Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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Tubulin/JAK2-IN-1
CAS:<p>Tubulin/JAK2-IN-1 (compound 7g) serves as a potent dual inhibitor targeting both Janus kinase 2 (JAK2) and microtubules, demonstrating significant</p>Fórmula:C22H20N6O3Forma y color:SolidPeso molecular:416.43RK-701
CAS:<p>RK-701: G9a inhibitor, IC50 23-27 nM, increases HbF/γ-Globin/BGLT3, decreases H3K9me2, inhibits BCL11A/ZBTB7A.</p>Fórmula:C26H30N4O3Forma y color:SolidPeso molecular:446.54DYRKs-IN-2
CAS:<p>DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM and 12.8 nM for DYRK1B and DYRK1A, respectively.</p>Fórmula:C32H38ClN9O3Pureza:98%Forma y color:SolidPeso molecular:632.16CLR-131
CAS:<p>CLR-131, a protein kinase B (PKB) inhibitor, is used potentially for the treatment of non small cell lung cancer, solid tumors.</p>Fórmula:C29H53INO4PPureza:98%Forma y color:SolidPeso molecular:641.62RG 14893
CAS:<p>RG 14893 is a antagonist of high-affinity leukotriene B4 receptor.</p>Fórmula:C29H27NO4Pureza:98%Forma y color:SolidPeso molecular:453.53Celiprolol hydrochloride
CAS:<p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>Fórmula:C20H33N3O4·HClForma y color:White Crystalline SolidPeso molecular:415.96(+)-Carbovir
CAS:<p>(+)-Carbovir is a nucleoside analog with increased chemical stability and increased metabolic stability.</p>Fórmula:C11H13N5O2Forma y color:SolidPeso molecular:247.25AAK1-IN-3
CAS:<p>AAK1-IN-3: Brain-penetrant AAK1 inhibitor for neuropathic pain research; IC50=11 nM.</p>Fórmula:C20H20N4Forma y color:SolidPeso molecular:316.4SC 53228
CAS:<p>SC 53228 is a specific leukotriene B4 receptor antagonist.</p>Fórmula:C31H41NO7Forma y color:SolidPeso molecular:539.66Muraglitazar glucuronide
CAS:<p>Muraglitazar glucuronide is a Peroxime Proliferator Activated (PPAR) Agonist that has glucose- and lipid-lowering activities.</p>Fórmula:C35H36N2O13Forma y color:SolidPeso molecular:692.67pppApG
CAS:<p>pppApG serves as an initial substrate for the synthesis of vRNA (viral RNA) and cRNA (complementary RNA), with applications in influenza virus research [1].</p>Fórmula:C20H28N10O20P4Forma y color:SolidPeso molecular:852.39L-739758
CAS:<p>L-739758 is a glycoprotein IIb/IIIa inhibitor.</p>Fórmula:C22H26N4O5S3Forma y color:SolidPeso molecular:522.66BR103354
CAS:<p>BR103354: potent FAP inhibitor, IC50 of 14 nM, oral bioavailability 48.4%, minimal hERG risk, potential anti-diabetic and anti-NASH agent.</p>Fórmula:C19H15F2N5O2SForma y color:SolidPeso molecular:415.42ZM 260384
CAS:<p>ZM 260384 is a potassium channel opener.</p>Fórmula:C15H11F4N3O4Forma y color:SolidPeso molecular:373.26HJC0152 free base
CAS:<p>HJC0152 (free base) is an orally active, potent STAT3 inhibitor that impedes cell cycle progression, induces apoptosis, and notably reduces MDA-MB-231 xenograft</p>Fórmula:C15H13Cl2N3O4Pureza:98%Forma y color:SolidPeso molecular:370.19(R)-MALT1-IN-7
CAS:<p>(R)-MALT1-IN-7 (compound 142a) is a potent inhibitor of MALT1 protease and has potential for cancer research.</p>Fórmula:C19H17F3N8O2SForma y color:SolidPeso molecular:478.45JAK-IN-24
CAS:<p>JAK-IN-24: JAK inhibitor, IC50: 0.534 nM (4 μM ATP), 24 nM (1mM ATP), STAT5 phosphorylation IC50: 86.171 nM.</p>Fórmula:C20H25N5O2Forma y color:SolidPeso molecular:367.44CGC 11093
CAS:<p>CGC 11093: A polyamine analog inhibiting human prostate tumor growth in mice; may help regress choroidal neovascularization.</p>Fórmula:C17H42Cl4N4Forma y color:SolidPeso molecular:444.35Avarofloxacin
CAS:<p>Avarofloxacin (JNJ-Q2) is a fluoroquinolone for treating bacterial skin infections and pneumonia.</p>Fórmula:C21H23F2N3O4Forma y color:SolidPeso molecular:419.42WAY-658494
CAS:<p>WAY-658494 is an (active) compound.</p>Fórmula:C13H13NO3S2Forma y color:SolidPeso molecular:295.38Glycolithocholic acid 3-sulfate disodium
CAS:<p>Glycolithocholic acid 3-sulfate (disodium) demonstrates inhibitory effects on in vitro HIV-1 replication and has potential applications in HIV infection and</p>Fórmula:C26H41NNa2O7SForma y color:SolidPeso molecular:557.65GIV3727
CAS:<p>GIV3727, a bitter taste receptor hTAS2R antagonist, inhibits the activation of hTAS2R31 by saccharin and acesulfame potassium, effectively diminishing the</p>Fórmula:C12H22O2Forma y color:SolidPeso molecular:198.3SARS-CoV-2-IN-66
CAS:<p>SARS-CoV-2-IN-66 (1), a derivative of vitamin K, functions as an inhibitor of SARS-CoV-2, exhibiting an effective concentration (EC50) of 70.8 μM in VeroE6/</p>Fórmula:C28H30O2Pureza:98%Forma y color:SolidPeso molecular:398.54BMS-763534
CAS:<p>BMS-763534 is a potent antagonist of corticotropin-releasing factor/hormone receptor 1 (CRHR-1).</p>Fórmula:C18H21ClF2N4O3Forma y color:SolidPeso molecular:414.83CID-50930756
CAS:<p>CID-50930756 is a novel HCV NS3 helicase catalyzed ATP hydrolysis stimulator.</p>Fórmula:C27H18N4O4S3Forma y color:SolidPeso molecular:558.6510-Chloroestra-1,4-diene-3,17-dione
CAS:<p>10-Chloroestra-1,4-diene-3,17-dione acts as an estrogen receptor α (ERα) agonist, enhancing reporter gene expression in S.</p>Fórmula:C18H21ClO2Forma y color:SolidPeso molecular:304.80Anticancer agent 127
CAS:<p>Anticancer agent 127 (142D6), an IAP inhibitor, covalently binds to the BIR3 domains of XIAP, cIAP1, and cIAP2, with IC50 values of 12 nM, 14 nM, and 9 nM,</p>Fórmula:C26H37FN4O6SPureza:98%Forma y color:SolidPeso molecular:552.66XR9051 Hydrochloride
CAS:<p>XR9051 Hydrochloride, a potent modulator of P-glycoprotein-mediated multidrug resistance (MDR), inhibits the binding of cytotoxics to P-glycoprotein.</p>Fórmula:C39H39ClN4O5Forma y color:SolidPeso molecular:679.21Inz-1
CAS:<p>Inz-1 is an effective and fungal-selective inhibitor of mitochondrial cytochrome bc1 with IC50s of 8.092 and 45.320 μM for yeast and human.</p>Fórmula:C16H14N2O2Pureza:99.55% - 99.88%Forma y color:SolidPeso molecular:266.29Mitochondria degrader-1
CAS:<p>Mitochondria degrader-1, a potent autophagy inducer, aids in neurodegenerative, cancer, and aging disease research.</p>Fórmula:C33H49ClFN7O8SForma y color:SolidPeso molecular:758.3Clobutinol hydrochloride
CAS:<p>Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in cough-related research [1] [2] [3].</p>Fórmula:C14H23Cl2NOPureza:98%Forma y color:SolidPeso molecular:292.25YM458
CAS:<p>YM458 inhibits EZH2 (490 nM) and BRD4 (34 nM), curbing tumor cell growth and inducing apoptosis.</p>Fórmula:C53H61ClN8O5SPureza:98%Forma y color:SolidPeso molecular:957.62ACHP Hydrochloride
CAS:<p>ACHP Hydrochloride (IKK-2 Inhibitor VIII) is a highly potent and selective IKK-β inhibitor with an IC50 of 8.5 nM.</p>Fórmula:C21H25ClN4O2Pureza:99.83%Forma y color:SolidPeso molecular:400.9Indacrinone
CAS:<p>Indacrinone is an investigational diuretic.</p>Fórmula:C18H14Cl2O4Pureza:98%Forma y color:SolidPeso molecular:365.21RP-001
CAS:<p>RP-001 is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.</p>Fórmula:C24H24N4O4Pureza:98%Forma y color:SolidPeso molecular:432.47(S)-FTY-720 Vinylphosphonate
CAS:<p>(S)-FTY-720 Vinylphosphonate blocks sphingosine kinase 1 and aids its breakdown in various human cancer cells.</p>Fórmula:C20H34NO4PForma y color:SolidPeso molecular:383.46AR-C117977
CAS:<p>AR-C117977: Potent MCT1 inhibitor, reduces immune response, extends graft survival, induces tolerance in vitro/in vivo.</p>Fórmula:C25H28N2O3S2Forma y color:SolidPeso molecular:468.632-Quinizarincarboxylic acid
CAS:<p>Compound 15, 2-Quinizarincarboxylic acid, functions as a glucose uptake inhibitor, demonstrating a 24.9% inhibition rate at a concentration of 50 μM [1].</p>Fórmula:C15H8O6Forma y color:SolidPeso molecular:284.22Mitemcinal
CAS:<p>Mitemcinal is a motilin agonist.</p>Fórmula:C40H69NO12Forma y color:SolidPeso molecular:755.98ICMT-IN-13
CAS:<p>ICMT-IN-13 (compound 49) functions as an inhibitor of ICMT, exhibiting an IC50 value of 0.47 μM [1].</p>Fórmula:C21H25ClFNOForma y color:SolidPeso molecular:361.88Thromboxane A2
CAS:<p>Thromboxane A2: unstable, leads to thromboxane B2, induces platelet aggregation, causes vasoconstriction.</p>Fórmula:C20H32O5Forma y color:SolidPeso molecular:352.47BMS-538158
CAS:<p>BMS-538158 is a bio-active chemical.</p>Fórmula:C15H16FNO5Forma y color:SolidPeso molecular:309.293RB-3
CAS:<p>RB-3, a PRC1 inhibitor, binds to RING1B-BMI1f , with a K d of 2.8 μM.</p>Fórmula:C24H20ClN3O2Forma y color:SolidPeso molecular:417.89FHND5071
CAS:<p>FHND5071, a potent and selective RET kinase inhibitor, exerts antitumor effects through the inhibition of RET autophosphorylation and may be utilized for tumor</p>Fórmula:C30H30D3N9OForma y color:SolidPeso molecular:538.66PD 128907
CAS:<p>PD 128907 - potent, selective dopamine D2/D3 agonist for researching receptor roles in the brain.</p>Fórmula:C14H19NO3Pureza:98%Forma y color:SolidPeso molecular:249.31FK 33-824
CAS:<p>FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.</p>Fórmula:C29H41N5O7SPureza:98%Forma y color:SolidPeso molecular:603.73AS6
CAS:<p>AS6 is an ABA-induced PYL-PP2C interaction antagonist in a dose-dependent manner.</p>Fórmula:C21H32O4SPureza:98%Forma y color:SolidPeso molecular:380.54GJH-166
CAS:<p>GJH-166 is an analog of dopamine that has been shown to inhibit adrenergic transmission in canines.</p>Fórmula:C14H19NO2Forma y color:SolidPeso molecular:233.31BP
<p>BP is a rare class enhancer of proteasomal activation in the absence of a heat shock response.</p>Fórmula:C33H47Cl2N5O10SForma y color:SolidPeso molecular:776.72KFM19
CAS:<p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>Fórmula:C16H22N4O3Pureza:98.62%Forma y color:SolidPeso molecular:318.37
