Otros inhibidores
Esta categoría abarca una amplia variedad de inhibidores que no encajan en las clasificaciones estándar, pero que son fundamentales para diversas investigaciones bioquímicas y farmacológicas. Estos inhibidores pueden dirigirse a vías, enzimas e interacciones moleculares únicas o menos estudiadas, proporcionando herramientas valiosas para áreas de investigación especializadas. En CymitQuimica, ofrecemos una selección diversa de inhibidores de alta calidad que abarcan múltiples objetivos biológicos y disciplinas de investigación, lo que le permite explorar nuevas vías terapéuticas y profundizar su comprensión de los procesos biológicos complejos.
Se han encontrado 36478 productos de "Otros inhibidores"
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HPK1-IN-18
CAS:<p>HPK1-IN-18: Potent, specific inhibitor of HPK1, a MAP4K enzyme, for cancer research and treatment.</p>Fórmula:C24H24N4Forma y color:LiquidPeso molecular:368.47Tifenazoxide
CAS:Tifenazoxide is an effective and SUR1/Kir6.2 selective KATP channels opener. Tifenazoxide has an anti-diabetic effect, can inhibit glucose-stimulated insulin release in vitro and in vivo.Fórmula:C9H10ClN3O2S2Pureza:98%Forma y color:SolidPeso molecular:291.78Cebranopadol ((1α,4α)stereoisomer)
CAS:<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Fórmula:C24H27FN2OPureza:98%Forma y color:SolidPeso molecular:378.48(E)-Crotylbarbital
CAS:<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Fórmula:C10H14N2O3Pureza:99.94%Forma y color:SolidPeso molecular:210.23Fosfonet sodium
CAS:Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.Fórmula:C2H4NaO5PForma y color:SolidPeso molecular:162.01PL265
CAS:<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Fórmula:C27H35N2O9PPureza:98%Forma y color:SolidPeso molecular:562.55PAD4-IN-2
CAS:<p>PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-</p>Fórmula:C20H23BClN7O6Forma y color:SolidPeso molecular:503.7Radafaxine hydrochloride
CAS:<p>Radafaxine hydrochloride is an inhibitor of DAT and NET transporters, and nAChR family modulator.</p>Fórmula:C13H19Cl2NO2Pureza:98%Peso molecular:292.2Aminobutane bisphosphonate
CAS:Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.Fórmula:C4H13NO6P2Forma y color:SolidPeso molecular:233.1KP372-1
CAS:<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Fórmula:C20H8N12O2Forma y color:SolidPeso molecular:448.36Butabindide oxalate
CAS:<p>CCK-inactivating serine protease (tripeptidyl peptidase II) inhibitor</p>Fórmula:C19H27N3O6Pureza:98%Forma y color:SolidPeso molecular:393.43Benzovindiflupyr
CAS:<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Fórmula:C18H15Cl2F2N3OForma y color:SolidPeso molecular:398.23CK176
CAS:CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.Fórmula:C21H12IN3O2Pureza:98%Forma y color:SolidPeso molecular:465.24(Rac)-LM11A-31 dihydrochloride
CAS:(Rac)-LM11A-31 dihydrochloride is an isomer of LM11A-31 dihydrochloride, a potent antagonist of proNGF (nerve growth factor).Fórmula:C12H27Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:316.268CH-100
CAS:CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.Fórmula:C14H22ClNO3Forma y color:SolidPeso molecular:287.78Trimetoquinol HCl hydrate
CAS:Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.Fórmula:C19H26ClNO6Forma y color:SolidPeso molecular:399.87Dioxifedrine
CAS:Dioxifedrine is a beta-2 -adrenergic agonist with bronchodilator activity.Fórmula:C10H15NO3Forma y color:SolidPeso molecular:197.23Saxitoxinol
CAS:<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Fórmula:C10H17N7O3Pureza:98%Forma y color:SolidPeso molecular:283.29Ref: TM-T68748
Producto descatalogadoIDX-375
CAS:IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.Fórmula:C29H50N5O7PSPureza:98%Forma y color:SolidPeso molecular:643.78PS372424 HCl
CAS:<p>PS372424 activates CXCR3, triggers ERK phosphorylation, and inhibits CXCL11's effect on CD45+ cell migration in humanized mice.</p>Fórmula:C33H45ClN6O4Forma y color:SolidPeso molecular:625.21FM-24 HCl
CAS:FM-24 HCl is a long acting beta-adrenergic receptor antagonist.Fórmula:C19H30ClNO2Forma y color:SolidPeso molecular:339.9D(-)-Octopamine CSA salt
CAS:D(-)-Octopamine CSA salt is an agonist of octopamine receptors.Fórmula:C18H27NO6SPureza:98%Forma y color:SolidPeso molecular:385.48BChE-IN-17
CAS:<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Fórmula:C23H23BrN2O4S2Forma y color:SolidPeso molecular:535.47Albuterol stearate
CAS:<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Fórmula:C31H57NO5Pureza:98%Forma y color:SolidPeso molecular:523.799Phenazolam
CAS:<p>Phenazolam is an analytical reference standard categorized as a benzodiazepine. [1] This product is intended for research and forensic applications.</p>Fórmula:C17H12BrClN4Forma y color:SolidPeso molecular:387.66Guancydine
CAS:Guancydine is an antihypertensive agent.Fórmula:C7H14N4Pureza:98%Forma y color:SolidPeso molecular:154.21Erythrityl Tetranitrate
CAS:Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."Fórmula:C4H6N4O12Forma y color:SolidPeso molecular:302.11Culmerciclib
CAS:<p>Culmerciclib is a cell cycle protein-dependent kinase (CDK) inhibitor that exhibits antitumour effects.</p>Fórmula:C24H27FN8Forma y color:SolidPeso molecular:446.52Phenamil methanesulfonate
CAS:TRPP3 channel inhibitorFórmula:C13H16ClN7O4SPureza:98%Forma y color:SolidPeso molecular:401.83DPX-3778
CAS:DPX-3778, a triethanolamine salt, boosts tobacco callus growth 4-5x at 0.124-2.48 μM and slows aging with IAA and kinetin.Fórmula:C16H23ClN4O6Forma y color:SolidPeso molecular:402.83Questiomycin A derivatives 18 TFA
<p>Questiomycin A derivative 18 TFA exhibits antibacterial, anticancer properties and inhibits GRP78.</p>Fórmula:C16H12F3N3O5Pureza:98.45%Forma y color:SoildPeso molecular:383.07Ref: TM-T67717L
Producto descatalogadoanti-TNBC agent-3
CAS:<p>Anti-TNBC agent-3 (compound 3g) is a compound that induces apoptosis and possesses anti-cancer cell proliferation properties.</p>Fórmula:C29H39F2N7OForma y color:SolidPeso molecular:539.66MDK-2959
CAS:MDK-2959 is a potent inhibitor of protein tyrosine phosphatase sigma (PTPsigma).Fórmula:C15H11N3O4Pureza:98%Forma y color:SolidPeso molecular:297.27Omeprazole acid
CAS:Omeprazole treats GERD, ulcers, Zollinger-Ellison syndrome, prevents GI bleeding; it's a proton pump inhibitor.Fórmula:C34H32N6Na2O10S2Forma y color:SolidPeso molecular:794.76FOXM1-IN-2
CAS:<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Fórmula:C48H47F4N7O12SForma y color:SolidPeso molecular:1021.99Civorebrutinib
CAS:<p>Civorebrutinib (WS-413) is an inhibitor of Bruton's tyrosine kinase that exhibits antineoplastic activity [1].</p>Fórmula:C23H22ClN7O2Forma y color:SolidPeso molecular:463.92I-BET282
CAS:<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Fórmula:C25H30N4O4Pureza:98%Forma y color:SolidPeso molecular:450.53LT-540-717
CAS:<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Fórmula:C24H24N8O2Forma y color:SolidPeso molecular:456.5LM2I
CAS:<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Fórmula:C47H77N3O11Forma y color:SolidPeso molecular:860.13PD1-PDL1-IN 2
CAS:<p>PD1-PDL1-IN 2 (ZE132) is a potent, selective inhibitor of PD-1/PD-L1, exhibiting significant anti-tumor activity in vivo. It enhances cytotoxic T-cell tumor infiltration and stimulates IL-2 expression, while also strongly inhibiting TGF-β [1] mRNA expression, showcasing its comprehensive immunotherapeutic potential.</p>Fórmula:C37H41ClN4O7SForma y color:SolidPeso molecular:721.26S-72
CAS:<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Fórmula:C20H22N4O3SForma y color:SolidPeso molecular:398.50Ref: TM-T83874
Producto descatalogadoAc4GalNAlk
CAS:<p>Ac4GalNAlk, a weakly alkyne-labeled reagent for metabolic oligosaccharide engineering (MOE), facilitates the detection of protein glycosylation by promoting nucleotide-sugar biosynthesis and enhancing bioorthogonal cell surface markers. It is activated by cellular biosynthetic machinery into nucleotide sugars, subsequently enabling the tracing of glycoproteins in bioorthogonal chemistry [1].</p>Fórmula:C19H25NO10Forma y color:SolidPeso molecular:427.4MDVN1003
CAS:MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.Fórmula:C22H20FN7OPureza:98%Forma y color:SolidPeso molecular:417.44IDO/Tubulin-IN-2
CAS:<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Fórmula:C48H40N6O10Forma y color:SolidPeso molecular:860.87ARN 077
CAS:ARN 077 is a selective N-acylethanolamine acid amidase (NAAA) inhibitor (IC50: 7 nM for human NAAA). ARN 077 significantly increases palmitoyl ethanolamine (PEA) levels within the CNS.Fórmula:C16H21NO4Forma y color:SolidPeso molecular:291.34Antibacterial agent 160
CAS:<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Fórmula:C29H27ClFN3O6Forma y color:SolidPeso molecular:567.99Sakura 6
CAS:<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Fórmula:C31H45N5O7Forma y color:SolidPeso molecular:599.73Anti-MI/R injury agent 1
CAS:<p>Anti-MI/R injury agent 1 (compound 18), derived from Panaxatriol, represents an orally administered, potent agent against myocardial ischemia/reperfusion (MI/R</p>Fórmula:C32H49NO6Forma y color:SolidPeso molecular:543.73Tauro-Obeticholic Acid sodium
CAS:<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Fórmula:C28H48NO6S·NaForma y color:SolidPeso molecular:549.74SHP2-IN-14
CAS:<p>SHP2-IN-14 (compound 27) is a potent, orally active allosteric inhibitor of SHP2, displaying strong anti-tumor activity with an IC50 of 7 nM.</p>Fórmula:C22H20Cl2N8OForma y color:SolidPeso molecular:483.35RIOK2-IN-2
CAS:<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Fórmula:C27H23F3N6O2Forma y color:SolidPeso molecular:520.51L 689037
CAS:L 689037 is an inhibitor of leukotriene biosynthesis.Fórmula:C36H37ClN2O4Pureza:98%Forma y color:SolidPeso molecular:597.14DDO-2213
CAS:<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Fórmula:C24H27ClFN7OForma y color:SolidPeso molecular:483.97DiaFluo
CAS:<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Fórmula:C32H32N4O9SForma y color:SolidPeso molecular:648.69Ref: TM-T31416
Producto descatalogadoAnd1-IN-1
CAS:<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Fórmula:C15H11BCl2O2Forma y color:SolidPeso molecular:304.96Antitumor agent-136
CAS:<p>Antitumor Agent-136 (Compound 17), a broad-spectrum antitumor agent and NAMPT inhibitor, exhibits potent activity with an IC50 of 9.5 nM. It efficiently lowers intracellular and extracellular NAMPT protein levels via the ubiquitin proteasome pathway, achieving effective tumor inhibition [1].</p>Fórmula:C58H76N10O11S3Forma y color:SolidPeso molecular:1185.48HPK1-IN-38
CAS:<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Fórmula:C29H29N5O3Forma y color:SolidPeso molecular:495.57Antitumor photosensitizer-1
CAS:<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Fórmula:C42H51N5O6Forma y color:SolidPeso molecular:721.88FAP-IN-2
CAS:<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Fórmula:C24H28F2N6O3Forma y color:SolidPeso molecular:486.51CYY292
CAS:<p>CYY292 is a chemical compound acting as an inhibitor of PDGFRα, PDGFRβ, FGFR1, -2, and -3, with respective IC50 values of 5.35, 4.6, 28, 28, and 78 nM.</p>Fórmula:C24H28N8OForma y color:SolidPeso molecular:444.53Immune cell migration-IN-1
CAS:<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Fórmula:C30H25ClN4O6SForma y color:SolidPeso molecular:605.06FLT3-IN-19
CAS:<p>FLT3-IN-19 (Comp 50) is a potent, selective inhibitor of FLT3, demonstrating an IC50 value of 0.213 nM, and is applicable in research pertaining to acute</p>Fórmula:C22H26N8OForma y color:SolidPeso molecular:418.49Antitumor photosensitizer-2
CAS:<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Fórmula:C40H47N5O7Forma y color:SolidPeso molecular:709.83Antibacterial agent 157
CAS:<p>Compound B12 (Antibacterial agent 157) is a fungicidal agent that can impact protein synthesis in Botrytis cinerea.</p>Fórmula:C26H23BrF4N2O3Forma y color:SolidPeso molecular:567.3780-O16B
CAS:<p>80-O16B, an ionizable cationic lipid featuring disulfide bonds, is utilized in the preparation of lipid nanoparticles (LNP) [1].</p>Fórmula:C39H78N2O4S4Forma y color:SolidPeso molecular:767.31HMR 1556
CAS:HMR 1556 is a chromanol derivative and is an IKs blocker (IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively).Fórmula:C17H24F3NO5SForma y color:SolidPeso molecular:411.44CIAC001
CAS:<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Fórmula:C20H25N3O2Forma y color:SolidPeso molecular:339.43URAT1 inhibitor 5
CAS:<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Fórmula:C18H14BrN3O2SForma y color:SolidPeso molecular:416.29Azilsartan mepixetil potassium
CAS:<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Fórmula:C36H33KN6O8Forma y color:SolidPeso molecular:716.78Ifetroban
CAS:<p>Ifetroban is a potent and selective TxA2/PGH2 receptor antagonist.</p>Fórmula:C25H32N2O5Forma y color:SolidPeso molecular:440.53BB-Cl-Amidine hydrochloride
CAS:BB-Cl-Amidine hydrochloride is an inhibitor of peptidylarginine deminase (PAD) [1].Fórmula:C26H27Cl2N5OPureza:98%Forma y color:SolidPeso molecular:496.43DG026
CAS:DG026 selectively inhibits IRAP, reducing its cross-presentation in dendritic cells without affecting ERAP1.Fórmula:C35H40N3O4PPureza:98%Forma y color:SolidPeso molecular:597.68Ifetroban sodium
CAS:<p>Ifetroban sodium (BMS-180291), oral TXA2/PGH2 antagonist for researching heart, stroke, BP, thrombosis.</p>Fórmula:C25H31N2NaO5Forma y color:SolidPeso molecular:462.522ALS-I-41
CAS:ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.Fórmula:C30H38FN3O6SPureza:98%Forma y color:SolidPeso molecular:587.7Cortivazol
CAS:Cortivazol is an Anti-Inflammatory Drug.Fórmula:C32H38N2O5Pureza:98%Forma y color:SolidPeso molecular:530.65Ref: TM-T25271
Producto descatalogadoBPH-628
CAS:<p>BPH-628 is a bioactive chemical.</p>Fórmula:C20H20O7P2Forma y color:SolidPeso molecular:434.329,10-Phenanthrenequinone
CAS:<p>9,10-Phenanthrenequinone is an inhibitor of claudin-5/CLDN5, which induces apoptosis via an NO synthase/ROS-dependent mechanism. It also promotes caspase activation and DNA fragmentation while reducing CLDN5 expression and proteasome proteolysis, contributing to endothelial barrier dysfunction.</p>Fórmula:C14H8O2Forma y color:SolidPeso molecular:208.21
