Sarafotoxin 6c
CAS: 121695-87-2
Ref. 3D-FS73598
1mg | A consultar | |
50µg | A consultar | |
100µg | A consultar | |
250µg | A consultar | |
500µg | A consultar |
Información del producto
- Srtx-C
- Sarafotoxin S6C (Atractaspis Engaddensis)
- Sarafotoxin S6C, Atractaspsis Engaddensis
- Sarafotoxin 6C
- Sarafotoxin C
- Sarafotoxin C (Atractaspis Engaddensis)
- Cys-Thr-Cys-Asn-Asp-Met-Thr-Asp-Glu-Glu-Cys-Leu-Asn-Phe-Cys-His-Gln-Asp-Val-Ile-Trp
Sarafotoxin 6c is a potent, selective, and noncompetitive endothelin-1 receptor antagonist. Sarafotoxin 6c binds to the extracellular domain of the endothelin-1 receptor and prevents endothelin-1 from binding, thereby inhibiting its activity. Sarafotoxin 6c has been shown to inhibit the production of intracellular Ca2+ in mesenteric artery cells. Sarafotoxin 6c also inhibits the enzymatic inactivation of endothelin-1 by carboxypeptidases and calpains. Sarafotoxin 6c has been shown to be effective against a number of infectious diseases including myocardial infarction.
Propiedades químicas
Consulta técnica sobre: 3D-FS73598 Sarafotoxin 6c
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