GSK1324726A

CAS: 1300031-52-0

Ref. 3D-ACC03152

Información del producto

• Nombre: GSK1324726A

Descripción

GSK1324726A is a small-molecule drug that can be used to treat cancer. It inhibits the HDAC enzyme, which is required for transcriptional repression of genes involved in tumorigenesis. GSK1324726A has been shown to inhibit the expression of suppressor genes and promote apoptosis in myeloid leukemia cells. This drug also potently inhibits HIV replication in vitro and has shown promising results in clinical studies involving patients with AIDS. GSK1324726A binds to bromodomain proteins, which are domains found on histone proteins that bind to acetylated lysine residues on DNA. These domains are known for their ability to regulate gene expression by binding to acetylated lysine residues on histone proteins and blocking transcriptional activation.

• Marca: Biosynth

Propiedades químicas

• Peso molecular: 434.92 g/mol
• Fórmula: C₂₅H₂₃ClN₂O₃
• Pureza: Min. 95%