Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.519 productos)
- Apoptosis(5.786 productos)
- Ciclo celular / Checkpoint(4.444 productos)
- Cromatina / Epigenética(2.235 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.823 productos)
- Endocrinología / Hormonas(3.499 productos)
- Enzima(3.639 productos)
- GPCR / proteína G(8.314 productos)
- Inmunología e inflamación(3.516 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.199 productos)
- Transportador de membrana / canal de iones(2.786 productos)
- Metabolismo(9.417 productos)
- Microbiología / Virología(6.967 productos)
- Neurociencia(9.920 productos)
- Otros inhibidores(37.931 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.596 productos)
- Células madre y Derivados(832 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.646 productos)
Mostrar 16 subcategorías más
Se han encontrado 66627 productos de "Inhibidores"
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Methacholine bromide
CAS:<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Fórmula:C8H18BrNO2Forma y color:SolidPeso molecular:240.141Flestolol sulfate
CAS:<p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>Fórmula:C15H24FN3O8SForma y color:SolidPeso molecular:425.43Lucidenic acid F
CAS:<p>Lucidenic acid F as a modulator of JNK and p38, it shows potent inhibitory effects on EBV-EA induction.</p>Fórmula:C27H36O6Pureza:98%Forma y color:SolidPeso molecular:456.57Quinterenol sulfate
CAS:<p>Quinoline sulfate has a bronchiectasis effect on patients with asthma.</p>Fórmula:C14H18N2O2H2O4SForma y color:SolidPeso molecular:295.35Cycrimine
CAS:<p>Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.</p>Fórmula:C19H29NOForma y color:SolidPeso molecular:287.44NMS-859
CAS:<p>NMS-859 is a covalent VCP/p97 inhibitor with IC50 of 0.37 μM (60 μM ATP) and 0.36 μM (1 mM ATP).</p>Fórmula:C15H12ClN3O3SPureza:98.20%Forma y color:SolidPeso molecular:349.79GW780056X
CAS:<p>GW780056X inhibits cyclin-dependent kinase, Yes1 kinase, and blocks Lassa Virus cell entry.</p>Fórmula:C21H23N7Pureza:98%Forma y color:SolidPeso molecular:373.45Pivalopril
CAS:<p>Pivalopril is a new orally active inhibitor of angiotensin-converting enzyme.</p>Fórmula:C16H27NO4SPureza:98%Forma y color:SolidPeso molecular:329.45Endochin
CAS:<p>Endochin is an experimental antimalarial. Endochin and analogues thereof are causal prophylactic and potent erythrocytic stage agents in avian models.</p>Fórmula:C18H25NO2Pureza:98%Forma y color:SolidPeso molecular:287.4PF00349412
CAS:<p>PF00349412 inhibits protozoan N-myristoyltransferases, a target for anti-fungal/trypanosome treatments.</p>Fórmula:C18H26N6SForma y color:SolidPeso molecular:358.5PDE10A-IN-8
CAS:<p>PDE10A-IN-8 is a potent inhibitor of PDE10A.</p>Fórmula:C23H19N3O2Pureza:98%Forma y color:SolidPeso molecular:369.42PBOX-15
CAS:<p>PBOX-15 induces apoptosis, regulates death receptors, enhances TRAIL effects, and inhibits T cell migration in myeloma cells.</p>Fórmula:C28H19NO3Forma y color:SolidPeso molecular:417.46SEP-363856
CAS:<p>SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.</p>Fórmula:C9H13NOSPureza:98%Forma y color:SolidPeso molecular:183.27COX-2-IN-24
CAS:<p>COX-2-IN-24 is an orally active COX-2 inhibitor (IC50: 0.17 μM) with anti-inflammatory and hypo-ulcerogenic effects.</p>Fórmula:C24H24BrN5O3S2Forma y color:SolidPeso molecular:574.51Dot1L-IN-2
CAS:<p>Dot1l-in-2 is an effective, selective and oral bioutilization inhibitor of histone methyltransferase Dot1L, with IC50 and Ki of 0.4 nM and 0.08 nM, respectively</p>Fórmula:C27H24N8OPureza:98%Forma y color:SolidPeso molecular:476.53hCAIX-IN-14
CAS:<p>hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .</p>Fórmula:C11H17ClN6O2SForma y color:SolidPeso molecular:332.81MDL-73811
CAS:<p>MDL-73811: Potent AdoMetDC blocker, anti-trypanosomal, cures mouse Brucella. Limited by fast plasma clearance, poor brain access.</p>Fórmula:C15H23N7O3Forma y color:SolidPeso molecular:349.39PI3K-IN-34
CAS:<p>PI3K-IN-34 targets PI3K-α/β/δ (IC50: 11.73/6.09/11.18 μM); potential leukemia research tool.</p>Fórmula:C23H22N6O3Forma y color:SolidPeso molecular:430.46CPI-455 HCl
CAS:<p>CPI-455: specific KDM5A inhibitor, IC50=10±1nM, increases H3K4me3, reduces DTPs in cancer cells.</p>Fórmula:C16H15ClN4OPureza:98%Forma y color:SolidPeso molecular:314.77Sarafloxacin
CAS:<p>Sarafloxacin (A56620) has antibacterial activities against Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H17F2N3O3Pureza:98.07% - 98.94%Forma y color:SolidPeso molecular:385.36Brofaromine
CAS:<p>Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).</p>Fórmula:C14H16BrNO2Forma y color:SolidPeso molecular:310.19BMY-25271
CAS:<p>BMY-25271 is an antagonist of histamine H2 receptor.</p>Fórmula:C12H19N5O2S2Pureza:98%Forma y color:SolidPeso molecular:329.44Cinalukast
CAS:<p>CysLT1 leukotriene receptor antagonist</p>Fórmula:C23H28N2O3SPureza:98%Forma y color:SolidPeso molecular:412.55GP17
CAS:<p>GP17 is a type II kinase inhibitor of the IRE1α endoribonuclease that acts by targeting the ATP-binding pocket of IRE1α.</p>Fórmula:C26H21F3N4OForma y color:SolidPeso molecular:462.47CB2R agonist 1
CAS:<p>CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.</p>Fórmula:C22H32N2OForma y color:SolidPeso molecular:340.5SCH529074
CAS:<p>SCH529074 is a selective activator of p53 (Ki = 1 μM) and can be used in studies about non-small-cell lung carcinoma.</p>Fórmula:C31H36Cl2N6Pureza:99.57%Forma y color:SolidPeso molecular:563.56SNT-207858 free base
CAS:<p>SNT-207858: selective MC-4 receptor antagonist, passes blood-brain barrier, orally active, IC50: 22 nM (binding), 11 nM (function).</p>Fórmula:C32H43Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:616.62HCV-IN-37
CAS:<p>HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.</p>Fórmula:C31H35F2N5Forma y color:SolidPeso molecular:515.64MRS2220
CAS:<p>MRS2220 is a selective enhancer of the ATP effects at fast desensitizing P2X (P2X1 and P2X3) receptors.</p>Fórmula:C13H12N3O11PS2Forma y color:SolidPeso molecular:481.35VUF-10214
CAS:<p>VUF-10214: H4 receptor ligand with anti-inflammatory effects in rat paw edema model.</p>Fórmula:C13H14Cl2N4OPureza:98%Forma y color:SolidPeso molecular:313.18CID1172084
CAS:<p>CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.</p>Fórmula:C23H18FN5O2S2Forma y color:SolidPeso molecular:479.55SPV106
CAS:<p>SPV106 is a ligand of lysine acetyltransferases (KATs).</p>Fórmula:C22H40O4Pureza:98%Forma y color:SolidPeso molecular:368.55Budralazine
CAS:<p>Budralazine is an agent of antihypertensive drug.</p>Fórmula:C14H16N4Pureza:98%Forma y color:SolidPeso molecular:240.3hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Fórmula:C12H12N4O5S2Forma y color:SolidPeso molecular:356.38A412997
CAS:<p>A412997 is a selective agonist of dopamine D4 receptor.</p>Fórmula:C19H23N3OPureza:98%Forma y color:SolidPeso molecular:309.41GEM144
CAS:<p>GEM144: oral POLA1/HDAC11 inhibitor; boosts p53, p21; halts G1/S cycle; triggers cell death.</p>Fórmula:C28H31NO5Forma y color:SolidPeso molecular:461.55CLE-030
CAS:<p>CLE-030, a KCNQ2 agonist, binds the central cavity, with its carbonyl oxygen influencing ions for activation.</p>Fórmula:C20H20Br2N4OS2Forma y color:SolidPeso molecular:556.34Trifenagrel
CAS:<p>Trifenagrel is an antithrombotic. It has been found to produce less gastric irritation and fecal blood loss in humans.</p>Fórmula:C25H25N3OPureza:98%Forma y color:SolidPeso molecular:383.49Alnespirone hydrochloride
CAS:<p>Alnespirone hydrochloride is a selective 5-HT1A receptor full agonist of the azapirone chemical class. It has both antidepressant and anxiolytic effects.</p>Fórmula:C26H39ClN2O4Forma y color:SolidPeso molecular:479.06CB1R Allosteric modulator 3
CAS:<p>CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.</p>Fórmula:C22H17ClN2O2Pureza:98.18%Forma y color:SolidPeso molecular:376.84NIC
CAS:<p>NIC is an inhibitor of host invasion. It is also an inhibitor of VEGF binding to immobilized heparin.</p>Fórmula:C15H16ClN3O3Pureza:98%Forma y color:SolidPeso molecular:321.76PAF (C16)
CAS:<p>PAF (C16) is a potent MAPK and MEK/ERK activator that induces increased vascular permeability.</p>Fórmula:C26H54NO7PPureza:98%Forma y color:SolidPeso molecular:523.68MK204
CAS:<p>MK204 is an inhibitor of AKR1B10, a tumor marker and promising antineoplastic target.</p>Fórmula:C16H9Br5ClNO4Pureza:98%Forma y color:SolidPeso molecular:714.22Bufetolol
CAS:<p>Bufetolol is an antagonist of beta-adrenoceptor.</p>Fórmula:C18H29NO4Pureza:98%Forma y color:SolidPeso molecular:323.43Antimycobacterial agent-1
CAS:<p>Compound 33: antimycobacterial, MIC 1 μg/ml vs M. tuberculosis H37Ra, low toxicity (IC50 143.2 μg/ml in Vero cells).</p>Fórmula:C18H12N4O5SForma y color:SolidPeso molecular:396.38LSP1-2111
CAS:<p>LSP1-2111 is a mGlu4 receptor subtype agonist.</p>Fórmula:C12H17N2O9PForma y color:SolidPeso molecular:364.25LKM38
CAS:<p>LKM38, a cholesterol probe, mimics cholesterol, supports resistant cell growth, and regulates homeostasis, aiding in cholesterol protein studies.</p>Fórmula:C28H44N2OPureza:97.75%Forma y color:SolidPeso molecular:424.66FGF/PDGF/VEGF RTK Inhibitor
CAS:<p>Potent, reversible ATP-competitive inhibitor for PDGFRβ, FGFR-1, VEGFR-2 (IC50: 20, 90, 240 nm); hinders VEGF-driven HMVEC growth (EC50: 420 nm).</p>Fórmula:C16H11N3O2Forma y color:SolidPeso molecular:277.28MDK8228
CAS:<p>MDK8228 is an inhibitor of CBP/p300 and BRD4 bromodomain. MDK8228 downregulates IL-6, IL-ß and IFN-ß in macrophages.</p>Fórmula:C31H41N5O3Forma y color:SolidPeso molecular:531.69Fasobegron
CAS:<p>Fasobegron is a agonist of β3-adrenoreceptor .</p>Fórmula:C24H24ClNO4Forma y color:SolidPeso molecular:425.91
