Sumatriptan N-oxide

CAS: 212069-94-8

Ref. 3D-FS27975

Información del producto

• Nombre: Sumatriptan N-oxide
• Sinónimos: 3-[2-(Dimethyloxidoamino)ethyl]-N-methyl-1H-indole-5-methanesulfonamideGR 112504

Descripción

Sumatriptan succinate is a triptan drug that is used to treat migraines. It has been shown to have high specificity for 5-HT1 receptors and low affinity for 5-HT2A, 5-HT2B, or 5-HT2C receptors. Sumatriptan succinate is rapidly metabolized by monoamine oxidase type A (MAO-A) in the liver to form sumatriptan. The major metabolite of sumatriptan is N-oxide (sumatriptan N-oxide). Sumatriptan N-oxide has been shown to be less potent than sumatriptan at inhibiting the release of inflammatory substances from mast cells in vitro.

• Marca: Biosynth

Propiedades químicas

• Peso molecular: 311.4 g/mol
• Fórmula: C₁₄H₂₁N₃O₃S
• Pureza: Min. 95%