Moduladores de enzimas
Los moduladores enzimáticos son compuestos que pueden aumentar o inhibir la actividad de las enzimas, regulando así la velocidad de las reacciones bioquímicas. Estos moduladores juegan un papel crítico en el control de las vías metabólicas, la señalización celular y diversos procesos fisiológicos. Los moduladores enzimáticos se utilizan ampliamente en la investigación y el desarrollo de fármacos para estudiar las funciones enzimáticas y desarrollar agentes terapéuticos. En CymitQuimica, ofrecemos una gama completa de moduladores enzimáticos de alta calidad para apoyar su investigación en la regulación enzimática y el descubrimiento de fármacos.
Subcategorías de "Moduladores de enzimas"
Se han encontrado 691 productos para "Moduladores de enzimas".
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Milrinone - Bio-X ™
CAS:Milrinone has an application for use in the treatment of heart failure. It has been shown to increase cardiac output and decrease left ventricular end diastolic pressure (LVEDP). Milrinone also increases the amount of oxygen delivered to the tissues by increasing cardiac contractility. Milrinone is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready to use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.Fórmula:C12H9N3OPureza:(%) Min. 95%Forma y color:PowderPeso molecular:211.22 g/molPravastatin sodium
CAS:HMG-CoA reductase inhibitor
Fórmula:C23H35NaO7Pureza:Min. 98 Area-%Forma y color:PowderPeso molecular:446.51 g/molCarfilzomib
CAS:Inhibits proteosomes of class peptide epoxyketone; antineoplastic
Fórmula:C40H57N5O7Pureza:Min. 95%Forma y color:PowderPeso molecular:719.91 g/molAbiraterone - Bio-X ™
CAS:Producto controladoAbiraterone is an anti-cancer drug that has been shown to be effective in treating prostate cancer. It works by blocking the production of testosterone by inhibiting androgen synthesis. Abiraterone does this by inhibiting CYP17A1, which converts cholesterol into pregnenolone, and then into progesterone and testosterone. Furthermore, it binds to the enzyme steroid 5-alpha reductase, which converts testosterone into dihydrotestosterone (DHT). Abiraterone is usually a last resort for patients who have stopped responding to other lines of hormone therapies, which is known as second-line therapy.
Fórmula:C24H31NOPureza:Min. 95%Forma y color:PowderPeso molecular:349.51 g/molNitazoxanide - Bio-X ™
CAS:Nitazoxanide acts as a noncompetitive inhibitor of the pyruvate: ferredoxin/flavodoxin oxidoreductases of various microorganism with Ki values between 2 and 10 μM. Nitazoxanide is clinically relevant for its broad-spectrum action to reduce the growth of bacteria, various parasites, and especially for its efficacy against the pathogen Helicobacter pylori. Nitazoxanide also has been shown to be effective in treating inflammatory bowel disease and acute enteritis caused by bacteria. In 2021, nitazoxanide was tested for the treatment of COVID-19 patients with mild symptoms due to its broad antiviral action.Fórmula:C12H9N3O5SPureza:Min. 90 Area-%Forma y color:PowderPeso molecular:307.28 g/mol4-5-(4-Pyridylmethylamino)pyrazolo1,5-apyrimidin-3-ylbenzamide
CAS:Selective inhibitor of the mutated RET variant RETV804M, which is the anticipated drug-resistant RET mutant that can occur in tumours treated with kinase inhibitors. The compound has a biochemical IC50 of 0.02 µM and selectivity for purified RETV804M over purified RET and KDR of 3.7 and 110, respectively. The efficacy of the compound was shown also in cell cultures with IC50 of 4.4 µM, and cell assay selectivity for RETV804M over RET and KDR of 0.89 and 2.3, respectively.Pureza:Min. 98 Area-%Forma y color:PowderPeso molecular:344.37 g/molA 1070722
CAS:High affinity inhibitor of glycogen synthase kinase GSK-3 with Ki of 0.6 nM. A 1070722 showed favourable characteristics for the penetration across blood brain barrier. A 1070722 was also shown to reduce the phosphorylation of microtubule-associated protein Tau.Fórmula:C17H13F3N4O2Pureza:Min. 95%Forma y color:SolidPeso molecular:362.31 g/molNintedanib ethanesulfonate
CAS:Used for treatment of idiopathic pulmonary fibrosisFórmula:C31H33N5O4•C2H6O3SPureza:Min. 98 Area-%Forma y color:PowderPeso molecular:649.76 g/molDiflunisal
CAS:Diflunisal is a nonsteroidal anti-inflammatory drug (NSAID), which is a synthetic derivative of salicylic acid. It is primarily sourced through chemical synthesis rather than extraction from natural elements. Diflunisal functions by inhibiting the cyclooxygenase (COX) enzymes, specifically COX-1 and COX-2, which play a crucial role in the biosynthesis of prostaglandins. This inhibition results in reduced production of prostaglandins, compounds involved in inflammation and pain signaling pathways.Fórmula:C13H8F2O3Pureza:Min. 98 Area-%Forma y color:White PowderPeso molecular:250.2 g/molBragsin 2
CAS:Inhibitor of BRAG2-mediated activation of Arf GTP-ase. In vitro experiments showed that Bragsin2 inhibits the Arf GTP-ase activation that is mediated by a nucleotide exchange factor BRAG2 in a membrane-dependent manner. Bragsin2 interacts with the PH domain of BRAG2 protein as well as membrane, which prevents the activation of lipidated Arf. Bragsin2 affects the trans-Golgi network and was shown to affect the tumour sphere in breast cancer cell lines.Fórmula:C11H6F3NO5Pureza:Min. 95%Forma y color:SolidPeso molecular:289.16 g/molTrametinib
CAS:Inhibitor of MEK kinase; anti-neoplasticFórmula:C26H23O4N5FIPureza:Min. 95%Forma y color:White PowderPeso molecular:615.39 g/molSD 0006
CAS:SD 0006 is a small-molecule inhibitor, which is synthesized through specialized chemical processes. It functions by selectively inhibiting the cyclooxygenase-2 (COX-2) enzyme, which plays a significant role in the inflammatory pathway. This inhibition reduces the production of pro-inflammatory prostaglandins, ultimately leading to a decrease in inflammation.Fórmula:C20H20ClN5O2Pureza:Min. 95%Peso molecular:397.86 g/molEverolimus
CAS:mTOR kinase inhibitor; rapamycin analog; immunosuppressantFórmula:C53H83NO14Pureza:90%Forma y color:White Off-White PowderPeso molecular:958.23 g/molPerindopril t-butylamine salt - Bio-X ™
CAS:Perindopril t-butylamine salt inhibits the angiotensin converting enzyme (ACE) to prevent the conversion of angiotensin I to angiotensin II. When used in drug formulations, it has been shown to decrease blood pressure in patients with congestive heart failure. Perindopril also has an effect on the renin-angiotensin system, which regulates blood pressure and fluid homeostasis by promoting vasoconstriction and increasing salt and water retention. Perindopril t-butylamine salt is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready to use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.Fórmula:C23H43N3O5Pureza:Min. 98 Area-%Forma y color:PowderPeso molecular:441.61 g/molGDC 0032
CAS:Inhibitor of PI3K kinase isoforms α, δ, and γFórmula:C24H28N8O2Pureza:Min. 95%Peso molecular:460.53 g/molOzagrel hydrochloride
CAS:Thromboxane A2 synthetase inhibitor
Fórmula:C13H12N2O2•HClPureza:Min. 95%Forma y color:PowderPeso molecular:264.71 g/molPitavastatin calcium
CAS:Inhibitor of HMG-CoA reductase
Fórmula:C50H46F2N2O8CaPureza:Min. 95%Forma y color:White Off-White PowderPeso molecular:880.98 g/molNiacinamide
CAS:Vitamin B3; antioxidant; favours cell repairFórmula:C6H6N2OPureza:98.5 To 101.5 Area-%Forma y color:White PowderPeso molecular:122.12 g/molFenoprofen calcium
CAS:Inhibitor of COX-1 and COX-2 cyclooxygenasesFórmula:C30H26CaO6Pureza:Min. 95%Forma y color:PowderPeso molecular:524.62 g/molPF 06409577
CAS:Potent agonist of a1β1γ1 5′-adenosine monophosphate-activated protein kinase (AMPK). It binds to the allosteric drug and metabolite (ADaM) site at the α- and β- subunit interface of AMPK. It has potential for the treatment of diabetic nephropathy. PF 06409577 reduces infections caused by flaviviruses, mediated by changes in the metabolism of lipids in host cells.
Fórmula:C19H16ClNO3Pureza:Min. 95%Forma y color:White/Off-White SolidPeso molecular:341.79 g/mol
