4,5,6,7-Tetrahydrofuro[3,2-c]pyridine
CAS: 150322-87-5
Ref. 3D-AGA32287
10mg | A consultar | ||
100mg | A consultar |
Información del producto
4,5,6,7-Tetrahydrofuro[3,2-c]pyridine is a potent and selective inhibitor of class I PI3K (PI3KCA) and class IIA PI3K (PI3KCG/PI3Kδ), which are enzymes that maintain the integrity of cellular membranes. It has been shown to inhibit the kinase activity of these enzymes. 4,5,6,7-Tetrahydrofuro[3,2-c]pyridine has been shown to have anti-cancer effects in vitro and in vivo in preclinical models. 4,5,6,7-Tetrahydrofuro[3,2-c]pyridine also inhibits Jak2 kinases and JAK1 with similar potency to its inhibition of PI3KCG/PI3Kδ. This compound has demonstrated high potency and selectivity over other kinases such as ER
Propiedades químicas
Consulta técnica sobre: 3D-AGA32287 4,5,6,7-Tetrahydrofuro[3,2-c]pyridine
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