Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65495 productos de "Derivados de Quinazolina y Quinolina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
2-(4-Chloro-3-difluoromethyl-5-methyl-pyrazol-1-yl)-propionic acid
CAS:Fórmula:C8H9ClF2N2O2Forma y color:SolidPeso molecular:238.62Methyl-(1-methyl-1H-pyrazol-3-ylmethyl)-amine
CAS:Pureza:95.0%Forma y color:Liquid, liquidPeso molecular:125.175003051757814-Amino-N-pyridin-3-ylmethylbenzamide
CAS:Fórmula:C13H13N3OPureza:97%Forma y color:SolidPeso molecular:227.2675-Difluoromethoxy-2-[(3,4-dimethoxy-2-pyridinyl)methyl]thio-1H-benzimidazole
CAS:Pureza:95.0%Peso molecular:367.36999511718752-[3-(4-nitrophenyl)-1-phenyl-1h-pyrazol-4-yl]acetic acid
CAS:Pureza:97%Peso molecular:323.30801391601564-(2-Pyrrolidinylmethyl)morpholine
CAS:Pureza:95.0%Forma y color:LiquidPeso molecular:170.255996704101563,5-Bis(trifluoromethyl)pyridine
CAS:Fórmula:C7H3F6NPureza:97%Forma y color:Solid, Low Melting SolidPeso molecular:215.0982-(3,4-Dimethoxy-phenyl)-quinoline-4-carboxylic acid hydrazide
CAS:Forma y color:SolidPeso molecular:323.351989746093751-Phenyl-2-pyrazin-2-yl ethanone
CAS:Fórmula:C12H10N2OPureza:95.0%Forma y color:SolidPeso molecular:198.225(3-Methoxypyridin-4-yl)boronic acid hydrate
CAS:Fórmula:C6H10BNO4Pureza:95.0%Forma y color:SolidPeso molecular:170.96(1H-Imidazol-2-yl)-thiophen-2-yl-methanone
CAS:Fórmula:C8H6N2OSForma y color:SolidPeso molecular:178.218-methyl-2-(5-methyl-2-furyl)quinoline-4-carboxylic acid
CAS:Pureza:95.0%Peso molecular:267.283996582031253-((3-(N-Cyclopropylsulfamoyl)-7-(2,4-dimethoxypyrimidin-5-yl)quinolin-4-yl)amino)-5-(3,5-difluorophenoxy)benzoic acid
CAS:Pureza:98%Peso molecular:649.630004882813Ref: 10-F867169
5mgA consultar10mgA consultar25mgA consultar50mgA consultar100mgA consultar250mgA consultarRef: 10-F794544
1gA consultar5gA consultar10mgA consultar25mgA consultar50mgA consultar100mgA consultar250mgA consultarDasatinib Dimeric Impurity
CAS:Producto controladoFórmula:C36H34Cl2N12O2S2Forma y color:White To BeigePeso molecular:801.77(S)-2-Hydroxy-3-methoxy-3,3-diphenylpropionic Acid
CAS:Producto controlado<p>Impurity Ambrisentan Hydroxy Acid Impurity<br>Applications (S)-2-Hydroxy-3-methoxy-3,3-diphenylpropionic Acid is used in analytical studies for chiral discrimination of α-functionalized acids. Ambrisentan Hydroxy Acid Impurity<br>References Jain, N., et al.: Tetrahedron, 70, 4343 (2014)<br></p>Fórmula:C16H16O4Forma y color:NeatPeso molecular:272.30rac Phenylephrine Hydrochloride
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Phenylephrine is a selective α1-adrenergic receptor agonist used as a decongestant. Phenylephrine lowers intraocular pressure and is used as an agent to dilate the pupil.<br>References Lorenzetti, O.J. et al.: Exp. Eye Res., 12, 80 (1971); Ando, J. et al.: Nip. Yakur. Zas., 61, 471 (1965);<br></p>Fórmula:C9H14ClNO2Forma y color:NeatPeso molecular:203.67[1-(2-Chloro-pyridine-3-carbonyl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester
CAS:Pureza:95.0%Peso molecular:353.8500061035156Tazarotene
CAS:<p>Applications An acetylenic retinoid prodrug converted to the active metabolite, Tazarotenic acid, with selective affinity for retinoic acid receptors RARβ and RARγ. Antiacne; antipsoriatic. Used in treatment of photodamaged skin.<br>References Tang-Liu, D.D.-S., et al.: Clin. Pharmacokinet., 37, 273 (1999), Roeder, A., et al.: Skin Pharmacol. Physiol., 17, 111 (2004),<br></p>Fórmula:C21H21NO2SForma y color:Light YellowPeso molecular:351.46Vadadustat
CAS:<p>Applications Vadadustat is a novel HIF (Hypoxia-inducible factor) stabilizer. It provides an effective anemia treatment in nondialysis-dependent chronic kidney disease.<br>References Pergola, P., et al.: Kidney Int., 90, 1115 (2016);<br></p>Fórmula:C14H11ClN2O4Forma y color:BeigePeso molecular:306.703-(1-benzofuran-2-yl)-1H-pyrazole
CAS:Pureza:95.0%Forma y color:Solid, Beige powderPeso molecular:184.197998046875Aminorex-d5
CAS:Producto controlado<p>Applications A labelled metabolite of Levamisole (L331100). Aminorex is an anorectic stimulant drug of the 2-amino-5-aryl oxazoline class. Aminorex has been shown to have locomotor stimulant effects similar to Methamphetamine (M258795).<br>References Poos, G., et al.: J. Med. Chem., 6, 266 (1963), Watson, A., et al.: Res. Vet. Sci., 45, 411 (1988), Russell, B., et al.: Pharmacol. Biochem. Behav., 51, 375 (1995),<br></p>Fórmula:C9D5H5N2OForma y color:NeatPeso molecular:167.219KAD-1229 Calcium Hydrate
CAS:Producto controladoFórmula:C19H24NO3·Ca·2H2OForma y color:NeatPeso molecular:704.916-Benzyloxy-7-methoxy-2-methyl-quinoline-3-carboxylic acid
Pureza:95.0%Peso molecular:323.3479919433594NAP 226-90
CAS:<p>Impurity Rivastigmine EP Impurity A; Rivastigmin USP Related Compound C<br>Applications NAP 226-90 (Rivastigmine EP Impurity A; Rivastigmin USP Related Compound C) is a S-Enantiomer metabolite of Rivastigmine, a brain selective acetylcholinesterase inhibitor.<br>References Rosler, M., et al.: Br. Med. J., 318, 633 (1999), Jann, M., et al.: Clin. Pharmacokinet., 41, 719 (2002), Frankfort, S., et al.: Int. J. Clin. Pract., 60, 646 (2006),<br></p>Fórmula:C10H15NOForma y color:WhitePeso molecular:165.23(R)-(+)-4’-Hydroxyphenyl Carvedilol
CAS:Producto controlado<p>Applications An optically active metabolite of Carvedilol (C184625), a nonselective ß-adrenergic blocker with α1-blocking activity.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., ET AL.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 10, 958 (1998),<br></p>Fórmula:C24H26N2O5Forma y color:NeatPeso molecular:422.47Telmisartan-d3 Acyl-β-D-glucuronide
CAS:Producto controlado<p>Applications Labelled Telmisartan Acyl-β-D-glucuronide (T017010). Telmisartan Acyl-β-D-glucuronide is a metabolite of Telmisartan (T017000).<br>References Abe, T., et al.: J. Biol. Chem., 274, 17159 (1999), Hirano, M., et al.: Drug Metab. Dispos., 34, 1229 (2006),<br></p>Fórmula:C39H35D3N4O8Forma y color:NeatPeso molecular:693.76Carprofen Glucuronide
CAS:<p>Stability Hygroscopic<br>Applications Carprofen Glucuronide is a derivative of Carprofen (C184350), a non steroidal anti-inflammatory that is used by veterinarians for the relief of arthritic systems in dogs. It can be used for joint pain or post operative inflammation. Carprofen, is also used for the relief from pain and inflammation associated with osteoarthritis, hip dysplasia and other joint issues.<br>References Randall, L.O., et al.: Arch. Int. Pharmacodyn., 220, 94 (1976), Yu, T.F., et al.: J. Clin. Pharmacol., 20, 347 (1980), O’Brien, W.M., et al.: Pharmacotherapy, 7, 16 (1987),<br></p>Fórmula:C21H20ClNO8Forma y color:Light BrownPeso molecular:449.843-Hydroxy Nevirapine
CAS:Producto controlado<p>Applications A metabolite of Nevirapine (N391275).<br>References Rettie, A., et al.: J. Biol. Chem., 263, 13733 (1988), Lamson, M., et al.: Biopharm. Drug Dispos., 20, 285 (1999), Guengerich, F., et al.: Chem. Res. Toxicol., 14, 611 (2001), Lu, W., et al.: Drug Metab. Dispos., 36, 1624 (2008),<br></p>Fórmula:C15H14N4O2Forma y color:NeatPeso molecular:282.301-(4-Bromophenyl)-5-methyl-1H-pyrazole-4-carboxylic acid hydrazide
CAS:Fórmula:C11H11BrN4OPureza:95.0%Peso molecular:295.144-Nitrophenethylamine Hydrochloride
CAS:Fórmula:C8H10N2O2·HClForma y color:Light BeigePeso molecular:166.18 + 36.46DL-Norepinephrine-d6 Hydrochloride, 85%
CAS:Producto controlado<p>Applications Antagonist of dibutyryl cyclic AMP in the regulation of narcosis. Norepinephrine modulates human dendritic cell activation by altering cytokine release.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Piguet, P., et al.: J. Exp. Med., 173, 673 (1991), Hosoi, J., et al.: Nature, 363, 159 (1993), Elenkov, I., et al.: Pharmacol. Rev., 52, 595 (2000), Kaplan, D., et al.: Immunity, 23, 611 (2005),<br></p>Fórmula:C82H6H5NO3·ClHPureza:85%Forma y color:NeatPeso molecular:211.685,10-Dihydro-2-methyl-4H-thieno[2,3-b][1,5]benzodiazepin-4-one (Olanzapine Impurity)
CAS:<p>Impurity Olanzapine EP Impurity B/ Olanzapeine USP Related Compound B<br>Applications Olanzapine impurity (Olanzapine EP Impurity B).<br>References Fenselau, C., et al.: Xenobiotica, 22, 1207 (1992), Moore, N., et al.: J. Pharmacol. Exper. Ther., 262, 545 (1992), Kassahun, K., et al.: Drug Metab. Dispos., 25, 81 (1997),<br></p>Fórmula:C12H10N2OSForma y color:NeatPeso molecular:230.292-Acetoxy-N-(2-thiazolyl)benzamide
CAS:Producto controlado<p>Applications 2-Acetoxy-N-(2-thiazolyl)-benzamide is used in the synthesis of thiazolides as novel antiviral agents. Used in the inhibition of hepatitis C virus replication. Nitazoxanide Impurity<br>References Edwards, G. et al.: J. Med. Chem., 54, 8670 (2011);<br></p>Fórmula:C12H10N2O3SForma y color:Off-WhitePeso molecular:262.28rac trans-Loxoprofen Alcohol
CAS:<p>Applications The cis-alcohol metabolite of Loxoprofen (L472900).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Terada, A., et al.: J. Med. Chem., 27, 212 (1984), Sugimoto, M., et al.: Biochem. Pharmacol., 42, 2363 (1991), Riendeau, D., et al.: Bioorg. Med. Chem. Lett., 14, 1201 (2004),<br></p>Fórmula:C15H20O3Forma y color:NeatPeso molecular:248.32Meloxicam
CAS:<p>Meloxicam (Metacam) is a Nonsteroidal Anti-inflammatory Drug.</p>Fórmula:C14H13N3O4S2Pureza:97.09% - 99.60%Forma y color:Light Yellow SolidPeso molecular:351.406-(4-Methoxyphenyl)-3-(pyridin-3-yl)pyrazolo[1,5-a]pyrimidine
CAS:Pureza:97.0%Peso molecular:302.33700561523444-(Trifluoromethyl)aniline
CAS:Producto controlado<p>Impurity Leflunomide EP Impurity A; Leflunomide USP Related Compound A<br>Applications 4-(Trifluoromethyl)aniline (Leflunomide EP Impurity A; Leflunomide USP Related Compound A) is a 4-Substituted aniline derivatives exert special hematotoxicity on the red blood cells and induce leukocytosis.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Weber, W., et al.: Pharmacol. Rev., 37, 25 (1985), Hein, D., et al.: Carcinogenesis, 14, 1633 (1993), Payton, M., et al.: Microbiology, 147, 1137 (2001), Mushtaq, A., et al.: J. Biol. Chem., 277, 12175 (2002),<br></p>Fórmula:C7H6F3NForma y color:NeatPeso molecular:161.124-(4-Morpholinyl)-1,2,5-thiadiazol-3(2H)-one 1-Oxide
CAS:Producto controlado<p>Impurity Timolol EP Impurity G; Timolol BP Impurity G<br>Stability Moisture Sensitive<br>Applications 4-(4-Morpholinyl)-1,2,5-thiadiazol-3(2H)-one 1-Oxide (Timolol EP Impurity G; Timolol BP Impurity G) is an impurity of Timolol (T4437005), an antihypertensive, an adrenergic blocking agent (1); antiarrhythmic (class II); antianginal; antiglaucoma (2) and antihypertensive (3) agent.<br>References 1. Wasson, B. et al.: J. Med. Chem. 1972 Jun;15(6):651-5.2. Heel, R. et al.: Drugs. 1979 Jan;17(1):38-55.3. Rofman, et al.: Hypertension. 1980 Sep-Oct;2(5):643-8.<br></p>Fórmula:C6H9N3O3SForma y color:WhitePeso molecular:203.224-OXO-5-(THIOPHEN-2-YLMETHYL)-4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE-3-CARBOXYLIC ACID
CAS:Pureza:95.0%Peso molecular:277.29998779296875R 84852
CAS:<p>Applications R 84852 is an impurity of paliperidone (P141000), a combined serotonin (5-HT2) and dopamine (D2) receptor antagonist.<br>References Solanki, P.V., et. al.: ACS Sustainable Chem. Eng., 1, 243 (2013)<br></p>Fórmula:C23H28FN3O4Forma y color:NeatPeso molecular:429.482-(((6-(Difluoromethoxy)-1H-benzo[d]imidazol-2-yl)sulfinyl)methyl)-3,4-dimethoxypyridine 1-oxide
CAS:Pureza:95.00%Peso molecular:399.3699951171875Nocodazole
CAS:<p>M05733 - Nocodazole</p>Fórmula:C14H11N3O3SPureza:98%Forma y color:Solid, Beige powderPeso molecular:301.32000732421875Ref: 10-M05733
1gA consultar1mgA consultar10mgA consultar50mgA consultar100mgA consultar250mgA consultar1-(4-Fluorophenyl)-5-(thiophen-2-yl)-1h-pyrazole-3-carboxylic acid
CAS:Pureza:95%Peso molecular:288.29998779296875Dasatinib monohydrate
CAS:Producto controladoFórmula:C22H26ClN7O2S·H2OForma y color:White To Off-WhitePeso molecular:506.02Aprepitant
CAS:Producto controlado<p>Applications Aprepitant is a neurokinin-1 antagonist and an antiemetic agent (1). It is used to prevent chemotherapy-induced nausea and vomiting (CINV) in colorectal cancer patients (2) Aprepitant has also been shown to induce apoptotic cell death and G1 arrest through Akt/p53 axis in pre-B acute lymphoblastic leukemia cells (3).<br>References (1) Takemoto, H., et al.: nt J Clin Oncol (2016) (2) Bayati, S., et al.: Eur J Pharmacol. 791, 274 (2016) (3) Navari, R.M.: Expert Rev Anticancer Ther. 4, 715 (2004)<br></p>Fórmula:C23H21F7N4O3Forma y color:Off-WhitePeso molecular:534.431-((4-Fluorophenyl)carbamoyl)cyclopropanecarboxylic Acid
CAS:Producto controladoFórmula:C11H10FNO3Forma y color:Off-WhitePeso molecular:223.2m-Ranolazine
CAS:Producto controlado<p>Applications m-Ranolazine is an impurity of Ranolazine Ethyl Dimer is an impurity of Ranolazine (R122500), an anti-ischemic agent which modulates myocardial metabolism. Antianginal.<br>References Chaitman, B.R., et al.: J. Am. Coll. Cardial., 43, 1375 (2004), McCormack, J.G., et al.: Gen. Pharmacol., 30, 639 (1998), Schofield, J.A.H., et al.: Expert Opin. Invest. Drugs, 11, 117 (2002),<br></p>Fórmula:C24H33N3O4Forma y color:NeatPeso molecular:427.536Benzyl (3-fluoro-4-(6-(2-methyl-2H-tetrazol-5-yl)pyridin-3-yl)phenyl)carbamate
CAS:Pureza:97%Peso molecular:404.4049987792969Chlorambucil
CAS:Producto controlado<p>Applications Chlorambucil is a alkylating agent that is used as an chemotherapy drug in the treatment of chronic lymphocytic leukemia. Chlorambucil is also used to treat non-Hodgkin's lymphoma (NHL) and Hodgkin's disease.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Cogia, A., et al.: Leuk. Lymph., 53, 1961 (2012); Tonino, S.H., et al.: Leuk. Lymph., 53, 1785 (2012); Smolej, L., et al.: Curr. Pharma. Design., 18, 3399 (2012);<br></p>Fórmula:C14H19Cl2NO2Forma y color:White To Light BeigePeso molecular:304.213-(5-Formylfuran-2-yl)-1-phenyl-1H-pyrazole-4-carbaldehyde
CAS:Pureza:98%Peso molecular:266.2560119628906Ambrisentan Methyl Ester
CAS:Producto controlado<p>Applications (S)-Methyl 2-((4,6-dimethylpyrimidin-2-yl)-oxy)-3-methoxy-3,3-diphenylpropanoate is a useful intermediate in the preparation of Ambrisentan. Ambrisentan is an Antihypertensive. Ambrisentan Impurity (A575860).<br>References Peng, X., et al.: J. Org. Chem., 77, 701 (2012), Riechers, H., et al.: J. Med. Chem., 39, 2123 (1996), Billman, G.E., et al.: Curr. Opin. Invest. Drugs, 3, 1483 (2002), Vatter, H., et al.: Clin. Neuropharmacol., 26, 73 (2003)<br></p>Fórmula:C23H24N2O4Forma y color:Off-WhitePeso molecular:392.45PTC-124
CAS:Producto controlado<p>Applications PTC-124 is a nonaminoglycoside that has been reported to induce ribosomes to read through premature nonsense stop signals on mRNA, allowing the production of full-length functional proteins,<br>References Yu, H. et al.: Int. J. Mol. Med., 33, 729 (2014); Aditya, S. et al.: J. Biomed. Pharm. Res., 2, 21 (2013);<br></p>Fórmula:C15H9FN2O3Forma y color:White To Off-WhitePeso molecular:284.244-Methoxy Moxonidine
CAS:Producto controladoFórmula:C10H15N5O2Forma y color:GreyPeso molecular:237.26Dipyridamole-d20 (Major)
CAS:Producto controlado<p>Applications Selective inhibitor of phosphodiesterase V (PDE 5); potent coronary vasodilator drug; adenosine transport inhibitor; inhibitor of platelet aggregation.A representative lot was: 36% d20; 25% d19; 13%d18; 24% d17; 1% d16.<br>References Buchalter, M.B., et al.: Postgrad. Med. J., 66, 531 (1990), Sundaram, M., et al.: J. Biol. Chem., 273, 21519 (1998), Denis, D., et al.: Eur. J. Pharmacol., 367, 343 (1999),<br></p>Fórmula:C24H20D20N8O4Forma y color:NeatPeso molecular:524.75Chlorpromazine N-Oxide
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Chlorpromazine N-Oxide is a metabolite of Chlorpromazine. Chlorpromazine exhibits antiadrenergic, antiserotonergic, anticholinergic, and antihistaminergic properties, and commonly used to treat schizophrenia.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Zhang, Z., et al.: Handbook of Metabolic Pathways of Xenobiotics, 3, 1102 (2014); Kigondu, E. M., et al.: MedChemComm, 5, 502 (2014); Yeung, P. K. F., et al.: Eur. J. Clin. Pharmacol., 45, 563 (1993)<br></p>Fórmula:C17H19ClN2OSForma y color:NeatPeso molecular:334.86N-Benzyl Salbutamon Hydrochloride
CAS:Producto controlado<p>Applications N-Benzyl Salbutamon Hydrochloride is an impurity of Albuterol (Salbutamol) (A514500), an β2-adrenoceptor agonist. Bronchodilator; tocolytic.<br>References 1. Collin, D. et al.: J. Med. Chem. 1970 Jul;13(4):674-80.2. Raidal, S. et al.: Vet. J. 2017 Apr;222:22-28.<br></p>Fórmula:C20H25NO3·ClHForma y color:NeatPeso molecular:363.88Intedanib
CAS:Producto controlado<p>Applications It is an indolinone derivative potently blocking VEGF-, PDGF-, and FGF-receptor kinases; an indolinone as triple angiokinase inhibitors. An antitumor agent.<br>References Sun, L., et al.: J. Med. Chem., 41, 2588 (1998); Xie, H., et al.: J. Med. Chem., 50, 4898 (2007); Hilberg, F., et al.: Cancer Res., 68, 4774 (2008); Roth, G., et al.: J. Med. Chem., 58, 1053 (2015)<br></p>Fórmula:C31H33N5O4Forma y color:NeatPeso molecular:539.62Gabapentin Related Compound D
CAS:<p>Impurity Gabapentin EP Impurity D; Gabapentin USP Related Compound D<br>Applications Gabapentin Related Compound D (Gabapentin EP Impurity D; Gabapentin USP Related Compound D) is a Gabapentin analogue.<br></p>Fórmula:C18H29NO3Forma y color:White To Off-WhitePeso molecular:307.43N-Desmethyl-N-cyclopentyl Tadalafil
CAS:Producto controlado<p>Applications N-Desmethyl-N-cyclopentyl Tadalafil is used as a reagent to synthesize tetracyclic cGMP-specific phosphodiesterase inhibitors, compounds that have potential to treat cardiovascular disorders and erectile dysfunction.<br>References Daugan, A. & Gellibert, F. Tetracyclic cGMP-specific Phosphodiesterase Inhibitors and Their Use in Disease Treatment. U.S. 6143746. Nov 7, 2000<br></p>Fórmula:C26H25N3O4Forma y color:NeatPeso molecular:443.49DL-Fenfluramine
CAS:Producto controlado<p>Applications Anorectic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Pinder, et al.: Drugs, 10, 241 (1975); Caccia, S., et al.: Eur. J. Clin. Pharmacol., 29, 221 (1985); Finner, N., et al.: Curr. Ther. Res., 38, 847 (1985);<br></p>Fórmula:C12H16F3NForma y color:NeatPeso molecular:231.26Tazarotene-d8
CAS:Producto controlado<p>Applications Labelled Tazarotene (T010050). An acetylenic retinoid prodrug converted to the active metabolite, Tazarotenic acid, with selective affinity for retinoic acid receptors RARβ and RARγ. Antiacne; antipsoriatic. Used in treatment of photodamaged skin.<br>References Tang-Liu, D.D.-S., et al.: Clin. Pharmacokinet., 37, 273 (1999), Roeder, A., et al.: Skin Pharmacol. Physiol., 17, 111 (2004),<br></p>Fórmula:C21H13D8NO2SForma y color:YellowPeso molecular:359.514-Nitro Lenalidomide
CAS:Producto controlado<p>Impurity Lenalidomide impurity<br>Applications Lenalidomide (L328000) analog. Lenalidomide impurity; Lenalidomide intermediate.<br>References Hashimoto, Y., et al.: Bioorg. Med. Chem., 10, 461 (2002),<br></p>Fórmula:C13H11N3O5Forma y color:NeatPeso molecular:289.24Dechloro-Rivaroxaban
CAS:Producto controlado<p>Applications Dechloro-Rivaroxaban is an impurity of Rivaroxaban (R538000), which is a novel antithrombotic agent. A highly potent and selective, direct FXa inhibitor.<br>References Ansell, J., et al.: Drugs, 64, 1 (2004), Eriksson, B., et al.: J. Thromb. Haemost., 3, 103 (2005), Kubitza, D., et al.: Clin. Pharmacol. Ther., 78, 412 (2005),<br></p>Fórmula:C19H19N3O5SForma y color:NeatPeso molecular:401.444-ethoxy-N-(pyridin-3-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Pureza:95.0%Peso molecular:285.3699951171875Maraviroc-d6
CAS:Producto controlado<p>Applications Potent, non-competitive CCR5 receptor antagonist; inhibits binding of HIV viral coat protein gp120. Antiviral.<br>References Fumero, E., et al.: Clin. Microbiol. Infect., 9, 1077 (2003), Walker, D.K., et al.: Drug Metab. Dispos., 33, 587 (2005), Wood, A., et al.: Prog. Med. Chem., 43, 239 (2005),<br></p>Fórmula:C29D6H35F2N5OForma y color:NeatPeso molecular:519.70(S)-Lisinopril Dimer
CAS:Producto controlado<p>Applications (S)-Lisinopril (L468985) impurity. Lisinopril Impurity G (Dimer Impurity)<br></p>Fórmula:C42H60N6O9Forma y color:WhitePeso molecular:792.96cis-(Z)-Flupentixol Dihydrochloride
CAS:Producto controlado<p>Applications Neuroleptic agent related structurally to thiothixene. Antipsychotic; neuroleptic agent; dopamine receptor antagonist.<br>References Nielsen, et al.: Acta Pharmacol. Toxicol., 32, 363 (1973), Post, M.L., et al.: Nature, 256, 342 (1975), Peuch, et al.: Neuropharmacology, 20, 1279 (1981),<br></p>Fórmula:C23H27Cl2F3N2OSForma y color:NeatPeso molecular:507.44rac-cis-N-Desmethyl Sertraline-d4 Hydrochloride
CAS:Producto controlado<p>Applications A labelled metabolite of Sertraline. N-Desmethyl Sertraline is significantly less active analogue as compared to the methylated compound, Sertraline.<br>References Welch, W.M., et al.: J. Med. Chem. 27, 1508 (1984)<br></p>Fórmula:C16H12D4Cl3NForma y color:NeatPeso molecular:332.69Flubendazole
CAS:<p>Applications An anthelmintic.<br>References Thienpont, D., et al.: Arzneimittel-Forsch., 28, 605 (1978), Vanparijs, O., et al.: Vet. Parasitol, 5, 237 (1979),<br></p>Fórmula:C16H12FN3O3Forma y color:ColourlessPeso molecular:313.282-[3,5-Dichloro-4-(4-chlorobenzoyl)phenyl]-1,2,4-triazine-3,5(2H,4H)-dione
CAS:Producto controlado<p>Applications An anticoccidal triazine used for the treatment of coccidiosis in chickens. An impurity of Diclazuril (D436200).<br>References McFarland, J. et al.: J. Med. Chem., 35, 2543 (1992);<br></p>Fórmula:C16H8Cl3N3O3Forma y color:NeatPeso molecular:396.61(3S,4S,3’S)-Ezetimibe
CAS:<p>Applications (3S,4S,3’S)-Ezetimbe is a 3-epimer impurity of Ezetimibe (E975000), a cholesterol absorption inhibitor.<br>References van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997), van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Fórmula:C24H21F2NO3Forma y color:Off-WhitePeso molecular:409.433-Hydroxy Imiquimod
CAS:Producto controlado<p>Applications 4-Amino-β-methyl-1H-imidazo[4,5-c]quinoline-1-propanol, is an aryl ether substituted imidazoquinolines, which can be used in the design of immunomodulating agents for use as vaccine adjuvants and anticancer treatments.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Shi, C., et al.: ACS Med. Chem. Lett., 3, 501 (2012);<br></p>Fórmula:C14H16N4OForma y color:NeatPeso molecular:256.34-Morpholin-4-ylmethyl-1H-quinolin-2-one
CAS:Pureza:97.0%Forma y color:SolidPeso molecular:244.29400634765625(3aR,4S,6R,6aS)-6-Aminotetrahydro-2,2-dimethyl-4H-cyclopenta-1,3-dioxol-4-ol
CAS:<p>Stability Hygroscopic<br>Applications (3aR,4S,6R,6aS)-6-Aminotetrahydro-2,2-dimethyl-4H-cyclopenta-1,3-dioxol-4-ol was used to preapare AZD6140 as an orally active reversible P2Y12 receptor antagonist for prevention of thrombosis.<br>References Zhang, H., et al.: Bioorg. Med. Chem. Lett., 22, 3598 (2012);<br></p>Fórmula:C8H15NO3Forma y color:NeatPeso molecular:173.21Tianeptine
CAS:<p>Applications Tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Antidepressant.<br>References Malen, C., et al.: Experientia, 28, 811 (1972), Safa, A., et al.: J. Biol. Chem., 262, 7884 (1987), Ford, J.M., et al.: Pharmacol. Rev., 42, 155, (1990), Pierre, A., et a.: Cancer Res., 51, 2312 (1991),<br></p>Fórmula:C21H25ClN2O4SForma y color:White To Off-WhitePeso molecular:436.95Levosimendan Triazene Impurity
CAS:<p>Stability Light Sensitive<br>Applications Levosimendan Triazene is an impurity of Levosimendan (L378000); a positive inotropic agent with vasodilating activity. Also cardiotonic.<br>References Sandell, E.-P., et al.: J. Cardiovasc. Pharmacol., 26, S57 (1995); Pagel, P.S., et al.: Cardiovasc. Drug Rev., 14, 286 (1996)<br></p>Fórmula:C22H23N7O2Forma y color:NeatPeso molecular:417.46
![5-Difluoromethoxy-2-[(3,4-dimethoxy-2-pyridinyl)methyl]thio-1H-benzimidazole](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF049541.webp&w=3840&q=75)
![2-[3-(4-nitrophenyl)-1-phenyl-1h-pyrazol-4-yl]acetic acid](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF652524.webp&w=3840&q=75)
![[1-(2-Chloro-pyridine-3-carbonyl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF089109.webp&w=3840&q=75)
![5,10-Dihydro-2-methyl-4H-thieno[2,3-b][1,5]benzodiazepin-4-one (Olanzapine Impurity)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FD449185.webp&w=3840&q=75)
![6-(4-Methoxyphenyl)-3-(pyridin-3-yl)pyrazolo[1,5-a]pyrimidine](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF053860.webp&w=3840&q=75)
![2-{[2-(4-chlorophenyl)quinazolin-4-yl]amino}ethanol](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF315194.webp&w=3840&q=75)
![4-OXO-5-(THIOPHEN-2-YLMETHYL)-4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE-3-CARBOXYLIC ACID](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF530938.webp&w=3840&q=75)
![2-(((6-(Difluoromethoxy)-1H-benzo[d]imidazol-2-yl)sulfinyl)methyl)-3,4-dimethoxypyridine 1-oxide](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF545011.webp&w=3840&q=75)
![2-[3,5-Dichloro-4-(4-chlorobenzoyl)phenyl]-1,2,4-triazine-3,5(2H,4H)-dione](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FD434005.webp&w=3840&q=75)
