Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65495 productos de "Derivados de Quinazolina y Quinolina"
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(Z)-Methyl 3-(hydroxy(phenyl)methylene)-2-oxoindoline-6-carboxylate
CAS:Fórmula:C17H13NO4Forma y color:NeatPeso molecular:295.29N-Ethoxycarbonyl Norfloxacin
CAS:Fórmula:C19H22FN3O5Forma y color:White To Off-WhitePeso molecular:391.391,1-Cyclohexanediacetic Acid Monoamide
CAS:Producto controlado<p>Applications 1,1-Cyclohexanediacetic acid monoamide is an impurity of Gabapentin (G117250), an amino acid structurally related to γ-Aminobutyric Acid (GABA), designed to cross the blood brain barrier. Gabapentin is used as an anticonvulsant.<br>References Vollmer, K.-O. et al.: Arzneimittel-Forshc., 36, 830 (1986), Saletu, B., et al.: Int. J. Clin. Pharmacol. Ther. Toxicol., 24, 362 (1986)<br></p>Fórmula:C10H17NO3Forma y color:White To Off-WhitePeso molecular:199.247N-Chloro Ethyl ThioTEPA
CAS:Producto controlado<p>Stability Hygroscopic, Moisture Sensitive<br>Applications N-Chloro Ethyl ThioTEPA is an impurity of ThioTEPA which is an alkylating agent used to treat cancer.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Maanen, M., et al.: Cancer Treatment Rev., 26, 257 (2000); Sykes, M., et al.: Cancer, 6, 142 (1953)<br></p>Fórmula:C6H13ClN3PSForma y color:White To Off-WhitePeso molecular:225.68Nimodipine
CAS:<p>Applications A dihydropyridine calcium channel blocker. It is used as a vasodilator (cerebral). Neuroprotective & Neuroresearch products.<br>References Allen, G.S., et al.: N. Engl. J. Med., 308, 619 (1983), Schluter, H.: Arzneim.-Forsch., 36, 1733 (1986), Deyo, R.A., et al.: Science, 243, 809 (1989),<br></p>Fórmula:C21H26N2O7Forma y color:NeatPeso molecular:418.44Vismodegib
CAS:Producto controlado<p>Applications Vismodegib targets the Hedgehog (Hh) pathway. Inhibition of the Hh signaling may be effective in the treatment and prevention of many types of human cancers. Potent Hedgehog inhibitor.<br>References Gupta, S. et al.: Ther. Advances in Med. Oncology 2,237(2010)<br></p>Fórmula:C19H14Cl2N2O3SForma y color:Off-WhitePeso molecular:421.30Alogliptin-d3
CAS:Producto controlado<p>Applications Labelled Alogliptin (A575425). It is an oral antihyperglycemic agent that is a selective inhibitor of the enzyme dipeptidyl peptidase-4 (DPP-4). Antidiabetic agent.<br>References Lynn, F., et al.: Diabetes, 50, 1004 (2001), Trumper, A., et al.: J. Endocrinol., 174, 233 (2002), Vollmer, K., et al.: J. Clin. Endocrinol. Metab., 94, 1379 (2009),<br></p>Fórmula:C182H3H18N5O2Forma y color:NeatPeso molecular:342.41Trametinib
CAS:Producto controlado<p>Applications Used in the systematic treatment of advanced cutaneous melanoma. An EGFR kinase inhibitor and potent MEK inhibitor.<br>References Ercan, D. et al.: Canc. Disc., 2, 934 (2012); Mackiewicz-Wysocka, M. et al.: Exp. Opin. Investig. Drugs., 22, 181 (2013);<br></p>Fórmula:C26H23FIN5O4Forma y color:Off-WhitePeso molecular:615.39Irbesartan-d4
CAS:Producto controlado<p>Applications Irbesartan-d4 is the labeled analogue of Irbesartan (I751000), an angiotensin II type 1 (AII1)-receptor antagonist.<br>References Gillis, J.C. and Markham, A.: Drugs, 54, 885 (1997); Chando, T.J., et al.: Drug. Metabol. Dispos., 26, 408 (1998); Massie, B., et al.: New Eng. J. Med., 359, 2456 (2008); Ren, X., et al.: Pharmacol., 83, 80 (2009)Aromatics, Heterocycles, Inhibitors, Isotope Labelled Compounds, Pharmaceuticals, Intermediates & Fine Chemicals<br></p>Fórmula:C25H24D4N6OForma y color:NeatPeso molecular:432.55Felbamate-d4
CAS:Producto controlado<p>Applications Antiepileptic, structurally similar to meprobamate.<br>References Swinyard, E.A., et al.: Epilepsia, 27, 27 (1986), Remmel, R.P., et al.: Ther. Drug Monit., 12, 90 (1990), Sofia, R.D., et al.: Epilepsy Res. Suppl., 3, 103 (1991),<br></p>Fórmula:C11H10D4N2O4Forma y color:NeatPeso molecular:242.267Vildagliptin Amide
CAS:Producto controlado<p>Impurity Vildagliptin Amide Impurity<br>Applications N-(3-Hydroxytricyclo[3.3.1.13,7]dec-1-yl)glycyl-L-prolinamide is an impurity of Vildagliptin (V305000) which is an oral anti-hyperglycemic agent that inhibit dipeptidyl peptidase 4 (DPP-4).<br>References Ahren, B., et al.: J. Clin. Endocrinol. Metab., 89, 2078 (2004), Ahren, B., et al.: Diabetes Care, 27, 2874 (2004), Barlocco, D., et al.: Curr. Opin. Invest. Drugs, 5, 1094 (2004),<br></p>Fórmula:C17H27N3O3Forma y color:Off-WhitePeso molecular:321.41Nifursol (~90%)
CAS:Producto controlado<p>Applications A medicinal, prophylactic additive in animal feeds, protecting poultry from histomoniasis.Environmental contaminants; Food contaminants; Heat processing contaminants<br>References Kowalski, P., et al.: J. Pharm. Biomed. Anal., 32, 937 (2003), Khlebnikov, A., et al.: Bioorg. Med. Chem., 16, 9302 (2008), Schepetkin, I., et al.: Mol. Pharmacol., 74, 392 (2008),<br></p>Fórmula:C12H7N5O9Pureza:~90%Forma y color:NeatPeso molecular:365.21Methyl 4’-[[2-n-Propyl-4-methyl-6-(1-methylbenzimidazol-2-yl)-benzimidazol-1-yl]methyl]biphenyl-2-ca
CAS:Fórmula:C34H32N4O2Forma y color:YellowPeso molecular:528.64Maraviroc
CAS:Producto controladoFórmula:C29H41F2N5OForma y color:White To Off-WhitePeso molecular:513.674-Anilino-4-oxobutanoic Acid
CAS:Producto controlado<p>Applications The metabolite (MII) of Suberoylanilide Hydroxamic Acid (S688700).<br>References Sun, W.S., et al.: J. Med. Chem., 46, 5619 (2003)<br></p>Fórmula:C10H11NO3Forma y color:NeatPeso molecular:193.201-(4-Aminophenyl)-5,6-dihydro-3-(4-morpholinyl)-2(1H)-pyridinone
CAS:Producto controlado<p>Applications 1-(4-Aminophenyl)-5,6-dihydro-3-(4-morpholinyl)-2(1H)-pyridinone is an intermediate in the synthesis of Apixaban (A726700), A potent, direct, selective, and orally active inhibitor of coagulation factor Xa. It is a potential new oral coagulant that may be useful prevention of venous thromboembolism in total hip, knee replacement orthopedic surgery and stroke in treatment of patient with venous thromboembolic disorder or with atrial fibrillation.<br>References Nevuluri, N. et al.: Monat. fuer Chem., 148, 1477 (2017);<br></p>Fórmula:C15H19N3O2Forma y color:NeatPeso molecular:273.33Flubendazole-d3
CAS:Producto controladoFórmula:C162H3H9FN3O3Forma y color:Off-WhitePeso molecular:316.302-Bromo-6-methoxynaphthalene (Naproxen Impurity N)
CAS:<p>Impurity Naproxen EP Impurity N<br>Applications Naproxen Impurity N.<br>References Markku, A., et al.: J. Pharm. Sci., 66, 433 (1977), Hamai, S., et al.: J. Phys. Chem., 99, 12109 (1995), Kearney, P., et al.: Br. Med. J., 332, 1302 (2006),<br></p>Fórmula:C11H9BrOForma y color:WhitePeso molecular:237.092-Amino-4-isopropylamino-6-chlorotriazine
CAS:Producto controlado<p>Applications Studies have shown compounds of this nature are of pharmacological interest. Also has been shown to inhibit the growth of plants.<br>References Pearlman, W.M., et al.: J.A.C.S. , 70, 3726 (1948), Thurston, J.T., et al.: J.A.C.S., 73, 7, 2981 (1951)<br></p>Fórmula:C6H10ClN5Forma y color:Off-WhitePeso molecular:187.63O-Desmethyl Felodipine
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications O-Desmethyl metabolite of the calcium channel blocker Felopidine (F232375).<br>References Uno, K. et al.: Yakub. Dotai, 7, 243 (1992);<br></p>Fórmula:C17H17Cl2NO4Forma y color:NeatPeso molecular:370.23Udenafil
CAS:Producto controlado<p>Applications Udenafil is an oral phosphodiesterase 5 inhibitor used for the treatment of erectile dysfunction.<br>References Kim, T. et al.: Br. J. Clin. Pharmacol., 68, 43 (2009); Lee, C. et al.: J. Sex Med., 7, 2564 (2010); Bae, S.K. et al.: Biomed. Chrom., 22, 939 (2008);<br></p>Fórmula:C25H36N6O4SForma y color:Off White SolidPeso molecular:516.66Ref: 10-F625925
1gA consultar5gA consultar10gA consultar100mgA consultar250mgA consultar500mgA consultar6β-Hydroxy Dutasteride
<p>Applications 6β-Hydroxy Dutasteride is a hydroxylated derivative of Dutasteride (D735000).<br></p>Fórmula:C27H30F6N2O3Forma y color:NeatPeso molecular:544.431-Phenyl-3-(thiophen-2-yl)-1h-pyrazole-4-carboxylic acid
CAS:Pureza:97%Peso molecular:270.30999755859375Levetiracetam
CAS:<p>Applications The (S)-enantiomer of Etiracetam (E932970) and the ethyl analog of Piracetam (P500800). Used as an anticonvulsant. Neuroprotective & Neuroresearch Product.<br>References Gower, A.J., et al.: Eur. J. Pharmacol., 222, 193 (1992); Kasteleijn-Noist Trenite, D.G.A., et al.: Epilepsy Res., 25, 225 (1996); Patsalos, P.N., et al.: Pharmacol. Ther., 85, 77 (2000)<br></p>Fórmula:C8H14N2O2Forma y color:NeatPeso molecular:170.21(2S,3S,5S)-5-Amino-1,6-diphenyl-2-([[thiazol-5-ylmethoxy)carbonyl]amino]hexan-3-yl 2-(3-((2-isopropylthiazol-4-yl)methyl)-3-methylureido)-3-methylbutanoate Hydrochloride
CAS:Producto controlado<p>Applications (2S,3S,5S)-5-amino-1,6-diphenyl-2-([[thiazol-5-ylmethoxy)carbonyl]amino]hexan-3-yl 2-(3-((2-isopropylthiazol-4-yl)methyl)-3-methylureido)-3-methylbutanoate Hydrochloride, is a prodrug of Ritonavir (R535000), which is a selective HIV protease inhibitor.<br>References Daluge, S., et al.: Antimicrob. Agents Chemother., 38, 1590 (1994), Ammaranond, P., et al.: J. Clin. Virol., 26, 153 (2003), Harrigan, P., et al.: J. Infect. Dis., 191, 339 (2005), Miller, J., et al.: Bioorg. Med. Chem. Lett., 16, 1788 (2006);<br></p>Fórmula:C37H48N6O5S2•xHClForma y color:NeatPeso molecular:720.944,5,6,7-Tetrahydro-1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxo-1-piperidinyl)phenyl]-1H-Pyrazolo[3,4-c]pyridine-3-carboxylic Acid Methyl Ester
CAS:Producto controladoFórmula:C26H26N4O5Forma y color:NeatPeso molecular:474.508N-(4-{[(Pyridin-4-ylmethyl)amino]methyl}phenyl)-acetamide
CAS:Fórmula:C15H17N3OPureza:98%Forma y color:SolidPeso molecular:255.3212,2'-Dithiobis[N-methyl-benzamide]
CAS:<p>Applications Benzamide, 2,2'-dithiobis[N-methyl- (cas# 2527-58-4) is a useful research chemical.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Fórmula:C16H16N2O2S2Forma y color:Light Yellow To Light BeigePeso molecular:332.445-Aminoimidazole-4-carboxamide
CAS:<p>Applications A metabolite of Temozolomide.<br>References Jaeken, J., et al.: Lancet, 2, 1058 (1984), Baggott, J., et al.: Biochem. J., 236, 193 (1986), Baggott, J., et al.: Arch. Dermatol., 135, 813 (1999),<br></p>Fórmula:C4H6N4OForma y color:White To Off-WhitePeso molecular:126.126-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole
CAS:Producto controlado<p>Applications An Intermediate in the synthesis of risperidone and iloperidone.<br></p>Fórmula:C12H13FN2OForma y color:NeatPeso molecular:220.24(S)-Naproxen
CAS:<p>Applications (S)-Naproxen is a a nonsteroidal anti-inflammatory compound with analgesic and antipyretic properties (1,2). (S)-Naproxen is also a potent COX1 inhibitor.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References (1) Harrison, I.T., et al.: J. Med. Chem., 13, 203 (1970)(2) Scott, W. W., et al.: World Neurosurg. 82, e633 (2014)<br></p>Fórmula:C14H14O3Forma y color:Off-WhitePeso molecular:230.26Dolutegravir O-b-D-Glucuronide Sodium salt
Fórmula:C26H26F2N3NaO11Forma y color:White To Off-WhitePeso molecular:617.49Celecoxib
CAS:Producto controlado<p>Applications Celecoxib is a selective cyclooxygenase-2 (COX-2) inhibitor. Anti-inflammatory. Used in treatment of familial adenomatous polyposis. Celecoxib is a nonsteroidal anti-inflammatory drug (NSAID). It works by reducing hormones that cause inflammation and pain in the body.Celecoxib is used to treat pain or inflammation caused by many conditions such as arthritis, ankylosing spondylitis, and menstrual pain. Celecoxib is also used in the treatment of hereditary polyps in the colon<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Simon, L.S., et al.: Arthritis Rheum., 41, 1591 (1998), Silverstein, F.E., et al.: J. Am. Med. Assoc., 284, 1247 (2000), Steinbach, G., et al.: N. Engl. J. Med., 342, 1946 (2000),<br></p>Fórmula:C17H14F3N3O2SForma y color:NeatPeso molecular:381.37Gabapentin-d4
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Amino acid structurally related to γ-Aminobutyric Acid (GABA), designed to cross the blood brain barrier. Used as an anticonvulsant.<br>References Vollmer, K.-O. et al.: Arzneimittel-Forshc., 36, 830 (1986), Saletu, B., et al.: Int. J. Clin. Pharmacol. Ther. Toxicol., 24, 362 (1986)<br></p>Fórmula:C9D4H13NO2Forma y color:Off-WhitePeso molecular:175.26Ezetimibe Diol Impurity
CAS:Producto controladoFórmula:C24H25F2NO3Forma y color:NeatPeso molecular:413.46cis Lacidipine
CAS:Producto controlado<p>Stability Light Sensitive<br>Applications Z-Isomer of Lacidipine; a dihydropyridine calcium channel blocker. Antihypertensive.<br>References Safar, M., et al.: Clin. Pharmacol. Ther., 46, 94 (1989), Kharat, V.R., et al.: J. Pharm. Biomed. Anal., 28, 789 (2002), McCormack, A.J., et al.: Drugs, 63, 2327 (2003),<br></p>Fórmula:C26H33NO6Forma y color:NeatPeso molecular:455.54Ezetimibe-d4 β-D-Glucuronide, >85%
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Phase-II labelled metabolite of Ezetimibe, an antihyperlipoproteinemic. A cholesterol absorption inhibitor.<br>References van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997), van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Fórmula:C30H25D4F2NO9Pureza:>85%Forma y color:NeatPeso molecular:589.57Perphenazine Sulfoxide
CAS:Producto controlado<p>Impurity Perphenazine EP Impurity A<br>Applications Perphenazine Sulfoxide (Perphenazine EP Impurity A) acts as a D2 dopamine receptor antagonist; α-adrenergic receptor antagonist and σ-receptor agonist; phenothiazine antipsychotic. Inhibits glutamate dehydrogenase in vitro. Antipsychotic.<br>References Gaertner, H.J., et al.: Drug Metab. Dispos., 3, 437 (1975), O Brien, S., et al.: J. Med. Chem., 48, 1287 (2005), Briggs, K., et al.: Toxicology, 231, 113 (2007), Toga, T., et al.: J. Pharmacol. Sci., 105, 207 (2007),<br></p>Fórmula:C21H26ClN3O2SForma y color:NeatPeso molecular:419.97Dasatinib Carboxylic Acid Ethyl Ester
CAS:Producto controlado<p>Applications Protected Dasatinib Carboxylic Acid (D193605). An oxidative metabolite of Dasatinib (M6 metabolite); used in the treatment of cancers and immune diseases. It is a COVID19-related research product.<br>References Jaworski, T., et al.: Xenobiotica, 21, 1451 (1991), Shah, N., et al.: Science, 305, 399 (2004), O'Hare, T., et al.: Cancer Res., 65, 4500 (2005), Das, J., et al.: J. Med. Chem., 49, 6819 (2006), Christopher, L., et al.: Drug Metab. Dispos., 36, 1341 (2008),<br></p>Fórmula:C24H28ClN7O3SForma y color:NeatPeso molecular:530.04N-Nitroso-N-methyl-4-aminobutyric Acid (200 μg/mL in Methanol)
CAS:Fórmula:C5H10N2O3Forma y color:ColourlessPeso molecular:146.14(R)-2-((4-Aminophenethyl)amino)-1-phenylethanol
CAS:Producto controladoFórmula:C16H20N2OForma y color:NeatPeso molecular:256.34Iso Loratadine
CAS:Producto controlado<p>Impurity Loratadine EP Impurity E<br>Applications Iso Loratadine (Loratadine EP Impurity E) is a Loratadine (L469575) impurity. An isomer of Loratadine used for preparation of tricyclic amides and ureas useful for inhibition of G-protein function and for treatment of proliferative diseases.<br>References Billah., et al.: Lipids, 26, 1172 (1991), Piwinski., et al.: J. Med. Chem., 34, 457 (1991),<br></p>Fórmula:C22H23ClN2O2Forma y color:NeatPeso molecular:382.88N-Desmethyl Diphenhydramine Hydrochloride
CAS:<p>Applications N-Desmethyl Diphenhydramine is an impurity of Diphenhydramine (D486900) with antihistaminic activity.<br>References Nauta, W. T. et al.: Med. Chem., Spec. Contrib. Int. Symp., 3rd, 125 (1973);<br></p>Fórmula:C16H19NO·ClHForma y color:White To Light BeigePeso molecular:277.794’-O-Benzyloxy Ezetimibe
CAS:Producto controlado<p>Impurity Ezetimibe Benzyl Ether Impurity<br>Applications Protected Ezetimibe, used for the synthesis of related derivatives.<br>References Raman, B., et al.: J. Pharm. Biomed. Anal., 52, 73 (2010),<br></p>Fórmula:C31H27F2NO3Forma y color:NeatPeso molecular:499.55N-Acetyldesloratadine
CAS:Producto controlado<p>Applications N-Acetyldesloratadine is an impurity in the synthesis of Desloratadine (D290250), Nonsedating-type histamine H1-receptor antagonist.<br>References Kreutner, W., et al.: Arzneimittel-Forsch., 50, 345 (2000); Salmun, L.M., et al.: Clin. Ther., 22, 613 (2000); Agrawal, D.K., et al.: Expert Opin. Invest. Drugs, 10, 547 (2001);<br></p>Fórmula:C21H21ClN2OForma y color:NeatPeso molecular:352.863-cyclopropyl-1-phenyl-1H-pyrazole-5-carboxylic acid
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:228.25100708007812(2S)-1-(2-Chloroacetyl)-2-9-pyrrolidinecarbonitrile
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications (2S)-1-(2-Chloroacetyl)-2-9-pyrrolidinecarbonitrile is a key intermediate for dipeptidyl peptidase IV inhibitor Vildagliptin (V305000).<br>References Singh, S.K., et al.: Beil. J. Org. Chem., 4, 20 (2008);<br></p>Fórmula:C7H9ClN2OForma y color:NeatPeso molecular:172.611-(3-Cyano-2-pyridyl)-4-methyl-2-phenylpiperazine
CAS:<p>Applications Used in the preparation of Mirtazapine (M365000) impurities.<br></p>Fórmula:C17H18N4Forma y color:Light Yellow To BrownPeso molecular:278.35Levomepromazine EP Impurity D
Producto controladoFórmula:C32H33N3O2S2Forma y color:NeatPeso molecular:555.82-Amino-4-thiazoleacetic Acid
CAS:Producto controladoFórmula:C5H6N2O2SForma y color:NeatPeso molecular:158.18Iso Sildenafil
CAS:Producto controlado<p>Applications Iso Sildenafil is the isomer of Sildenafil methylated at N-2 position of the pyrazolo[4,3-d]pyrimidin-7-one nucleus.<br>References Sheldrick, G., et al.: Acta Crystallogr., A46, 467 (1990), Terrett, N., et al.: Bioorg. Med. Chem. Lett., 6, 1819 (1996),<br></p>Fórmula:C22H30N6O4SForma y color:NeatPeso molecular:474.58(S)-(-)-4’-Hydroxyphenyl Carvedilol
CAS:Producto controlado<p>Applications An optically active metabolite of Carvedilol (C184625), a nonselective ß-adrenergic blocker with α1-blocking activity.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., ET AL.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 10, 958 (1998),<br></p>Fórmula:C24H26N2O5Forma y color:NeatPeso molecular:422.472-(1-Nitroso-4-piperidinyl)-1H-benzimidazole
CAS:Producto controladoFórmula:C12H14N4OForma y color:NeatPeso molecular:230.2661-(4-Chlorophenyl)-5-(furan-2-yl)-1h-pyrazole-3-carboxylic acid
CAS:Pureza:95%Peso molecular:288.69000244140625Risperidone EP Impurity J
CAS:<p>Impurity Risperidone EP Impurity J<br>Applications 3-[2-[4-[(Z)-(4-Fluoro-2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)piperidin-1-yl)phenyl](hydroxyimino)methyl]piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one (Risperidone EP Impurity J) is a Risperidone (R525000) impurity.<br></p>Fórmula:C35H40F2N6O3Forma y color:White To YellowPeso molecular:630.7273Meloxicam
CAS:<p>Applications Preferential cyclooxygenase (COX-2) inhibitor. Sudoxicam and Meloxicam are nonsteroidal anti-inflammatory drugs (NSAIDs) from the enol-carboxamide class.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hawkey, C., et al.: Br. J. Rheumatol., 35, Suppl. 1, 1 (1996), Fleischmann, R., et al.: Expert Opin. Pharmacother., 3, 1501 (2002),<br></p>Fórmula:C14H13N3O4S2Forma y color:Light YellowPeso molecular:351.40rac-trans-Ambroxol-d5
CAS:Producto controlado<p>Applications A labelled metabolite of Bromohexine. Ambroxol Hydrochloride is a bronchosecretolytic drug.<br>References Jauch, R., et al.: Arzneim-Forsch., 13, 474 (1963)<br></p>Fórmula:C13H13D5Br2N2OForma y color:NeatPeso molecular:383.13Aripiprazole-d8 (Butyl-d8)
CAS:Producto controladoFórmula:C232H8H19Cl2N3O2Forma y color:White To Off-WhitePeso molecular:456.434-(2-(4-CHLORO-5H-PYRROLO[2,3-D]PYRIMIDIN-7(6H)-YL)ETHYL)MORPHOLINE
CAS:Pureza:95.0%Peso molecular:268.75Vildagliptin Racemic
CAS:<p>Applications Vildagliptin Racemic is an impurity of Vildagliptin (V305000),a class of oral anti-hyperglycemic agents that inhibit dipeptidyl peptidase 4 (DPP-4), which can act as a serine exopeptidase. Aside from their use in type 2 diabetes, gliptins have positive cardiovascular and anti-inflammtatory effects. Antidiabetic.<br>References Ahren, B., et al.: J. Clin. Endocrinol. Metab., 89, 2078 (2004), Ahren, B., et al.: Diabetes Care, 27, 2874 (2004), Barlocco, D., et al.: Curr. Opin. Invest. Drugs, 5, 1094 (2004),<br></p>Fórmula:C17H25N3O2Forma y color:NeatPeso molecular:303.399Risperidone Carboxylate Impurity
CAS:Producto controlado<p>Impurity Risperidone EP Impurity F<br>Applications Risperidone Carboxylate Impurity (Risperidone EP Impurity F) is a Risperidone (R525000) impurity.<br></p>Fórmula:C24H27FN4O4Forma y color:NeatPeso molecular:454.494’-Hydroxyphenyl Carvedilol-d3
CAS:Producto controlado<p>Applications A labelled metabolite of Carvedilol (C184625). It is used in the treatment of hypertension.<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., ET AL.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 10, 958 (1998),<br></p>Fórmula:C242H3H23N2O5Forma y color:NeatPeso molecular:425.49Sulindac Acyl-β-D-Glucuronide
CAS:Producto controlado<p>Applications Sulindac Acyl-β-D-Glucuronide is the major metabolite of the non-steroidal anti-inflammatory drug Sulindac (S699215) in plasma and urine.<br>References Hucker, H.B., et al.: Drug Metab. Dispos., 1, 721 (1973),<br></p>Fórmula:C26H25FO9SForma y color:NeatPeso molecular:532.533-Methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinemethanol
CAS:Producto controladoFórmula:C9H10F3NO2Forma y color:Light Beige To Light BrownPeso molecular:221.07DL-Erythro Ritalinic Acid
CAS:Producto controlado<p>Applications A major metabolite of Methylphenidate.<br>References Redalieu, E., et al.: Drug Metab. Dispos., 10, 708 (1982), Brewer, E., et al.: J. Pharm. Sci., 87, 395 (1998), Shah, V., et al.: Pharm. Res., 17, 1551 (2000), Tanaka, N., et al.: Anal. Chem., 73, 420 (2001),<br></p>Fórmula:C13H17NO2Forma y color:WhitePeso molecular:219.28Aprepitant-d4
CAS:Producto controlado<p>Applications Aprepitant-d4 is a labeled analogue of Aprepitant (A729800), A novel selective neurokinin-1 (NK-1) receptor antagonist. In vitro studies using human liver microsomes indicate that Aprepitant is metabolised primarily by CYP3A4 with minor metabolism by CYP1A2 and CYP2C19, and no metabolism by CYP2D6, CYP2C9, or CYP2E1. Aprepitant-d4 is a potential treatment for chemotherapy induced nausea and vomiting.<br>References Hale, J.J., et al.: J. Med. Chem., 41, 4607 (1998); Campos, D., et al.: J. Clin. Oncol., 19, 1759 (2001); Van Belle, S., et al.: Cancer, 94, 3032 (2002); Majumdar, A.K., et al.: J. Clin. Pharmacol., 46, 291 (2006)<br></p>Fórmula:C23H17D4F7N4O3Forma y color:NeatPeso molecular:538.45Rebamipide 3-Chloro Impurity (>80%)
CAS:Producto controlado<p>Applications Rebamipide 3-Chloro Impurity (CAS# 90098-05-8) is a useful research chemical compound.<br></p>Fórmula:C19H15ClN2O4Pureza:>80%Forma y color:White To Off-WhitePeso molecular:370.7864rac-Epinephrine-3-O-sulfate
CAS:Fórmula:C9H13NO6SForma y color:White To Off-WhitePeso molecular:263.268Baricitinib
CAS:Producto controlado<p>Applications Baricitinib is a JAK1 and JAK2 inhibitor and have been used as a promising treatment for rheumatoid arthritis.<br>References Greenwald, L.J., et al.: Int. J. Clin. Rheumatol., 6, 401 (2011); Fridman, J.S., et al.: J. Immunol., 184, 5298 (2010);<br></p>Fórmula:C16H17N7O2SForma y color:White SolidPeso molecular:371.42N-[1-(1H-1,2,3-Benzotriazol-1-yl)-3-phenylpropyl]pyridine-4-carboxamide
Peso molecular:357.4169921875N1-Ethylcarbamoyl Cabergoline (>90%)
CAS:Fórmula:C29H42N6O3Forma y color:Off White SolidPeso molecular:522.68(S)-Pramipexole-d5 Dihydrochloride
CAS:Producto controlado<p>Applications (S)-Pramipexole-d5 Dihydrochloride is a labeled analogue of (S)-Pramipexole Dihydrochloride (P700755), a dopamine-D2-receptor agonist. Antiparkinsonian.<br>References Schilling, J.C., et al.: Clin. Pharmacol. Ther., 51, 541 (1992); Kieburtz, K., et al.: J. Am. Med. Assoc., 278, 125 (1997)<br></p>Fórmula:C10H14D5Cl2N3SForma y color:Off White SolidPeso molecular:289.28Desidustat
CAS:<p>Stability Hygroscopic<br>Applications Desidustat, is an HIF hydroxylase inhibitor.<br></p>Fórmula:C16H16N2O6Forma y color:NeatPeso molecular:332.31(R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic Acid Hydrochloride
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications (R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic Acid Hydrochloride is an intermediate in the synthesis of the new antidiabetic drug Sitagliptine (S491000); a trizolopyrazine dipeptidyl peptidase IV inhibitor.<br>References Tasnadi, G., et al.: Org. Biomol. Chem., 8, 793 (2010); Kim, D., et al.: J. Med. Chem. 48, 141 (2005); Ahren, B., et al.: Eur. J. Pharmacol. 521 164 (2005); Bergman, A., et al: Clin. Ther. 28, 55 (2006)<br></p>Fórmula:C10H10F3NO2·ClHForma y color:White To Off-WhitePeso molecular:269.65Topiramate
CAS:<p>Applications Used as an anticonvulsant.<br>References Maryanoff, B.E., et al.: J. Med. Chem., 30, 880 (1987); Bialer, M.: Clin. Pharmacokinet., 24(6), 441-52 (1993)<br></p>Fórmula:C12H21NO8SForma y color:White To Off-WhitePeso molecular:339.36Anastrozole Diamide
CAS:Producto controlado<p>Impurity Anastrozole Diamide Impurity<br>Applications Anastrozole Diamide is a derivative of Anastrozole (A637425), an aromatase inhibitor. Used as an antineoplastic. Anastrozole Diamide Impurity<br>References Plourde, P.V., et al.: Breast Cancer Res. Treat., 30, 103 (1994), Buzdar, A.U., et al.: Cancer, 79, 730 (1997)<br></p>Fórmula:C17H23N5O2Forma y color:WhitePeso molecular:329.403-Hydroxyagomelatine
CAS:<p>Impurity Agomelatine Impurity 11/ Agomelatine 3-Hydroxy Impurity<br>Applications 3-Hydroxyagomelatine is an intermediate in the synthesis of 1-(aminoethyl)naphthalene derivative with potential binding affinity for melatonin receptors. Agomelatine Impurity 11<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Simonin, G., et al.: J. Pharma. Biomed. Anal., 21, 591 (1999)<br></p>Fórmula:C15H17NO3Forma y color:NeatPeso molecular:259.3
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