N2-Methyl-N4-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine

CAS: 2407433-00-3

Ref. 3D-HWD43300

Información del producto

• Nombre: N2-Methyl-N4-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine
• Marca: Biosynth

Descripción

N2-Methyl-N4-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine is an inhibitor of the alpha subunit of the protein phosphatase 2A. This drug binds to the active site and inhibits the dephosphorylation of phosphoprotein substrates. N2-Methyl-N4-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-- diamine has been shown to inhibit ion channels that are regulated by Ca++ concentration. It also inhibits the activation of protein kinase C by phorbol esters and has been used in pharmacological studies as a ligand for receptor binding studies.

Propiedades químicas

• Peso molecular: 382.42 g/mol
• Fórmula: C₂₁H₁₈N₈
• Pureza: Min. 95%