
Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.787 productos)
- Ciclo celular / Checkpoint(4.446 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.824 productos)
- Endocrinología / Hormonas(3.500 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.318 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.200 productos)
- Transportador de membrana / canal de iones(2.787 productos)
- Metabolismo(9.416 productos)
- Microbiología / Virología(6.968 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.928 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(831 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.649 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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ELOVL6-IN-2
CAS:<p>ELOVL6-IN-2 is a orally active and selective ELOVL6 inhibitor.</p>Fórmula:C28H23F6N3O4Pureza:99.43%Forma y color:SolidPeso molecular:579.49C-021
CAS:<p>C 021 dihydrochloride is a potent CCR4 antagonist.</p>Fórmula:C27H41N5O2Pureza:99.74% - 99.90%Forma y color:SolidPeso molecular:467.65123C4
CAS:<p>123C4 is a potent, selective and competitive agonist of the receptor tyrosine kinase EPHA4 (Ki=0.65 μM)[1].</p>Fórmula:C43H47ClN8O6Pureza:98.94%Forma y color:SolidPeso molecular:807.34Vacuolin-1
CAS:<p>Vacuolin-1 is a cell-permeable inhibitor of Ca2+ dependent fusion of lysosomes to the cell membrane.</p>Fórmula:C26H24IN7OPureza:97.20% - 98.45%Forma y color:SolidPeso molecular:577.42(+)-Isocorydine hydrochloride
CAS:<p>(+)-Isocorydine hydrochloride (Isocorydine HCl) is a eukaryote protein kinases Inhibitor.</p>Fórmula:C20H24ClNO4Pureza:98% - >99.99%Forma y color:SolidPeso molecular:377.873-hydroxycephem
CAS:<p>3-hydroxycephem is a useful organic compound for research related to life sciences. The catalog number is T4581 and the CAS number is 54639-48-4.</p>Fórmula:C28H24N2O5SPureza:98.74%Forma y color:White Or Off-White Crysalline PowderPeso molecular:500.572'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Fórmula:C16H14O4Pureza:98.75%Forma y color:SolidPeso molecular:270.28Sultopride hydrochloride
CAS:<p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>Fórmula:C17H27ClN2O4SPureza:≥95%Forma y color:White Or Yellowish PowderPeso molecular:390.93Pneumocandin B0
CAS:<p>Pneumocandin B0 (L-688786) is a natural product and a key intermediate in the synthesis of the antifungal agent.</p>Fórmula:C50H80N8O17Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:1065.21Isavuconazole
CAS:<p>Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.</p>Fórmula:C22H17F2N5OSPureza:99.74% - >99.99%Forma y color:SolidPeso molecular:437.47UNC0064-12 hydrochloride (1430089-64-7(free base))
<p>UNC0064-12 hydrochloride is an inhibitor of VEGFR2.</p>Fórmula:C19H25ClN8Pureza:99.52%Forma y color:SolidPeso molecular:400.91Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Fórmula:C19H20N2O3Pureza:99.84% - 99.86%Forma y color:White PowderPeso molecular:324.37Hexahydrocurcumin
CAS:<p>Hexahydrocurcumin is a selective, orally active COX-2 inhibitor and inactive against COX-1.</p>Fórmula:C21H26O6Pureza:99.43% - 99.88%Forma y color:SolidPeso molecular:374.43FMoc-Val-Cit-PAB-PNP
CAS:<p>Fmoc-Val-Cit-PAB-PNP is a linker for Antibody-Drug-Conjugation (ADC).</p>Fórmula:C40H42N6O10Pureza:98.05% - 98.46%Forma y color:SolidPeso molecular:766.8AS-252424
CAS:<p>AS-252424 is a potent and selective inhibitor of PI3Kγ with IC50 of 33 nM; >10 fold selectivity for PI3Kγ versus PI3Kα.</p>Fórmula:C14H8FNO4SPureza:99.06% - 99.09%Forma y color:SolidPeso molecular:305.28Delanzomib
CAS:<p>Delanzomib (CEP-18770) is an oral proteasome inhibitor with an IC50 of 3.8 nM, targeting chymotrypsin-like activity with minimal effect on other activities.</p>Fórmula:C21H28BN3O5Pureza:95.52% - 99.46%Forma y color:SolidPeso molecular:413.28Temsavir
CAS:<p>Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.</p>Fórmula:C24H23N7O4Pureza:99.14%Forma y color:SolidPeso molecular:473.482-hexyl-4-Pentynoic Acid
CAS:<p>2-hexyl-4-Pentynoic Acid, a valproic acid (VPA) derivatives, is a potent and robust HDACs inhibitor with IC50 value of 13 μM.</p>Fórmula:C11H18O2Pureza:98%Forma y color:SolidPeso molecular:182.26BMS986260
CAS:<p>BMS-986260 is a selective, and orally bioavailable TGFβR1 inhibitor(IC50 = 1.6 nM).</p>Fórmula:C18H12ClFN6OPureza:97.67%Forma y color:SolidPeso molecular:382.78Enavogliflozin
CAS:<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Fórmula:C24H27ClO6Pureza:97.37%Forma y color:SolidPeso molecular:446.92(±)-Methyl Jasmonate
CAS:<p>Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate ((±)-Jasmonic Acid methyl ester)induces the synthesis of proteinase inhibitors in plant leaves.</p>Fórmula:C13H20O3Pureza:98.95% - 99.39%Forma y color:Colorless Liquid Clear To Pale Yellow LiquidPeso molecular:224.3Hemin
CAS:<p>Hemin (Hemin chloride) is a chlorinated iron-containing porphyrin, a heme oxygenase (HO)-1 inducer.</p>Fórmula:C34H32ClFeN4O4Pureza:97.169% - 99.59%Forma y color:Dark Purple Crystalline PowderPeso molecular:651.94Boc-GABA-OH
CAS:<p>Boc-GABA-OH serves as a PROTAC linker essential for synthesizing UNC6852, an EED-targeted PROTAC[1].</p>Fórmula:C9H17NO4Pureza:99%Forma y color:White Crystalline PowderPeso molecular:203.24Daclatasvir dihydrochloride
CAS:<p>Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.</p>Fórmula:C40H52Cl2N8O6Pureza:99.67%Forma y color:SolidPeso molecular:811.8BIBR 1532
CAS:<p>BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay).</p>Fórmula:C21H17NO3Pureza:98.49% - 98.90%Forma y color:SolidPeso molecular:331.36AMD 3465 hexahydrobromide
CAS:<p>AMD 3465 hexahydrobromide (GENZ-644494 (hexahydrobromide)) is a CXCR4 receptor antagonist with potential anticancer and anti-HIV activity.</p>Fórmula:C24H44Br6N6Pureza:99.39%Forma y color:SolidPeso molecular:896.07Sudan IV
CAS:<p>Sudan IV (Solvent Red 24) is a lysochrome (fat-soluble dye) diazo dye used for the staining of triglycerides,lipids and lipoproteins on frozen paraffin sections</p>Fórmula:C24H20N4OForma y color:Dark Red Solid PowderPeso molecular:380.44Glycyrrhetic acid 3-O-β-D-glucuronide
CAS:<p>Glycyrrhetic acid 3-O-β-D-glucuronide is a potent sweetener (relative sweetness to sucrose: x 941).</p>Fórmula:C36H54O10Pureza:99.04% - 99.86%Forma y color:SolidPeso molecular:646.81Grazoprevir hydrate
CAS:<p>Grazoprevir: Hepatitis C protease inhibitor effective against various genotypes, including drug-resistant strains.</p>Fórmula:C38H52N6O10SPureza:98%Forma y color:SolidPeso molecular:784.92Cloquintocet-mexyl
CAS:<p>Cloquintocet-mexyl, a herbicide, targets and controls coarse annual grasses within the Poaceae family.</p>Fórmula:C18H22ClNO3Pureza:98.69%Forma y color:Light Brown Solid PowderPeso molecular:335.83ω-Pentadecalactone
CAS:<p>ω-Pentadecalactone (Exaltolide) is the fragrance structural group macrocyclic lactone and lactide derivatives used as a fragrance ingredient.</p>Fórmula:C15H28O2Pureza:98%Forma y color:Liquid OthersolidPeso molecular:240.38Feruloylputrescine
CAS:<p>Feruloylputrescine is a natural product.</p>Fórmula:C14H20N2O3Pureza:97.7% - 99.71%Forma y color:SolidPeso molecular:264.32Esculentoside A
CAS:<p>Esculentoside A dampens inflammation in ALI, modulates T cells, and could treat autoimmune diseases and BXSB mice by adjusting cytokines and renal cells.</p>Fórmula:C42H66O16Pureza:98% - 99.85%Forma y color:SolidPeso molecular:826.96Chrysosplenol D
CAS:<p>Chrysosplenol D, an efflux pump inhibitor that can potentiate the activity of commercially important antibiotics and antimalarials.</p>Fórmula:C18H16O8Pureza:97.87% - 99.98%Forma y color:SolidPeso molecular:360.31(Z)-4-Amino-4-oxobut-2-enoic acid
CAS:<p>(Z)-4-Amino-4-oxobut-2-enoic acid (Maleamic acid) is a useful research chemical.</p>Fórmula:C4H5NO3Pureza:98.25%Forma y color:SolidPeso molecular:115.097β-Hydroxylathyrol
CAS:<p>7β-Hydroxylathyrol is a diterpenoid extract from the seed oil of Caper Spurge and displays P-gp inhibition resulting in cytotoxic properties.</p>Fórmula:C20H30O5Pureza:97.49% - ≥95%Forma y color:SolidPeso molecular:350.452-Aminooctadecane-1,3,4-Triol
CAS:<p>2-Aminooctadecane-1,3,4-Triol (Phytosphingosine) is a natural product.</p>Fórmula:C18H39NO3Pureza:≥98%Forma y color:SolidPeso molecular:317.51Talnetant
CAS:<p>Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.</p>Fórmula:C25H22N2O2Pureza:97.88%Forma y color:SolidPeso molecular:382.45Spinorphin
CAS:<p>Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.</p>Fórmula:C45H64N8O10Pureza:99.68%Forma y color:SolidPeso molecular:877Bradykinin (acetate)
CAS:<p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>Fórmula:C52H77N15O13Pureza:>99.99%Forma y color:SolidPeso molecular:1120.26Telaprevir
CAS:<p>Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).</p>Fórmula:C36H53N7O6Pureza:96.9% - 98.89%Forma y color:SolidPeso molecular:679.85ELR510444
CAS:<p>ELR510444 (LR510444) is a novel microtubule disruptor; inhibits MDA-MB-231 cell proliferation with IC50 of 30.9 nM.</p>Fórmula:C19H16N2O2S2Pureza:97.67% - 98.69%Forma y color:SolidPeso molecular:368.47Tetrahydropalmatine hydrochloride
CAS:<p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>Fórmula:C21H26ClNO4Pureza:98% - 99.59%Forma y color:SolidPeso molecular:391.888LY3200882
CAS:<p>LY3200882 is a highly selective inhibitor of TGF-β receptor type 1 (TGFβRI).</p>Fórmula:C24H29N5O3Pureza:99.46% - 99.63%Forma y color:SolidPeso molecular:435.52GLPG2938
CAS:<p>GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and</p>Fórmula:C20H19F6N7O2Pureza:98.25%Forma y color:SolidPeso molecular:503.4Taurochenodeoxycholic Acid
CAS:<p>Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) is one of the main bioactive substances of animals' bile acid.</p>Fórmula:C26H45NO6SPureza:99.53% - 99.86%Forma y color:SolidPeso molecular:499.7trans-Coniferyl aldehyde
CAS:<p>Coniferaldehyde hinders Oenococcus oeni growth and exhibits anti-inflammatory effects by inducing HO-1.</p>Fórmula:C10H10O3Pureza:98%Forma y color:SolidPeso molecular:178.18ABT-639 hydrochloride
CAS:<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Fórmula:C20H21Cl2F2N3O3SForma y color:SolidPeso molecular:492.36Pyrintegrin
CAS:<p>Pyrintegrin: β1-integrin agonist, boosts embryonic stem cell survival, and podocyte protection, improves cell-matrix adhesion.</p>Fórmula:C23H25N5O3SPureza:99.19%Forma y color:SolidPeso molecular:451.54S-Adenosyl-L-methionine disulfate tosylate
CAS:<p>S-Adenosyl-L-methionine disulfate tosylate is an orally active methyl donor. anti-proliferation. High-Quality, Low-Cost!</p>Fórmula:C22H34N6O16S4Pureza:97.02% - 98.61%Forma y color:White PowderPeso molecular:766.8
