Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
HAPSBC
CAS:<p>HAPSBC, an S-benzyl iron chelator, modulates the intracellular distribution of ^59Fe [1].</p>Fórmula:C15H15N3S2Forma y color:SolidPeso molecular:301.43N-Demethyl Mifepristone
CAS:<p>N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone'</p>Fórmula:C28H33NO2Pureza:98%Forma y color:SolidPeso molecular:415.57ANN33840
CAS:<p>ANN33840: Selective 5-HT2C agonist, 300x vs 5-HT2B, 70x vs 5-HT2A; cuts rat food intake.</p>Fórmula:C14H15F3N2OForma y color:SolidPeso molecular:284.28Bcl-2-IN-12
CAS:<p>Bcl-2-IN-12 (Compound 1) is a potent Bcl-2 inhibitor with an IC50 value of 6 nM, utilized in cancer research [1].</p>Fórmula:C47H41ClN4O6SForma y color:SolidPeso molecular:825.37BMT-124110
CAS:<p>BMT-124110: AAK1 inhibitor, IC50=0.9 nM, pain relief. BMT-090605: BIKE inhibitor, IC50=17 nM; GAK inhibitor, IC50=99 nM.</p>Fórmula:C21H27N3O3Pureza:98.07%Forma y color:SolidPeso molecular:369.46BT424
CAS:<p>BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation and renal fibrosis in the UUO model [1].</p>Fórmula:C22H15BCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:421.08GGTI-297
CAS:<p>GGTI-297 is a potent, cell-permeable, and selective peptidomimetic inhibitor of GGTase I compared to Farnesyl Transferase (FTase).</p>Fórmula:C26H31N3O3SForma y color:SolidPeso molecular:465.61BMS-189664 HCl
CAS:<p>BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.</p>Fórmula:C22H35ClN6O4SPureza:98%Forma y color:SolidPeso molecular:515.07NLX-204
CAS:<p>NLX-204 is a selective, potent agonist of ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor with pKi value of 10.19.</p>Fórmula:C20H22ClF2N3O2Pureza:98%Forma y color:SolidPeso molecular:409.86FPTQ
CAS:<p>FPTQ is a highly effective antagonist of mGluR 1, displaying IC50 values of 6 nM and 1.4 nM for human and mouse mGluR1 respectively [1].</p>Fórmula:C17H12FN5Pureza:99.68% - 99.88%Forma y color:SolidPeso molecular:305.31JNJ-46281222
CAS:<p>JNJ-46281222: mGlu2-selective, potent PAM, Kd = 1.7 nM, pEC50 = 7.71.</p>Fórmula:C23H25F3N4Forma y color:SolidPeso molecular:414.47Lifirafenib
CAS:<p>Lifirafenib (Beigene-283) is a potent inhibitor of RAF family kinases and EGFR in biochemical assays with IC50 of 23, 29 and 495 nM for the recombinant</p>Fórmula:C25H17F3N4O3Pureza:98% - 98.25%Forma y color:SolidPeso molecular:478.42MLN-3897
CAS:<p>MLN-3897 is an oral CCR1 antagonist, Ki 2.3 nM, blocks 125I-MIP-1α binding, and inhibits Akt signaling in MM cells.</p>Fórmula:C30H31ClN2O4Pureza:98.62%Forma y color:SolidPeso molecular:519.03Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Fórmula:C38H43ClN4O6Pureza:98%Forma y color:SolidPeso molecular:687.22Duocarmycin MA
CAS:<p>Duocarmycin MA: ADCs toxin for multi-drug resistant cells; DNA alkylating agent binding in DNA minor groove.</p>Fórmula:C34H31ClN4O5Pureza:98%Forma y color:SolidPeso molecular:611.09Crisdesalazine
CAS:<p>Crisdesalazine (AAD 2004) is an inhibitor of microsomal prostaglandin E2 synthase-1 (mPGES-1).</p>Fórmula:C16H14F3NO3Pureza:98.96%Forma y color:SolidPeso molecular:325.28RSV L-protein-IN-2
CAS:<p>RSV L-protein-IN-2 (Compound A), a noncompetitive inhibitor of the RSV polymerase (IC50: 4.5 μM), exhibits antiviral activity against long RSV strains (EC50: 1.</p>Fórmula:C32H36N4O5Pureza:98%Forma y color:SolidPeso molecular:556.65Quorum Sensing-IN-2
CAS:<p>Quorum Sensing-IN-2 (compound 23e) is a quorum sensing inhibitor that curtails bacterial pathogenicity without impeding growth.</p>Fórmula:C19H13F2NO3Forma y color:SolidPeso molecular:341.31JAK2-IN-4
CAS:<p>JAK2-IN-4 is a selective JAK2/JAK3 inhibitor, with IC50 values of 0.7 nM and 23.2 nM for JAK2 and JAK3, respectively.</p>Fórmula:C23H27N5O4SPureza:98%Forma y color:SolidPeso molecular:469.56PCSK9-IN-14
CAS:<p>PCSK9-IN-14, also known as compound Ia-8, is a potent inhibitor of PCSK9 [1].</p>Fórmula:C15H10F6N4O2Forma y color:SolidPeso molecular:392.26H3B-6545 Hydrochloride
CAS:<p>H3B-6545 Hydrochloride is a selective, oral estrogen receptor covalent antagonist (SERCA).</p>Fórmula:C30H30ClF4N5O2Forma y color:SolidPeso molecular:604.04TAS2R14 agonist-2
CAS:<p>Compound 28.1, also known as TAS2R14 agonist-2, is a potent and selective inhibitor of TAS2R14, exhibiting an EC50 of 72 nM [1].</p>Fórmula:C13H10F3N7Forma y color:SolidPeso molecular:321.26Tedalinab
CAS:<p>Tedalinab is an effective and selective cannabinoid receptor 2 agonist.</p>Fórmula:C19H21F2N3OPureza:98%Forma y color:SolidPeso molecular:345.39Cbl-b-IN-7
CAS:<p>Cbl-b-IN-7 (Compound 248) is an inhibitor of casitas B-lineage lymphoma-b (Cbl-b) and c-Cbl, exhibiting inhibitory half-maximal inhibitory concentrations (IC50s</p>Fórmula:C29H31F4N5O2Pureza:98%Forma y color:SolidPeso molecular:557.58Skp2 inhibitor 2
CAS:<p>Skp2 inhibitor 2 (14f) impedes the F-box protein S-phase kinase-associated protein 2 (Skp2), demonstrating an IC50 of 10.2 μM against Skp2-Cks1.</p>Fórmula:C27H32N4OPureza:98%Forma y color:SolidPeso molecular:428.57Phenoxan
CAS:<p>Phenoxan is isolated from Polyangium; inhibits electron transport at NADH-ubiquinone oxidoreductase.</p>Fórmula:C23H25NO4Forma y color:SolidPeso molecular:379.45ERX-41
CAS:<p>ERX-41 is an orally active, stereospecific small molecule that targets lysosomal acid lipase A (LIPA).</p>Fórmula:C38H48N4O9Pureza:98%Forma y color:SolidPeso molecular:704.81NUC-7738
CAS:<p>NUC-7738 is a 5'-aryloxyphosphoamidoester prodrug of 3'-dA, which regulates 尾-catenin signaling and can be used in cancer research.</p>Fórmula:C26H29N6O7PPureza:97.32% - 97.32%Forma y color:SolidPeso molecular:568.52LY 134046
CAS:<p>LY 134046 is an inhibitor of phenylethanolamine-N-methyltransferase (PNMT).</p>Fórmula:C10H11Cl2NPureza:98%Forma y color:SolidPeso molecular:216.11FX-06
CAS:<p>FX-06 (Fibrin-derived peptide Bβ15-42) is a peptide derived from the fibrin Bbeta chain.</p>Fórmula:C133H216N44O38Forma y color:SolidPeso molecular:3039.41MI-888 free base
CAS:<p>MI-888 is the most potent MDM2 inhibitor (Ki = 0.44 nM), with high oral efficacy in human cancer models and optimal pharmacokinetics.</p>Fórmula:C28H32Cl2FN3O3Forma y color:SolidPeso molecular:548.48IWP-051
CAS:<p>IWP-051: potent oral sGC stimulator, >99% protein bound, stable, permeable, no Caco-2 efflux, potential for daily dose.</p>Fórmula:C17H11F2N5O2Forma y color:SolidPeso molecular:355.3Lingdolinurad
CAS:<p>Lingdolinurad is a uric acid transporter protein inhibitor targeting hURAT1 for the study of hyperuricemia or gout.</p>Fórmula:C17H12BrN3O2Pureza:96.26%Forma y color:SolidPeso molecular:370.2Orexin receptor modulator-1
CAS:<p>Orexin Receptor Modulator-1 is a compound utilized in the study of various conditions including substance addiction, panic disorder, anxiety, post-traumatic</p>Fórmula:C23H22ClF5N6OForma y color:SolidPeso molecular:528.91NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal)
CAS:<p>Compound 40, a cyclic Ape13 analogue and potent APJ agonist (Ki 5.7 nM), shows Gα12-bias and longer half-life.</p>Fórmula:C49H73N13O11Forma y color:SolidPeso molecular:1020.18FGFR3-IN-7
CAS:<p>FGFR3-IN-7 is a potent, selective inhibitor of FGFR 3, demonstrating an IC50 value of less than 350 nM , and is utilized in cancer research [1].</p>Fórmula:C25H24FN9OPureza:98%Forma y color:SolidPeso molecular:485.52PBB3
CAS:<p>PBB3 is a tau-specific PET tracer.</p>Fórmula:C17H15N3OSForma y color:SolidPeso molecular:309.39Afizagabar
CAS:<p>Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.</p>Fórmula:C19H12FN3O2SForma y color:SolidPeso molecular:365.383-Hydroxy-2-(palmitoyloxy)propyl stearat
CAS:<p>3-Hydroxy-2-(palmitoyloxy)propyl stearate is a non-volatile compound isolated from the less polar fractions of the brown macroalga Fucus virsoides J.</p>Fórmula:C37H72O5Forma y color:SolidPeso molecular:596.96RCB16007
CAS:<p>RCB16007 is a Yellow Fever Virus (YFV) inhibitor that also demonstrates inhibitory action against the West Nile virus with an effective concentration (EC50) of</p>Fórmula:C18H14ClN5O2SForma y color:SolidPeso molecular:399.85BMS-604992
CAS:<p>EX-1314 (BMS-604992) is a growth hormone secretagogue receptor (GHSR) agonist.</p>Fórmula:C24H32ClN7O5Forma y color:SolidPeso molecular:534.01RIPK1-IN-8
CAS:<p>RIPK1-IN-8 is an aminoimidazolopyridine and is a selective and potent inhibitor of RIPK1 (IC50: 4 nM).RIPK1-IN-8 has research potential in inflammatory diseases</p>Fórmula:C26H24F2N6O3Forma y color:SolidPeso molecular:506.5Antioxidant agent-15
CAS:<p>Antioxidant agent-15 (Compound 4) demonstrates potent antioxidant inhibition activity, exhibiting an IC50 value of 15.44 nM.</p>Fórmula:C19H14O2Pureza:98%Forma y color:SolidPeso molecular:274.31IDH1 Inhibitor 7
CAS:<p>IDH1 Inhibitor 7 is an IDH1 inhibitor with an IC 50 of less than 100 nM .</p>Fórmula:C22H24F3N7OForma y color:SolidPeso molecular:459.47Cindunistat HCl maleate
CAS:<p>Cindunistat, a potent oral iNOS inhibitor for symptomatic knee osteoarthritis.</p>Fórmula:C20H39ClN6O8S2Forma y color:SolidPeso molecular:591.14Flucythrinate
CAS:<p>Flucythrinate is an insecticide.</p>Fórmula:C26H23F2NO4Forma y color:Viscous Liquid SolidPeso molecular:451.46GPR120 Agonist 1
CAS:<p>GPR120 Agonist 1 selectively activates human/mouse GPR120 with EC50 of 42/77 nM in HEK293 cells.</p>Fórmula:C20H12ClF6NO3SPureza:98%Forma y color:SolidPeso molecular:495.82H4R antagonist 2
CAS:<p>H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid</p>Fórmula:C13H17N5OPureza:98%Forma y color:SolidPeso molecular:259.31Indacrinone
CAS:<p>Indacrinone is an investigational diuretic.</p>Fórmula:C18H14Cl2O4Pureza:98%Forma y color:SolidPeso molecular:365.21LY2922083
CAS:<p>LY2922083: Potent, selective GPR40 agonist; lowers glucose, boosts insulin and GLP-1.</p>Fórmula:C31H33NO3SForma y color:SolidPeso molecular:499.66
