Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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(3S,4S)-Tivantinib
CAS:<p>(3S,4S)-Tivantinib, a potent and highly selective inhibitor of the receptor tyrosine kinase c-MET, targets GSK3α and GSK3β—two novel enzymes implicated in the</p>Fórmula:C23H19N3O2Forma y color:SolidPeso molecular:369.42L 363851
CAS:<p>L 363851 is a neurokinin B agonist.</p>Fórmula:C38H51N7O7SForma y color:SolidPeso molecular:749.93LY-426965
CAS:<p>LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.</p>Fórmula:C28H38N2O2Forma y color:SolidPeso molecular:434.61CD08108
CAS:<p>CD08108 is a MC1R agonist.</p>Fórmula:C31H38N4O4Forma y color:SolidPeso molecular:530.66α7β1 integrin modulator-1
CAS:<p>α7β1 Integrin Modulator-1 is a potent modulator with research potential for muscular dystrophy [1].</p>Fórmula:C23H29N3O6SPureza:98%Forma y color:SolidPeso molecular:475.56β-Tocotrienol
CAS:<p>Beta-Tocotrienol to serve as a new anticancer agent for treating human lung and brain cancers.</p>Fórmula:C28H42O2Pureza:98%Forma y color:SolidPeso molecular:410.63Akt-I-1,2
CAS:<p>Akt-I-1,2 is a selective inhibitor of Akt1 and Akt2.</p>Fórmula:C23H22ClN3Pureza:99.95%Forma y color:SolidPeso molecular:375.89PSMA-Val-Cit-PAB-MMAE
CAS:<p>PSMA-Val-Cit-PAB-MMAE is a novel PSMA-targeted small-molecule conjugate leveraging monomethyl auristatin E (MMAE) for prostate cancer chemotherapy.</p>Fórmula:C114H165ClN20O26Forma y color:SolidPeso molecular:2267.1T338C Src-IN-1
CAS:<p>T338C Src-IN-1 is a potent mutant-Src T338C inhibitor(T338C,IC50=111 nM relative to WT c-Src (10-fold increase)).</p>Fórmula:C17H20N6O2SPureza:98%Forma y color:SolidPeso molecular:372.44Gly-Gly-Phe-Gly-NH-CH2-O-CH2COOH
CAS:<p>Gly-Gly-Phe-Gly-NH-CH2-O-CH2COOH is an ADC linker utilized in the synthesis of drug-linker conjugates specific to ADCs, notably for creating Deruxtecan, a</p>Fórmula:C18H25N5O7Forma y color:SolidPeso molecular:423.42SKF-86002 dihydrochloride
CAS:<p>p38 MAP kinase inhibitor</p>Fórmula:C16H14Cl2FN3SPureza:98%Forma y color:SolidPeso molecular:370.27A-849519
CAS:<p>A-849519 is a reversible MetAP2 inhibitor with anti-angiogenic and anticancer properties, tested against prostate cancer and compared to TNP-470.</p>Fórmula:C22H25FN2O4SForma y color:SolidPeso molecular:432.51MN-05
CAS:<p>MN-05 is a neuroprotective and vasodilator for neurodegenerative diseases.</p>Fórmula:C13H22N2O3Forma y color:SolidPeso molecular:254.33AAK1-IN-3
CAS:<p>AAK1-IN-3: Brain-penetrant AAK1 inhibitor for neuropathic pain research; IC50=11 nM.</p>Fórmula:C20H20N4Forma y color:SolidPeso molecular:316.4Palinavir
CAS:<p>Palinavir is an antiviral, it inhibits HIV-1 protease.</p>Fórmula:C41H52N6O5Pureza:98%Forma y color:SolidPeso molecular:708.89CUR61414
CAS:<p>CUR61414 is a cell-permeable inhibitor of Hedgehog signaling pathway (IC50 =100-200 nM) and selectively binds to smoothened (Ki = 44 nM).</p>Fórmula:C31H42N4O5Pureza:97.34% - 98%Forma y color:SolidPeso molecular:550.69SC-50605
CAS:<p>SC-50605 is a second-generation LTB4 receptor antagonist.</p>Fórmula:C30H35NO6SForma y color:SolidPeso molecular:537.67Methyl 2-amino-5-bromobenzoate
CAS:<p>Methyl 2-amino-5-bromobenzoate (Methyl 5-Bromoanthranilate) is an HCV NS5b RNA polymerase inhibitor with antimicrobial activity.</p>Fórmula:C8H8BrNO2Pureza:98.05%Forma y color:SolidPeso molecular:230.06PD-1/PD-L1-IN-26
CAS:<p>PD-1/PD-L1-IN-26 is a strong inhibitor with IC50 of 0.0380 μM that may boost immune response in cancer by aiding CD4+ T cell entry to tumors.</p>Fórmula:C43H52N4O8Pureza:98%Forma y color:SolidPeso molecular:752.89MDK-0757
CAS:<p>MDK-0757 is a novel inhibitor of heat shock protein 90 (Hsp90).</p>Fórmula:C20H18FN5OPureza:98%Forma y color:SolidPeso molecular:363.39LY2922083
CAS:<p>LY2922083: Potent, selective GPR40 agonist; lowers glucose, boosts insulin and GLP-1.</p>Fórmula:C31H33NO3SForma y color:SolidPeso molecular:499.66Falcarindiol
CAS:<p>Falcarindiol: Activates PPARγ, boosts ABCA1, induces apoptosis/autophagy, has anti-inflammatory/anticancer effects.</p>Fórmula:C17H24O2Forma y color:SolidPeso molecular:260.37Xenognosin
CAS:<p>Xenognosin is a biochemical.</p>Fórmula:C16H16O3Forma y color:SolidPeso molecular:256.3Celiprolol hydrochloride
CAS:<p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>Fórmula:C20H33N3O4·HClForma y color:White Crystalline SolidPeso molecular:415.96HBV-IN-8
CAS:<p>HBV-IN-6 is a potent inhibitor of HBV (EC50: 287.9 nM).</p>Fórmula:C21H25ClFN5O5S2Forma y color:SolidPeso molecular:546.04Biotin-PEG7-Maleimide
CAS:<p>Biotin-PEG7-Maleimide is a biotinylation agent that selectively binds to thiol (SH) groups and is utilized in the synthesis of Drug-Linker Conjugates for</p>Fórmula:C33H55N5O12SForma y color:SolidPeso molecular:745.88ER degrader 1
CAS:<p>ER degrader 1 targets estrogen receptor, crucial for cell regulation; shows promise in cancer therapy. (Patent WO2021139756A1, compound 11)</p>Fórmula:C26H32F4N4O3Forma y color:SolidPeso molecular:524.55CR-6086
CAS:<p>CR6086: potent EP4 antagonist with DMARD effects, low Ki (16.6 nM), and specific anti-inflammatory action.</p>Fórmula:C26H27F3N2O3Forma y color:SolidPeso molecular:472.5CHF 2819
CAS:<p>CHF 2819 is a novel orally active acetylcholinesterase inhibitor (AChE) developed for the treatment of Alzheimer's disease (AD).</p>Fórmula:C21H26ClN3O3Forma y color:SolidPeso molecular:403.9(+)-Apogossypol
CAS:<p>(+)-Apogossypol is an antagonist of pan-BCL-2. (+)-Apogossypol binds to Mcl-1(Bcl-2 and Bcl-xL with EC50s of 2.6, 2.8 and 3.69 μM, respectively).</p>Fórmula:C28H30O6Pureza:98%Forma y color:SolidPeso molecular:462.53DU172
CAS:<p>DU172 is the tyrosine-targeted covalent adenosine A1 receptor antagonist.</p>Fórmula:C24H30FN5O5SForma y color:SolidPeso molecular:519.59eIF4A3-IN-17
CAS:<p>eIF4A3-IN-17, a silvestrol analogue, disrupts eIF4F assembly; EC50: 0.9-15 nM. Used in cancer pathogenesis research.</p>Fórmula:C28H25NO7Forma y color:SolidPeso molecular:487.5AAK1-IN-4
CAS:<p>AAK1-IN-4 selectively inhibits AAK1 with IC50 of 4.6 nM; penetrates CNS, oral bioactive, potential for studying neuropathic pain.</p>Fórmula:C20H28N4O3Forma y color:SolidPeso molecular:372.46A 53693
CAS:<p>A 53693 is a rigid catecholamine and a selective adrenergic agonist. A 53693 has affinity to certain alpha receptor subtypes in rat alpha-2 receptors.</p>Fórmula:C13H17NO2Pureza:98%Forma y color:SolidPeso molecular:219.28Streptovitacin A
CAS:<p>Streptovitacin A boosts growth inhibition against fungi.</p>Fórmula:C15H23NO5Pureza:98%Forma y color:SolidPeso molecular:297.35Casein Kinase II Inhibitor IV
CAS:<p>Casein kinase II inhibitor IV is an effective small molecule inducer, which can be used to induce epidermal keratinocyte differentiation.</p>Fórmula:C24H23N5O3Pureza:99.65% - 99.75%Forma y color:SolidPeso molecular:429.47KRAS G12C inhibitor 53
CAS:<p>KRAS G12C inhibitor 53 (Compound 1) is a KRAS G12C inhibitor.</p>Fórmula:C21H14ClF2N5O2Forma y color:SolidPeso molecular:441.82WAY-612453
CAS:<p>WAY-612453 is an active compound utilized in researching amyloid diseases and synucleinopathies.</p>Fórmula:C9H8Cl2N4SForma y color:SolidPeso molecular:275.16Valtorcitabine dihydrochloride
CAS:<p>Valtorcitabine dihydrochloride, a DNA polymerase inhibitor, is used potentially for the treatment of HBV infection.</p>Fórmula:C14H24Cl2N4O5Forma y color:SolidPeso molecular:399.27K145 hydrochloride
CAS:<p>K145 hydrochloride is a selective sphk2 inhibitor with substrate competitiveness and oral activity, with IC50 of 4.3 µM and Ki of 6.4 µM.</p>Fórmula:C18H25ClN2O3SPureza:99.8%Forma y color:SolidPeso molecular:384.92PDE1-IN-1
CAS:<p>PDE1-IN-1 boosts cAMP/cGMP, enhancing neuronal plasticity and neuroprotection, with potential as a neurological therapeutic.</p>Fórmula:C32H31N5OForma y color:SolidPeso molecular:501.62BMS-654457
CAS:<p>BMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa; Kis: 0.2 and 0.42 nM for human and rabbit FXIa).</p>Fórmula:C36H37N5O4Pureza:98%Forma y color:SolidPeso molecular:603.71MC-EVCit-PAB-MMAE
CAS:<p>MC-EVCit-PAB-MMAE (Linker-Payload 11), a conjugate utilized in antibody-drug conjugates (ADCs), comprises the MC-EVCit-PAB linker attached to the powerful</p>Fórmula:C73H112N12O18Forma y color:SolidPeso molecular:1445.74Arrhythmias-Targeting Compound 1
CAS:<p>Arrhythmias-Targeting Compound 1 is a compound. It is used in the research of arrhythmias.</p>Fórmula:C22H32N4O2Pureza:98%Forma y color:SolidPeso molecular:384.52ALK/EGFR-IN-2
CAS:<p>ALK/EGFR-IN-2 is a potent dual inhibitor targeting ALK and EGFR, promoting apoptosis and G0/G1 cell cycle arrest in cancer cells.</p>Fórmula:C27H34ClN7O3SForma y color:SolidPeso molecular:572.12Docebenone
CAS:<p>Docebenone is a selective and orally active inhibitor of 5-LO.</p>Fórmula:C21H26O3Forma y color:SolidPeso molecular:326.43L-159884
CAS:<p>L-159884 is a radiolabelled, nonpeptide angiotensin II antagonist that is useful for angiotensin II, AT1 receptor imaging</p>Fórmula:C31H30N4O4SForma y color:SolidPeso molecular:554.66GTPγS tetralithium
CAS:<p>GTPγS tetralithium (Guanosine 5'-[γ-thio]triphosphate tetralithium) is a G-protein activator and a non-hydrolyzable GTP analog.</p>Fórmula:C10H12Li4N5O13P3SPureza:75%Forma y color:SolidPeso molecular:562.98Clavulanic Acid Methyl Ester
CAS:<p>Clavulanic Acid Methyl Ester is a substituted Clavulanic acid and β-lactamase inhibitor.</p>Fórmula:C9H11NO5Forma y color:SolidPeso molecular:213.19PDE4-IN-8
CAS:<p>PDE4-IN-8 is a potent PDE4 inhibitor with IC50 0.93 nM for PDE4B2 and minor impact on IL13, IL4, IFNy (IC50: 4.04, 36.33, 2394 nM).</p>Fórmula:C18H22BNO4Forma y color:SolidPeso molecular:327.18
