
Receptores acoplados de proteína G y receptores 7-TM
Los receptores acoplados a proteínas G (GPCR) y los receptores de 7 dominios transmembrana (7-TM) son una gran familia de proteínas de membrana que desempeñan un papel clave en la comunicación celular y la transducción de señales. Estos receptores están involucrados en una amplia gama de procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la regulación hormonal. Los GPCR son objetivos principales en el descubrimiento de fármacos, lo que los convierte en esenciales para la investigación en farmacología y medicina. En CymitQuimica, ofrecemos una amplia selección de reactivos y compuestos de alta calidad relacionados con los GPCR y los receptores 7-TM para apoyar su investigación y esfuerzos en el desarrollo de medicamentos.
Se han encontrado 5973 productos para "Receptores acoplados de proteína G y receptores 7-TM".
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Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Fórmula:C17H30ClN5O2SForma y color:SolidPeso molecular:403.97PSA1 (141-150)
CAS:This Prostate Specific Antigen 1 peptide was used in the immunotherapy of cancer experiments.Fórmula:C55H93N13O13SPureza:98%Forma y color:SolidPeso molecular:1176.47Zovaglutide
CAS:Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.Forma y color:SolidDesmethyl Mirtazapine (hydrochloride)
CAS:Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Fórmula:C16H18ClN3Forma y color:SolidPeso molecular:287.79ELA-32(human)
CAS:Potent apelin receptor agonist with IC50 = 0.27 nM; does not bind GPR15/GPR25. Boosts hESC self-renewal and angiogenesis.Fórmula:C170H289N63O39S4Pureza:98%Forma y color:SolidPeso molecular:3967.8Substance P, Free Acid
CAS:Substance P, Free Acid is a synthetic analog of native Substance P, however, it lacks the biological activity exhibited by Substance P.Fórmula:C63H97N17O14SPureza:98%Forma y color:SolidPeso molecular:1348.61AL12180
CAS:AL12180 is a bioactive chemical.Fórmula:C21H27ClO6Forma y color:SolidPeso molecular:410.89Formoterol O-β-D-Glucuronide
CAS:Formoterol O-β-D-glucuronide is a metabolite of formoterol .Fórmula:C25H32N2O10Forma y color:SolidPeso molecular:520.535(-)-Eseroline fumarate
CAS:(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.Fórmula:C17H22N2O5Forma y color:SolidPeso molecular:334.37GRPP (human)
CAS:GRPP (human), a 30-amino-acid peptide derived from Gcg, modestly elevates plasma insulin levels while reducing plasma glucagon concentrations.Fórmula:C136H215N41O58SForma y color:SolidPeso molecular:3384.47sGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Fórmula:C64H83N17O12Forma y color:SolidPeso molecular:1282.4516-phenoxy tetranor Prostaglandin F2α isopropyl ester
CAS:Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.Fórmula:C25H36O6Forma y color:SolidPeso molecular:432.557GUB03385
GUB03385 is a long-acting PrRP31 analogue and an effective dual agonist for GPR10 (full agonist, EC50: 0.4 nM) and NPFF2R (partial agonist, EC50: 20 nM), with anti-obesity properties.Fórmula:C198H322N60O52SPeso molecular:4404.41173(p-Iodo-Phe7)-ACTH (4-10)
CAS:(p-Iodo-Phe7)-ACTH (4-10), an ACTH derivative and MC receptor antagonist, inhibits α-MSH-induced grooming in rats.Fórmula:C44H58IN13O10SForma y color:SolidPeso molecular:1087.98Glucagon receptor antagonists-1
CAS:Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.Fórmula:C29H34FNO2Pureza:98%Forma y color:SolidPeso molecular:447.5815(S)-HpEPE
CAS:15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.Fórmula:C20H30O4Forma y color:SolidPeso molecular:334.456TH023
TH023 is an inhibitor of the TLR4 signaling pathway, specifically targeting the formation of TLR4 homodimers. In HEK-Blue hTLR4 cells, TH023 suppresses the secretion of embryonic alkaline phosphatase with an IC50 of 0.354 μM and inhibits NO expression in RAW264.7 cells, with an IC50 of 1.61 μM. Additionally, TH023 inhibits the activation of NF-κB and reduces the nuclear translocation of NF-κB p65. The compound demonstrates anti-inflammatory effects in a mouse model of LPS-induced acute sepsis and improves lung injury in mice.Fórmula:C22H21ClF2N4OForma y color:SolidPeso molecular:430.88Vensemaglutide
CAS:Vensemaglutide is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in research related to diabetes or other metabolic disorders.Fórmula:C214H337N49O67Forma y color:SolidPeso molecular:4668.25Bz-Dab(nbd)-awfpp-nle-NH2
CAS:Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.Fórmula:C56H65N13O11Forma y color:SolidPeso molecular:1096.2[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS:'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.Fórmula:C39H64N8O10Forma y color:SolidPeso molecular:804.97

