast).</p>Fórmula:C4H4N2O2Forma y color:SolidPeso molecular:112.087Melithiazole C
CAS:<p>Melithiazol C is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA) with antifungal properties.</p>Fórmula:C16H21NO5SForma y color:SolidPeso molecular:339.407Saframycin B
CAS:<p>Saframycin B exhibits activity against Gram-positive bacteria and has weaker efficacy against mycobacteria.</p>Fórmula:C28H31N3O8Forma y color:SolidPeso molecular:537.5616"'-Deamino-6"'-hydroxyneomycin B
CAS:<p>6"'-Deamino-6"'-hydroxyneomycin B is an aminoglycoside antibiotic produced by [Streptomyces fradiaeUC 75]. It is effective against both Gram-positive and Gram-negative bacteria and serves as an intermediate in the biosynthesis of neomycin.</p>Fórmula:C23H45N5O14Forma y color:SolidPeso molecular:615.628Epoxyquinomicin C
CAS:<p>Epoxyquinomicin C is an antibiotic that can be isolated from Amycolatopsis sp. It exhibits anti-inflammatory properties against collagen-induced arthritis and is also utilized in the synthesis of the NF-κB inhibitor DHMEQ.</p>Fórmula:C14H13NO6Forma y color:SolidPeso molecular:291.256Nemotinic acid
CAS:<p>Nemotinic acid exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while also displaying weaker activity against Gram-negative bacteria.</p>Fórmula:C11H10O3Forma y color:SolidPeso molecular:190.195trans-Doxercalciferol
CAS:<p>trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.</p>Fórmula:C28H44O2Pureza:98%Forma y color:SolidPeso molecular:412.65Steroid sulfatase/17β-HSD1-IN-4
<p>Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).</p>Fórmula:C18H17N3O4S2Forma y color:SolidPeso molecular:403.48Novokinin
CAS:<p>Angiotensin AT2 receptor agonist</p>Fórmula:C39H61N11O7Pureza:98%Forma y color:SolidPeso molecular:795.97SAR107375
CAS:<p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>Fórmula:C24H30ClN5O5S2Forma y color:SolidPeso molecular:568.11Ici D1542
CAS:<p>Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.</p>Fórmula:C25H30N2O7Pureza:98%Forma y color:SolidPeso molecular:470.515,6-Dihydro-4-methoxy-2H-pyran-2-one
CAS:<p>5,6-Dihydro-4-methoxy-2H-pyran-2-one is produced by the Penicillium italicum strain MRC 1360.</p>Fórmula:C6H8O3Peso molecular:128.13Inactone
CAS:<p>Inactone is a biologically active molecule with a 3-pentanoylimino group that inhibits the large ribosomal subunit.</p>Fórmula:C15H21NO4Forma y color:SolidPeso molecular:279.332Cuevaene B
CAS:<p>Cuevaene B can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. This compound exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and shows moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>Fórmula:C21H24O7Forma y color:SolidPeso molecular:388.411Cirramycin B1
CAS:<p>Cirramycin B1 exhibits activity against both Gram-positive bacteria, Gram-negative bacteria, and mycoplasmas.</p>Fórmula:C37H59NO12Forma y color:SolidPeso molecular:709.864Korormicin
CAS:<p>Korormicin is effective against marine Gram-negative bacteria but does not work against marine Gram-positive bacteria or common bacteria.</p>Fórmula:C25H39NO5Forma y color:SolidPeso molecular:433.581Galactostatin
CAS:<p>Galactostatin is an inhibitor of β-galactosidase.</p>Fórmula:C6H13NO5Forma y color:SolidPeso molecular:179.171Phenazostatin A
CAS:<p>Phenazostatin A is a phenazine compound known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. Phenazostatin A inhibits glutamate toxicity in N18-RE-105 cells with an EC50 of 0.34 μg/mL.</p>Fórmula:C28H20N4O3Forma y color:SolidPeso molecular:460.48Menoxymycin B
CAS:<p>Menoxymycin B is an antibiotic with cytotoxic properties, inhibiting KB and N18-RE-105 cells with IC50 values of 0.22 μM and 0.023 μM, respectively.</p>Fórmula:C25H31NO9Forma y color:SolidPeso molecular:489.5152-Hydroxygentamicin C2
CAS:<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H41N5O8Forma y color:SolidPeso molecular:479.568Epihygromycin
CAS:<p>Epihygromycin is a glycoside antibiotic with relatively weak activity against Gram-positive bacteria.</p>Fórmula:C23H29NO12Forma y color:SolidPeso molecular:511.476Glucopiericidin B
CAS:<p>Glucopiericidin B exhibits antibacterial activity.</p>Fórmula:C31H47NO9Forma y color:SolidPeso molecular:577.706MRS4738
<p>MRS4738 is a potent antagonist with high affinity for the P2Y14R receptor. It demonstrates in vivo anti-hyperallodynic and antiasthmatic activity [1].</p>Fórmula:C30H24F3NO2Forma y color:SolidPeso molecular:487.51Lobaric acid
CAS:<p>Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.</p>Fórmula:C25H28O8Forma y color:SolidPeso molecular:456.48Plumbemycin A
CAS:<p>Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Fórmula:C12H20N3O9PForma y color:SolidPeso molecular:381.28Clavamycin A
CAS:<p>Clavamycin A displays notable antifungal activity against Candida species, with its effects being antagonized by dipeptides or tripeptides, although not by amino acids. It lacks antibacterial properties and does not inhibit β-lactamase.</p>Fórmula:C16H22N4O9Forma y color:SolidPeso molecular:414.367ZL-Pin13
CAS:<p>ZL-Pin13: potent Pin1 inhibitor (IC50: 67 nM), halts MDA-MB-231 cell growth, reduces Pin1 substrates.</p>Fórmula:C24H23ClN2O3SForma y color:SoildPeso molecular:454.97Resorcinomycin B
CAS:<p>Resorcinomycin B is an antibiotic found in [Streptoverticillum roseoverticillatum].</p>Fórmula:C13H18N4O5Forma y color:SolidPeso molecular:310.306Dinalbuphine sebacate
CAS:<p>Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.</p>Fórmula:C52H68N2O10Forma y color:SolidPeso molecular:881.1FXIa-IN-10
<p>FXIa-IN-10 is a potent, orally bioavailable inhibitor of Activator XI (FXIa) (Ki: 0.17 nM).</p>Fórmula:C23H18Cl2F3N9O2Forma y color:SolidPeso molecular:580.35T-3861174
CAS:<p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>Fórmula:C26H25FN6O2Forma y color:SolidPeso molecular:472.51DGY-08-097
CAS:<p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>Fórmula:C60H76N10O14Forma y color:SolidPeso molecular:1161.3METTL3-IN-2
CAS:<p>METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.</p>Fórmula:C25H26N8OForma y color:SolidPeso molecular:454.53Anticancer agent 12
<p>Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.</p>Fórmula:C16H17BrN4O2SForma y color:SolidPeso molecular:409.3Defucogilvocarcin V
CAS:<p>Defucogilvocarcin V is an antibiotic with activity against Gram-positive bacteria.</p>Fórmula:C21H16O5Forma y color:SolidPeso molecular:348.349AT-IAP
CAS:AT-IAP is an effective dual antagonist of XIAP and cIAP1.Fórmula:C29H40FN5O2Pureza:98%Forma y color:SolidPeso molecular:509.66Mimocine
CAS:<p>Mimosine, a plant amino acid, is known to act as a normoxic inducer of hypoxia-inducible factor (HIF).</p>Fórmula:C15H14N2O5Forma y color:SolidPeso molecular:302.28Dehatrine
CAS:<p>Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.</p>Fórmula:C37H38N2O6Forma y color:SolidPeso molecular:606.71nNOS-IN-25
CAS:<p>nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.</p>Fórmula:C21H22N4Pureza:98%Forma y color:SolidPeso molecular:330.43Theophylline EP impurity C
CAS:<p>Theophylline EP impurity C, an alkaloid with anti-bronchospasm activity, is employed to assess the purity and quality of compounds. This substance also holds potential clinical value in the management of asthma and chronic obstructive pulmonary disease (COPD).</p>Fórmula:C7H10N4O3Forma y color:SolidPeso molecular:198.18AFP-07 free acid
CAS:<p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>Fórmula:C22H30F2O5Pureza:98%Forma y color:SolidPeso molecular:412.47PPARγ agonist 1
<p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>Fórmula:C34H39NO3Forma y color:SolidPeso molecular:509.68BDZ-h
CAS:<p>BDZ-h inhibits both closed/open states of all 4 homomeric & 2 GluA2R-complex AMPA receptors.</p>Fórmula:C21H21N5O3SForma y color:SolidPeso molecular:423.49Pulvilloric acid
CAS:<p>Pulvilloric acid is an antifungal antibiotic produced by the organism Pen. pulvillorum 504.</p>Fórmula:C15H18O5Forma y color:SolidPeso molecular:278.30Propizepine
CAS:<p>Propizepine is a tricyclic antidepressant compound.</p>Fórmula:C17H20N4OForma y color:SolidPeso molecular:296.37Antitrypanosomal agent 6
<p>Compound 18a: potent vs. T. brucei (IC50: 0.47 μM), >2x efficacy compared to Nifurtimox, good ADME, binds AT-rich DNA.</p>Fórmula:C22H29Cl2N5OForma y color:SolidPeso molecular:450.4PF-06815345 hydrochloride
CAS:<p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>Fórmula:C27H30Cl2FN9O4Forma y color:SolidPeso molecular:634.49Polvitolimod
CAS:<p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>Fórmula:C13H14FN5O4Forma y color:SolidPeso molecular:323.28SLC4101431
<p>SLC4101431 is a potent SphK2 inhibitor with Ki value of 90 nM.</p>Fórmula:C29H28ClN7OSForma y color:SolidPeso molecular:558.1Lp-PLA2-IN-6
CAS:<p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>Fórmula:C25H21F5N4O3Forma y color:SolidPeso molecular:520.45SML-10-70-1
CAS:<p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>Fórmula:C25H42ClN7O13P2Forma y color:SolidPeso molecular:746.04Combretastatin A1 phosphate
CAS:<p>Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.</p>Fórmula:C18H22O12P2Forma y color:SolidPeso molecular:492.31YKL-04-085
CAS:<p>YKL-04-085 inhibits viral translation effectively, with strong antiviral action at much lower doses than those affecting host-cell growth.</p>Fórmula:C30H29N5O2Forma y color:SolidPeso molecular:491.6SID 125240931
CAS:<p>SID 125240931 is a regulator of fluorine-activated proteins (FAPs). This compound disrupts the binding between fluoride and FAPs.</p>Fórmula:C19H24N4O3SForma y color:SolidPeso molecular:388.48Plumbemycin B
CAS:<p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Fórmula:C12H21N4O8PForma y color:SolidPeso molecular:380.29(25S)-δ7-Dafachronic acid
CAS:<p>(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.</p>Fórmula:C27H42O3Pureza:98%Forma y color:SolidPeso molecular:414.62NAZ2329
CAS:<p>NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.</p>Fórmula:C21H18F3NO4S3Forma y color:SoildPeso molecular:501.56Cilobamine mesylate
CAS:<p>Cilobamine mesylate is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.</p>Fórmula:C18H27Cl2NO4SForma y color:SolidPeso molecular:424.38CHNQD-01255
CAS:<p>CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).</p>Fórmula:C23H29NO6Forma y color:SolidPeso molecular:415.48YEATS4 binder-1
<p>YEATS4 binder-1(4e) is an effective and selective compound that targets the KAc recognition site within the YEATS structural domain, exhibiting a binding</p>Fórmula:C23H34N4O3Forma y color:SolidPeso molecular:414.54EICAR
CAS:<p>EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.</p>Fórmula:C11H13N3O5Forma y color:SolidPeso molecular:267.24LRH-1 modulator-1
CAS:<p>LRH-1 modulator-1: potent agonist, boosts IL-10, reduces IL-1b/TNFa, anti-inflammatory in gut.</p>Fórmula:C28H36N2O2SForma y color:SolidPeso molecular:464.66A1-Phytoprostane-I
CAS:<p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.</p>Fórmula:C18H28O4Forma y color:SolidPeso molecular:308.41Latrunculin M
CAS:<p>Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.</p>Fórmula:C21H33NO5SForma y color:SolidPeso molecular:411.55VRT-18858
CAS:<p>VRT-18858 is a metabolite of VX-740.</p>Fórmula:C24H25N5O7Forma y color:SolidPeso molecular:495.489(S)-HEPE
CAS:<p>9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.</p>Fórmula:C20H30O3Forma y color:SolidPeso molecular:318.45CYP121A1-IN-1
<p>CYP121A1-IN-1: Strong inhibitor for CYP121A1, hinders Mycobacterium tuberculosis growth (MIC 90 ~6.25 μM), reduces mycocyclosin synthesis.</p>Fórmula:C22H20N4OForma y color:SolidPeso molecular:356.42SphK2-IN-2
<p>SphK2-IN-2 (21g) is a potent and selective inhibitor of SphK2 (IC50: 0.23 μM).</p>Fórmula:C21H25ClN10OForma y color:SolidPeso molecular:468.94FWM-1
<p>FWM-1 blocks SARS-CoV-2 NSP13, hinders ATP binding, with -328.6 kcal/mol binding energy.</p>Fórmula:C15H11ClN4O4S2Forma y color:SolidPeso molecular:410.86M-COPA
CAS:<p>M-COPA disrupts Golgi, blocks MET & Arf1 activation, and inhibits angiogenesis via VEGFR & NF-kB pathways.</p>Fórmula:C25H34N2O2Forma y color:SolidPeso molecular:394.55NTPDase-IN-3
CAS:<p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>Fórmula:C22H24ClN3OS2Forma y color:SolidPeso molecular:446.03TRK-IN-19
<p>TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) & TRKAG595R (5.3 nM), promising for cancer research.</p>Fórmula:C22H26FN5O2Forma y color:SolidPeso molecular:411.47Pradimicin Q
CAS:<p>Pradimicin Q is an antibiotic exhibiting cytotoxicity against human colon HCT-116 cells and mouse melanoma B16-F10 cells, with IC50 values of 75 μg/mL and 100 μg/mL, respectively.</p>Fórmula:C24H16O10Forma y color:SolidPeso molecular:464.378AN-12-H5
CAS:<p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>Fórmula:C24H23N3O4S3Forma y color:SolidPeso molecular:513.6513-Hydroxyglucopiericidin A
CAS:<p>13-Hydroxyglucopiericidin A is an antibiotic with potent antitumor cell activity.</p>Fórmula:C31H47NO10Forma y color:SolidPeso molecular:593.706Detajmium
CAS:<p>Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.</p>Fórmula:C27H42N3O3Pureza:98%Forma y color:SolidPeso molecular:456.64Tauro-ω-muricholic acid sodium
<p>Tauro-ω-muricholic acid sodium (TωMCA sodium) is an analogue of tauro-α-muricholic acid, a bile acid of hepatic origin.</p>Fórmula:C26H44NNaO7SForma y color:SolidPeso molecular:537.68Pyruvate Carboxylase-IN-2
CAS:<p>Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.</p>Fórmula:C21H22O8Forma y color:SolidPeso molecular:402.39Pyrromycin
CAS:<p>Pyrromycin is a monosaccharide anthracycline which can be used to inhibit cellular RNA synthesis.</p>Fórmula:C30H35NO11Forma y color:SolidPeso molecular:585.60Glycocinnasperimicin D
CAS:<p>Glycocinnasperimicin D is a glycoside cinnamoyl iminohistamine antibiotic. It exhibits activity against both Gram-positive and Gram-negative bacteria. Additionally, Glycocinnasperimicin D inhibits leukemia L1210 cells, with an IC50 of 2.0 μg/mL.</p>Fórmula:C30H50N10O9Forma y color:SolidPeso molecular:694.78Brostallicin HCl
CAS:<p>Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.</p>Fórmula:C30H36BrClN12O5Forma y color:SolidPeso molecular:760.04ABT 491 Hydrochloride
CAS:<p>ABT-491 hydrochloride is an active platelet activator receptor (PAF-R) antagonist with good selectivity and oral administration.</p>Fórmula:C28H23ClFN5O2Forma y color:SolidPeso molecular:515.97Leukotriene F-4 sulfone
CAS:<p>Leukotriene F-4 sulfone induces vascular permeability changes.</p>Fórmula:C28H44N2O10SForma y color:SolidPeso molecular:600.72MRS2279 diammonium
CAS:<p>MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.</p>Fórmula:C13H24ClN7O8P2Forma y color:SolidPeso molecular:503.77L-2,5-Dihydrophenylalanine
CAS:<p>L-2,5-Dihydrophenylalanine can induce apoptosis in human medulloblastoma leukemia cells [HL-60].</p>Fórmula:C9H13NO2Forma y color:SolidPeso molecular:167.21Glutaminyl cyclases-IN-1
<p>Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.</p>Fórmula:C25H30N6O2SForma y color:SolidPeso molecular:478.61mPGES1-IN-5
CAS:<p>mPGES1-IN-5 (compound 18) is a multi-substituted pyrimidine compound that acts as a submicromolar inhibitor of PGE2 production. It primarily exerts its anti-inflammatory effects by inhibiting mPGES-1 and demonstrates significant inhibitory activity in vivo against acute inflammation models.</p>Fórmula:C27H27N3OForma y color:SolidPeso molecular:409.5217β-HSD1-IN-1
<p>17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.</p>Fórmula:C21H21NO3Forma y color:SolidPeso molecular:335.4CLR01 sodium
CAS:<p>CLR01 is a tweezer reducing α-synuclein in MSA, inhibits SOD1 in ALS, blocks Ebola/Zika, stabilizes proteins, and lessens mutant p53 toxicity.</p>Fórmula:C42H30Na2O8P2Forma y color:SolidPeso molecular:770.6211PF1070A
CAS:<p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>Fórmula:C31H44N4O6Forma y color:SolidPeso molecular:568.7MF-592
CAS:<p>MF-592: EP4 receptor antagonist, hEP4 IC50 3 nM, hWB IC50 78 nM, great oral PK, rat arthritis ED50 0.1 mg/kg/day, promising for development.</p>Fórmula:C34H33Cl2N3O6SForma y color:SolidPeso molecular:682.61
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