Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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Indeloxazine hydrochloride
CAS:<p>Indeloxazine HCl: Serotonin releaser, NE reuptake inhibitor, NMDA antagonist; antidepressant that boosts acetylcholine in rats.</p>Fórmula:C14H18ClNO2Pureza:98%Forma y color:SolidPeso molecular:267.75GGTI2417
CAS:<p>GGTI2417 blocks Geranylgeranyltransferase I, targeting RalB for apoptosis and RalA to stop growth.</p>Fórmula:C24H33N5O4Forma y color:SolidPeso molecular:455.55Uplarafenib
CAS:<p>Uplarafenib (B-Raf IN 10), a potent BRAF inhibitor (IC50: 50-100 nM), exhibits antitumor effects on solid cancers.</p>Fórmula:C22H21F3N4O4SPureza:99.85%Forma y color:SolidPeso molecular:494.49PPO-IN-2
CAS:<p>PPO-IN-2 is a protoporphyrinogen IX oxidase inhibitor, exhibiting a Ki value of 16 nM [1].</p>Fórmula:C17H15ClFN3O2S2Forma y color:SolidPeso molecular:411.9Heclin
CAS:<p>Heclin is an inhibitor of HECT E3 ubiquitin ligase that acts by inhibiting Smurf2, Nedd4, and WWP1 with IC50 values of 6.8, 6.3, and 6.9 μM, respectively.</p>Fórmula:C17H17NO3Pureza:95.79%Forma y color:SolidPeso molecular:283.32ISPA-28
CAS:<p>ISPA-28: reversible PSAC antagonist via direct CLAG3 binding.</p>Fórmula:C21H24N6O3Forma y color:SolidPeso molecular:408.45BMS-695735
CAS:<p>BMS-695735: benzimidazole, inhibits IGF-1 receptor, broad antitumor effects, affects CYP3A4, low solubility, binds plasma proteins.</p>Fórmula:C26H31ClFN7OForma y color:SolidPeso molecular:512.021,8-Dichloroanthraquinone
CAS:<p>1,8-Dichloroanthraquinone, a derivative of anthraquinone, effectively inhibits sulfide production in sulfate-reducing bacteria [1].</p>Fórmula:C14H6Cl2O2Forma y color:SolidPeso molecular:277.1ROCK-IN-8
CAS:<p>ROCK-IN-8 (Example 4), a ROCK inhibitor, exhibits anti-inflammatory properties and is suitable for respiratory and gastro-intestinal disease research,</p>Fórmula:C30H25FN4O4SPureza:98%Forma y color:SolidPeso molecular:556.61SCS
CAS:<p>SCS is a GABAA receptor antagonist.</p>Fórmula:C14H12N2O3Pureza:99.73%Forma y color:SolidPeso molecular:256.26NITD008
CAS:<p>NITD008 (7-Deaza-2'-C-acetylene-adenosine) is an adenosine nucleoside inhibitor with antiviral activity that inhibits dengue and Zika viruses.</p>Fórmula:C13H14N4O4Pureza:98.04%Forma y color:SolidPeso molecular:290.27Limocrocin
CAS:<p>Limocrocin is an inhibitor of reverse transcriptase.</p>Fórmula:C26H26N2O6Pureza:98%Forma y color:SolidPeso molecular:462.49SHP2/CDK4-IN-1
CAS:<p>SHP2/CDK4-IN-1: dual inhibitor, oral, potent (IC50: SHP2 4.3 nM, CDK4 18.2 nM), hinders TNBC growth, strong antitumor effects in mice.</p>Fórmula:C33H35ClF2N10OSForma y color:SolidPeso molecular:693.21FXR antagonist 1
CAS:<p>"Oral FXR antagonist 1 selectively blocks intestinal FXR, with IC50 of 2.1 μM, aiding in NASH research by improving liver health."</p>Fórmula:C36H59NO5Forma y color:SolidPeso molecular:585.86INX-SM-6
CAS:<p>INX-SM-6, a chemical compound, serves as a targeted delivery vehicle for anti-inflammatory agents and has shown efficacy in suppressing LPS-induced IL-1β</p>Fórmula:C32H36N2O6SForma y color:SolidPeso molecular:576.7WAY-300570
CAS:<p>N-(4-Chlorophenyl)-3-(4-oxo-5-(thiophen-2-ylmethylene)-2-thioxothiazolidin-3-yl)propanamide is an active chemical compound characterized by its complex</p>Fórmula:C17H13ClN2O2S3Forma y color:SolidPeso molecular:408.95EGFR-IN-33
CAS:<p>EGFR-IN-33, a low-toxicity acrylamide, inhibits EGFR, aiding against cancer, especially NSCLC (from WO2021185348A1, comp. 13).</p>Fórmula:C26H25ClN6O2Forma y color:SolidPeso molecular:488.97KY386
CAS:<p>KY386 is a potent and selective DHX33 helicase inhibitor with an IC50 value of 19 nM.</p>Fórmula:C21H19N5O2SForma y color:SolidPeso molecular:405.47FTI 276
CAS:<p>FTI-276 is an inhibitor of protein farnesyltransferase (PFT) (IC50s: 0.9 and 0.5 nM for Plasmodium falciparum and human).</p>Fórmula:C21H27N3O3S2Pureza:98%Forma y color:SolidPeso molecular:433.59DQP-26
CAS:<p>DQP-26, a potent negative allosteric modulator of NMDA receptors (NMDARs), exhibits IC50 values of 0.77 μM for GluN2C and 0.44 μM for GluN2D subunits,</p>Fórmula:C28H21Cl2N3O4Pureza:98%Forma y color:SolidPeso molecular:534.39DGKα-IN-7
CAS:<p>DGKα-IN-7 is a potent DGKα inhibitor with an IC50 value of 6.225 nM and potential applications in cancer research.</p>Fórmula:C23H17F5N6Forma y color:SolidPeso molecular:472.415'-ODMT cEt N-Bzm5 C Phosphoramidite (Amidite)
CAS:<p>5'-ODMT cEt N-Bzm5 C Phosphoramidite is a strong modified nucleic acid analog for antisense oligos.</p>Fórmula:C49H56N5O9PForma y color:SolidPeso molecular:889.97PAK1-IN-1
CAS:<p>PAK1-IN-1: PAK1 inhibitor, IC50 9.8 nM, hinders tumor cell migration and invasion dose-dependently.</p>Fórmula:C26H20ClN5O2Forma y color:SolidPeso molecular:469.92Fiduxosin hydrochloride
CAS:<p>Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.</p>Fórmula:C30H30ClN5O4SForma y color:SolidPeso molecular:592.11PIK-inhibitors
CAS:<p>PIK-inhibitors (MDK34597) is a pan PI3K inhibitors, an analog of PI-103.</p>Fórmula:C19H17N5O2Pureza:96.98%Forma y color:SolidPeso molecular:347.37LAS191859
CAS:<p>LAS191859, a CRTH2 antagonist, IC50: 7.6-15.5nM across species, 21h half-life for sustained in vivo effect.</p>Fórmula:C24H24F3N3O3Pureza:98%Forma y color:SolidPeso molecular:459.46RTI-13951-33
CAS:<p>RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).</p>Fórmula:C28H33N3O3Pureza:98%Forma y color:SolidPeso molecular:459.58PD-1/PD-L1-IN-33
CAS:<p>PD-1/PD-L1-IN-33 (Compound N11), a PD-1/PD-L1 inhibitor, effectively impedes the interaction between PD-1 and PD-L1 with an IC50 of 6.3 nM.</p>Fórmula:C26H27N5OPureza:98%Forma y color:SolidPeso molecular:425.53BAY-784
CAS:<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Fórmula:C29H26ClF4N3O5S2Pureza:98%Forma y color:SolidPeso molecular:672.11KPZ560
CAS:<p>KPZ560, a potent HDAC 1 and HDAC 2 inhibitor, exhibits IC50 values of 12 nM and 68 nM, respectively.</p>Fórmula:C26H21N5O3S2Pureza:98%Forma y color:SolidPeso molecular:515.61Rosoxacin
CAS:<p>Rosoxacin (Acrosoxacin) shows antibacterial activities against a broad spectrum of Gram-negative bacteria including Neisseria gonorrhoeae (MIC90 = 0.03mg/ml).</p>Fórmula:C17H14N2O3Pureza:99.1%Forma y color:SolidPeso molecular:294.3SARS-CoV-2-IN-44
CAS:<p>SARS-CoV-2-IN-44, an inhibitor of SARS-CoV-2, effectively suppresses viral replication with an EC50 value of 0.6μM and exhibits negligible cytotoxicity in Calu-</p>Fórmula:C18H16O5Pureza:98%Forma y color:SolidPeso molecular:312.32MK-1421
CAS:<p>MK-1421 is a potent and selective sstr3 antagonist.</p>Fórmula:C27H24FN9O2Forma y color:SolidPeso molecular:525.54C-6 NBD-dihydro-Ceramide
CAS:<p>C-6 NBD-dihydro-Ceramide, a biologically active, fluorescent analog of short-chain ceramides, features membrane permeability.</p>Fórmula:C30H49N5O6Forma y color:SolidPeso molecular:575.74Acorafloxacin HCl
CAS:<p>Acorafloxacin: broad-spectrum fluoroquinolone antibacterial for acute skin infections and pneumonia.</p>Fórmula:C21H24ClF2N3O4Pureza:98%Forma y color:SolidPeso molecular:455.88STING-IN-7
CAS:<p>STING-IN-7 (compound 21) serves as a potent inhibitor of the stimulator of interferon genes (STING) pathway, demonstrating an inhibitory concentration (IC50) of</p>Fórmula:C16H14ClN3OPureza:98%Forma y color:SolidPeso molecular:299.76CBP/p300-IN-5
CAS:<p>P300/CBP-IN-5 is a potent inhibitor of p300/CBP histone acetyltransferase (IC50 of 18.8 nM).</p>Fórmula:C29H27F5N6O4Pureza:98%Forma y color:SolidPeso molecular:618.55ICMT-IN-25
CAS:<p>ICMT-IN-25 (compound 37) serves as a potent inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting an IC50 value of 0.025 μM [1].</p>Fórmula:C21H26ClNOForma y color:SolidPeso molecular:343.89Tenalisib R Enantiomer
CAS:<p>Tenalisib R Enantiomer is an R enantiomer of Tenalisib .</p>Fórmula:C23H18FN5O2Pureza:98%Forma y color:SolidPeso molecular:415.428-bromo NAD+ sodium
CAS:<p>8-Bromo NAD+ serves as a prodrug for the cyclic ADP-ribose (cADPR) inhibitor, 8-bromo cADPR, undergoing conversion to its active form by the enzyme CD38.</p>Fórmula:C21H25BrN7O14P2·NaForma y color:SolidPeso molecular:764.30SOS1-IN-7
CAS:<p>SOS1-IN-7 (compound 18-p1) is a potent inhibitor of SOS1 and acts on SOS1-G12D (IC50: 20 nM) and SOS1-G12V (IC50: 67 nM).</p>Fórmula:C23H25F3N4O3Forma y color:SolidPeso molecular:462.46PZ-1190
CAS:<p>PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents [1].</p>Fórmula:C27H30N4O2S2Pureza:98%Forma y color:SolidPeso molecular:506.68Chroman 1
CAS:<p>Chroman 1 is a potent inhibitor of ROCK1 (IC50 = 52 pM) and ROCK2 (IC50 = 1 pM).</p>Fórmula:C24H28N4O4Pureza:99.67% - 99.84%Forma y color:SolidPeso molecular:436.5LY-311727
CAS:<p>secreted phospholipase A2 (sPLA2) inhibitor</p>Fórmula:C22H27N2O5PPureza:98%Forma y color:SolidPeso molecular:430.43ent-Entecavir
CAS:<p>Ent-Entecavir, an enantiomeric impurity of Entecavir (an oral HBV drug), inhibits HBV replication as a reverse transcriptase inhibitor.</p>Fórmula:C12H15N5O3Forma y color:SolidPeso molecular:277.28(S,R)-WT IDH1 Inhibitor 2
CAS:<p>(S,R)-WT IDH1 Inhibitor 2: selectively targets mutant IDH1; IC50 - R132G: 2.9 nM, R132C: 3.8 nM, R132H: 4.6 nM, WT: 46 nM; potential for AML treatment.</p>Fórmula:C28H28FN5O3Forma y color:SolidPeso molecular:501.55Moxestrol
CAS:<p>Moxestrol, a synthetic estrogen, treats menopause and menstrual issues in Europe.</p>Fórmula:C21H26O3Pureza:98%Forma y color:SolidPeso molecular:326.43NS5A-IN-3
CAS:<p>NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.</p>Fórmula:C44H44N6O8Pureza:98%Forma y color:SolidPeso molecular:784.86Alpelisib hydrochloride
CAS:<p>Alpelisib hydrochloride (BYL-719) is an oral, selective PI3Kα inhibitor with anticancer properties.</p>Fórmula:C19H23ClF3N5O2SPureza:98%Forma y color:SolidPeso molecular:477.93Acitretin sodium
CAS:<p>Acitretin sodium is a second-generation, systemic retinoid. It is also has been used in the treatment of psoriasis.</p>Fórmula:C21H26NaO3Pureza:98%Forma y color:SolidPeso molecular:349.42
