Pitolisant hydrochloride

CAS: 903576-44-3

Ref. 3D-FC153335

Información del producto

• Nombre: Pitolisant hydrochloride
• Sinónimos: 1-[3-[3-(4-Chlorophenyl)propoxy]propyl]piperidine hydrochloride, Ciproxidine, Bf2649
• CAS: 903576-44-3

Descripción

Pitolisant is an inverse agonist and antagonist of the histamine (H3) receptor. It acts as an allosteric modulator of the H3 receptor to increase the activity of histamine at the M1 receptor. Pitolisant has been used in the treatment of narcolepsy, schizophrenia and Alzheimer's disease. Its mechanism of action involves binding to the amide group on histamine, which increases its affinity for the H3 receptor and enhances its activity at this site. Pitolisant has been shown to improve cognitive ability and reduce fatigue in patients with Alzheimer's disease.

• Marca: Biosynth

Propiedades químicas

• Peso molecular: 332.31 g/mol
• Fórmula: C₁₇H₂₆ClNO·HCl
• Pureza: Min. 95%
• Color/Forma: White Off-White Powder