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Señalización citoesquelética

Señalización citoesquelética

Los inhibidores de la señalización del citoesqueleto son compuestos que interrumpen las vías de señalización que regulan el citoesqueleto, crucial para la forma celular, la motilidad, la división y el transporte intracelular. Estos inhibidores se utilizan para estudiar la dinámica de las proteínas del citoesqueleto, como la actina y la tubulina, y su papel en procesos como la migración celular, la adhesión y la metástasis del cáncer. Los inhibidores de la señalización del citoesqueleto son valiosos en la investigación sobre biología celular, cáncer y neurobiología. En CymitQuimica, ofrecemos una amplia gama de inhibidores de la señalización del citoesqueleto de alta calidad para apoyar su investigación en estas áreas.

Se han encontrado 1381 productos de "Señalización citoesquelética"

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  • ER degrader 7

    CAS:
    <p>ER degrader 7 (Compound 35t) is a selective degrader of both ERα and ERβ, and possesses activity as a tubulin polymerization inhibitor.</p>
    Fórmula:C33H31F4N3O5SSe
    Forma y color:Solid
    Peso molecular:736.63
  • CCT251455

    CAS:
    <p>CCT251455, the mitotic kinase monopolar spindle 1 (MPS1/TTK) inhibitor, is a potent (IC50=3 nM) and specific chemical tool.</p>
    Fórmula:C26H26ClN7O2
    Pureza:99.1% - 99.1%
    Forma y color:Solid
    Peso molecular:503.98
  • TC-I 15

    CAS:
    α2β1 integrin inhibitor
    Fórmula:C23H28N4O6S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:520.62
  • SB-267268

    CAS:
    <p>SB-267268: αvβ3 inhibitor (IC50: 0.68 nM human, 0.29 nM mouse), blocks αvβ3/αvβ5 integrins (Ki: 0.9 nM human, 0.5 nM monkey αvβ3, 0.7 nM human αvβ5).</p>
    Fórmula:C22H24F3N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:451.44
  • HSP90-IN-27

    CAS:
    <p>HSP90-IN-27, also known as compound 19, is an inhibitor of HSP90 [1].</p>
    Fórmula:C18H21N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:343.44
  • ALM301

    CAS:
    <p>ALM301: oral AKT inhibitor targeting AKT1, AKT2, AKT3; blocks AKT phosphorylation, curbs cancer cell growth.</p>
    Fórmula:C25H25N3O3
    Forma y color:Solid
    Peso molecular:415.48
  • PKC-θ inhibitor 1

    CAS:
    <p>PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)</p>
    Fórmula:C17H15F3N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:348.32
  • PAK1-IN-1

    CAS:
    <p>PAK1-IN-1: PAK1 inhibitor, IC50 9.8 nM, hinders tumor cell migration and invasion dose-dependently.</p>
    Fórmula:C26H20ClN5O2
    Forma y color:Solid
    Peso molecular:469.92
  • JNJ-26076713

    CAS:
    <p>JNJ-26076713, an oral alpha V integrin blocker, may treat macular edema, AMD, and diabetic retinopathy.</p>
    Fórmula:C29H38N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:490.64
  • HSP90-IN-19

    CAS:
    <p>HSP90-IN-19: potent Hsp90 inhibitor, IC50 = 0.27 μM, used in research on viral diseases, neurodegeneration, inflammation.</p>
    Fórmula:C29H38O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:498.61
  • Antitumor agent-86

    CAS:
    <p>Antitumor agent-86 targets MCF-7 cells with 2.62 µM IC50, induces apoptosis, and disrupts RAS/PI3K/Akt/JNK pathways.</p>
    Fórmula:C29H31N5O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:513.65
  • α7β1 integrin modulator-1

    CAS:
    <p>α7β1 Integrin Modulator-1 is a potent modulator with research potential for muscular dystrophy [1].</p>
    Fórmula:C23H29N3O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:475.56
  • Phenamacril

    CAS:
    <p>Phenamacril (JS39919) is acyanoacrylate fungicide, has powerful inhibition against Fusarium species, especially to Fusarium graminearum.</p>
    Fórmula:C12H12N2O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:216.24
  • β-Catenin modulator-5

    CAS:
    <p>β-Catenin Modulator-5 (Compound IIa-84), an oxazole and thiazole-based compound, serves as a potent and selective modulator of β-Catenin [1].</p>
    Fórmula:C21H22N2O2S
    Forma y color:Solid
    Peso molecular:366.48
  • UU-T01

    CAS:
    <p>UU-T01 inhibits β-catenin/Tcf4 with Ki of 3.14 µM, binds β-catenin directly with KD of 0.531 µM.</p>
    Fórmula:C10H10N6O
    Forma y color:Solid
    Peso molecular:230.23
  • Pivanex

    CAS:
    <p>Pivanex, an oral HDAC inhibitor, targets metastasis, angiogenesis, reduces Bcr-Abl protein, and promotes apoptosis.</p>
    Fórmula:C10H18O4
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:202.25
  • Synstatin (92-119)

    CAS:
    <p>Synstatin (92-119) serves as an anti-tumor agent by suppressing angiogenesis and cancer cell invasion, chiefly through the down-regulation of integrin αvβ3 and</p>
    Fórmula:C133H207N35O46
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3032.27
  • G-5555

    CAS:
    <p>G-5555 is a potent inhibitor of p21-activated kinase 1 (PAK1) (Kis: 3.7 nM and 11 nM for PAK1 and PAK2, respectively).</p>
    Fórmula:C25H25ClN6O3
    Pureza:99.76% - 99.84%
    Forma y color:Solid
    Peso molecular:492.96
  • AKT-I-1

    CAS:
    <p>AKT-I-1 is a selective and reversible inhibitor of Akt1.</p>
    Fórmula:C22H30N6
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:378.51
  • TAS0612

    CAS:
    <p>TAS0612, a novel oral inhibitor of RSK, AKT, and S6K, exhibits broad-spectrum antitumor activity by impeding cell growth [1].</p>
    Fórmula:C27H34F3N9O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:573.61