Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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PDK1-IN-RS2
CAS:<p>PDK1-IN-RS2, a PIFtide mimic, selectively inhibits PDK1, blocking S6K1 activation (Kd: 9 μM).</p>Fórmula:C15H9ClN2O2S3Pureza:98%Forma y color:SolidPeso molecular:380.89Ref: TM-T16450
Producto descatalogadoGolgicide A-2
CAS:<p>GCA-2 is a potent enantiomer of GCA, selectively and efficiently kills An. stephensi larvae, useful for dengue research.</p>Fórmula:C17H14F2N2Forma y color:SolidPeso molecular:284.31SEMBL
CAS:<p>SEMBL, a novel inhibitor of DNA binding of NF-kappaB component p65 in vitro, inhibits NF-kappaB and cellular invasion in ovarian carcinoma ES-2 cells.</p>Fórmula:C12H11NO4Pureza:98%Forma y color:SolidPeso molecular:233.22Phosal 50 PG
CAS:<p>Phosal 50 PG is a co-solvent used as an emulsifier and stabilizer in the pharmaceutical and cosmetic industries.Phosal 50 PG is used as a dietary supplement.</p>Pureza:98%Forma y color:Solid3-Methylcrotonylglycine
CAS:<p>3-Methylcrotonylglycine is an acyl glycine, a normal amino acid metabolite found in urine.</p>Fórmula:C7H11NO3Pureza:98%Forma y color:SolidPeso molecular:157.17HT-2 Toxin
CAS:<p>HT-2 Toxin, a deacetylated metabolite of T-2 toxin, impairs protein synthesis and hinders cell proliferation in plants.</p>Fórmula:C22H32O8Pureza:98%Forma y color:SolidPeso molecular:424.49Ref: TM-T13726
Producto descatalogadoCanagliflozin-d4
CAS:<p>Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.</p>Fórmula:C24H25FO5SPureza:98%Forma y color:SolidPeso molecular:448.54Ref: TM-T10669
Producto descatalogadoPIH
CAS:<p>PIH inhibits ciliogenesis by destabilizing microtubules and blocking Hh signaling, hindering cilia formation and alpha-tubulin disassembly.</p>Fórmula:C20H19N5SPureza:98%Forma y color:SolidPeso molecular:361.46Cysteinylglycine TFA
CAS:<p>Cysteinylglycine TFA is an endogenous metabolite. It is used in disease diagnosis.</p>Fórmula:C7H11F3N2O5SForma y color:SolidPeso molecular:292.23(Rac)-Rotigotine hydrochloride
CAS:<p>(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.</p>Fórmula:C19H26ClNOSForma y color:SolidPeso molecular:351.93Muzolimine
CAS:<p>Muzolimine: a long-acting, high-capacity diuretic for kidney failure/hypertension; withdrawn due to serious neurological side effects.</p>Fórmula:C11H11Cl2N3OForma y color:SolidPeso molecular:272.13Indium(III) isopropoxide
CAS:<p>Indium(III) Isopropoxide: a catalyst for Oppenauer oxidation, turns benzylic alcohols to aldehydes/ketones.</p>Fórmula:C3H8InOPureza:98%Forma y color:SolidPeso molecular:174.914Ref: TM-T19372
Producto descatalogadoValiloxibic acid
CAS:<p>Valiloxibic acid is a prodrug for GHB, a natural psychoactive neurotransmitter and weak GABAB agonist.</p>Fórmula:C9H17NO4Forma y color:SolidPeso molecular:203.238(S)-Rasagiline
CAS:<p>(S)-Rasagiline is rasagiline S-isomer, and is an agent of anti-Parkinson.</p>Fórmula:C12H13NForma y color:SolidPeso molecular:171.24Ref: TM-T13252
Producto descatalogado2-Nitrosopyridine
CAS:<p>2-Nitrosopyridine: used in antibiotic synthesis, Click/Diels-Alder reactions, excellent dienophile.</p>Fórmula:C5H4N2OForma y color:SolidPeso molecular:108.1Golgicide A-1
CAS:<p>Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction.</p>Fórmula:C17H14F2N2Forma y color:SolidPeso molecular:284.31Loviride
CAS:<p>Loviride, a reverse transcriptase inhibitor with IC50 of 0.3 μM, blocks HIV-1/2 and SIV in MT-4 cells.</p>Fórmula:C17H16Cl2N2O2Forma y color:SolidPeso molecular:351.23Ref: TM-T15776
Producto descatalogado5-OxoETE
CAS:<p>5-OxoETE, a dehydrogenase-oxidized 5-HETE, raises neutrophil Ca²⁺ (EC50=2nM) & drives eosinophil migration & MAPK pathway.</p>Fórmula:C20H30O3Pureza:98.59%Forma y color:SolidPeso molecular:318.45Aniline-2,4-diphosphonic acid tetraethyl ester;
CAS:<p>Intermediates and building blocks - phosphorous compounds; nucleophile</p>Fórmula:C14H25NO6P2Forma y color:SolidPeso molecular:365.3L-690330
CAS:<p>L-690330 inhibits human/bovine inositol monophosphatase; Ki: 0.19-0.42 μM. 10x potency vs. mouse/rat IMPase.</p>Fórmula:C8H12O8P2Forma y color:SolidPeso molecular:298.12Ref: TM-T15685
Producto descatalogadoSIRT-IN-3
CAS:<p>SIRT-IN-3: potent SIRT1 inhibitor (IC50=17μM), 4x selective over SIRT2, 14x over SIRT3 (IC50s: 74μM & 235μM).</p>Fórmula:C13H12N2OForma y color:SolidPeso molecular:212.25STING agonist-23
CAS:<p>CF502 (STING agonist-23) is a non-nucleotide that activates STING pathway, boosts immune responses, and shows activity against SARS-CoV.</p>Fórmula:C33H35N13O4Forma y color:SolidPeso molecular:677.72(S,S)-Valifenalate
CAS:<p>(S,S)-Valifenalate is an acylamino acid fungicide and is used to control a wide range of fungi belonging to the class of Oomycetes.</p>Fórmula:C19H27ClN2O5Forma y color:SolidPeso molecular:398.88TD-106
CAS:<p>TD-106 is a modulator of cereblon (CRBN), and can be used for targeted protein degradation. BRD4 PROTACs with TD-106 induce BRD4 degradation.</p>Fórmula:C12H11N5O3Pureza:98%Forma y color:SolidPeso molecular:273.25Ref: TM-T13104
Producto descatalogadoDeoxypseudouridine
CAS:<p>Deoxypseudouridine is a nucleotide analog.</p>Fórmula:C9H12N2O5Forma y color:SolidPeso molecular:228.2Ref: TM-T13645
Producto descatalogadoAlminoprofen
CAS:<p>Alminoprofen: NSAID; reduces anaphylactic bronchoconstriction at 30 mg/kg intraduodenally.</p>Fórmula:C13H17NO2Forma y color:SolidPeso molecular:219.283-Hydroxyhippuric acid
CAS:<p>3-Hydroxyhippuric acid is an acyl glycine, which are normally minor metabolites of fatty acids.</p>Fórmula:C9H9NO4Forma y color:SolidPeso molecular:195.17GRK2 Inhibitor
CAS:<p>GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).</p>Fórmula:C12H9NO6Forma y color:SolidPeso molecular:263.2N-Octylmaleimide
CAS:<p>N-Octylmaleimide is an alkylmaleimide, which can inhibit rat liver glucose 6-phosphatase.</p>Fórmula:C12H19NO2Forma y color:SolidPeso molecular:209.287-Methoxy-1-tetralone
CAS:<p>7-Methoxy-1-tetralone may have insecticidal activity.</p>Fórmula:C11H12O2Pureza:99.93%Forma y color:White CrystalPeso molecular:176.21Elamipretide
CAS:<p>Elamipretide (SS-31, MTP-131, Bendavia) is a mitochondria-focused peptide that curbs toxic ROS and stabilizes cardiolipin.</p>Fórmula:C32H49N9O5Pureza:98.53% - 99.85%Forma y color:SolidPeso molecular:639.79Desidustat
CAS:<p>Desidustat is an inhibitor of HIF hydroxylase.</p>Fórmula:C16H16N2O6Pureza:98%Forma y color:SolidPeso molecular:332.31Rosmanol
CAS:<p>Rosmanol has antioxidant, anti-inflammatory, CNS effects; induces apoptosis in cancer cells; modulates GABAA receptors.</p>Fórmula:C20H26O5Pureza:98.82% - 99.79%Forma y color:SolidPeso molecular:346.42Oxindole
CAS:<p>Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.</p>Fórmula:C8H7NOPureza:99.34%Forma y color:Off-White Crystalline PowderPeso molecular:133.15AM-2232
CAS:<p>AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.</p>Fórmula:C24H20N2OPureza:99.37%Forma y color:SolidPeso molecular:352.43Cebranopadol
CAS:<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Fórmula:C24H27FN2OPureza:98.32% - 99.78%Forma y color:SolidPeso molecular:378.48L-(+)-Abrine
CAS:<p>L-(+)-Abrine (L-N-Methyltryptophan) is a toxic protein found in the jequirity seed.,can be used as a biomarker for abrin exposure.</p>Fórmula:C12H14N2O2Pureza:98.71% - ≥95%Forma y color:White PowderPeso molecular:218.25Compound T69202(SC)
CAS:<p>NBQX (FG9202), an AMPA/kainate receptor blocker, counters glutamate toxicity; water-soluble as disodium salt, has anticonvulsant properties.</p>Fórmula:C12H6N4Na2O6SForma y color:SolidPeso molecular:380.2415Ref: TM-T69202
Producto descatalogadoMTP 131 acetate
CAS:<p>MTP 131 (acetate) is a small mitochondrially-targeted tetrapeptide.</p>Fórmula:C34H53N9O7Pureza:99.9%Forma y color:SolidPeso molecular:699.84Danoprevir sodium
CAS:<p>Danoprevir sodium is an NS3/4A protease inhibitor used in the treatment of Hepatitis C</p>Fórmula:C35H45FN5NaO9SForma y color:SolidPeso molecular:753.82Elamipretide 2TFA
CAS:<p>Elamipretide 2TFA (RX-31 2TFA) is a novel mitochondrion-targeted antioxidant.</p>Fórmula:C36H51F6N9O9Pureza:>99.99%Forma y color:SolidPeso molecular:867.84Ref: TM-T8831
Producto descatalogadoEthyl 4-hydroxyphenylacetate
CAS:<p>Ethyl 4-hydroxyphenylacetate is a selective inhibitor of monoamine oxidase A.</p>Fórmula:C10H12O3Pureza:99.89%Forma y color:Slightly Yellow LiquidPeso molecular:180.2SR17018
CAS:<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Fórmula:C19H18Cl3N3OPureza:99.89%Forma y color:SolidPeso molecular:410.72Decyl-TPP bromide
CAS:<p>Decyl-TPP bromide ((1-Decyl)triphenylphosphonium bromide) may be used as an intermediate for chemical synthesis and an inactive control or as a reference to</p>Fórmula:C28H36BrPPureza:98%Forma y color:SolidPeso molecular:483.46CTB
CAS:<p>CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.</p>Fórmula:C16H13ClF3NO2Pureza:99.82%Forma y color:SolidPeso molecular:343.73Lupinine
CAS:<p>Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin.</p>Fórmula:C10H19NOPureza:99.95%Forma y color:SolidPeso molecular:169.26p-Toluic Acid
CAS:<p>p-Toluic Acid (4-Methylbenzoic acid) belongs to the class of organic compounds known as benzoic acids. 4-Methylbenzoic acid has been primarily detected in saliva. Within the cell, 4-methylbenzoic acid is primarily located in the cytoplasm.</p>Fórmula:C8H8O2Pureza:99.44%Forma y color:Physical Description White Powder Sublimes (Ntp 1992)Peso molecular:136.15Dimethylamine hydrochloride
CAS:<p>Dimethylamine hydrochloride, found in urine, comes from food compound TMAO and NO synthesis inhibitor ADMA, processed by DDAH enzyme.</p>Fórmula:C2H8ClNPureza:98% - 99.89%Forma y color:White Solid CrystallinePeso molecular:81.542-Methyl-5-HT hydrochloride
CAS:<p>2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.</p>Fórmula:C11H15ClN2OPureza:98%Forma y color:SolidPeso molecular:226.74-Hydroxy-6-methylcoumarin
CAS:<p>4-Hydroxy-6-methylcoumarin (4-HMC) is a naturally occurring phenolic compound, a derivative of coumarin, found in a variety of plants, fungi, and bacteria. It has anti-inflammatory and anti-tumor activity.4-HMC is used as a flavoring agent, preservative and antioxidant in the food industry.</p>Fórmula:C10H8O3Pureza:99.95%Forma y color:White PowderPeso molecular:176.17Coumaran
CAS:<p>Coumaran (2,3-Dihydrobenzofuran) is an acetylcholinesterase (AChE) inhibitor isolated from leaves of L. camara. Coumaran(2,3-Dihydrobenzofuran) can be used as a biopesticide. 2,3-dihydrobenzofuran is a member of the class of 1-benzofurans that is the 2,3-dihydroderivative of benzofuran. It has a role as a metabolite.</p>Fórmula:C8H8OPureza:99.61%Forma y color:LiquidPeso molecular:120.15Sculponeatin O
CAS:<p>Sculponeatin O may have protective effects on the lipid peroxidation-damaged live cells.</p>Fórmula:C28H40O4Pureza:95.00%Forma y color:SolidPeso molecular:440.61NLX-204 hydrochloride(2170405-10-2 free base)
<p>NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).</p>Fórmula:C20H23Cl2F2N3O2Pureza:99.59%Forma y color:SolidPeso molecular:446.32Elamipretide Triacetate
CAS:<p>Elamipretide TriTFA, a tetrapeptide, targets mitochondria, associates with cardiolipin, studied for treating Leber's Optic Neuropathy.</p>Fórmula:C38H61N9O11Pureza:>99.99%Forma y color:SolidPeso molecular:819.944-Methoxycoumarine
CAS:<p>4-Methoxycoumarine has antitumour effects.</p>Fórmula:C10H8O3Pureza:99.88%Forma y color:SolidPeso molecular:176.17TFLLR-NH2 2TFA(197794-83-5(free base))
<p>TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).</p>Fórmula:C35H55F6N9O10Pureza:99.56%Forma y color:SolidPeso molecular:875.87Isonicotinic acid
CAS:<p>Isonicotinic acid is a metabolite of Isoniazid.Isonicotinic acid is a useful isomer of nicotinic acid. Isoniazid is converted to Isonicotinic acid by hydrazinolysis, with the biotransformation also to be catalyzed by cytochrome P450 enzymes, such as CYP2C.</p>Fórmula:C6H5NO2Pureza:99.68%Forma y color:White To Off-White Crystalline SolidPeso molecular:123.114-Hydroxybenzyl cyanide
CAS:<p>4-Hydroxybenzyl cyanide (4-Hydroxyphenylacetonitrile) shows strong antioxidative activity.</p>Fórmula:C8H7NOPureza:98.13%Forma y color:Light Brown SolidPeso molecular:133.1510Z-Nonadecenoic acid
CAS:<p>10Z-Nonadecenoic acid is a long-chain fatty acid with anti-tumor activity.</p>Fórmula:C19H36O2Pureza:99.43%Forma y color:SolidPeso molecular:296.49Tropinone
CAS:<p>Tropinone used as an intermediate in the synthesis of atropine sulfate, and is a decane alkaloid.</p>Fórmula:C8H13NOPureza:99.90%Forma y color:Beige To Brown Crystalline PowderPeso molecular:139.19Pamoic acid
CAS:<p>Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.</p>Fórmula:C23H16O6Pureza:99.99%Forma y color:Fine Yellow PowderPeso molecular:388.37SR-4370
CAS:<p>SR-4370 is an HDAC inhibitor. SR- 4370 exhibited IC50 values of 0.5 μM, 0.1 μM and 0.06 μM towards HDAC1, HDAC2 and HDAC3, resp.</p>Fórmula:C17H18F2N2OPureza:99.50%Forma y color:SolidPeso molecular:304.33IGFBP-1 Protein, Rat, Recombinant
<p>IGF-binding proteins prolong the half-life of the IGFs and have been shown to either inhibit or stimulate the growth promoting effects of the IGFs on cell culture. They alter the interaction of IGFs with their cell surface receptors. Promotes cell migration. IGFBP-1 Protein, Rat, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.9 kDa and the accession number is P21743.</p>Peso molecular:26.9 kDa (predicted)ARGX-112
CAS:<p>Temtokibart is a humanized IgG1 λ2 antibody that specifically targets IL22RA1, and is expressed by cells that are deficient in the glutamine synthetase gene.</p>Forma y color:Odour LiquidCOR-001
CAS:<p>Ziltivekimab (COR-001) is a human IL-6 antibody, lowers CRP, and may treat inflammation and heart issues in CKD.</p>Pureza:95%Forma y color:Odour LiquidOkadaic acid
CAS:<p>Okadaic acid, a polyether marine toxin, is a highly potent and selective protein phosphatase (PP) inhibitor.</p>Fórmula:C44H68O13Pureza:98%Forma y color:White Crystals Or PowderPeso molecular:805DprE1-IN-8
CAS:<p>DprE1-IN-8 is a potent inhibitor of DprE1, exhibiting an IC50 of less than 0.75 μM.</p>Fórmula:C19H12F3N5O4SPureza:98%Forma y color:SolidPeso molecular:463.39Ref: TM-T79628
Producto descatalogado(S)-Coriolic acid
CAS:<p>(S)-Coriolic acid, a 15-LOX metabolite and signaling molecule, modulates cell growth, tumor adhesion, receptor expression, and can cause mitochondrial damage.</p>Fórmula:C18H32O3Pureza:97.67% - 98.04%Forma y color:SolidPeso molecular:296.44D(-)-Octopamine CSA salt
CAS:<p>D(-)-Octopamine CSA salt is an agonist of octopamine receptors.</p>Fórmula:C18H27NO6SPureza:98%Forma y color:SolidPeso molecular:385.48Anti-NASH agent 1
CAS:<p>Anti-NASH Agent 1 (Compound 3d), derived from Elafibranor, serves as a strong PPAR-α/δ agonist aimed at treating nonalcoholic steatohepatitis (NASH).</p>Fórmula:C26H33NO4Pureza:98%Forma y color:SolidPeso molecular:423.54Ref: TM-T79454
Producto descatalogadoCH-100
CAS:<p>CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.</p>Fórmula:C14H22ClNO3Forma y color:SolidPeso molecular:287.78SR14150
CAS:<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Fórmula:C21H30N2OPureza:98%Forma y color:SolidPeso molecular:326.48GR 218,231
CAS:<p>GR 218,231 is a selective antagonist of D3 dopamine receptor.</p>Fórmula:C24H33NO3SPureza:98%Forma y color:SolidPeso molecular:415.59Benzovindiflupyr
CAS:<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Fórmula:C18H15Cl2F2N3OForma y color:SolidPeso molecular:398.23UBP1112
CAS:<p>group III mGlu receptor antagonist</p>Fórmula:C10H14NO5PPureza:98%Forma y color:SolidPeso molecular:259.2Cebranopadol ((1α,4α)stereoisomer)
CAS:<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Fórmula:C24H27FN2OPureza:98%Forma y color:SolidPeso molecular:378.48IDX-375
CAS:<p>IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.</p>Fórmula:C29H50N5O7PSPureza:98%Forma y color:SolidPeso molecular:643.78SB251023
CAS:<p>SB251023 is an agonist of β3-adrenoceptor.</p>Fórmula:C28H34NO6PForma y color:SolidPeso molecular:511.55BChE-IN-17
CAS:<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Fórmula:C23H23BrN2O4S2Forma y color:SolidPeso molecular:535.47Glutaminyl Cyclase Inhibitor 4
CAS:<p>Glutaminyl Cyclase Inhibitor 4 is a potent, selective glutaminyl cyclase (QC) inhibitor (IC50: 6.1 nM). It is a potent anti-Alzheimer’s agent.</p>Fórmula:C22H33N5O3Pureza:98%Forma y color:SolidPeso molecular:415.53Saxitoxinol
CAS:<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Fórmula:C10H17N7O3Pureza:98%Forma y color:SolidPeso molecular:283.29Ref: TM-T68748
Producto descatalogadoAKOS-22
CAS:<p>AKOS-22: potent VDAC1 inhibitor, Kd=15.4 μM; prevents mitochondrial dysfunction and apoptosis.</p>Fórmula:C22H21ClF3N3O3Pureza:98%Forma y color:SolidPeso molecular:467.87Erythrityl Tetranitrate
CAS:<p>Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."</p>Fórmula:C4H6N4O12Forma y color:SolidPeso molecular:302.11PKUMDL-LTQ-301
CAS:<p>PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.</p>Fórmula:C30H28N2O4Pureza:98%Forma y color:SolidPeso molecular:480.55MEN11467
CAS:<p>MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.</p>Fórmula:C38H40N4O3Pureza:>99.99%Forma y color:SolidPeso molecular:600.75FGFR1 inhibitor-10
CAS:<p>FGFR1 inhibitor-10 (Compound 4i), with an IC50 of 28 nM, effectively inhibits FGFR1 phosphorylation.</p>Fórmula:C26H30F3N7O2SPureza:98%Forma y color:SolidPeso molecular:561.62Ref: TM-T79686
Producto descatalogadoAlbuterol stearate
CAS:<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Fórmula:C31H57NO5Pureza:98%Forma y color:SolidPeso molecular:523.799EGFR-IN-82
CAS:<p>EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of 0.09 nM for EGFR L858R/T790M/C797S and 0.06 nM for EGFR Del19/</p>Fórmula:C32H41BrN9O2PPureza:98%Forma y color:SolidPeso molecular:694.6Ref: TM-T78788
Producto descatalogadoCXCR4-IN-1
CAS:<p>CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, applicable for the research of various conditions such as cancer, HIV, diabetic</p>Fórmula:C23H32N6Pureza:98%Forma y color:SolidPeso molecular:392.54Ref: TM-T79059
Producto descatalogadoPL265
CAS:<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Fórmula:C27H35N2O9PPureza:98%Forma y color:SolidPeso molecular:562.55(E)-Crotylbarbital
CAS:<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Fórmula:C10H14N2O3Pureza:99.94%Forma y color:SolidPeso molecular:210.23Trimetoquinol HCl hydrate
CAS:<p>Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.</p>Fórmula:C19H26ClNO6Forma y color:SolidPeso molecular:399.87Aminobutane bisphosphonate
CAS:<p>Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.</p>Fórmula:C4H13NO6P2Forma y color:SolidPeso molecular:233.1Lp-PLA2-IN-16
CAS:<p>Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].</p>Fórmula:C22H17F5N4O3Pureza:98%Forma y color:SolidPeso molecular:480.39Ref: TM-T79076
Producto descatalogadoHBV-IN-34
CAS:<p>HBV-IN-34 (compound 17i) is a potent inhibitor of HBsAg production, demonstrating remarkable in vitro anti-HBV efficacy with EC50 values of 0.018 μM for HBV DNA</p>Fórmula:C21H19F2N7Pureza:98%Forma y color:SolidPeso molecular:407.42Ref: TM-T79469
Producto descatalogadoGacyclidine
CAS:<p>Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.</p>Fórmula:C16H25NSPureza:99.85% - 99.92%Forma y color:SolidPeso molecular:263.44KP372-1
CAS:<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Fórmula:C20H8N12O2Forma y color:SolidPeso molecular:448.36Fosfonet sodium
CAS:<p>Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.</p>Fórmula:C2H4NaO5PForma y color:SolidPeso molecular:162.01JAK2-IN-9
CAS:<p>Compound A8, known as JAK2-IN-9, is a selective JAK2 inhibitor with an IC50 of 5 nM.</p>Fórmula:C20H24N6O2SPureza:98%Forma y color:SolidPeso molecular:412.51Ref: TM-T79581
Producto descatalogadoCK176
CAS:<p>CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.</p>Fórmula:C21H12IN3O2Pureza:98%Forma y color:SolidPeso molecular:465.24
