Moduladores de enzimas
Los moduladores enzimáticos son compuestos que pueden aumentar o inhibir la actividad de las enzimas, regulando así la velocidad de las reacciones bioquímicas. Estos moduladores juegan un papel crítico en el control de las vías metabólicas, la señalización celular y diversos procesos fisiológicos. Los moduladores enzimáticos se utilizan ampliamente en la investigación y el desarrollo de fármacos para estudiar las funciones enzimáticas y desarrollar agentes terapéuticos. En CymitQuimica, ofrecemos una gama completa de moduladores enzimáticos de alta calidad para apoyar su investigación en la regulación enzimática y el descubrimiento de fármacos.
Subcategorías de "Moduladores de enzimas"
Se han encontrado 693 productos de "Moduladores de enzimas"
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Licofelone
CAS:Dual COX/5-LO inhibitor; anti-inflammatory; analgesic
Fórmula:C23H22ClNO2Pureza:Min. 95%Forma y color:PowderPeso molecular:379.88 g/molGefitinib hydrochloride
CAS:RIPK2 protein kinase inhibitor; EGFR inhibitorFórmula:C22H24ClFN4O3·HClPureza:Min. 95%Forma y color:PowderPeso molecular:483.36 g/molAZD 1152
CAS:AZD 1152 is an Aurora kinase inhibitor, which is a type of small-molecule therapeutic agent. It is derived from the pharmaceutical research conducted by AstraZeneca. Its primary mode of action involves the selective inhibition of Aurora B kinase, an enzyme crucial for the regulation of mitosis. By interfering with this enzyme, AZD 1152 disrupts the normal progression of cell division, leading to the inhibition of proliferation and induction of apoptosis in rapidly dividing cells.Fórmula:C26H31FN7O6PPureza:Min. 97 Area-%Forma y color:Slightly Yellow PowderPeso molecular:587.54 g/molCerivastatin sodium
CAS:An inhibitor of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase that reduces total cholesterol and low-density lipoprotein (LDL). Cerivastatin is cardioprotective and anti-atherosclerotic. Cerivastatin inhibits the expression of the atherosclerotic genes monocyte chemoattractant protein-1 (MCP-1) and C-C chemokine receptor type 2 (CCR2), whilst inducing the expression of Kruppel-like factor 2 (KLF2).Fórmula:C26H33FNNaO5Pureza:Min. 98 Area-%Forma y color:PowderPeso molecular:481.53 g/molSU 11274
CAS:MET tyrosine kinase inhibitor; anti-proliferative; pro-apoptoticFórmula:C28H30ClN5O4SPureza:Min. 95%Forma y color:Yellow To Orange SolidPeso molecular:568.09 g/molOmeprazole - Bio-X ™
CAS:Omeprazole is a proton pump inhibitor (PPI) that inhibits the production of gastric acid in the stomach. This is due to Omeprazole binding through a stable disulphide bond to the H+/K+ ATPase enzyme found on parietal cells, and preventing hydrogen ion transport. Consequently, gastric acid secretion is supressed. As a PPI, Omerprazole can be used to treat disorders where gastric acid is over-secreted. Examples of these disorders are gastroesophageal reflux disease (GERD) and peptic ulcer disease.Fórmula:C17H19N3O3SPureza:Min. 95%Forma y color:PowderPeso molecular:345.42 g/molAceclofenac - Bio-X ™
CAS:Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.Fórmula:C16H13Cl2NO4Pureza:Min. 95%Forma y color:PowderPeso molecular:354.18 g/molUNC 4203
CAS:Potent and specific inhibitor of the tyrosine protein kinase Mer precursor (MERTK) with 38-fold selectivity over the FMS-like protein kinase FLT3. UNC 4203 inhibits MERTK with an IC50 value of 2.4 nM and shows favourable pharmacokinetic properties. In vivo experiments in mice showed that UNC 4203 dramatically decreased the phosphorylation of MERTK in bone marrow leukemia cells.Fórmula:C30H44N6OPureza:Min. 95%Forma y color:Yellow PowderPeso molecular:504.71 g/molIrsogladine maleate - Bio-X ™
CAS:Irsogladine is a gastroprotective drug that is used for the treatment of GERD and gastric ulcers. This drug also has antioxidant properties. Irsogladine is a phosphodiesterase-4 inhibitor and increases levels of cAMP. It helps to prevent and heal damage to the stomach lining.Fórmula:C13H11Cl2N5O4Pureza:Min. 95%Forma y color:PowderPeso molecular:372.16 g/molChymostatin
CAS:Inhibitor of chymotrypsinFórmula:C31H41N7O6Forma y color:White To Yellowish SolidPeso molecular:607.7 g/molBAY 607550
CAS:A selective and potent inhibitor of phosphodiesterase 2 (PDE2). Raises cAMP and cGMP levels in neurons, improves social recognition and object memory in murine animals. Reverses anxiolytic effects induced by oxidative stress in mice by blocking cGMP-PKG signaling.
Fórmula:C27H32N4O4Pureza:Min. 95%Forma y color:PowderPeso molecular:476.24236Zotarolimus
CAS:Inhibitor of immunophilin FKBP12 and mTOR signalling with immunosuppressant activity. Zotarolimus inhibits proliferation of endothelial cells and smooth muscle cells and is employed in vascular interventional therapies.Fórmula:C52H79N5O12Pureza:Min. 95%Forma y color:White PowderPeso molecular:966.21 g/molRebamipide - Bio-X ™
CAS:Rebamipide is a gastroprotective agent that is used to treat various gastrointestinal disorders such as gastric ulcers and GERD. This drug’s mechanism of action is not fully understood however, it is thought to exert its effects by promoting the secretion of protective mucus in the stomach and intestine, which helps to create a barrier against stomach acid and other irritants. Additionally, it has antioxidant and anti-inflammatory properties that can help reduce tissue damage.Fórmula:C19H15ClN2O4Pureza:Min. 95%Forma y color:PowderPeso molecular:370.79 g/molThioglycosyl Naphthalimide
CAS:Thioglycosyl Naphthalimide is a highly potent human O-GlcNAcase (hOGA) inhibitor with good selectivity against human β-N-acetylhexosaminidase B (HsHexB).Fórmula:C30H40N4O7SPureza:Min. 95%Peso molecular:600.73 g/molGilteritinib
CAS:Inhibitor of FLT3 and AXL tyrosine kinasesFórmula:C29H44N8O3Pureza:Min. 95%Forma y color:PowderPeso molecular:552.71 g/mol(-)-Huperzine A
CAS:Acetylcholinesterase inhibitor; therapy for Alzheimer's diseaseFórmula:C15H18N2OPureza:(%) Min. 98%Forma y color:PowderPeso molecular:242.32 g/molLY 411575
CAS:Potent inhibitor of γ-secretase. LY 411575 inhibited production of amyloid β (Aβ) peptides with IC50 of 0.078 nM in vitro as well as decreased levels of Aβ40 and Aβ42 amyloids in brain of a mouse model for Alzheimer’s disease. In vitro studies confirmed that LY 411575 inhibited cleavage of Notch receptor at S3 site with IC50 of 0.39 nM, which blocked Notch activation and downstream signalling, leading to apoptosis in primary and immortalized Kaposi's sarcoma cells.Fórmula:C26H23F2N3O4Pureza:Min. 95%Forma y color:SolidPeso molecular:479.48 g/molLovastatin - Bio-X ™
CAS:Lovastatin is an HMG-CoA reductase inhibitor that is used to lower LDL cholesterol levels and to aid in the management of cardiovascular diseases. Animal studies have demonstrated that this drug has vasculoprotective properties.Fórmula:C24H36O5Pureza:Min. 95%Forma y color:PowderPeso molecular:404.54 g/molMRK 560
CAS:γ-secretase inhibitor; reduces amyloid-β in brainÂ
Fórmula:C19H17ClF5NO4S2Pureza:Min. 95%Peso molecular:517.92 g/molRofecoxib - Bio-X ™
CAS:Producto controladoRofecoxib is a non-steroidal anti-inflammatory drug that is used to treat osteoarthritis, acute pain and migraine attacks. This drug is also a COX-2 inhibitor. As a result, it reduces inflammation and pain.Fórmula:C17H14O4SPureza:Min. 95%Forma y color:PowderPeso molecular:314.36 g/mol
