Otros inhibidores
Esta categoría abarca una amplia variedad de inhibidores que no encajan en las clasificaciones estándar, pero que son fundamentales para diversas investigaciones bioquímicas y farmacológicas. Estos inhibidores pueden dirigirse a vías, enzimas e interacciones moleculares únicas o menos estudiadas, proporcionando herramientas valiosas para áreas de investigación especializadas. En CymitQuimica, ofrecemos una selección diversa de inhibidores de alta calidad que abarcan múltiples objetivos biológicos y disciplinas de investigación, lo que le permite explorar nuevas vías terapéuticas y profundizar su comprensión de los procesos biológicos complejos.
Se han encontrado 36533 productos de "Otros inhibidores"
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Antitumor agent-136
CAS:<p>Antitumor Agent-136 (Compound 17), a broad-spectrum antitumor agent and NAMPT inhibitor, exhibits potent activity with an IC50 of 9.5 nM. It efficiently lowers intracellular and extracellular NAMPT protein levels via the ubiquitin proteasome pathway, achieving effective tumor inhibition [1].</p>Fórmula:C58H76N10O11S3Forma y color:SolidPeso molecular:1185.48Civorebrutinib
CAS:<p>Civorebrutinib (WS-413) is an inhibitor of Bruton's tyrosine kinase that exhibits antineoplastic activity [1].</p>Fórmula:C23H22ClN7O2Forma y color:SolidPeso molecular:463.92DDO-2213
CAS:<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Fórmula:C24H27ClFN7OForma y color:SolidPeso molecular:483.97And1-IN-1
CAS:<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Fórmula:C15H11BCl2O2Forma y color:SolidPeso molecular:304.96LM2I
CAS:<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Fórmula:C47H77N3O11Forma y color:SolidPeso molecular:860.13DiaFluo
CAS:<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Fórmula:C32H32N4O9SForma y color:SolidPeso molecular:648.69Ref: TM-T31416
Producto descatalogadoCIAC001
CAS:<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Fórmula:C20H25N3O2Forma y color:SolidPeso molecular:339.43LT-540-717
CAS:<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Fórmula:C24H24N8O2Forma y color:SolidPeso molecular:456.5FOXM1-IN-2
CAS:<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Fórmula:C48H47F4N7O12SForma y color:SolidPeso molecular:1021.99Antitumor photosensitizer-2
CAS:<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Fórmula:C40H47N5O7Forma y color:SolidPeso molecular:709.83HMR 1556
CAS:HMR 1556 is a chromanol derivative and is an IKs blocker (IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively).Fórmula:C17H24F3NO5SForma y color:SolidPeso molecular:411.4480-O16B
CAS:<p>80-O16B, an ionizable cationic lipid featuring disulfide bonds, is utilized in the preparation of lipid nanoparticles (LNP) [1].</p>Fórmula:C39H78N2O4S4Forma y color:SolidPeso molecular:767.31Immune cell migration-IN-1
CAS:<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Fórmula:C30H25ClN4O6SForma y color:SolidPeso molecular:605.06CYY292
CAS:<p>CYY292 is a chemical compound acting as an inhibitor of PDGFRα, PDGFRβ, FGFR1, -2, and -3, with respective IC50 values of 5.35, 4.6, 28, 28, and 78 nM.</p>Fórmula:C24H28N8OForma y color:SolidPeso molecular:444.53I-BET282
CAS:<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Fórmula:C25H30N4O4Pureza:98%Forma y color:SolidPeso molecular:450.53S-72
CAS:<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Fórmula:C20H22N4O3SForma y color:SolidPeso molecular:398.50Ref: TM-T83874
Producto descatalogadoL 689037
CAS:L 689037 is an inhibitor of leukotriene biosynthesis.Fórmula:C36H37ClN2O4Pureza:98%Forma y color:SolidPeso molecular:597.14FAP-IN-2
CAS:<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Fórmula:C24H28F2N6O3Forma y color:SolidPeso molecular:486.51Sakura 6
CAS:<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Fórmula:C31H45N5O7Forma y color:SolidPeso molecular:599.73MDVN1003
CAS:MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.Fórmula:C22H20FN7OPureza:98%Forma y color:SolidPeso molecular:417.44HPK1-IN-38
CAS:<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Fórmula:C29H29N5O3Forma y color:SolidPeso molecular:495.57ARN 077
CAS:ARN 077 is a selective N-acylethanolamine acid amidase (NAAA) inhibitor (IC50: 7 nM for human NAAA). ARN 077 significantly increases palmitoyl ethanolamine (PEA) levels within the CNS.Fórmula:C16H21NO4Forma y color:SolidPeso molecular:291.34IDO/Tubulin-IN-2
CAS:<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Fórmula:C48H40N6O10Forma y color:SolidPeso molecular:860.87Antitumor photosensitizer-1
CAS:<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Fórmula:C42H51N5O6Forma y color:SolidPeso molecular:721.88PD1-PDL1-IN 2
CAS:<p>PD1-PDL1-IN 2 (ZE132) is a potent, selective inhibitor of PD-1/PD-L1, exhibiting significant anti-tumor activity in vivo. It enhances cytotoxic T-cell tumor infiltration and stimulates IL-2 expression, while also strongly inhibiting TGF-β [1] mRNA expression, showcasing its comprehensive immunotherapeutic potential.</p>Fórmula:C37H41ClN4O7SForma y color:SolidPeso molecular:721.26ALS-I-41
CAS:ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.Fórmula:C30H38FN3O6SPureza:98%Forma y color:SolidPeso molecular:587.7Ifetroban sodium
CAS:<p>Ifetroban sodium (BMS-180291), oral TXA2/PGH2 antagonist for researching heart, stroke, BP, thrombosis.</p>Fórmula:C25H31N2NaO5Forma y color:SolidPeso molecular:462.522BPH-628
CAS:<p>BPH-628 is a bioactive chemical.</p>Fórmula:C20H20O7P2Forma y color:SolidPeso molecular:434.32DG026
CAS:DG026 selectively inhibits IRAP, reducing its cross-presentation in dendritic cells without affecting ERAP1.Fórmula:C35H40N3O4PPureza:98%Forma y color:SolidPeso molecular:597.68Ifetroban
CAS:<p>Ifetroban is a potent and selective TxA2/PGH2 receptor antagonist.</p>Fórmula:C25H32N2O5Forma y color:SolidPeso molecular:440.53BB-Cl-Amidine hydrochloride
CAS:BB-Cl-Amidine hydrochloride is an inhibitor of peptidylarginine deminase (PAD) [1].Fórmula:C26H27Cl2N5OPureza:98%Forma y color:SolidPeso molecular:496.43Cortivazol
CAS:Cortivazol is an Anti-Inflammatory Drug.Fórmula:C32H38N2O5Pureza:98%Forma y color:SolidPeso molecular:530.65Ref: TM-T25271
Producto descatalogado9,10-Phenanthrenequinone
CAS:<p>9,10-Phenanthrenequinone is an inhibitor of claudin-5/CLDN5, which induces apoptosis via an NO synthase/ROS-dependent mechanism. It also promotes caspase activation and DNA fragmentation while reducing CLDN5 expression and proteasome proteolysis, contributing to endothelial barrier dysfunction.</p>Fórmula:C14H8O2Forma y color:SolidPeso molecular:208.21
