Receptores acoplados de proteína G y receptores 7-TM

Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It …

Silodosin is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic …

Droperidol is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a …

ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)

Anandamide, an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but also …

Dapoxetine HCl is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature …

Rimonabant hydrochloride is a cannabinoid receptor antagonist, binding selectively to central cannabinoid receptors (CB1) with …

Alverine Citrate is utilized in functional gastrointestinal disorders.

TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).

Loratadine is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis …

Quinacrine Hydrochloride is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and …

BP 897 is a potent and selective agonist of dopamine D3 receptor and it is …

FTBMT is a selective GPR52 agonist (EC50: 75 nM) and it also has antipsychotic and …

Molindone hydrochloride is an indole derivative effective in schizophrenia and other psychoses by blocking the …

Seratrodast (INN), a thromboxane A2 (TXA2) receptor (TP receptor) antagonist, is mainly used in the …

DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular …

Citalopram, a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, …

Dyphylline is a xanthine derivative. Dyphilline exerts bronchodilator effects and to a lesser extent vasodilator …

Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, …

Olanzapine is an atypical antipsychotic that is used currently in the treatment of schizophrenia and …

AH 6809 is an antagonist of EP and DP receptor(with Kis of 1217, 1150, 1597, …

Paroxetine hydrochloride is a serotonin uptake inhibitor that is effective in the treatment of depression.

Bromopride is a dopamine antagonist with prokinetic properties closely related to metoclopramide, and is widely …

2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 …

Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .

Pentoxifylline modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits …

Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).

Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors …

AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].

Tripelennamine hydrochloride is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.

Vincamine is a major alkaloid of Vinca minor L., Apocynaceae. It has been used therapeutically …

METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.

N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with …

2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.

Asenapine is a second generation (atypical) antipsychotic agent that is taken sublingually and used in …

Palonosetron is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and …

Matrine, an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.

Penfluridol is a highly potent antipsychotic.

[Leu5]-Enkephalin is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid …

Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment …

S1RA(E-52862) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM) antagonist, showed good selectivity against …

Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and …

Clorprenaline Hydrochloride is a beta-2 adrenergic agonist with bronchodilator activity.

Sotalol Hydrochloride is the hydrochloride salt form of sotalol, an ethanolamine derivative with Class III …

Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.

Pranoprofen (INN) is a non-steroidal anti-inflammatory drug used in ophthalmology.

Jatrorrhizine chloride is a potent and orally active uptake-2 transporter inhibitor. It exhibits a critical …

Bromperidol is a butyrophenone derivative and it is a potent and long-acting neuroleptic. Which is …

Ursodeoxycholic acid can be used to dissolve gallstones and reduce cholesterol absorption.

Promazine hydrochloride is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. …

Levodropropizine is a histamine receptor inhibitor. It is used as an effective and very well …

Sodium Butyrate is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short …

Almorexant HCl (ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor …

Tandospirone (SM-3997) is a selective partial agonist of 5-HT1A receptor (Ki: 27 nM) that displays …

Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL …

Ticlopidine hydrochloride is an effective inhibitor of platelet aggregation commonly used in the placement of …