Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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KAT modulator-1
CAS:<p>KAT modulator-1 (Compound 3), an epigenetics research tool, selectively interacts with the full-length p300 protein but not its catalytic domain [1].</p>Fórmula:C20H36O2Pureza:98%Forma y color:SolidPeso molecular:308.5PARP7-probe-1
CAS:<p>PARP7-probe-1: biotinylated, chemiluminescent PARP7 active site probe for research use.</p>Fórmula:C36H49F3N8O5SForma y color:SolidPeso molecular:762.89BMS-187308
CAS:<p>BMS-187308 is an endothelin-A (ETA) selective antagonist.</p>Fórmula:C21H25N3O3SForma y color:SolidPeso molecular:399.51ICMT-IN-29
CAS:<p>ICMT-IN-29, also known as compound 66, effectively inhibits ICMT with an IC50 value of 0.019 μM [1].</p>Fórmula:C20H27NO2SForma y color:SolidPeso molecular:345.5(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Fórmula:C21H20ClNO6Pureza:98%Forma y color:SolidPeso molecular:417.84EGFR-IN-30
CAS:<p>EGFR-IN-30 is an EGFR inhibitor (IC50: 1-10 nM, <1 nM WT/mutants) with potential in cancer research.</p>Fórmula:C28H33BrN7O2PForma y color:SolidPeso molecular:610.49A-371191
CAS:<p>A-371191 is an antagonist of Bcl-XL.</p>Fórmula:C36H47N5O5S2Pureza:98%Forma y color:SolidPeso molecular:693.9210-Chloroestra-1,4-diene-3,17-dione
CAS:<p>10-Chloroestra-1,4-diene-3,17-dione acts as an estrogen receptor α (ERα) agonist, enhancing reporter gene expression in S.</p>Fórmula:C18H21ClO2Forma y color:SolidPeso molecular:304.80Tomicorat
CAS:<p>Tomicorat is an anti-inflammatory agent.</p>Fórmula:C32H30FNO5Forma y color:SolidPeso molecular:527.58Anticancer agent 86
CAS:<p>Compound 6i, an anticancer agent, exhibits promising activity against breast adenocarcinoma [1].</p>Fórmula:C31H23Cl2N3O5Forma y color:SolidPeso molecular:588.44GLX481304
CAS:<p>GLX481304 is a selective Nox-2 and Nox-4 inhibitor, exhibiting IC50 values of 1.25 μM.</p>Fórmula:C23H29N7OForma y color:SolidPeso molecular:419.52MK-8153
CAS:<p>MK-8153: Selective, potent ROMK inhibitor, orally active, IC50: ROMK EP 5 μM, hERG EP 34 μM; potential diuretic.</p>Fórmula:C24H28N2O6Forma y color:SolidPeso molecular:440.49BRD7-IN-1
CAS:<p>BRD7-IN-1, a BI7273 derivative, forms PROTAC VZ185, targeting BRD7/9 with DC50s of 4.5/1.8 nM via VHL ligand linkage.</p>Fórmula:C22H28Cl2N4O3Pureza:98.95%Forma y color:SolidPeso molecular:467.39Keap1-Nrf2-IN-15
CAS:<p>Keap1-Nrf2-IN-15 (Compound 24a) is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction, displaying IC50 values of 77 nM in a fluorescence</p>Fórmula:C39H35N3O12S2Forma y color:SolidPeso molecular:801.84Androgen receptor degrader-2
CAS:<p>Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].</p>Fórmula:C16H16ClN3O4Pureza:98%Forma y color:SolidPeso molecular:349.77NVP-SAA164
CAS:<p>NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.</p>Fórmula:C36H45N5O5SPureza:98%Forma y color:SolidPeso molecular:659.84TASP 0277308
CAS:<p>NH2-UAMC1110 TFA is an aminobutoxy derivative of UAMC1110 used in the synthesis of FAPI-QS. UAMC1110 is a fibroblast activating protein (fap) inhibitor.</p>Fórmula:C23H28Cl2N6O3SForma y color:SolidPeso molecular:539.48BMT-108908
CAS:<p>BMT-108908 is a Negative Allosteric Modulator. It is selective for the NR2B Subtype of The NMDA Receptor Impair Cognition in Multiple Domains.</p>Fórmula:C22H25FN2O2Forma y color:SolidPeso molecular:368.44ON 108600
CAS:<p>ON 108600 is a chemical inhibitor targeting CK2 (Casein Kinase 2), TNIK, and DYRK1, demonstrating IC50 values of 0.016 μM and 0.007 μM for DYRK1A and DYRK1B, 0.</p>Fórmula:C22H14Cl2N2O6S2Pureza:98%Forma y color:SolidPeso molecular:537.39KRAS G12C inhibitor 51
CAS:<p>KRAS G12C inhibitor 51 is a KRAS G12C inhibitor.</p>Fórmula:C33H35FN6O3Forma y color:SolidPeso molecular:582.67VT-1598 tosylate
CAS:<p>VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.</p>Fórmula:C38H28F4N6O5SForma y color:SolidPeso molecular:756.72CP 154,526
CAS:<p>CP 154,526 is a selective CRF1 receptor antagonist (Ki = 2.7 nM). CP 154,526 blocks CRF-induced activation of adenylate cyclase and the HPA axis.</p>Fórmula:C23H32N4Forma y color:SolidPeso molecular:364.53QM 7184
CAS:<p>QM 7184 is a thiophene analogue of taclamine with potent alpha-adrenoceptor blocking activity.</p>Fórmula:C19H21NSForma y color:SolidPeso molecular:295.44Type II TRK inhibitor 1
CAS:<p>Type II TRK Inhibitor 1 is a potent inhibitor targeting multiple tropomyosin receptor kinase (TRK) fusion protein variants as well as the wild type.</p>Fórmula:C35H33F3N8O3Pureza:98%Forma y color:SolidPeso molecular:670.68(Rac)-Neurodegenerative Disorder-Targeting Compound 1
CAS:<p>(Rac)-Neurodegenerative Disorder-Targeting Compound 1 is a calpain inhibitor.</p>Fórmula:C28H28N4O4Forma y color:SolidPeso molecular:484.55HL23
CAS:<p>HL23 is a histone deacetylase (HDAC) inhibitor that effectively targets hepatocellular carcinoma (HCC).</p>Fórmula:C44H44N2O7Pureza:98%Forma y color:SolidPeso molecular:712.83TrkA-IN-4
<p>TrkA-IN-4, a potent, orally active and allosteric TrkA inhibitor, is a prodrug of TrkA-IN-3 . TrkA-IN-4 exhibits potent antinociceptive effects [1] .</p>Fórmula:C27H21F3N4O5Forma y color:SolidPeso molecular:538.47ML-099
CAS:<p>ML-099 is a pan Ras-related GTPases activator that activates Rac1, Ras, GTP-binding protein (Rab7), Rab2A and cell division cycle 42.</p>Fórmula:C14H13NO2SPureza:99.73%Forma y color:SolidPeso molecular:259.32FXa-IN-1
CAS:<p>FXa-IN-1, an FXa blocker: IC50=3 nM, Ki=0.7 nM, orally available, long half-life, for thrombosis research.</p>Fórmula:C24H18F5N5OForma y color:SolidPeso molecular:487.42Rp-Adenosine-5'-O-(1-thiodiphosphate) sodium
CAS:<p>Rp-Adenosine-5'-O-(1-thiodiphosphate) (Rp-ADP-α-S), a sulfur-containing isomer of the nucleotide derivative ADP-α-S, acts as an inhibitor of phosphorylase</p>Fórmula:C10H12N5O9P2S·3NaForma y color:SolidPeso molecular:509.21TLR8 agonist 5
CAS:<p>TLR8 Agonist 5, exhibiting potent efficacy as a TLR8 agonist, demonstrates an EC50 of 20 nM in HEK-Blue hTLR8, effectively activating the immune response.</p>Fórmula:C31H40N6O5Forma y color:SolidPeso molecular:576.69Org-21465
CAS:<p>Org-21465, a gamma-aminobutyric acid (GABA) receptor agonist, is used potentially for the use of anesthesia.</p>Fórmula:C27H43NO4Pureza:98%Forma y color:SolidPeso molecular:445.63SB-743921 free base
CAS:<p>SB-743921, a kinesin spindle protein (KSP) inhibitor, is used potentially for the treatment of non-Hodgkin's lymphoma (NHL).</p>Fórmula:C31H33ClN2O3Pureza:98%Forma y color:SolidPeso molecular:517.06GIV3727
CAS:<p>GIV3727, a bitter taste receptor hTAS2R antagonist, inhibits the activation of hTAS2R31 by saccharin and acesulfame potassium, effectively diminishing the</p>Fórmula:C12H22O2Forma y color:SolidPeso molecular:198.3BRD4 Inhibitor-23
CAS:<p>BRD4 Inhibitor-23: potent, oral, IC50: BRD4 BD-1 6.21 nM, BD-2 1.44 nM. See WO2022033542A1 Example 1.</p>Fórmula:C22H19F2N3O4SForma y color:SolidPeso molecular:459.47MeOSuc-AAPV-CMK
CAS:<p>MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediated</p>Fórmula:C22H35ClN4O7Forma y color:SolidPeso molecular:502.99Merodantoin
CAS:<p>Merodantoin induces apoptosis in KRAS-mutant cancer cells via ROS-autophagy and Akt pathway.</p>Fórmula:C11H18N2O2SPureza:99.8%Forma y color:SolidPeso molecular:242.34Org 43553
CAS:<p>Org 43553: oral LMW LH-R agonist; targets LH (EC50: 3.7nM) & FSH (EC50: 110nM); useful for endocrine research.</p>Fórmula:C24H30N6O3S2Forma y color:SolidPeso molecular:514.66FT206
CAS:<p>FT206 is a carboxamide inhibitor of ubiquitin-specific protease[1].</p>Fórmula:C25H29N5OSForma y color:SolidPeso molecular:447.6TR antagonist 1
CAS:<p>TR antagonist 1 is a highly potent thyroid hormone receptor (TR) antagonist that can be used to study diseases caused by endocrine abnormalities.</p>Fórmula:C25H23Br2NO4Pureza:99.57%Forma y color:SolidPeso molecular:561.26JTE-952
CAS:<p>JTE-952: oral, selective Type II CSF-1R inhibitor, IC50 = 13 nM for CSF1R, 261 nM for TrkA, effective in mouse arthritis model.</p>Fórmula:C30H34N2O6Pureza:98%Forma y color:SolidPeso molecular:518.6Anticancer agent 101
CAS:<p>Anticancer Agent 101, a tetracaine derivative, exhibits anti-cancer activity [1].</p>Fórmula:C19H20F3N3OForma y color:SolidPeso molecular:363.38KH-3
CAS:<p>KH-3: HuR inhibitor, IC50 0.35 μM, halts cell growth, blocks HuR-FOXQ1 mRNA, curbs breast cancer invasion, slows lung colony growth.</p>Fórmula:C21H22N2O4S2Forma y color:SolidPeso molecular:430.54MDL-27467A
CAS:<p>MDL-27467A is an ester derivative of a potent angiotensin converting enzyme inhibitor.</p>Fórmula:C40H42N2O5Forma y color:SolidPeso molecular:630.77Englitazone sodium
CAS:<p>Englitazone sodium is an antidiabetic agent and a novel NSCA and KATP channel blocker.</p>Fórmula:C20H19NNaO3SForma y color:SolidPeso molecular:376.43G4/HDAC-IN-1
<p>G4/HDAC-IN-1, a G4/HDAC dual inhibitor, IC50 1.1 µM, blocks TNBC growth, useful in cancer research.</p>Fórmula:C36H49ClFN7O4Forma y color:SolidPeso molecular:698.27αvβ1 integrin-IN-2
CAS:<p>αvβ1 integrin-IN-2 (compound 32) is a potent inhibitor of ανβ1 and α5β1 integrins, exhibiting IC50 values of 0.9 nM and 33 nM, respectively.</p>Fórmula:C29H38N4O4Pureza:98%Forma y color:SolidPeso molecular:506.64VT-1598
CAS:<p>VT-1598 is a novel, selective, orally active fungal CYP51 inhibitor. VT-1598 exhibits antifungal effects against Candida albicans.</p>Fórmula:C31H20F4N6O2Forma y color:SolidPeso molecular:584.52Flamprop-methyl
CAS:<p>Flamprop-methyl is a post-emergence herbicide, it is usually used on wild oats.</p>Fórmula:C17H15ClFNO3Pureza:98%Forma y color:SolidPeso molecular:335.76ARQ-736
CAS:<p>ARQ 736 effectively targets and inhibits BRAF, crucial in MAPK pathway, beneficial for treating melanomas and certain colon cancers.</p>Fórmula:C25H25N8Na2O8PSForma y color:SolidPeso molecular:674.54
